Download - ChemInform Abstract: A Novel and Efficient 2,4,6-Trisubstituted Pyridine Ring Synthesis via α-Benzotriazolyl Ketones.

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2000 pyridine derivatives

pyridine derivativesR 0380

11 - 140A Novel and Efficient 2,4,6-Trisubstituted Pyridine Ring Synthesisvia α-Benzotriazolyl Ketones. — Reaction of chalcones (I) withα-benzotriazolylketones yields 2,4,6-triarylated pyridines. The proposedintermediate 1,5-diketone type (VIII) can be prepared independently. — (KA-TRITZKY, ALAN R.; ABDEL-FATTAH, ASHRAF A. A.; TYMOSHENKO,DMYTRO O.; ESSAWY, SAMY A.; Synthesis (1999) 12, 2114-2118; Dep.Chem., Univ. Fla., Gainesville, FL 32611, USA; EN)

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