DE LA OCIEDAD ESPAÑOLA QUÍMICA ERAPÉUTICA30-13:45 Patricia M. R. Pereira (University of Aveiro,...
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9:00-9:30 REGISTRATION 9:30-9:45 OPENING CEREMONY 9:45-10:15 Inaugural Lecture (Coaching) Dr. Óscar Delgado (Janssen, Spain) “Chasing drugs instead of molecules: chemistry and the pharmaceutical industry” 10:15-10:30 Carles Galdeano (University of Dundee, UK) “Targeting the VHL: HIF-1 α protein-protein interaction with small-molecules chemical probes” 10:30-10:45 Eleni Pitta (University of Antwerp, Belgium & GSK, Spain) “Hit to lead optimization of novel quinoloxyacetamide derivatives against mycobacterium tuberculosis” 10:45-11:00 Ana María García (Centro de Investigaciones Biológicas, CSIC, Spain) “Sulfide-like PDE7 inhibitors: in vitro metabolic oxidation study using rat liver microsomes” 11:00-11:15 María Gómez Cañas (Universidad Complutense Madrid, Spain) “Biological characterization of PM226, achromenoisoxazole, as a selective CB 2 receptor agonist with antiinflammatory/neuroprotective profile” 11:15-12:15 POSTER SESSION/COFFEE BREAK 12:15-12:45 Invited Lecture Dr. Manuel Guzmán (Universidad Complutense Madrid, Spain) “Cannabinoid receptors as potential antitumor targets” 12:45-13:00 Laura Aramburu (Universidad de Salamanca, Spain) “Novel sulfoxides and sulfones as tubulin polymerization inhibitors” 13:00-13:15 Marta Acebron (Centro Nacional de Investigaciones Oncológicas, CSIC, Spain) “Fragment based ligand discovery for local adhesion kinase” 13:15-13:30 Sofía Salazar (University of Porto, Portugal) “New potential selective activators of caspase-7 identified using the yeast screening assay” II SIMPOSIO DE JÓVENES INVESTIGADORES DE LA SOCIEDAD ESPAÑOLA DE QUÍMICA TERAPÉUTICA 12 de junio de 2015, 09:00h Salón de actos de la Sede Central CSIC c/ Serrano 117, Madrid Scientific committee
Transcript of DE LA OCIEDAD ESPAÑOLA QUÍMICA ERAPÉUTICA30-13:45 Patricia M. R. Pereira (University of Aveiro,...
9:00-9:30 REGISTRATION
9:30-9:45 OPENING CEREMONY
9:45-10:15
Inaugural
Lecture
(Coaching)
Dr. Óscar Delgado (Janssen, Spain)
“Chasing drugs instead of molecules: chemistry and the pharmaceutical industry”
10:15-10:30 Carles Galdeano (University of Dundee, UK)
“Targeting the VHL: HIF-1α protein-protein interaction with small-molecules chemical probes”
10:30-10:45
Eleni Pitta (University of Antwerp, Belgium & GSK, Spain)
“Hit to lead optimization of novel quinoloxyacetamide derivatives against mycobacterium
tuberculosis”
10:45-11:00 Ana María García (Centro de Investigaciones Biológicas, CSIC, Spain)
“Sulfide-like PDE7 inhibitors: in vitro metabolic oxidation study using rat liver microsomes”
11:00-11:15
María Gómez Cañas (Universidad Complutense Madrid, Spain)
“Biological characterization of PM226, achromenoisoxazole, as a selective CB2receptor
agonist with antiinflammatory/neuroprotective profile”
11:15-12:15 POSTER SESSION/COFFEE BREAK
12:15-12:45
Invited
Lecture
Dr. Manuel Guzmán (Universidad Complutense Madrid, Spain)
“Cannabinoid receptors as potential antitumor targets”
12:45-13:00 Laura Aramburu (Universidad de Salamanca, Spain)
“Novel sulfoxides and sulfones as tubulin polymerization inhibitors”
13:00-13:15 Marta Acebron (Centro Nacional de Investigaciones Oncológicas, CSIC, Spain)
“Fragment based ligand discovery for local adhesion kinase”
13:15-13:30 Sofía Salazar (University of Porto, Portugal)
“New potential selective activators of caspase-7 identified using the yeast screening assay”
II SIMPOSIO DE JÓVENES INVESTIGADORES DE LA SOCIEDAD ESPAÑOLA DE QUÍMICA TERAPÉUTICA
12 de junio de 2015, 09:00h
Salón de actos de la Sede Central CSIC
c/ Serrano 117, Madrid Scientific committee
13:30-13:45
Patricia M. R. Pereira (University of Aveiro, Portugal)
“The dual functionality of phosphonate-appended phthalocyanines: inhibitors of urokinase
plasminogen activator and anticancer photodynamic agents”
13:45-14:00 Ana C. S. Lobo (University of Coimbra, Portugal)
“The effect of photodynamic therapy with LUZ11 on tumour metastases”
14:00-14:15
Clara Pérez Peinado (Universitat Pompeu Fabra, Spain)
“Structure-activity studies of crotalicidin and analogs, antimicrobial and antitumoral peptides
from rattlesnake venom”
14:15-16:00 LUNCH BREAK
16:00-16:15
Mery Santivañez Veliz (Universidad de Navarra, Spain)
“Structure-activity studies of crotalicidin and analogs, antimicrobial and antitumoral peptides
from rattlesnake venom”
16:15-16:30 Alejandra Carriles Linares (Instituto Química Física Rocasolano, CSIC, Spain)
“Novel drug design strategies for trypanosomatid-causing diseases: a structural approach”
16:30-16:45
Ana María Gamo Albero (Instituto Química Médica, CSIC, Spain)
“α/β3-peptide foldamers: potent dimerization inhibitors of Leishmania infantum trypanothione
reductase with improved proteolytic stability”
16:45-17:00
Montserrat Nácher (Centro de Investigaciones Biológicas, CSIC, Spain)
“Photodynamic therapy as an alternative for cutaneous leishmaniasis. Metal-organic Ru(II)
complexes as new photosensitizer leads”
17:00-17:45 POSTER SESSION
17:45-18:00
Verónica Ortiz de Elguea (Universidad del País Vasco, Spain)
“Ready access to biologically active heterocycles via palladium-catalyzed alkenylation
reactions”
18:00-18:15
Jennifer Enrich Bengoa (University of Aix-Marseille, France)
“MicroRNA involvement in the Hutchinson-Gliford progeria physiopathology by the inhibition of
autophagic progerin degradation?”
18:15-18:30 Alejandro Escobar Peso (Instituto Química Orgánica General, CSIC, Spain)
“New drugs for ageing related diseases”
18:30-19:00 FINAL REMARKS & AWARDS
19:00 CLOSING EVENT: drinks and tapas
La duración de las comunicaciones orales será de
10 min de exposición + 5 min para preguntas.
Location
Salón de actos de la Sede Central del CSIC C/Serrano, 117 28006, Madrid
República Argentina, línea 6 Gregorio Marañón, líneas 7 y 10
C/ Serrano 111, líneas 16, 19 y 51
