SYNTHESIS Vol 41 - 2009
SPIS TREŚCI
No 1
1 Enantioselective Preparation of β2-Amino Acid Derivatives for β-Peptide Synthesis D Seebach A K Beck S Capone G Deniau U Grošelj E Zass
33 Discoveries from the Abyss The Abyssomicins and Their Total Synthesis K C Nicolaou S T Harrison J S Chen
43 α-Metallated O-2-Alkenyl Carbamates Synthetic Equivalents of Chiral Homoenolates and Materials for Asymmetric Homoaldol Reaction D Hoppe
56 Direct CarbonndashCarbon Bond Formation via Soft Enolization of Thioesters An Operationally Simple Mannich Addition Reaction J M Yost M R Garnsey M C Kohler D M Coltart
59 Synthesis of Norbornane-Bridged Diporphyrins via Palladium-Catalyzed [3+2] Annulation Strategy M Mizumura H Shinokubo A Osuka
62 Synthesis and Olfactory Evaluation of (4aR8aR)-118a-Trimethyldecahydronaphthalen-4a-ol A cis-Decalol Intersection Structure of (ndash)-Patchoulol and (5R6S)-116-Trimethylspiro[45]decan-6-ol A Jahnke C Burschka R Tacke P Kraft
69 Synthesis of Novel Halogenated 4(1H)-Quinolones by Thermolysis of Arylaminomethylene-13-dioxane-46-diones S Rotzoll H Reinke C Fischer P Langer
79 Synthesis of Functionalized Oligophenylenes and Oligoarylenes Bearing Heteroaryl Groups I Wallmann G Schnakenburg A Luumltzen
85 Synthesis of Benzo[b]furans by PalladiumndashNHC Catalyzed Ring Closure of o-Bromobenzyl Ketones J Faragoacute A Kotschy
91 Intermolecular CndashH and SindashH Insertion Reactions with Halodiazoacetates H T Bonge T Hansen
97 The Direct Synthesis of Unsymmetrical Vicinal Diamines from Terminal Alkynes A Tandem Sequential Approach for the Synthesis of Imidazolidinones A V Lee M Sajitz L L Schafer
105 Synthesis of 2-Deoxyuridine and 2-Deoxycytidine Nucleosides Bearing Bipyridine and Terpyridine Ligands at Position 5 L Kalachova R Pohl M Hocek
113 Inverse-Electron-Demand DielsndashAlder Reactions of N-(Heteroarylsulfonyl)-1-aza-13-dienes Catalyzed by Chiral Lewis Acids J Esquivias I Alonso R Goacutemez Arrayaacutes J C Carretero
127 Coordination-Induced Intramolecular Double Cyclization Synthesis of Boron-Bridged Dipyridylvinylenes and Dithiazolylvinylenes Q Zhao H Zhang A Wakamiya S Yamaguchi
133 An Enantiospecific Approach to Triazolylalanine Derivatives C E Jamookeeah C D Beadle J P A Harrity
138 Double Couplings of Dibromothiophenes Using Boronic Acids and Boronates S Varello S T Handy
143 Synthesis of Fmoc-Pro-Hyp(TBDPS)-Gly-OH and Its Application as a Versatile Building Block for the Preparation of Collagen Model Peptides R S Erdmann H Wennemers
148 Complementary Reactions of Allylic Carbamates Using Palladium(II) Formation of Oxazolidinones or Allylic Amides from a Common Precursor S D R Christie A D Warrington C J Lunniss
155 Thermal Amination of 26-Dihalopyridines by Sterically Demanding Amines A Faust O Wolff S R Waldvogel
160 The Thermal Amidation of Carboxylic Acids Revisited L J Gooszligen D M Ohlmann P P Lange
XVII Instructions for Authors XXIII Forthcoming Articles
No 2 165 Selected Synthetic Strategies to Spirocyclics S Kotha A C Deb
K Lahiri E Manivannan 194 Effective Catalytic Activity of the Hydrated Gold Catalyst NaAuCl42H2O To
Construct Highly Fused Cyclopentenones S Karmakar A Kim C H Oh
199 Efficient Synthesis of an Allose-Containing Analogue of the Phytoalexin-Elicitor Glucohexaose and Its Dodecyl Glycoside H Ma D Qiu X Mei J Ning Q Zhao Y Li
205 Synthesis of 14-Benzodiazepine-25-diones Using an Ionic Liquid as a Soluble Support H Xie C Lu G Yang Z Chen
211 A Facile Synthesis of Thioalkyl- and Di(thioalkyl)-Substituted Bipyridines D Chen R De D L Mohler
217 Diastereoselective Synthesis of Dimethyl (4R4aR7aR)-1-Aryl-6-benzoyl-4a-methyl-5-oxo-144a556-hexahydrospiro[pyrazole-47-pyrrolo[34-c]pyridazine]-37a(1H)-dicarboxylates U Uršič U Grošelj A Meden J Svete B Stanovnik
227 Synthesis of 3-Acylpyrroles 3-(Alkoxycarbonyl)pyrroles 1567-Tetrahydro-4H-indol-4-ones and 3-Benzoylpyridines Based on StaudingerndashAza-Wittig Reactions of 13-Dicarbonyl Compounds with 2- and 3-Azido-11-dialkoxyalkanes E Bellur M A Yawer I Hussain A Riahi O Fatunsin C Fischer P Langer
243 Regioselective Synthesis of Functionalized Biaryls Based on the First [3+3] Cyclocondensations of 4-Aryl-13-bis(trimethylsilyloxy)buta-13-dienes M Adeel M A Rashid N Rasool R Ahmad A Villinger H Reinke C Fischer P Langer
251 Synthesis of Functionalized Bicyclic Precursors of Heptulosonic Acid Analogues H Filali S Ballereau F O Chahdi M Baltas
257 Efficient Regio- and Stereoselective Synthesis of 5-Alkyl(aryl)idene- and 5-[Iodoalkyl(aryl)idene]-1H-pyrrol-2(5H)-ones via Electrophilic Cyclization K Cherry A Duchecircne J Thibonnet J-L Parrain E Anselmi M Abarbri
271 PdCu-Catalyzed Oxidative CndashH Alkenylation of Imidazo[12-α]pyridines J Koubachi S Berteina-Raboin A Mouaddib G Guillaumet
277 A Convenient Synthesis of Unsymmetrical Pinacols by Coupling of Structurally Similar Aromatic Aldehydes Mediated by Low-Valent Titanium X-F Duan J-X Feng G-F Zi Z-B Zhang
283 A Method for the Selective Protection of Aromatic Amines in the Presence of Aliphatic Amines V Perron S Abbott N Moreau D Lee C Penney B Zacharie
290 Synthesis and Antiviral Evaluation of (ndash)-3-Methylcarbovir (ndash)-3-Methylabacavir and Modified Purine Analogues P Breacutemond G Audran H Monti E De Clercq C Pannecouque
297 Regioselective Synthesis of 2-(Aryloxythio)benzoates by the First [3+3] Cyclizations of 3-Aryloxythio-1-silyloxybuta-13-dienes with 3-Alkoxy-2-en-1-ones I Iqbal M Imran A Villinger P Langer
306 Molybdenum(VI) Dichloride Dioxide Catalyzed Conversion of b-Hydroxycarbonyls into a-Bromo 13-Dicarbonyls by N-Bromosuccinimide K Jeyakumar D K Chand
311 A Short Route to the Synthesis of Pyrrolocoumarin and Pyrroloquinolone Derivatives by Sonogashira Cross-Coupling and Gold-Catalyzed Cycloisomerization of Acetylenic Amines K C Majumdar B Chattopadhyay S Samanta
318 Aspects of the Synthesis of an Exceptionally Preorganized Self-Immolative SpacerndashPhenolate Unit M Waibel X-B Zhang J Hasserodt
325 Design and Efficient Synthesis of Amino Acid Derived 2-Substituted Imidazoles by Palladium-Catalyzed Cross-Coupling Reactions A Marek J Kulhaacutenek F Bureš
332 A Convenient Preparation of Di-p-chlorobenzyl Azodicarboxylate (DCAD) for Mitsunobu Couplings B R Taft E C Swift B H Lipshutz
335 Enantioselective Rhodium-Catalyzed Alkylative Desymmetrization of 35-Dimethylglutaric Anhydride M J Cook T Rovis
XIII Forthcoming Articles
No 3 339 Intermolecular Addition Reactions of N-Acyliminium Ions (Part I)
A Yazici S G Pyne 369 Desulfurization of Thioamides into Amides with H2O2ZrCl4 Reagent System
K Bahrami M M Khodaei Y Tirandaz 372 Total Synthesis of (plusmn)-1345-Tetragalloylapiitol R M Patel
N P Argade 375 A Convenient Synthesis of 4-Hydroxy-2-oxo-12-dihydro-18-
naphthyridine-3-carboxamide Derivatives K Kobayashi D Iitsuka S Fukamachi H Konishi
379 Intramolecular Ketalization of Functionalized 7-Norbornenols L A Paquette J D Pettigrew
385 Ring Contraction of 12-Dihydronaphthalenes Promoted by Thallium(III) in Acetonitrile A Diastereoselective Approach to Indanes H M C Ferraz V M T Carneiro L F Silva Jr
389 Regio-Controlled Nucleophilic Attack of 3-Thiaisatoic Anhydride by α-Amino Acids One-Pot Synthesis of 3-(2-Thienyl)imidazolidine-24-dione and 34-Substituted Thieno[23-e][14]diazepine-25-dione Analogues Y Brouillette G Sujol J Martinez V Lisowski
395 The Unprecedented Cobalt-Catalysed Oxidative Glaser Coupling under Reductive Conditions G Hilt C Hengst M Arndt
399 Nucleophilic Addition of 4-Hydroxycoumarin to BaylisndashHillman Acetate Adducts C Raji Reddy N Kiranmai K Johny M Pendke P Naresh
403 Palladium-Mediated Heck Reaction to the Synthesis of 3-Substituted Indoles and Indolones K C Majumdar S Chakravorty P K Shyam A Taher
409 Synthesis of Bicyclo[310]hexan-2-ones by Manganese(III) Oxidation in Ethanol K Asahi H Nishino
424 High Regio- and Stereoselective Synthesis of (Z)- or (E)-N-Acryl Butenedioic Monoimide Derivatives by a Multicomponent Reaction F Sha Y Lin X Huang
431 The First Synthesis of Allyl Isonitriles from BaylisndashHillman Adducts and Their Application in the Synthesis of Substituted Imidazo[12-α]pyridines and Tetraazadibenzoazulenes M Nayak S Kanojiya S Batra
438 One-Pot Three-Step Synthesis of Pyrazinothienopyrimidines Using Tandem Aza-WittigElectrocyclic Ring Closure G Blanco A Fernaacutendez-Mato J M Quintela C Peinador
445 Synthesis of Biaryls Fluorenones Cyclopenta[def]phenanthren-4-ones and Benzophenones Based on Formal [3+3] Cyclocondensations of 13-Bis(silyloxy)buta-13-dienes with 3-(Silyloxy)-2-en-1-ones S Reim M Lau M Adeel I Hussain M A Yawer A Riahi Z Ahmed C Fischer H Reinke P Langer
464 Diastereoselective Synthesis of α-Stabilized Phosphorus Ylides via a Four-Component Reaction A Alizadeh N Zohreh L-G Zhu
469 Stereoselective Synthesis of Alkynyl Vinyl Chalcogenides via HornerndashWittig Reaction C C Silveira F Rinaldi R C Guadagnin A L Braga
474 Stereoselective Preparation of C1ndashC10 and C11ndashO14 Fragments of Narbonolide Exploiting the Versatility of Thiazolidinethione Chiral Auxiliary C P Narasimhulu P Das
483 Efficient Catalytic Activity of CopperAluminum Hydrotalcite in Diaryl Ether Synthesis B Sreedhar R Arundhathi M A Reddy M L Kanatm
488 On-Resin Click-Glycoconjugation of Peptoids A S Norgren C Budke Z Majer C Heggemann T Koop N Sewald
495 A Simple and Efficient Preparation of Novel Formaldehyde Derivatives R Hartung G Golz S Schlaf G Silvennoinen K Polborn P Mayer H R Pfaendler
502 2-Oxazol-5-ylethanones by Consecutive Three-Component AmidationndashCouplingndashCycloisomerization (ACCI) Sequence E Merkul O Grotkopp T J J Muumlller
508 SuzukindashMiyaura Cross-Couplings Mediated by trans-PdBr(N-Succ)(PPh3)2 A Convenient Synthetic Method for Diarylmethanes and Aryl(heteroaryl)-methanes I J S Fairlamb P Sehnal R J K Taylor
511 Modern Reduction Methods Edited by P G Andersson and I J Munslow Reviewed by Siegfried R Waldvogel
512 Addendum and Erratum XIII Forthcoming Articles
No 4 513 Intermolecular Addition Reactions of N-Acyliminium Ions (Part II)
A Yazici S G Pyne 542 A Simple Practical Method for the Synthesis of 46-Dimethoxy-135-
triazin-2(1H)-one Using Dimethylamine-Functionalized Solid-Phase Reagents K Hioki K Ohshima Y Sota M Tanaka M Kunishima
545 Conjugation-Amenable Tetrasaccharide of the Side Chain of the Major Glycoprotein of the Bacillus anthracis Exosporium A Large-Scale Preparation S Hou P Kovaacuteč
551 Reductive Amination ndash A Convenient Method for Generating Diverse Mono-Functionalised 5101520-Tetraphenyl Porphyrins C Welch S J Archibald R W Boyle
557 Highly Regioselective Preparation of 13-Dioxolane-4-methanol Derivatives from Glycerol Using Phosphomolybdic Acid N W Fadnavis R Gowrisankar G Ramakrishna M K Mishra G Sheelu
561 Rapid Synthesis of 3-Aminoisoquinoline-5-sulfonamides Using the BuchwaldndashHartwig Reaction N Proisy S Taylor A Nelson I Collins
567 Synthesis of Divalent 22-Linked Mannose Derivatives by Homodimerization F S Ekholm M Polaacutekovaacute A J Pawłowicz R Leino
577 Efficient Synthesis of Substituted Cyclic α-Aminophosphonates I L Odinets O I Artyushin N Shevchenko P V Petrovskii V G Nenajdenko G-V Roumlschenthaler
583 Methylated Imidazolinium-Dithiocarboxylates Two Representatives of a New Class of Ionic Liquids A Blanrue R Wilhelm
587 An Efficient Route to 1-Vinylpyrrole-2-carbaldehydes A I Mikhaleva A V Ivanov E V Skitalrsquotseva I A Ushakov A M Vasilrsquotsov B A Trofimov
591 A Regioselective Route to 5-Substituted Isoxazole- and Isoxazoline-3-phosphonates P Conti A Pinto L Tamborini P Dunkel V Gambaro G L Visconti C De Micheli
597 Solvent-Free One-Pot Conjugate Addition of Benzyl Bromides to β-Nitroalkenes Mediated by Magnesium Powder W Shi J-X Wang
602 Synthesis of 234-Trideoxy-44-difluoro-D-ribo-hexopyranose Adenosines J Xu X Zhang X-L Qiu F-L Qing
609 Synthesis of anti-27-Disubstituted Norbornadienes G C Tsui P Le Marquand A Allen W Tam
620 Novel Peptide Mimetic Inhibitors of Hepatitis C Serine Protease Derived from Isomannide T G Barros S Pinheiro J S Williamson A Tanuri H S Pereira R M Brindeiro J B A Neto O A C Antunes E M F Muri
627 A Practical Synthesis of α-Substituted tert-Butyl Acrylates from Meldrumrsquos Acid and Aldehydes C G Frost S D Penrose R Gleave
636 A New Class of Troumlgerrsquos Base Analogues Bearing Spiro[45] Lactone Straps A B Mahon D C Craig A C Try
643 A New Approach to Di- and Tetrasubstituted 23-Dihydropyridin-4(1H)-ones through Aza-DielsndashAlder Reaction Promoted by Silicon Tetrachloride A Massa V de Sio R Villano M R Acocella L Palombi G Sellitto A Peduto R Filosa P De Capraris A Scettri
650 Palladium-Catalysed Direct Arylation of Sydnones A Rodriguez W J Moran
655 Synthesis of (ndash)-Monomorine I R W Bates P Song 660 Cobalt(II) Chloride HexahydratendashDiisopropylamine Catalyzed Mild and
Chemoselective Reduction of Carboxylic Esters with Sodium Borohydride A R Jagdale A S Paraskar A Sudalai
665 Synthesis of Bi- and Tricyclic αβ-Unsaturated Lactams as Potential Michael Acceptors Starting from Heterocyclic Imines K Schulz M Watzke K Johannes P Ullrich J Martens
674 An Expedient Synthesis of Bis-Fused Benzofuran and a Two-Directional Ring-Closing Metathesis for the Synthesis of Bisbenzoxepines and Bisbenzoxocines K C Majumdar B Chattopadhyay S Chakravorty
681 Palladium-Catalyzed Cross-Couplings of Unsaturated Halides Bearing Relatively Acidic Hydrogen Atoms with Organozinc Reagents Z Dong G Manolikakes J Li P Knochel
687 Synthesis of Enantioenriched aa-Disubstituted Cyclopentenes Catalyzed by N-Heterocyclic Carbenes E M Phillips M Wadamoto K A Scheidt
XVII Forthcoming Articles
No 5 691 Transannulation Reactions in the Synthesis of Natural Products
P A Clarke A T Reeder J Winn 710 Synthesis of DL-erythro-Sphingosine Using a Tethered
Aminohydroxylation Reaction as the Key Step J A Morales-Serna Y Diacuteaz M I Matheu S Castilloacuten
713 Convenient Multigram Synthesis of 4-Chloropyridine-26-dicarbonyl Dichloride K Mitsui J R Parquette
715 A Novel and Efficient Synthesis of Dihydrexidine J P Cueva D E Nichols
721 Synthesis of 57-Dichloro-6-azaindoles and Functionalization via a Highly Selective LithiumndashChlorine Exchange N Lachance L-P Bonhomme-Beaulieu P Joly
731 A Convenient Synthesis of Fluorinated Pyrazolo[34-b]pyridine and Pyrazolo[34-d]pyrimidine Nucleosides V O Iaroshenko D V Sevenard A Kotljarov D M Volochnyuk A O Tolmachev V Y Sosnovskikh
741 Diastereoselective Synthesis of γ-Amino Acids and Their Derivatives from Nitroethane via Intermediacy of 56-Dihydro-4H-12-oxazines Bearing the CH2CH(CO2Me)2 Substituent at C3 A Y Sukhorukov A V Lesiv Y A Khomutova S L Ioffe
755 Synthesis of a New Pyrrolopyridoindole and Its Pyrrolopyridobenzimidazole Regioisomer F Bouchikhi M Sassatelli F Anizon M Prudhomme P Moreau
759 Practical Syntheses of Sphingosine-1-Phosphate and Analogues V Blot U Jacquemard H-U Reissig B Kleuser
767 A Facile Synthetic Route towards Substituted Thieno[32-e]indoles W Van Snick W Nulens S Jambon W Dehaen
775 Microwave-Assisted One-Pot Synthesis of (Aminoalkyl)naphthols and (Aminoalkyl)quinolinols by Using Ammonium Carbamate or Ammonium Hydrogen Carbonate as Solid Ammonia Source I Szatmaacuteri F Fuumlloumlp
779 Enantioselective Synthesis of Flavan-3-ols Using a Mitsunobu Cyclization K Krohn I Ahmed M John 787 Synthesis of a Novel γ-Folic AcidndashNτ-Histidine Conjugate Suitable for
Labeling with 99mTc and 188Re C Sparr U Michel R E Marti C Muumlller R Schibli R Moser V Groehn
793 Palladium-Catalyzed Intramolecular Biaryl Coupling A Highly Efficient Avenue for Benzannulated Pyranoquinolines and Julolidine Derivatives K C Majumdar A Taher P Debnath
801 Preparation of NN-Dimethyl-N-Arylureas Using SS-Dimethyl Dithiocarbonate as a Carbonylating Reagent I Degani R Fochi C Magistris M Migliaccio
809 Versatile Selective α-Carboxylic Acid Esterification of N-Protected Amino Acids and Peptides by Alcalase T Nuijens C Cusan J A W Kruijtzer D T S Rijkers R M J Liskamp P J L M Quaedflieg
815 Efficient Palladium-Catalyzed Amination of Aryl Chlorides Using Dicyclohexylamino[(26-dimethyl)morpholino]phenylphosphine as a PN2 Ligand S-E Park S B Kang K-J Jung J-E Won S-G Lee Y-J Yoon
824 A Clean Facile and Stereospecific Synthesis of α-Oxoketene OS-Acetals in Water Y Li Q Zhang X Cheng Q Liu X Xu
829 Sonogashira Cross-Coupling Reactions and Construction of the Indole Ring System Using a Robust Silica-Supported Palladium Catalyst E Tyrrell L Whiteman N Williams
836 Synthesis of Angular 78-Pyridazinocoumarins via the Transformation of a Hydroxy Group into a Carbonyl Group A Kotali I S Lafazanis P A Harris
841 Synthesis of New Cyclic and Acyclic 5-Halouridine Derivatives as Potential Antiviral Agents M F Elshehry J Balzarini C Meier
848 Dendritic Triphenylmethylium and Tetraphenylmethane Compounds H Meier S Kim A Oehlhof
853 Synthesis of Homoallylic Alcohols via Lewis Acid Assisted Enantioselective Desymmetrization B Yu F Menad N Isono M Lautens
860 Diastereoselective Synthesis of 123-Trisubstituted Indanes via Rhodium(I)-Catalyzed Tandem Conjugate Additions C Navarro A G Csaacutekyuml
864 Bakerrsquos Yeast for Sweet Dough Enables Large-Scale Synthesis of Enantiomerically Pure Bicyclo[331]nonane-26-dione C J Wallentin E Orentas E Butkus K Waumlrnmark
868 Addendum and Erratum XV Forthcoming Articles
No 6 869 Stereoselective Transformations of meso Bicyclic Hydrazines Versatile
Access to Functionalized Aminocyclopentanes C Bournaud F Chung A P Luna M Pasco G Errasti T Lecourt L Micouin
888 Synthesis of Glycoaminoxy Acids as Novel Sugar Building Blocks A Malapelle R Ramozzi J Xie
891 Electrophilic ipso-Halocyclization of N-Arylpropynamides with Polyfluoroalkyl Alcohols Selective Synthesis of 8-(Polyfluoroalkoxy) azaspiro[45]trienes Z-Q Wang B-X Tang H-P Zhang F Wang J-H Li
903 Electrooxidation of Alcohols in N-Oxyl-Immobilized Silica GelWater Disperse System Approach to Totally Closed System M Kuroboshi K Goto H Tanaka
909 Synthetic Routes to Aminotriamantanes Topological Analogues of the Neuroprotector Memantinereg A A Fokin A Merz N A Fokina H Schwertfeger S L Liu J E P Dahl R K M Carlson P R Schreiner
913 Parallel Synthesis of Drug-like 5-Amino-Substituted 124-Thiadiazole Libraries Using Cyclization Reactions of a Carboxamidine Dithiocarbamate Linker J Y Park I A Ryu J H Park D C Ha Y-D Gong
921 Copper-Catalyzed Selective S-Arylation of 12-Bis(o-amino-1H-pyrazolyl) Disulfides with Arylboronic Acids P-S Luo F Wang J-H Li R-Y Tang P Zhong
929 2-Iodoxybenzoic AcidTetraethylammonium BromideWater An Efficient Combination for Oxidative Cleavage of Acetals C Kuhakarn W Panchan S Chiampanichayakul N Samakkanad M Pohmakotr V Reutrakul T Jaipetch
935 Synthesis of Quinonoid Analogues of Diospyrin S Sagar I R Green 941 A One-Pot Method for the Iodination of Aryl Amines via Stable Aryl
Diazonium Silica Sulfates Under Solvent-Free Conditions A Zaroi A R Hajipour L Khazdooz
945 Poly(NN-dichloro-N-ethylbenzene-13-disulfonamide) and NNNN-Tetrachlorobenzene-13-disulfonamide as Novel Reagents for the Synthesis of N-Chloroamines Nitriles and Aldehydes R Ghorbani-Vaghei H Veisi
951 Synthesis of an (R)-Garner-type Aldehyde from L-Serine Useful Building Block for a (+)-Furanomycin Derivative G Bartoli G Di Antonio R Fiocchi S Giuli E Marcantoni M Marcolini
957 An Efficient and Highly Selective Synthesis of (Z)-Fluoroenol Phosphates from Hydroxy Difluorophosphonates P Beier R Pohl A V Alexandrova
963 Iodine-Catalyzed Three-Component Reaction A Rapid Synthesis of α-Alkoxy Azides and Homoallyl Ethers J S Yadav B V S Reddy G M Reddy R Narender
969 Rhodium(I)-Catalyzed Cycloisomerization of 13-Dienes with Alkenes in a Tether Y Oonishi A Saito M Mori Y Sato
980 Synthesis of New Optically Active D-GlucosaminendashPyrrole Derivatives B A Frontana-Uribe M V Escaacutercega-Bobadilla J Juaacuterez-Lagunas R A Toscano G A Garciacutea de la Mora M Salmoacuten
985 Partially Saturated Indeno[12-b]indole Derivatives via Deoxygenation of Heterocyclic α-Hydroxy-NO-hemiaminals H-J Hemmerling G Reiss
1000 Light-Induced Synthesis of Π-Extended Tetrathiafulvalenes Incorporating Ferrocenes An Efficient Route for the Synthesis of Electron-Donor Materials A A O Sarhan C Bolm
1007 Preparation of Nβ-Fmoc-Protected Aza-β3-Amino Acids with Nonproteinogenic Hydrophobic Side Chains for Solid-Phase Syntheses of Pseudopeptides M Laurencin P Bauchat M Baudy-Flocrsquoh
1014 Diastereomeric (η4-diene)Fe(CO)3 Complexes Containing Chiral Amide Groups A Convenient Method for the Resolution of Amino Acids M Schumacher G Coste L Miesch
1021 Palladium-Catalysed Heck Reactions of Alk-1-en-3-ones with Aryl Bromides A Very Simple Access to (E)-1-Arylalk-1-en-3-ones M Lemhadri Y Fall H Doucet M Santelli
1036 An Improved Process for the Synthesis of 4H-Imidazo[15-α][14]benzodiazepines J Yang Y Teng S Ara S Rallapalli J M Cook
1041 Meta- and Para-Difunctionalization of Arenes via an Ortho-Magnesiation and a Subsequent SulfoxidendashMagnesium Exchange L Melzig C B Rauhut P Knochel
XIII Forthcoming Articles
No 7 1049 Catalytic Transformations of Benzylic Carboxylates and Carbonates
R Kuwano 1062 A Simple and Practical Method for the Oxidation of Thebaine to 14-
Hydroxycodeinone by V2O5ndashH2O2 S Das Sharma D Konwar 1065 Umpolung with Sulfur Dioxide CarbonndashCarbon Cross-Coupling of Electron-
Rich 13-Dienes and Alkenes Application to the Enantioselective Synthesis of Long-Chain Polyketide Fragments M Turks C J Exner C Hamel P Vogel
1075 One-Pot Synthesis of 14-Diarylnaphthalenes via a WittigndashHorner Reaction[4+2] CycloadditionDehydrogenation Sequence Z Chen W Shou Y Wang
1081 A Novel and General Method for the Formation of S-Aryl Se-Aryl and Te-Aryl Phosphorochalcogenoates Y-X Gao G Tang Y Cao Y-F Zhao
1087 A Remarkable Access to γ-Fluoroalkylated Propargylamine Derivatives or Fluoroalkylated Dihydroisoxazoles via the Reaction of Fluoroalkylated Acetylides with Various Nitrones T Konno K Moriyasu T Ishihara
1095 Short and Practical Syntheses of (S)-(+)-3-(p-Tolylsulfinyl)furan-2(5H)-one and (S)-(+)-3-(p-Tolylsulfinyl)-56-dihydropyran-2-one D Cruz Cruz A Hernaacutendez Linares F Yuste M R Martiacuten J L Garciacutea Ruano
1099 Decarboxylative Aldol-Type Reaction of 2-(Trifluoroacetyl)-13-diazoles with Activated Acetic Acids P V Khodakovskiy D M Volochnyuk A A Tolmachev
1105 Synthesis of 2-[(Arylmethylene)amino]cyclopropanecarbonitriles via a Two-Step Ring Transformation of 2-(Cyanomethyl)aziridines S Mangelinckx M Drsquohooghe S Peeters N De Kimpe
1113 Synthesis of Dendrimeric Tumor-Associated Mucin-Type Glycopeptide Antigens T Becker A Kaiser H Kunz
1123 A Simple and Efficient Oxidation Procedure for the Synthesis of Acid-Sensitive Epoxides O Bortolini G Fantin M Fogagnolo
1127 Rapid Chemoselective Deprotection of Benzyl Esters by Nickel Boride J M Khurana R Arora
1131 Three-Component Coupling of Isoquinoline Activated Alkyne and Nitromethane A Facile Synthesis of Nitromethyl Derivatives of 12-Dihydroisoquinolines J S Yadav B V S Reddy N N Yadav M K Gupta
1137 Palladium Supported on a Polyionic Resin as an Efficient Ligand-Free and Recyclable Catalyst for Heck SuzukindashMiyaura and Sonogashira Reactions B Basu S Das P Das B Mandal D Banerjee F Almqvist
1147 Oxidation of 25-Dialkylpyrrole Derivatives with Cerium(IV) Ammonium Nitrate R Voloshchuk M Gałęzowski D T Gryko
1153 Practical Syntheses of Enantiomerically Pure Key Intermediates of Opioid Receptor-like 1 (ORL1) Antagonists T Yoshizumi A Ohno T Tsujita H Takahashi O Okamoto I Hayakawa H Kigoshi
1163 An Environmentally Benign TEMPO-Catalyzed Efficient Alcohol Oxidation System with a Recyclable Hypervalent Iodine(III) Reagent and Its Facile Preparation X-Q Li C Zhang
1170 Efficient and Stereoselective Rearrangement of BaylisndashHillman Acetates Catalyzed by Gold(I) ChlorideSilver(I) Trifluoromethanesulfonate Y Liu D Mao J Qian S Lou Z Xu Y Zhang
1175 The First Total Synthesis of Kynapcin-24 by Palladium Catalysis L-Y Yang C-F Chang Y-C Huang Y-J Lee C-C Hu T-H Tseng
1180 Enantioselective Synthesis of N-Protected α-Amino Acid Hydrazides M Bibian S El-Habnouni J Martinez J-A Fehrentz
1185 Synthesis of 11H-Indolo[32-c]quinoline-6-carboxylic Acids by Cascade AutoxidationndashRing Contractions A Becker S Kohfeld T Pies K Wieking L Preu C Kunick
1190 Reaction of N-Nonaflylbenzotriazole with Silyl Enol Ethers M Uhde T Ziegler
1195 2-(Benzoylimino)thiazolidin-4-ones Formation by an Alternative Ring Closure and Analysis of Rotational Barriers H-G Haumlcker P W Elsinghorst S Michels J Daniels G Schnakenburg M Guumltschow
1204 Microwave-Assisted Synthesis and Functionalization of Selenolopyrimidines S Hesse C Chenet D Thomae G Kirsch
1209 12-Disubstituted 4-Quinolones via Copper-Catalyzed Cyclization of 1-(2-Halophenyl)-2-en-3-amin-1-ones R Bernini S Cacchi G Fabrizi A Sferrazza
1220 A New Atom-Economical and Selective Synthesis of Secondary and Tertiary Alkylamines by Means of CpIridium Complex Catalyzed Multiple N-Alkylation of Ammonium Salts with Alcohols without Solvent R Yamaguchi Z Mingwen S Kawagoe C Asai K-i Fujita
1224 Synthesis of Regioisomerically Pure 5-Functionalized 27-Dichlorofluoresceins J C Castro A Malakhov K Burgess
XIII Forthcoming Articles
No 8 1227 Michael Additions to Activated Vinylphosphonates T Janecki J Kędzia
T Wąsek 1255 A Facile and General Synthesis of 2β-Aminosteroids X Ke H Hu
D Zhou W Xu Q Zhu N P Reddy X Hu 1261 Efficacious Preparation of Oppolzerrsquos Glycylsultam via the Deleacutepine
Reaction A Isleyen C Gonsky R C Ronald P Garner 1265 Synthesis of Masked Vicinal Amino Aldehydes of Pyrrolizine and Pyrrolo
[12-c]thiazole Series A V Tverdokhlebov A V Denisenko A A Tolmachev Y M Volovenko S V Shishkina O V Shishkin
1271 Preparation of 9-Substituted Pyridine-Stretched Adenines and Hypoxanthines J A Crawford W Fraser C A Ramsden
1279 A Versatile Synthesis of Heterocyclic Analogues of Neoflavonoids from Enamino Ketones V S Moskvina V P Khilya O V Turov U M Groth
1287 New Stereoselective Synthesis of Paeonilactone B F G Gatti S Serra 1291 The Use of NN-Dialkyltrimethylsilylamines in the Synthesis of
Pentamethinium Salts M Kořiacutenek M Rybaacutečkovaacute Boumlhm 1297 Synthesis of Triazoles via Regioselective Reactions of Aryl Azides with
Cyanoacetyl Pyrroles and Indoles N T Pokhodylo V S Matiychuk M D Obushak
1301 Gallium(III) Chloride Catalyzed Hydroarylation of Arylacetylenes with Naphthols and Phenols A Facile Synthesis of Vinylarenes J S Yadav B V S Reddy S Sengupta S K Biswas
1305 Electrophilic Bromination of meta-Substituted Anilines with N-Bromosuccinimide Regioselectivity and Solvent Effect S Bartoli A Cipollone A Squarcia A Madami D Fattori
1309 Cross-Coupling Reactions of Halopurines with Aryl- and Alkyltrifluoroborates The Scope and Limitations in the Synthesis of Modified Purines Z Hasniacutek R Pohl M Hocek
1318 A Convenient Method for Converting Hydroxyacetophenones into Their Ethylene or Trimethylene Acetals F Ono H Takenaka T Fujikawa M Mori T Sato
1323 γ-Chloromagnesio γ-Lactones and δ-Chloromagnesio δ-Lactones Generation Properties and Synthetic Uses H Shimizu S Fukuda S Sugiyama T Satoh
1336 Click Reactions with Nitroxides T Kaacutelai W L Hubbell K Hideg 1341 Synthesis of Novel 14-Benzoquinone-Containing 123-Triazoles An Entry
Into a New Library F Algi M Balci 1348 Efficient Synthesis of Two Sialylated Tetrasaccharides Found in Goat Milk
P K Mandal A K Misra 1355 Dendrimers of Vaccines Consisting of Tumor-Associated Glycopeptide
Antigens and T Cell Epitope Peptides S Keil A Kaiser F Syed H Kunz
1370 IBXTBAB-Mediated Oxidation of Primary Amines to Nitriles F Drouet P Fontaine G Masson J Zhu
1375 Chemoselectivity of Multicomponent Condensations of Barbituric Acids 5-Aminopyrazoles and Aldehydes E A Muravyova S V Shishkina V I Musatov I V Knyazeva O V Shishkin S M Desenko V A Chebanov
1386 Stereoselective Total Syntheses of Leiocarpin A and (ndash)-Galantinic Acid Starting from D-Mannitol K Nagaiah D Sreenu K V Purnima R S Rao J S Yadav
1393 A Facile Mild Deprotection Protocol for 13-Dithianes and 13-Dithiolanes with 30 Hydrogen Peroxide and Iodine Catalyst in Aqueous Micellar System N C Ganguly S K Barik
1400 Rhodium-Catalyzed Gram-Scale Synthesis of Highly Substituted Pyridine Derivatives K Parthasarathy C-H Cheng
1403 Enantioselective Synthesis of (R)-Propylene Carbonate from Ethyl (S)-Lactate J M Whitaker R C Ronald
XIII Forthcoming Articles
no 9 1405 Transition-Metal-Catalyzed Site-Selective Cross-Coupling of Di- and
Polyhalogenated Compounds J-R Wang K Manabe 1428 An Improved Synthesis of (4-4-Hydroxy-3-isopropyl-5-[(4-nitrophenyl)
ethynyl]benzyl-35-dimethylphenoxy)acetic Acid (NH-3) M B Gopinathan K S Rehder
1431 Copper-Catalyzed Tandem CndashN Bond Formation Reaction Selective Synthesis of 2-(Trifluoromethyl)benzimidazoles M-W Chen X-G Zhang P Zhong M-L Hu
1437 Synthesis and Thermochemical Properties of Stereoisomeric Dihydroxy- and Tetrahydroxyalkylammonium Salts M Thomas L Rothman J Hatcher P Agarkar R Ramkirath S Lall-Ramnarine R Engel
1445 Preparation of 5-Substituted 2-(2-Alkylaryl-1H-imidazol-4-yl)oxazoles and 5-Substituted 2-(2-Alkylarylthiazol-4-yl)oxazoles by Utilizing 5-Substituted 2-(2-Bromo-11-diethoxyethyl)oxazole as a Synthon D R St Laurent J L Romine
1459 Novel and Efficient Methods for the Synthesis of Symmetrical Trisulfides A Kertmen S Lach J Rachon D Witt
1463 An Environmentally Benign Electrochemical Process for the Reduction of Carboxylic Acid Hydrazides to Amides M Mentel M J Beier R Breinbauer
1469 Synthesis of 1-Chloroalkynes from Alkynylsilanes Using Trichloroisocyanuric Acid as Chlorinating Agent M H Vilhelmsen A S Andersson M B Nielsen
1473 A Convenient Approach to Enantioenriched Cyclopropanes Bearing Electron-Withdrawing Functionalities H Krawczyń K Wąsek J Kędzia
1477 Synthesis of Cyclopropenes via 12-Elimination of Bromocyclopropanes Catalyzed by Crown Ether W M Sherrill R Kim M Rubin
1485 A Base-Catalysed One-Pot Three-Component Coupling Reaction Leading to Nitrosubstituted Pyrroles I R Baxendale C D Buckle S V Ley L Tamborini
1494 Synthesis of 4-Alkylidene-4H-31-benzoxazine Derivatives by Acid-Catalyzed Cyclization of 2-Isocyanophenyl Ketones in the Presence of a Vinyl Ether K Kobayashi Y Okamura H Konishi
1499 Synthesis of Higher Helicenes via Olefin Metathesis and CndashH Activation J Cocircteacute S K Collins
1506 Azido- and Ethynyl-Substituted 2262-Terpyridines as Suitable Substrates for Click Reactions A Winter A Wild R Hoogenboom M W M Fijten M D Hager R-A Fallahpour U S Schubert
1513 Synthesis of 2-(Arylamino)ethanethiols via Lewis Acid Catalyzed Aminolysis of 22-Dimethylthiirane as Precursors of the 14-Benzothiazine Nucleus R Spogli S Sabatini G Manfroni O Tabarrini V Cecchetti
1520 Iron(III) Chloride A Versatile Catalyst for the Practical Synthesis of 3-Sulfenylindoles J S Yadav B V S Reddy Y J Reddy K Praneeth
1525 Organocatalytic Enantioselective Conjugate Addition of 2-Fluoromalonate to Nitroolefins Direct Synthesis of Chiral Fluorinated γ-Nitro Carboxylic Acid Derivatives H Li L Zu H Xie W Wang
1531 Asymmetric Transfer Hydrogenation of Ketimines with Trichlorosilane Structural Studies Z Zhang P Rooshenas H Hausmann P R Schreiner
1545 Prolinol Sulfinyl Ester Derivatives Organocatalytic Michael Addition of Ketones to Nitroolefins under Neat Conditions X Zeng G Zhong
1551 Asymmetric Oxidations of Electron-Poor Alkenes Promoted by the β-Amino AlcoholTBHP System A Russo A Lattanzi
1557 Enantioselectivity Switch in Direct Asymmetric Aminoxylation Catalyzed by Binaphthyl-Based Chiral Secondary Amines T Kano A Yamamoto F Shirozu K Maruoka
1564 Enantioselective Conjugate Addition of N-Heterocycles to αβ-Unsaturated Ketones Catalyzed by Chiral Primary Amines G Luo S Zhang W Duan W Wang
1573 Sulfonyl Hydrazine as New Functionality in Organocatalysis Camphorsulfonyl Hydrazine Catalyzed Enantioselective Aza-Michael Addition L-Y Chen H He B-J Pei W-H Chan A W M Lee
1578 Conversion of Primary Alcohols and Aldehydes into Methyl Esters by Ruthenium-Catalysed Hydrogen Transfer Reactions N A Owston T D Nixon A J Parker M K Whittlesey J M J Williams
1582 Addendum and Erratum XVII Forthcoming Articles
no 10 1583 Organocatalytic Formation of Quaternary Stereocenters M Bella
T Gasperi 1615 Regioselective Synthesis of 5H-Thiazolo[32-a]pyrimidin-5-ones from
MoritandashBaylisndashHillman Adduct Acetates under Solvent-Free and Base-Free Conditions W Zhong B Guo F Lin Y Liu W Su
1623 First Synthesis of 5-Cyanosalicylates by Formal [3+3] Cyclocondensations of 13-Bis(silyloxy)-13-butadienes A Riahi O Fatunsin M Shkoor R Dede H Reinke C Fischer P Langer
1635 Reaction of Isocyanides Dialkyl Acetylenedicarboxylates and a-Keto Lactones Unexpected Participation of an Ester Carbonyl Group in the Isocyanide-Based Three-Component Reaction A A Esmaeili H Vesalipoor
1639 An Efficient and Chemoselective Synthesis of 16-Naphthyridines and Pyrano[32-c]pyridines under Microwave Irradiation Z-G Han S-J Tu B Jiang S Yan X-H Zhang S-S Wu W-J Hao X-D Cao F Shi G Zhang N Ma
1647 N-Activation of N-Arylimidazoles Facile Syntheses of N-Alkyl-N-arylimidazolium Iodides from Less Expensive Chloro Substrates A M Oertel V Ritleng M J Chetcuti
1651 Synthesis of Polyhalogenated 2-(Phenylamino)pyridines by Thermal Amination Reactions S R Waldvogel A Faust W Barkmann R Froumlhlich O Wolff
1655 Cyanide Ion Promoted Addition of Acylphosphonates to Diethyl Cyanophosphonate Synthesis of Phosphonocyanohydrin O-Phosphates A S Demir A Aybey M Emrullahoglu
1659 Straightforward and Scalable Synthesis of Orthogonally Protected 37-Diazabicyclo[410]heptane H Schramm M Pavlova C Hoenke J Christoffers
1663 Hypervalent Iodine Mediated Oxidation of 12-Diaminobenzimidazole and Its Schiff Bases Efficient Synthesis of 3-Amino-124-benzotriazine and 2-Aryl-124-triazolo[15-a]benzimidazoles A Kumar M Parshad R K Gupta D Kumar
1667 Synthesis of the Reported Protoberberine Gusanlung D P B Wakchaure S Easwar N P Argade
1673 2-(Azidomethyl)arylboronic Acids in the Synthesis of Coumarin-Type Compounds M I Naumov A V Nuchev N S Sitnikov Y B Malysheva A S Shavyrin I P Beletskaya A E Gavryushin S Combes A Y Fedorov
1683 Asymmetric Synthesis of 12-anti-Disubstituted Taurine Derivatives D Enders D Iffland G Raabe
1689 A Novel One-Pot Three-Component Synthesis of 5-Imino-2358-tetrahydropyrazolo[12-a]pyridazin-1-one Derivatives B Qian M-J Fan Y-X Xie L-Y Wu Y Shi Y-M Liang
1694 One-Portion Synthesis of 2-Acetoxy Carbonyl Compounds from Aldehydes by Using an Acetylated Masked Acyl Cyanide H Nemoto T Kawamura K Kitasaki K Yatsuzuka M Kamiya Y Yoshioka
1703 Synthesis of 9-Anthryl Ethers from trans-910-Dihydro-910-dimethoxyanthracene by Acid-Catalyzed Transetherification K S Jang H Y Shin D Y Chi
1708 Efficient Synthesis of Azo Dye Labeled Terpenes Sugars and Steroids Using N-(4-Arylazobenzoyl)-1H-benzotriazoles A R Katritzky S R Tala N E Abo-Dya Z K Abdel-Samii
1715 Tandem CH-ActivationndashImine-Formation Reaction A New Route to Imidazo[21-a]phthalazines A Heim-Riether K R Gipson
1720 A Convenient and Efficient α-Sulfenylation of Carbonyl Compounds E Okragla S Demkowicz J Rachon D Witt
1725 Stereoselective Synthesis of β-Branched Phenylalanine Derivatives via Chelate-Claisen Rearrangement C Quirin U Kazmaier
1732 Catalyst-Free and Base-Free Water-Promoted SNAr Reaction of Heteroaryl Halides with Thiols B Sreedhar P S Reddy M A Reddy
1739 Convenient Methods for Synthesis of C2-Symmetric Diphenyltetrahydrothiophenes M Periasamy G Ramani G P Muthukumaragopal
1744 Highly Diastereoselective Conjugate AdditionndashElimination of Chiral Nickel(II) Glycinate with Activated Allylic Acetates for Asymmetric Synthesis of Glutamic Acid Derivatives J Wang J Shi X Zhang D Lin H Jiang H Liu
1753 Synthesis of 36-Dimethoxybenzene-12-diamine and of 47-Dimethoxy-2-methyl-1H-benzimidazole T Besset C Morin
1757 An Inexpensive Procedure for Reductive Aminations Using Dimethylamineborane on Millimolar and Molar Scale R Ortmann M Schlitzer
1760 Classics in Stereoselective Synthesis Edited by E M Carreira L Kvaerno Reviewed by Rolf Breinbauer
XV Forthcoming Articles
no 11 1761 Transition-Metal-Catalyzed Enantioselective Synthesis of Compounds with
Non-Centrochirality M Ogasawara S Watanabe 1786 One-Pot Synthesis of 3-Acyl-2-(alkylsulfanyl)indoles and 2-(Alkylsulfanyl)-
indole-3-carboxylates from (2-Isocyanophenyl)methyl Ketones or (2-Isocyanophenyl)acetates S Fukamachi H Konishi K Kobayashi
1791 Efficient and Recyclable Phthalocyanine-Based Sensitizers for Photooxygenation Reactions H Xu W-K Chan D K P Ng
1797 A Facile and Practical One-Pot Synthesis of β-Oxo Thioamides from β-Oxo Amides and Isothiocyanates P Huang D Xiang Y Zhou Y Liang T Na D Dong
1801 Microwave-Promoted Solid-Acid-Catalyzed One-Pot Synthesis of Phthalazinones V M Outerbridge S M Landge H Tamaki B Toumlroumlk
1807 Benzylic Brominations with N-Bromosuccinimide in (Trifluoromethyl)-benzene D Suarez G Laval S-M Tu D Jiang C L Robinson R Scott B T Golding
1811 Synthesis of Thioflavanone and Flavanone Derivatives by Cyclization of Chalcones W Konieczny M Konieczny
1815 A New and Expedient Total Synthesis of Ochratoxin A and d5-Ochratoxin A B Gabriele M Attya A Fazio L Di Donna P Plastina G Sindona
1821 Synthesis of Benzopyrrolizidinones by NorrishndashYang Cyclization of 3-(Acylmethyl)-2-alkylisoindol-1-ones J Wu W Zhang C Wang
1829 Reactions of MoritandashBaylisndashHillman Acetates with Huisgen Zwitterions A Novel Strategy for the Synthesis of β-Amino Acid Derivatives A Jose R R Paul R Mohan S C Mathew A T Biju E Suresh V Nair
1834 Peracetylated β-Allyl C-Glycosides of D-Ribofuranose and 2-Deoxy- D-ribofuranose in the Chemical Literature Until Now Mirages in the Literature H Otero Martinez H Reinke D Michalik C Vogel
1841 Core-Tetrasubstituted Naphthalene Diimides by Stille Cross-Coupling Reactions and Characterization of Their Optical and Redox Properties S-L Suraru F Wuumlrthner
1846 A Practical Synthesis of Indole-Based Heterocycles Using an Amidoaluminum-Mediated Strategy R Todd M M Hossain
1851 Synthesis of Fluorinated Pyrrolo[23-b]pyridine and Pyrrolo[23-d]pyrimidine Nucleosides V O Iaroshenko Y Wang D V Sevenard D M Volochnyuk
1858 Recyclization Reactions of 5-Formyl-13-dimethyluracil with Electron-Rich Amino Heterocycles A P Mityuk D M Volochnyuk S V Ryabukhin A S Plaskon A Shivanyuk A A Tolmachev
1865 Facile Synthesis of Fluorinated 1-Desazapurines V O Iaroshenko D V Sevenard D M Volochnyuk Y Wang A Martiloga A O Tolmachev
1876 A Practical Synthesis of 3-Diethoxyphosphoryl-12-pyridazine Derivatives J-C Monbaliu J Marchand-Brynaert
1881 Enantioselective Reduction of Prochiral Ketones Employing Sprouted Pisum sativa as Biocatalyst J S Yadav B V S Reddy C Sreelakshmi A B Rao
1886 Application of Phenolate Ion Mediated Intramolecular Epoxide Ring Opening in the Enantioselective Synthesis of Functionalized 23-Dihydrobenzofurans and 1-Benzopyrans S K Dinda S K Das G Panda
1897 Complementary Synthetic Approaches to Constitutionally Diverse N-Aminoalkylated Isoindolinones Application to the Synthesis of Falipamil and 5-HT1A Receptor Ligand Analogues M Lorion A Couture E Deniau P Grandclaudon
1904 Selective Deprotection of Silyl Ethers with Sodium Periodate J Li D Menche
1909 Micellar Solution of Sodium Dodecyl Sulfate (SDS) Catalyzes KabacknikndashFields Reaction in Aqueous Media S Sobhani A Vafaee
1916 Convenient Methods for the Synthesis of a Library of Hemilabile Phosphines M V Jimeacutenez J J Peacuterez-Torrente M I Bartolomeacute L A Oro
1923 Terminal Aziridines by Addition of Grignard Reagents or Organoceriums to an (α-Chloro)sulfinylimine D M Hodgson J Kloesges B Evans
1933 A Robust Synthesis of Nε-(Carboxymethyl)-L-lysine (CML) R Csuk S Stark A Barthel R Kluge D Stroumlhl
1935 One-Pot Curtius Rearrangement Processes from Carboxylic Acids O Leogane H Lebel
XV Forthcoming Articles
no 12 1941 The Chemistry of Deprotonated α-Aminonitriles T Opatz 1960 An Efficient Synthesis of Tetraalkyl 2345-Thiophenetetracarboxylate
Derivatives A Alizadeh R Hosseinpour 1963 Facile Deprotection of Bulky (Trialkylsilyl)acetylenes with Silver Fluoride
S Kim B Kim J In 1969 Highly Efficient and Reusable Ionic Liquids for the Catalyzed
Hydroamination of Alkenes with Sulfonamides Carbamates and Carboxamides L Yang L-W Xu C-G Xia
1975 Synthesis of 2391016172324-Octasubstituted Phthalocyaninatozinc(II) Complexes Mediated by Reductive Agents G A Gauna A C Monsalvo J Awruch
1979 A Short and Efficient Synthesis of 3-2-[2-(Bromomethyl)thiazol-4-yl]-ethynyl-5-fluorobenzonitrile A Precursor for PET Radioligand [18F]SP203 M B Gopinathan C Jin K S Rehder
1983 Synthesis of a Substituted Benzazepin-2-one Dihydrate S K Boini R K Vaid K P Moder D Mitchell
1987 Synthesis of Novel Trisubstituted Imidazolines F J Lakner M A Parker B Rogovoy A Khvat A Ivachtchenko
1991 A Novel Synthesis of N-But-3-enyl-α- and β-Amino Acids T T Van Nguyen R T C Brownlee A B Hughes
1999 Synthesis of Substituted 5-(3-Hydroxypropyl)pyrrolidin-2-ones and Pyrrolizidinones from Nitroethane via C3 Functionalized 56-Dihydro-4H-12-oxazines A Novel Approach to Some Analogues of the Antidepressant Rolipram A Yu Sukhorukov A V Lesiv Y A Khomutova S L Ioffe V A Tartakovsky
2009 Chiral Cyclobutanols and Cyclopentane Dimers via Samarium(II) Iodide Induced Keto-Olefin Cyclisations of Carbohydrate-Derived Unsaturated Ketones D B G Williams J Caddy K Blann J J C Groveacute C W Holzapfel
2015 Synthesis of Perfluoroalkylthio-Substituted Ferrocenes C Rhode J Lemke M Lieb N Metzler-Nolte
2019 Functionalization of Polyhedral Oligomeric Silsesquioxane (POSS) via Nucleophilic Substitution M Dutkiewicz H Maciejewski B Marciniec
2025 A Novel Synthesis of Aryl Mesylates via One-Pot DemethylationndashMesylation of Aryl Methyl Ethers Using a Mixture of Phosphorus Pentoxide in Methanesulfonic Acid B Kaboudin Y Abedi
2029 Anionic Cyclization of (NN-Dimethylamino)[2-(prop-2-yn-1-yloxy)aryl]-acetonitriles T Zdrojewski J Musielak A Jończyk
2035 Strecker-Type Reaction Catalyzed by Carboxylic Acids in Aqueous Media Z Xie G Li G Zhao J Wang
2040 Synthesis of Novel Structurally Simplified Estrogen Analogues with Electron-Donating Groups in Ring A L F Tietze C A Vock I K Krimmelbein L Nacke
2061 On the Resolution of Secondary Phosphine Oxides via Diastereomeric Complex Formation The Case of tert-Butylphenylphosphine Oxide J Holt A M Maj E P Schudde K M Pietrusiewicz L Sieroń W Wieczorek T Jerphagnon I W C E Arends U Hanefeld A J Minnaard
2066 Enantioselective Copper-Catalyzed Conjugate Addition of Dimethylzinc to 5-(1-Arylalkylidene) Meldrumrsquos Acids A Wilsily T Lou E Fillion
2073 SuzukindashMiyaura Coupling Reactions Using Phosphite Ligands M Jang Y Jo I-K Oh H M Jung S Lee
2076 Synthesis of 2-Methylindoline- and 2-Methyl-1234-tetrahydroquinoline-Derived Phosphoramidites and Their Applications in Iridium-Catalyzed Allylic Alkylation of Indoles W-B Liu H He L-X Dai S-L You
2083 Stereocontrolled Synthesis of 13-Amino Alcohols by Reduction of Substituted 2-1-[(tert-Butylsulfinyl)amino]alkylcyclohexanones J C Gonzaacutelez-Goacutemez F Foubelo M Yus
2089 Tunable Phosphoramidite Ligands for Asymmetric Hydrovinylation Ligands par excellence for Generation of All-Carbon Quaternary Centers C R Smith H J Lim A ZhangT V RajanBabu
2101 Copper-Catalyzed Asymmetric Ring-Opening Reaction of Oxabenzonorbornadienes with Grignard and Aluminum Reagents R Millet L Gremaud T Bernardez L Palais A Alexakis
2113 A Simplified Synthesis of Takemotorsquos Catalyst A Berkessel B Seelig 2116 Pharmaceutical Substances Syntheses Patents and Applications of the
Most Relevant AIPs Edited by Axel Kleeman Juumlrgen Engel Bernhard Kutscher Dietmar Reichert Reviewed by I Agranat
XV Forthcoming Articles
no 13 2117 Recent Advances in the Aza-Claisen Rearrangement K C Majumdar
T Bhattacharyya B Chattopadhyay B Sinha 2143 A Novel and Convenient Synthesis of lsquoReversedrsquo Diamidino 25-Aryl- and
25-Azaheterocycle-Substituted Furans L Hu D W Boykin 2146 Efficient and General Preparation of Pyranostilbenes First Total Synthesis
of Artocarbene and Pawhuskin B B H Park Y R Lee W S Lyoo 2155 Mild Oxidation of Diarylacetylenes to 12-Diketones Using Oxone in
Trifluoroacetic Acid J-H Chu Y-J Chen M-J Wu 2163 One-Pot Microwave-Assisted Selective Azido ReductionTandem Cyclization
in Condensed and Solid Phase with Nickel Boride N Shankaraiah N Markandeya M Espinoza-Moraga C Arancibia A Kamal L Silva Santos
2171 Pyrrolo[321-ij]quinolin-4-one and Pyrrolo[321-ij]quinolin-6-one H McNab D J Nelson E J Rozgowska
2175 Practical Synthesis of 5-Substituted Tetrazoles under Microwave Irradiation J Roh T V Artamonova K Vaacutevrovaacute G I Koldobskii A Hrabaacutelek
2179 A Simple Method for the Synthesis of 3-Arylthieno[23-b]pyridines via Iodine-Mediated Cyclization of 3-(1-Arylalkenyl)-2-[(1-phenylethyl)sulfanyl]pyridines K Kobayashi D Nakamura Y Shiroyama S Fukamachi H Konishi
2184 Synthesis of Four Lysine-Linked Cereulide Analogues Showing Ionophoric Activity Towards Potassium Cations as Lead Compounds for Emetic Toxin-Detection by Immunoassays A Makarasen T Nishikawa M Isobe
2205 Synthesis of α-Aliphatic and β-Aromatic Substituted Taurines via Regioselective Ring Opening of Thiiranes with Ammonia H Yu S Cao L Zhang G Liu J Xu
2210 Stability of 5(6)-Carboxyfluorescein in Microwave-Assisted Synthesis of Fluorescein-Labelled O-Dimannosylated Peptides R Kowalczyk P W R Harris R P Dunbar M A Brimble
2223 Diversity-Oriented Synthesis of Functionalized Diaryl Sulfones by Regioselective [3+3] Cyclizations of 13-Bis(siloxy)buta-13-dienes with 2-(Arylsulfonyl)-3-ethoxy-2-en-1-ones Scope and Limitations M Shkoor A Riahi O Fatunsin H Reinke C Fischer P Langer
2236 Synthesis of Functionalized Salicylates by Formal [3+3] Cyclocondensation of 13-Bis(silyloxy)buta-13-dienes with 3-Alkoxy-2-en-1-ones G Mroszlig S Ladzik H Reinke A Spannenberg C Fischer P Langer
2249 Synthetic Approach to Alkoxy-β-(trifluoromethyl)styrenes and Their Application in the Synthesis of New Trifluoromethylated Heterocycles V M Muzalevskiy V G Nenajdenko A V Shastin E S Balenkova G Haufe
2260 o-Benzenedisulfonimide as a Powerful and Recyclable Organocatalyst for the Nazarov Reaction M Barbero S Cadamuro A Deagostino S Dughera P Larini E G Occhiato C Prandi S Tabasso R Vulcano P Venturello
2267 The Catalytic Potential of 4-Guanidinylpyridines in Acylation Reactions I Held E Larionov C Bozler F Wagner H Zipse
2278 Iron(III) Chloride in EthanolndashWater Highly Efficient Catalytic System for the Synthesis of Garcia Gonzalez Polyhydroxyalkyl- and C-Glycosylfurans L Nagarapu M V Chary A Satyender B Supriya R Bantu
2283 Ruthenium-Catalyzed Addition of Primary Amides to Alkynes A Stereoselective Synthesis of Secondary Enamides L J Gooszligen M Blanchot K S M Salih K Gooszligen
2289 Binaphthyl-Modified Quaternary Phosphonium Salts as Chiral Phase Transfer Catalysts Application to Asymmetric Amination of β-Keto Esters R He K Maruoka
X Table of Contents XI Forthcoming Articles
no 14 2293 Direct Methods for Stereoselective Polypropionate Synthesis A Survey
J Li D Menche 2316 Synthesis of Symmetrical Ketones from Grignard Reagents and
11-Carbonyldiimidazole D Bottalico V Fiandanese G Marchese A Punzi
2319 Synthesis of 45-Substituted Imidazoles by a Fast Condensation of 12-Diketones and Urotropine in Heterogeneous Medium G Bratulescu
2321 (Arylsulfonyl)acetones and -acetonitriles New Activated Methylenic Building Blocks for Synthesis of 123-Triazoles N T Pokhodylo V S Matiychuk M D Obushak
2324 A Safe Convenient and Efficient One-Pot Synthesis of α-Chloroketone Acetals Directly from Ketones Using Iodobenzene Dichloride J Yu C Zhang
2329 An Efficient Oxidative Conversion of Aldehydes into 2-Substituted 2-Oxazolines Using 13-Diiodo-55-dimethylhydantoin S Takahashi H Togo
2333 A Novel Procedure for the Synthesis of Benzo[b][18]naphthyridine-3-carboxylate Derivatives from MoritandashBaylisndashHillman Adduct Acetates W Zhong F Lin R Chen W Su
2341 An Improved Synthesis of 147-Triazacyclononanes (tacns) and 14710-Tetraazacyclododecanes (cyclens) J Huang Z Zhou T H Chan
2345 The Ullmann Coupling between 2-Chlorobenzoic Acids and Amino Acids A Valuable Reaction for Preparing 2-Substituted 1-Acetyl-1H-indol-3-yl Acetates J C Rodriguez Dominguez X Gang G Kirsch
2349 gem-Dibromomethyl Aromatics Efficient Aldehyde Equivalents in the KnoevenagelndashDoebner Reaction J K Augustine Y A Naik S Poojari N Chowdappa B S Sherigara K Areppa
2357 Synthesis of Novel α-Aminophosphonates Containing Adamantyl Fragment M M Kabachnik L I Minaeva I P Beletskaya
2361 Efficient Fluoride-Mediated Synthesis of 5-Amino-Substituted Isothiazoles Y S Zubenko V I Potkin
2365 Phosphine-Catalyzed Reaction of Cyanohydrins with Activated Alkynes A Siby O Loreau F Taran
2371 Sulfanyl-Substituted [3]Cumulenes and Buta-13-dienes from a Tetrakis(pyridinium)-Substituted Butadiene A Schmidt A Rahimi M Gjikaj
2379 Efficient Synthesis of 2-Substituted Pyrido[32-d]pyrimidines Involving SNAr and Palladium-Catalyzed Cross-Coupling Reactions A Tikad S Routier M Akssira J-M Leacuteger C Jarry G Guillaumet
2385 Novel Synthesis of Medium-Sized Heterocycles by Palladium-Catalyzed Intramolecular Heck Reaction via 9-endo-trig Mode of Cyclization K C Majumdar B Chattopadhyay
2393 Facile Synthesis of Fluorinated Benzofuro- and Benzothieno[23-b]pyridines α-Carbolines and Nucleosides Containing the α-Carboline Framework V O Iaroshenko Y Wang B Zhang D Volochnyuk V Ya Sosnovskikh
2403 Synthesis of Functionalized N-Vinyl Nitrogen-Containing Heterocycles S M M Lopes A M Beja M Ramos Silva J A Paixatildeo F Palacios T M V D Pinho e Melo
2408 Kumada Cross-Coupling of Aryl Grignard Reagents with Aryl Halides Catalyzed by an Immobilized Nickel Catalyst X Chen L Wang J Liu
2413 Highly Enantioselective Synthesis of Heteroaromatic Alcohols Catalyzed by Chiral DiaminodiphosphinendashRuthenium(II) Complexes W-Y Shen Y-Y Li Z-R Dong J-X Gao
2418 Concise Total Synthesis of (+)-Disparlure and its trans-Isomer Using Asymmetric Organocatalysis S-G Kim
2423 Rhodium Carbenoid Induced [12]-Migration in an L-Lyxo-Configured α-Diazo β-Keto Ester Synthesis of a New Griseolic Acid Analogue N N Bhujbal K S A Kumar D D Dhavale
2430 Synthesis of 5-Arylthio-3-hydroxyphthalates by the First [4+2] Cycloadditions of 3-Arylthio-1-silyloxy-13-butadienes with Dimethyl Acetylenedicarboxylate I Iqbal M Imran P Langer
2435 Synthesis of Highly Functionalized Proline Derivatives via a One-Pot MichaelSN-AdditionCyclization Approach U Kazmaier C Schmidt
2440 RhodiumGraphite-Catalyzed Hydrogenation of Carbocyclic and Heterocyclic Aromatic Compounds G Falini A Gualandi D Savoia
2447 Potassium [1-(tert-Butoxycarbonyl)-1H-indol-2-yl]trifluoroborate as an Efficient Building Block in Palladium-Catalyzed SuzukindashMiyaura Cross Couplings P Kassis V Beacuteneacuteteau J-Y Meacuterour S Routier
2454 Syntheses of Substituted Furans and Pyrroles by Platinum-Catalyzed Cyclizations of Propargylic Oxiranes and Aziridines in Aqueous Media M Yoshida M Al-Amin K Shishido
2467 Transition-Metal-Free Oxidative Homocoupling of Aryl Alkenyl and Alkynyl Grignard Reagents with TEMPO M S Maji A Studer
XIII Forthcoming Articles
no 15 2471 Advances in Synthetic Approaches for the Preparation of Combretastatin-
Based Anti-Cancer Agents R Singh H Kaur 2492 Synthesis of Unsymmetrical Ureas by Sulfur-Assisted Carbonylation with
Carbon Monoxide and Oxidation with Molecular Oxygen under Mild Conditions T Mizuno T Nakai M Mihara
2497 Ring-OpeningRecyclization Reactions of (Dimethylamino)propenoyl-Substituted Cyclopropanes Facile Synthesis of Halogenated Pyridin-2(1H)-ones R Zhang Y Zhou Y Liang Z Jiang D Dong
2501 Facile and Efficient Total Synthesis of Taspine B Cheng S Zhang L Zhu J Zhang Q Li A Shan L He
2505 Oligomeric Iodosylbenzene Sulfate A Convenient Hypervalent Iodine Reagent for Oxidation of Organic Sulfides and Alkenes M S Yusubov R Y Yusubova T V Funk K-W Chi V V Zhdankin
2509 Pyrrolidine-Based Organocatalysts for Enantioselective Michael Addition of Cyclohexanone to trans-β-Nitrostyrene A P Carley S Dixon J D Kilburn
2517 CundashAl Hydrotalcite An Efficient and Reusable Ligand-Free Catalyst for the Coupling of Aryl Chlorides with Aliphatic Aromatic and N(H)-Heterocyclic Amines B Sreedhar R Arundhathi P L Reddy M A Reddy M L Kantam
2523 Highly Efficient Synthesis of trans-βγ-Unsaturated a-Keto Amides C Allais T Constantieux J Rodriguez
2531 Gas-Phase Synthesis of N-Unsubstituted 3-Hydroxypyrroles and 1H-Pyrrol-3(2H)-ones L Hill G A Hunter S H Imam H McNab W J OrsquoNeill
2535 3-Hydroxy-1H-pyrrole L Hill S H Imam H McNab W J OrsquoNeill 2539 123-Thiadiazoles with Unsaturated Side Chains Synthesis
Polymerization and Photocrosslinking M Al-Smadi N Hanold H Kalbitz H Meier
2547 Synthesis of 1112-Didehydrodibenzo[ae]cycloocten-5(6H)-one A Strained Eight-Membered Alkyne S C Kornmayer F Rominger R Gleiter
2553 Stannous Chloride Dihydrate A Novel and Efficient Catalyst for the Synthesis of gem-Dihydroperoxides from Ketones and Aldehydes D Azarifar K Khosravi F Soleimanei
2557 Synthesis of a Novel Class of Azacrown Macrocycles and Lariat Crown Ethers Containing Two 124-Triazole Rings as Subunits N Foroughifar A Mobinikhaledi S Ebrahimi
2561 Enantioselective Synthesis of the 3C-Protease Inhibitor (ndash)-Thysanone by a StauntonndashWeinreb Annulation Strategy J Sperry T Y Yuen M A Brimble
2570 Stereoselective Synthesis of Unnatural β-Amino Acids from Nitroethane via 56-Dihydro-4H-12-oxazin-3-ylacetates A Yu Sukhorukov A V Lesiv O L Eliseev Y A Khomutova S L Ioffe
2579 A Versatile Unexpected One-Pot Regioselective Synthesis of a New Class of 13-Diazepinoindolones by Reaction of Pyranoindolones with Monosubstituted Ureas D Livadiotou C A Tsoleridis J Stephanidou-Stephanatou
2584 Synthesis of a Trisaccharide and a Tetrasaccharide from the Cell-Wall Lipopolysaccharides of Azospirillum brasilense S17 S Pandey S Ghosh A K Misra
2591 Synthesis of Isoindoline Nitroxides by Electrocyclic Reactions T Kaacutelai J Jekı K Hideg
2596 Glycosylations of Tertiary Alcohols Synthesis of Fully Protected Disaccharides with Sterically Demanding Groups Attached to the Sugar Core A Holkenbrink J B Vicente D B Werz
2605 Copper-Catalyzed [13]-Dipolar Cycloaddition for the Synthesis of Macrocycles Containing Acyclic Aromatic and Steroidal Moieties G V Latyshev M S Baranom A V Kazantsev A D Averin N V Lukashev I P Beletskaya
2616 Aryl Ring Migration Reaction in the Synthesis of 24-Diaryl-4H-31-benzothiazines A V Butin F A Tsiunchik V T Abaev A V Gutnov D A Cheshkov
2627 Hydrogenation of β-N-Substituted and β-NN-Disubstituted Enamino Esters in the Presence of Iridium(I) Catalyst H Hebbache Z Hank C Bruneau J-L Renaud
2634 Stereoselective Olefination Reactions Promoted by Rieke Manganese J M Concelloacuten H Rodriacuteguez-Solla V del Amo P Diacuteaz
2646 Synthesis of Piperidinones through a Radical Cascade E Godineau Y Landais
2650 Asymmetric Organic Synthesis with Enzymes Edited by V Gotor I Alfonso E Garciacutea-Urdiales Reviewed by Steve Collier
XVII Forthcoming Articles
no 16 2651 Synthesis of Spirocyclic Ethers S Rosenberg R Leino 2674 Bimetallic PalladiumndashPlatinum-on-Carbon-Catalyzed HndashD Exchange
Reaction Synergistic Effect on Multiple Deuterium Incorporation T Maegawa N Ito K Oono Y Monguchi H Sajiki
2679 Efficient Copper-Catalyzed Synthesis of 2-Amino-4(3H)-quinazolinone and 2-Aminoquinazoline Derivatives X Huang H Yang H Fu R Qiao Y Zhao
2689 Synthesis and Chemoselective N- and O-Alkylation of Thiadiazolopyrimidine Nucleosides and Uridines A M L Hossion R Islam R K Kandahary T Nagamatsu
2697 Facile and Efficient Synthesis of a New Class of Indole-Substituted Pyridine Derivatives via One-Pot Multicomponent Reactions K Zhao X-P Xu S-L Zhu D-Q Shi Y Zhang S-J Ji
2709 Studies toward a Total Synthesis of Rhizoxin D Stereoselective Preparation of the C11ndashC19 Fragment S Padakanti C K Kumar E Ashok P Das
2715 A Short Synthesis of Enantiomeric Phytoprostanes B1 Type I W Perlikowska M Mikołajczyk
2719 Chemistry of Polyhalogenated Nitrobutadienes Part 7 A Novel Synthetic Access to Chlorinated Nitrile Oxides E Nutz V A Zapolrsquoskii D E Kaufmann
2725 Microwave-Assisted Silver(I)-Mediated Selective O-Alkylation of Aromatic Imidate Systems B K Singh C Cavalluzzo M De Maeyer Z Debyser V S Parmar E Van der Eycken
2729 Iodogen A Novel Reagent for the Oxidation of Urazoles under Heterogeneous Conditions A Khoramabadi A Shiri M A Zolfigol S Mallakpour
2733 An Unprecedented Synthesis of Eight-Membered-Ring Cyclic Thioimidic Esters by a Three-Component Reaction A Alizadeh R Hosseinpour
2737 A Novel Diastereoselective Synthesis of β-Phosphonato Unsaturated Thioimidates A Alizadeh N Zohreh
2741 Synthesis of 21-Benzisoxazoles by Nucleophilic Substitution of Hydrogen in Nitroarenes Activated by the Azole Ring N T Pokhodylo Y O Teslenko V S Matiychuk M D Obushak
2749 A Facile Synthesis of Two Series of Multifunctional Carbon Compounds from αα-Dihalo Ketones Using Allylsamarium Bromide X Liu S Zhang J Di
2756 Stereocontrolled Formation of Protected Aminodeoxyalditols from Simple Carbohydrate Precursors by Debenzylating Cycloetherification Y Jiang Z Fang Q Zheng H Jia J Cheng B Zheng
2761 trans-Stilbene as a Starting Material for the Synthesis of Tamoxifen Based on Palladium-Catalyzed Cross-Coupling Reactions C M Nunes J Limberger S Poersch M Seferin A L Monteiro
2766 Synthesis and Biological Evaluation of 6-Substituted Purinylcarbanucleosides with a Cyclopenta[b]thiophene Pseudosugar P Abeijoacuten J M Blanco O Caamantildeo F Fernaacutendez M D Garciacutea X Garciacutea-Mera J E Rodriacuteguez-Borges J Balzarini E De Clercq
2773 Synthesis and Electrochemical Signature of Novel Norbornyl-ferrocene Hybrids F A Khan S K Upadhyay
2778 A Regioselective TsujindashTrost Pentadienylation of 3-Allyltetronic Acid R Schobert B Barnickel
2785 Copper(I)-Catalyzed CarylndashCalkynyl Bond Formation of Aryl Iodides with Terminal Alkynes K G Thakur G Sekar
2790 Aminolysis of Epoxides Using Iridium Trichloride as an Efficient Catalyst J Agarwal A Duley R Rani R K Peddinti
2797 Preparation of Several Active N-Chloro Compounds from Trichloroisocyanuric Acid A Shiri A Khoramabadi-zad
2802 The First Mineral-Catalyzed One-Pot [3+1+2] Coupling Protocol for Multifunctionalized Fused-Ring Pyrimidines L D S Yadav A Rai
2809 Efficient Synthesis of Tetrahydro-β-carbolin-1-one and Dihydroisoquinolin-1-one Derivatives as Versatile Intermediates K E Judd M F Mahon L Caggiano
2818 A Concise Synthesis of ortho-Iodobenzyl Alcohols via Addition of ortho-Iodophenyl Grignard Reagent to Aldehydes and Ketones J Cvengroš D Stolz A Togni
XIII Forthcoming Articles
no 17 2825 Reactivity of Oxazol-5-(4H)-ones and Their Application toward Natural
Product Synthesis N M Hewlett C D Hupp J J Tepe 2840 Towards the Total Synthesis of 3-Hydroxyvibsanin E B D Schwartz
J R Denton P V Bernhardt H M L Davies C M Williams 2847 Structure Investigations of (ent)-Cladospolide D by De Novo Synthesis and
Kinetic and Thermodynamic Isomerization Y Xing J H Penn G A OrsquoDoherty
2855 New Applications of PhI(OAc)2 in Synthesis Total Synthesis and SAR Development of Potent Antitumor Natural Product PsymberinIrciniastatin A N Shao X Huang A Palani R Aslanian A Buevich J Piwinski R Huryk C Seidel-Dugan
2873 Total Synthesis of Largazole ndash Devolution of a Novel Synthetic Strategy B Wang C J Forsyth
2881 Formal Total Synthesis of Palmerolide A J Jaumlgel M E Maier 2893 Total Synthesis of Bongkrekic Acid via Sequential SuzukindashMiyaura Coupling
Reactions M Kanematsu M Shindo M Yoshida K Shishido 2905 Stereodivergent Approach to Both C28a-syn and C28a-anti Relative
Stereochemical Manifolds in the Lepadin Family via a TiCl4-Promoted G Li L J Carlson I K Sagamanova B W Slafer R P Hsung C Gilardi H M Sklenicka N Sydorenko
2915 Enantioselective Aldol Reaction of Tetrasubstituted Ketene Silyl Acetals with Achiral Aldehydes for the Construction of Asymmetric Tertiary Alcohols An Application for the Divergent Total Syntheses of Buergerinins F and G I Shiina T Iizumi Y-s Yamai Y-i Kawakita K Yokoyama Y-k Yamada
2927 Second-Generation Biomimetic Total Synthesis of Chaetominine A Coste G Karthikeyan F Couty G Evano
2935 Total Synthesis of (+)-Fostriecin and (+)-Phoslactomycin B S Shibahara M Fujino Y Tashiro N Okamoto T Esumi K Takahashi J Ishihara S Hatakeyama
2954 Stereochemical Assignments of the Chlorinated Residues in Victorin C A C Durow C Butts C L Willis
2963 Studies of the Asymmetric Total Synthesis of Clavilactone D by the lsquoLariatrsquo Cyclization Strategy T Yoshimitsu S Nojima M Hashimoto K Tsukamoto T Tanaka
2970 Total Synthesis of the Leucetta-Derived Alkaloid Calcaridine A P B Koswatta R Sivappa H V R Dias C J Lovely
2983 Formal Synthesis of Salinosporamide A Starting from D-Glucose T Momose Y Kaiya J-i Hasegawa T Sato N Chida
2992 Synthesis of Bioactive Natural Products by Asymmetric syn- and anti-Aldol Reactions A K Ghosh Z L Dawson
no 18 3003 Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural
Products B M Trost M K Brennan 3026 One-Pot Synthesis of Furo[34-b]pyridin-5(7H)-ones from 2-
Bromopyridine-3-carboxylic Acid and Carbonyl Compounds K Kobayashi T Kozuki H Konishi
3029 Iodocyclization of N-[2-(Methylthio)phenyl]propiolamides Selective Synthesis of 3-Iodo-15-benzothiazepin-4-ones T-S Jiang X-G Zhang J-H Li
3039 A Facile Synthetic Method for Fluorine-Containing 17-Phenanthrolines Pyridine-Ring Formation Reaction of N-Propargyl-68-bis(trifluoroacetyl)-quinolin-5-amine with Various Nucleophiles D Shibata E Okada M Hinoshita M Meacutedebielle
3047 Enantiotopic Discrimination in Palladium-Mediated Nucleophilic Substitutions on Achiral Substrates Chiral Ligand versus Chiral Nucleophile O Jacquet F Charnay J-C Fiaud J Ollivier
3051 Studies on the Chemistry of 2-[3-(2-Nitrophenyl)-2-oxopropyl]benzaldehydes Novel Syntheses of 5H-Benzo[b]carbazole-611-diones and Indolo[12-b]isoquinoline-611-diones M Fernaacutendez
3061 Studies on the C22ndashC23 Aldol Coupling of Spirangien M Lorenz N Bluhm M Kalesse
3067 One-Pot Synthesis of N-Alkyl Purine Pyrimidine and Azole Derivatives from Alcohols using Ph3PCCl4 A Rapid Route to Carboacyclic Nucleoside Synthesis M N Soltani Rad A Khalafi-Nezhad S Behrouz Z Asrari M Behrouz Z Amini
3077 Synthesis of 2-Amino-34-dihydroquinazolines and Imidazo[21-b]quinazoline-2-ones A Mishra S Batra
3089 Studies on the Reaction of Diimines with Thiourea Synthesis and Solvent-Induced cistrans-Isomerization of 135-Triazinane-2-thiones B Kaboudin T Ghasemi T Yokomatsu
3094 Suzuki Coupling of Heteroaromatic Chlorides Using Highly Electron-Donating ClickPhos Ligands S M Spinella Z-H Guan J Chen X Zhang
3099 Reaction of NN-Dioxyenamines with Anhydrides of Carboxylic and Sulfonic Acids A New Method for the Synthesis of a-Hydroxyoxime Derivatives A A Tabolin A V Lesiv S L Ioffe
3106 Directed ortho Metallation Chemistry and Phosphine Synthesis New Ligands for the SuzukindashMiyaura Reaction D B G Williams S J Evans H de Bod M S Mokhadinyana T Hughes
3113 New Functional Derivatives of 9-Phenylquinine P J Boratyński J SkarŜewski
3120 On the Synthesis of Asymmetric and Dissymmetric Amino Analogues of Troumlgerrsquos Base J Artacho K Waumlrnmark
3127 Synthesis of Polycyclic Sultams by Palladium-Catalyzed Intramolecular Cyclization K C Majumdar S Mondal N De
3136 Synthesis of Functionalized L-Cysteine and L-Methionine by Reaction with Electron-Deficient Acetylenes B A Trofimov A G Malrsquokina O A Shemyakina V V Nosyreva A P Borisova S S Khutsishvili L B Krivdin
3143 A lsquoClickrsquo Approach to the Synthesis of 3-[2-(1-Alkyltriazol-4-yl)ethyl]indoles M Petrini R R Shaikh
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
148 Complementary Reactions of Allylic Carbamates Using Palladium(II) Formation of Oxazolidinones or Allylic Amides from a Common Precursor S D R Christie A D Warrington C J Lunniss
155 Thermal Amination of 26-Dihalopyridines by Sterically Demanding Amines A Faust O Wolff S R Waldvogel
160 The Thermal Amidation of Carboxylic Acids Revisited L J Gooszligen D M Ohlmann P P Lange
XVII Instructions for Authors XXIII Forthcoming Articles
No 2 165 Selected Synthetic Strategies to Spirocyclics S Kotha A C Deb
K Lahiri E Manivannan 194 Effective Catalytic Activity of the Hydrated Gold Catalyst NaAuCl42H2O To
Construct Highly Fused Cyclopentenones S Karmakar A Kim C H Oh
199 Efficient Synthesis of an Allose-Containing Analogue of the Phytoalexin-Elicitor Glucohexaose and Its Dodecyl Glycoside H Ma D Qiu X Mei J Ning Q Zhao Y Li
205 Synthesis of 14-Benzodiazepine-25-diones Using an Ionic Liquid as a Soluble Support H Xie C Lu G Yang Z Chen
211 A Facile Synthesis of Thioalkyl- and Di(thioalkyl)-Substituted Bipyridines D Chen R De D L Mohler
217 Diastereoselective Synthesis of Dimethyl (4R4aR7aR)-1-Aryl-6-benzoyl-4a-methyl-5-oxo-144a556-hexahydrospiro[pyrazole-47-pyrrolo[34-c]pyridazine]-37a(1H)-dicarboxylates U Uršič U Grošelj A Meden J Svete B Stanovnik
227 Synthesis of 3-Acylpyrroles 3-(Alkoxycarbonyl)pyrroles 1567-Tetrahydro-4H-indol-4-ones and 3-Benzoylpyridines Based on StaudingerndashAza-Wittig Reactions of 13-Dicarbonyl Compounds with 2- and 3-Azido-11-dialkoxyalkanes E Bellur M A Yawer I Hussain A Riahi O Fatunsin C Fischer P Langer
243 Regioselective Synthesis of Functionalized Biaryls Based on the First [3+3] Cyclocondensations of 4-Aryl-13-bis(trimethylsilyloxy)buta-13-dienes M Adeel M A Rashid N Rasool R Ahmad A Villinger H Reinke C Fischer P Langer
251 Synthesis of Functionalized Bicyclic Precursors of Heptulosonic Acid Analogues H Filali S Ballereau F O Chahdi M Baltas
257 Efficient Regio- and Stereoselective Synthesis of 5-Alkyl(aryl)idene- and 5-[Iodoalkyl(aryl)idene]-1H-pyrrol-2(5H)-ones via Electrophilic Cyclization K Cherry A Duchecircne J Thibonnet J-L Parrain E Anselmi M Abarbri
271 PdCu-Catalyzed Oxidative CndashH Alkenylation of Imidazo[12-α]pyridines J Koubachi S Berteina-Raboin A Mouaddib G Guillaumet
277 A Convenient Synthesis of Unsymmetrical Pinacols by Coupling of Structurally Similar Aromatic Aldehydes Mediated by Low-Valent Titanium X-F Duan J-X Feng G-F Zi Z-B Zhang
283 A Method for the Selective Protection of Aromatic Amines in the Presence of Aliphatic Amines V Perron S Abbott N Moreau D Lee C Penney B Zacharie
290 Synthesis and Antiviral Evaluation of (ndash)-3-Methylcarbovir (ndash)-3-Methylabacavir and Modified Purine Analogues P Breacutemond G Audran H Monti E De Clercq C Pannecouque
297 Regioselective Synthesis of 2-(Aryloxythio)benzoates by the First [3+3] Cyclizations of 3-Aryloxythio-1-silyloxybuta-13-dienes with 3-Alkoxy-2-en-1-ones I Iqbal M Imran A Villinger P Langer
306 Molybdenum(VI) Dichloride Dioxide Catalyzed Conversion of b-Hydroxycarbonyls into a-Bromo 13-Dicarbonyls by N-Bromosuccinimide K Jeyakumar D K Chand
311 A Short Route to the Synthesis of Pyrrolocoumarin and Pyrroloquinolone Derivatives by Sonogashira Cross-Coupling and Gold-Catalyzed Cycloisomerization of Acetylenic Amines K C Majumdar B Chattopadhyay S Samanta
318 Aspects of the Synthesis of an Exceptionally Preorganized Self-Immolative SpacerndashPhenolate Unit M Waibel X-B Zhang J Hasserodt
325 Design and Efficient Synthesis of Amino Acid Derived 2-Substituted Imidazoles by Palladium-Catalyzed Cross-Coupling Reactions A Marek J Kulhaacutenek F Bureš
332 A Convenient Preparation of Di-p-chlorobenzyl Azodicarboxylate (DCAD) for Mitsunobu Couplings B R Taft E C Swift B H Lipshutz
335 Enantioselective Rhodium-Catalyzed Alkylative Desymmetrization of 35-Dimethylglutaric Anhydride M J Cook T Rovis
XIII Forthcoming Articles
No 3 339 Intermolecular Addition Reactions of N-Acyliminium Ions (Part I)
A Yazici S G Pyne 369 Desulfurization of Thioamides into Amides with H2O2ZrCl4 Reagent System
K Bahrami M M Khodaei Y Tirandaz 372 Total Synthesis of (plusmn)-1345-Tetragalloylapiitol R M Patel
N P Argade 375 A Convenient Synthesis of 4-Hydroxy-2-oxo-12-dihydro-18-
naphthyridine-3-carboxamide Derivatives K Kobayashi D Iitsuka S Fukamachi H Konishi
379 Intramolecular Ketalization of Functionalized 7-Norbornenols L A Paquette J D Pettigrew
385 Ring Contraction of 12-Dihydronaphthalenes Promoted by Thallium(III) in Acetonitrile A Diastereoselective Approach to Indanes H M C Ferraz V M T Carneiro L F Silva Jr
389 Regio-Controlled Nucleophilic Attack of 3-Thiaisatoic Anhydride by α-Amino Acids One-Pot Synthesis of 3-(2-Thienyl)imidazolidine-24-dione and 34-Substituted Thieno[23-e][14]diazepine-25-dione Analogues Y Brouillette G Sujol J Martinez V Lisowski
395 The Unprecedented Cobalt-Catalysed Oxidative Glaser Coupling under Reductive Conditions G Hilt C Hengst M Arndt
399 Nucleophilic Addition of 4-Hydroxycoumarin to BaylisndashHillman Acetate Adducts C Raji Reddy N Kiranmai K Johny M Pendke P Naresh
403 Palladium-Mediated Heck Reaction to the Synthesis of 3-Substituted Indoles and Indolones K C Majumdar S Chakravorty P K Shyam A Taher
409 Synthesis of Bicyclo[310]hexan-2-ones by Manganese(III) Oxidation in Ethanol K Asahi H Nishino
424 High Regio- and Stereoselective Synthesis of (Z)- or (E)-N-Acryl Butenedioic Monoimide Derivatives by a Multicomponent Reaction F Sha Y Lin X Huang
431 The First Synthesis of Allyl Isonitriles from BaylisndashHillman Adducts and Their Application in the Synthesis of Substituted Imidazo[12-α]pyridines and Tetraazadibenzoazulenes M Nayak S Kanojiya S Batra
438 One-Pot Three-Step Synthesis of Pyrazinothienopyrimidines Using Tandem Aza-WittigElectrocyclic Ring Closure G Blanco A Fernaacutendez-Mato J M Quintela C Peinador
445 Synthesis of Biaryls Fluorenones Cyclopenta[def]phenanthren-4-ones and Benzophenones Based on Formal [3+3] Cyclocondensations of 13-Bis(silyloxy)buta-13-dienes with 3-(Silyloxy)-2-en-1-ones S Reim M Lau M Adeel I Hussain M A Yawer A Riahi Z Ahmed C Fischer H Reinke P Langer
464 Diastereoselective Synthesis of α-Stabilized Phosphorus Ylides via a Four-Component Reaction A Alizadeh N Zohreh L-G Zhu
469 Stereoselective Synthesis of Alkynyl Vinyl Chalcogenides via HornerndashWittig Reaction C C Silveira F Rinaldi R C Guadagnin A L Braga
474 Stereoselective Preparation of C1ndashC10 and C11ndashO14 Fragments of Narbonolide Exploiting the Versatility of Thiazolidinethione Chiral Auxiliary C P Narasimhulu P Das
483 Efficient Catalytic Activity of CopperAluminum Hydrotalcite in Diaryl Ether Synthesis B Sreedhar R Arundhathi M A Reddy M L Kanatm
488 On-Resin Click-Glycoconjugation of Peptoids A S Norgren C Budke Z Majer C Heggemann T Koop N Sewald
495 A Simple and Efficient Preparation of Novel Formaldehyde Derivatives R Hartung G Golz S Schlaf G Silvennoinen K Polborn P Mayer H R Pfaendler
502 2-Oxazol-5-ylethanones by Consecutive Three-Component AmidationndashCouplingndashCycloisomerization (ACCI) Sequence E Merkul O Grotkopp T J J Muumlller
508 SuzukindashMiyaura Cross-Couplings Mediated by trans-PdBr(N-Succ)(PPh3)2 A Convenient Synthetic Method for Diarylmethanes and Aryl(heteroaryl)-methanes I J S Fairlamb P Sehnal R J K Taylor
511 Modern Reduction Methods Edited by P G Andersson and I J Munslow Reviewed by Siegfried R Waldvogel
512 Addendum and Erratum XIII Forthcoming Articles
No 4 513 Intermolecular Addition Reactions of N-Acyliminium Ions (Part II)
A Yazici S G Pyne 542 A Simple Practical Method for the Synthesis of 46-Dimethoxy-135-
triazin-2(1H)-one Using Dimethylamine-Functionalized Solid-Phase Reagents K Hioki K Ohshima Y Sota M Tanaka M Kunishima
545 Conjugation-Amenable Tetrasaccharide of the Side Chain of the Major Glycoprotein of the Bacillus anthracis Exosporium A Large-Scale Preparation S Hou P Kovaacuteč
551 Reductive Amination ndash A Convenient Method for Generating Diverse Mono-Functionalised 5101520-Tetraphenyl Porphyrins C Welch S J Archibald R W Boyle
557 Highly Regioselective Preparation of 13-Dioxolane-4-methanol Derivatives from Glycerol Using Phosphomolybdic Acid N W Fadnavis R Gowrisankar G Ramakrishna M K Mishra G Sheelu
561 Rapid Synthesis of 3-Aminoisoquinoline-5-sulfonamides Using the BuchwaldndashHartwig Reaction N Proisy S Taylor A Nelson I Collins
567 Synthesis of Divalent 22-Linked Mannose Derivatives by Homodimerization F S Ekholm M Polaacutekovaacute A J Pawłowicz R Leino
577 Efficient Synthesis of Substituted Cyclic α-Aminophosphonates I L Odinets O I Artyushin N Shevchenko P V Petrovskii V G Nenajdenko G-V Roumlschenthaler
583 Methylated Imidazolinium-Dithiocarboxylates Two Representatives of a New Class of Ionic Liquids A Blanrue R Wilhelm
587 An Efficient Route to 1-Vinylpyrrole-2-carbaldehydes A I Mikhaleva A V Ivanov E V Skitalrsquotseva I A Ushakov A M Vasilrsquotsov B A Trofimov
591 A Regioselective Route to 5-Substituted Isoxazole- and Isoxazoline-3-phosphonates P Conti A Pinto L Tamborini P Dunkel V Gambaro G L Visconti C De Micheli
597 Solvent-Free One-Pot Conjugate Addition of Benzyl Bromides to β-Nitroalkenes Mediated by Magnesium Powder W Shi J-X Wang
602 Synthesis of 234-Trideoxy-44-difluoro-D-ribo-hexopyranose Adenosines J Xu X Zhang X-L Qiu F-L Qing
609 Synthesis of anti-27-Disubstituted Norbornadienes G C Tsui P Le Marquand A Allen W Tam
620 Novel Peptide Mimetic Inhibitors of Hepatitis C Serine Protease Derived from Isomannide T G Barros S Pinheiro J S Williamson A Tanuri H S Pereira R M Brindeiro J B A Neto O A C Antunes E M F Muri
627 A Practical Synthesis of α-Substituted tert-Butyl Acrylates from Meldrumrsquos Acid and Aldehydes C G Frost S D Penrose R Gleave
636 A New Class of Troumlgerrsquos Base Analogues Bearing Spiro[45] Lactone Straps A B Mahon D C Craig A C Try
643 A New Approach to Di- and Tetrasubstituted 23-Dihydropyridin-4(1H)-ones through Aza-DielsndashAlder Reaction Promoted by Silicon Tetrachloride A Massa V de Sio R Villano M R Acocella L Palombi G Sellitto A Peduto R Filosa P De Capraris A Scettri
650 Palladium-Catalysed Direct Arylation of Sydnones A Rodriguez W J Moran
655 Synthesis of (ndash)-Monomorine I R W Bates P Song 660 Cobalt(II) Chloride HexahydratendashDiisopropylamine Catalyzed Mild and
Chemoselective Reduction of Carboxylic Esters with Sodium Borohydride A R Jagdale A S Paraskar A Sudalai
665 Synthesis of Bi- and Tricyclic αβ-Unsaturated Lactams as Potential Michael Acceptors Starting from Heterocyclic Imines K Schulz M Watzke K Johannes P Ullrich J Martens
674 An Expedient Synthesis of Bis-Fused Benzofuran and a Two-Directional Ring-Closing Metathesis for the Synthesis of Bisbenzoxepines and Bisbenzoxocines K C Majumdar B Chattopadhyay S Chakravorty
681 Palladium-Catalyzed Cross-Couplings of Unsaturated Halides Bearing Relatively Acidic Hydrogen Atoms with Organozinc Reagents Z Dong G Manolikakes J Li P Knochel
687 Synthesis of Enantioenriched aa-Disubstituted Cyclopentenes Catalyzed by N-Heterocyclic Carbenes E M Phillips M Wadamoto K A Scheidt
XVII Forthcoming Articles
No 5 691 Transannulation Reactions in the Synthesis of Natural Products
P A Clarke A T Reeder J Winn 710 Synthesis of DL-erythro-Sphingosine Using a Tethered
Aminohydroxylation Reaction as the Key Step J A Morales-Serna Y Diacuteaz M I Matheu S Castilloacuten
713 Convenient Multigram Synthesis of 4-Chloropyridine-26-dicarbonyl Dichloride K Mitsui J R Parquette
715 A Novel and Efficient Synthesis of Dihydrexidine J P Cueva D E Nichols
721 Synthesis of 57-Dichloro-6-azaindoles and Functionalization via a Highly Selective LithiumndashChlorine Exchange N Lachance L-P Bonhomme-Beaulieu P Joly
731 A Convenient Synthesis of Fluorinated Pyrazolo[34-b]pyridine and Pyrazolo[34-d]pyrimidine Nucleosides V O Iaroshenko D V Sevenard A Kotljarov D M Volochnyuk A O Tolmachev V Y Sosnovskikh
741 Diastereoselective Synthesis of γ-Amino Acids and Their Derivatives from Nitroethane via Intermediacy of 56-Dihydro-4H-12-oxazines Bearing the CH2CH(CO2Me)2 Substituent at C3 A Y Sukhorukov A V Lesiv Y A Khomutova S L Ioffe
755 Synthesis of a New Pyrrolopyridoindole and Its Pyrrolopyridobenzimidazole Regioisomer F Bouchikhi M Sassatelli F Anizon M Prudhomme P Moreau
759 Practical Syntheses of Sphingosine-1-Phosphate and Analogues V Blot U Jacquemard H-U Reissig B Kleuser
767 A Facile Synthetic Route towards Substituted Thieno[32-e]indoles W Van Snick W Nulens S Jambon W Dehaen
775 Microwave-Assisted One-Pot Synthesis of (Aminoalkyl)naphthols and (Aminoalkyl)quinolinols by Using Ammonium Carbamate or Ammonium Hydrogen Carbonate as Solid Ammonia Source I Szatmaacuteri F Fuumlloumlp
779 Enantioselective Synthesis of Flavan-3-ols Using a Mitsunobu Cyclization K Krohn I Ahmed M John 787 Synthesis of a Novel γ-Folic AcidndashNτ-Histidine Conjugate Suitable for
Labeling with 99mTc and 188Re C Sparr U Michel R E Marti C Muumlller R Schibli R Moser V Groehn
793 Palladium-Catalyzed Intramolecular Biaryl Coupling A Highly Efficient Avenue for Benzannulated Pyranoquinolines and Julolidine Derivatives K C Majumdar A Taher P Debnath
801 Preparation of NN-Dimethyl-N-Arylureas Using SS-Dimethyl Dithiocarbonate as a Carbonylating Reagent I Degani R Fochi C Magistris M Migliaccio
809 Versatile Selective α-Carboxylic Acid Esterification of N-Protected Amino Acids and Peptides by Alcalase T Nuijens C Cusan J A W Kruijtzer D T S Rijkers R M J Liskamp P J L M Quaedflieg
815 Efficient Palladium-Catalyzed Amination of Aryl Chlorides Using Dicyclohexylamino[(26-dimethyl)morpholino]phenylphosphine as a PN2 Ligand S-E Park S B Kang K-J Jung J-E Won S-G Lee Y-J Yoon
824 A Clean Facile and Stereospecific Synthesis of α-Oxoketene OS-Acetals in Water Y Li Q Zhang X Cheng Q Liu X Xu
829 Sonogashira Cross-Coupling Reactions and Construction of the Indole Ring System Using a Robust Silica-Supported Palladium Catalyst E Tyrrell L Whiteman N Williams
836 Synthesis of Angular 78-Pyridazinocoumarins via the Transformation of a Hydroxy Group into a Carbonyl Group A Kotali I S Lafazanis P A Harris
841 Synthesis of New Cyclic and Acyclic 5-Halouridine Derivatives as Potential Antiviral Agents M F Elshehry J Balzarini C Meier
848 Dendritic Triphenylmethylium and Tetraphenylmethane Compounds H Meier S Kim A Oehlhof
853 Synthesis of Homoallylic Alcohols via Lewis Acid Assisted Enantioselective Desymmetrization B Yu F Menad N Isono M Lautens
860 Diastereoselective Synthesis of 123-Trisubstituted Indanes via Rhodium(I)-Catalyzed Tandem Conjugate Additions C Navarro A G Csaacutekyuml
864 Bakerrsquos Yeast for Sweet Dough Enables Large-Scale Synthesis of Enantiomerically Pure Bicyclo[331]nonane-26-dione C J Wallentin E Orentas E Butkus K Waumlrnmark
868 Addendum and Erratum XV Forthcoming Articles
No 6 869 Stereoselective Transformations of meso Bicyclic Hydrazines Versatile
Access to Functionalized Aminocyclopentanes C Bournaud F Chung A P Luna M Pasco G Errasti T Lecourt L Micouin
888 Synthesis of Glycoaminoxy Acids as Novel Sugar Building Blocks A Malapelle R Ramozzi J Xie
891 Electrophilic ipso-Halocyclization of N-Arylpropynamides with Polyfluoroalkyl Alcohols Selective Synthesis of 8-(Polyfluoroalkoxy) azaspiro[45]trienes Z-Q Wang B-X Tang H-P Zhang F Wang J-H Li
903 Electrooxidation of Alcohols in N-Oxyl-Immobilized Silica GelWater Disperse System Approach to Totally Closed System M Kuroboshi K Goto H Tanaka
909 Synthetic Routes to Aminotriamantanes Topological Analogues of the Neuroprotector Memantinereg A A Fokin A Merz N A Fokina H Schwertfeger S L Liu J E P Dahl R K M Carlson P R Schreiner
913 Parallel Synthesis of Drug-like 5-Amino-Substituted 124-Thiadiazole Libraries Using Cyclization Reactions of a Carboxamidine Dithiocarbamate Linker J Y Park I A Ryu J H Park D C Ha Y-D Gong
921 Copper-Catalyzed Selective S-Arylation of 12-Bis(o-amino-1H-pyrazolyl) Disulfides with Arylboronic Acids P-S Luo F Wang J-H Li R-Y Tang P Zhong
929 2-Iodoxybenzoic AcidTetraethylammonium BromideWater An Efficient Combination for Oxidative Cleavage of Acetals C Kuhakarn W Panchan S Chiampanichayakul N Samakkanad M Pohmakotr V Reutrakul T Jaipetch
935 Synthesis of Quinonoid Analogues of Diospyrin S Sagar I R Green 941 A One-Pot Method for the Iodination of Aryl Amines via Stable Aryl
Diazonium Silica Sulfates Under Solvent-Free Conditions A Zaroi A R Hajipour L Khazdooz
945 Poly(NN-dichloro-N-ethylbenzene-13-disulfonamide) and NNNN-Tetrachlorobenzene-13-disulfonamide as Novel Reagents for the Synthesis of N-Chloroamines Nitriles and Aldehydes R Ghorbani-Vaghei H Veisi
951 Synthesis of an (R)-Garner-type Aldehyde from L-Serine Useful Building Block for a (+)-Furanomycin Derivative G Bartoli G Di Antonio R Fiocchi S Giuli E Marcantoni M Marcolini
957 An Efficient and Highly Selective Synthesis of (Z)-Fluoroenol Phosphates from Hydroxy Difluorophosphonates P Beier R Pohl A V Alexandrova
963 Iodine-Catalyzed Three-Component Reaction A Rapid Synthesis of α-Alkoxy Azides and Homoallyl Ethers J S Yadav B V S Reddy G M Reddy R Narender
969 Rhodium(I)-Catalyzed Cycloisomerization of 13-Dienes with Alkenes in a Tether Y Oonishi A Saito M Mori Y Sato
980 Synthesis of New Optically Active D-GlucosaminendashPyrrole Derivatives B A Frontana-Uribe M V Escaacutercega-Bobadilla J Juaacuterez-Lagunas R A Toscano G A Garciacutea de la Mora M Salmoacuten
985 Partially Saturated Indeno[12-b]indole Derivatives via Deoxygenation of Heterocyclic α-Hydroxy-NO-hemiaminals H-J Hemmerling G Reiss
1000 Light-Induced Synthesis of Π-Extended Tetrathiafulvalenes Incorporating Ferrocenes An Efficient Route for the Synthesis of Electron-Donor Materials A A O Sarhan C Bolm
1007 Preparation of Nβ-Fmoc-Protected Aza-β3-Amino Acids with Nonproteinogenic Hydrophobic Side Chains for Solid-Phase Syntheses of Pseudopeptides M Laurencin P Bauchat M Baudy-Flocrsquoh
1014 Diastereomeric (η4-diene)Fe(CO)3 Complexes Containing Chiral Amide Groups A Convenient Method for the Resolution of Amino Acids M Schumacher G Coste L Miesch
1021 Palladium-Catalysed Heck Reactions of Alk-1-en-3-ones with Aryl Bromides A Very Simple Access to (E)-1-Arylalk-1-en-3-ones M Lemhadri Y Fall H Doucet M Santelli
1036 An Improved Process for the Synthesis of 4H-Imidazo[15-α][14]benzodiazepines J Yang Y Teng S Ara S Rallapalli J M Cook
1041 Meta- and Para-Difunctionalization of Arenes via an Ortho-Magnesiation and a Subsequent SulfoxidendashMagnesium Exchange L Melzig C B Rauhut P Knochel
XIII Forthcoming Articles
No 7 1049 Catalytic Transformations of Benzylic Carboxylates and Carbonates
R Kuwano 1062 A Simple and Practical Method for the Oxidation of Thebaine to 14-
Hydroxycodeinone by V2O5ndashH2O2 S Das Sharma D Konwar 1065 Umpolung with Sulfur Dioxide CarbonndashCarbon Cross-Coupling of Electron-
Rich 13-Dienes and Alkenes Application to the Enantioselective Synthesis of Long-Chain Polyketide Fragments M Turks C J Exner C Hamel P Vogel
1075 One-Pot Synthesis of 14-Diarylnaphthalenes via a WittigndashHorner Reaction[4+2] CycloadditionDehydrogenation Sequence Z Chen W Shou Y Wang
1081 A Novel and General Method for the Formation of S-Aryl Se-Aryl and Te-Aryl Phosphorochalcogenoates Y-X Gao G Tang Y Cao Y-F Zhao
1087 A Remarkable Access to γ-Fluoroalkylated Propargylamine Derivatives or Fluoroalkylated Dihydroisoxazoles via the Reaction of Fluoroalkylated Acetylides with Various Nitrones T Konno K Moriyasu T Ishihara
1095 Short and Practical Syntheses of (S)-(+)-3-(p-Tolylsulfinyl)furan-2(5H)-one and (S)-(+)-3-(p-Tolylsulfinyl)-56-dihydropyran-2-one D Cruz Cruz A Hernaacutendez Linares F Yuste M R Martiacuten J L Garciacutea Ruano
1099 Decarboxylative Aldol-Type Reaction of 2-(Trifluoroacetyl)-13-diazoles with Activated Acetic Acids P V Khodakovskiy D M Volochnyuk A A Tolmachev
1105 Synthesis of 2-[(Arylmethylene)amino]cyclopropanecarbonitriles via a Two-Step Ring Transformation of 2-(Cyanomethyl)aziridines S Mangelinckx M Drsquohooghe S Peeters N De Kimpe
1113 Synthesis of Dendrimeric Tumor-Associated Mucin-Type Glycopeptide Antigens T Becker A Kaiser H Kunz
1123 A Simple and Efficient Oxidation Procedure for the Synthesis of Acid-Sensitive Epoxides O Bortolini G Fantin M Fogagnolo
1127 Rapid Chemoselective Deprotection of Benzyl Esters by Nickel Boride J M Khurana R Arora
1131 Three-Component Coupling of Isoquinoline Activated Alkyne and Nitromethane A Facile Synthesis of Nitromethyl Derivatives of 12-Dihydroisoquinolines J S Yadav B V S Reddy N N Yadav M K Gupta
1137 Palladium Supported on a Polyionic Resin as an Efficient Ligand-Free and Recyclable Catalyst for Heck SuzukindashMiyaura and Sonogashira Reactions B Basu S Das P Das B Mandal D Banerjee F Almqvist
1147 Oxidation of 25-Dialkylpyrrole Derivatives with Cerium(IV) Ammonium Nitrate R Voloshchuk M Gałęzowski D T Gryko
1153 Practical Syntheses of Enantiomerically Pure Key Intermediates of Opioid Receptor-like 1 (ORL1) Antagonists T Yoshizumi A Ohno T Tsujita H Takahashi O Okamoto I Hayakawa H Kigoshi
1163 An Environmentally Benign TEMPO-Catalyzed Efficient Alcohol Oxidation System with a Recyclable Hypervalent Iodine(III) Reagent and Its Facile Preparation X-Q Li C Zhang
1170 Efficient and Stereoselective Rearrangement of BaylisndashHillman Acetates Catalyzed by Gold(I) ChlorideSilver(I) Trifluoromethanesulfonate Y Liu D Mao J Qian S Lou Z Xu Y Zhang
1175 The First Total Synthesis of Kynapcin-24 by Palladium Catalysis L-Y Yang C-F Chang Y-C Huang Y-J Lee C-C Hu T-H Tseng
1180 Enantioselective Synthesis of N-Protected α-Amino Acid Hydrazides M Bibian S El-Habnouni J Martinez J-A Fehrentz
1185 Synthesis of 11H-Indolo[32-c]quinoline-6-carboxylic Acids by Cascade AutoxidationndashRing Contractions A Becker S Kohfeld T Pies K Wieking L Preu C Kunick
1190 Reaction of N-Nonaflylbenzotriazole with Silyl Enol Ethers M Uhde T Ziegler
1195 2-(Benzoylimino)thiazolidin-4-ones Formation by an Alternative Ring Closure and Analysis of Rotational Barriers H-G Haumlcker P W Elsinghorst S Michels J Daniels G Schnakenburg M Guumltschow
1204 Microwave-Assisted Synthesis and Functionalization of Selenolopyrimidines S Hesse C Chenet D Thomae G Kirsch
1209 12-Disubstituted 4-Quinolones via Copper-Catalyzed Cyclization of 1-(2-Halophenyl)-2-en-3-amin-1-ones R Bernini S Cacchi G Fabrizi A Sferrazza
1220 A New Atom-Economical and Selective Synthesis of Secondary and Tertiary Alkylamines by Means of CpIridium Complex Catalyzed Multiple N-Alkylation of Ammonium Salts with Alcohols without Solvent R Yamaguchi Z Mingwen S Kawagoe C Asai K-i Fujita
1224 Synthesis of Regioisomerically Pure 5-Functionalized 27-Dichlorofluoresceins J C Castro A Malakhov K Burgess
XIII Forthcoming Articles
No 8 1227 Michael Additions to Activated Vinylphosphonates T Janecki J Kędzia
T Wąsek 1255 A Facile and General Synthesis of 2β-Aminosteroids X Ke H Hu
D Zhou W Xu Q Zhu N P Reddy X Hu 1261 Efficacious Preparation of Oppolzerrsquos Glycylsultam via the Deleacutepine
Reaction A Isleyen C Gonsky R C Ronald P Garner 1265 Synthesis of Masked Vicinal Amino Aldehydes of Pyrrolizine and Pyrrolo
[12-c]thiazole Series A V Tverdokhlebov A V Denisenko A A Tolmachev Y M Volovenko S V Shishkina O V Shishkin
1271 Preparation of 9-Substituted Pyridine-Stretched Adenines and Hypoxanthines J A Crawford W Fraser C A Ramsden
1279 A Versatile Synthesis of Heterocyclic Analogues of Neoflavonoids from Enamino Ketones V S Moskvina V P Khilya O V Turov U M Groth
1287 New Stereoselective Synthesis of Paeonilactone B F G Gatti S Serra 1291 The Use of NN-Dialkyltrimethylsilylamines in the Synthesis of
Pentamethinium Salts M Kořiacutenek M Rybaacutečkovaacute Boumlhm 1297 Synthesis of Triazoles via Regioselective Reactions of Aryl Azides with
Cyanoacetyl Pyrroles and Indoles N T Pokhodylo V S Matiychuk M D Obushak
1301 Gallium(III) Chloride Catalyzed Hydroarylation of Arylacetylenes with Naphthols and Phenols A Facile Synthesis of Vinylarenes J S Yadav B V S Reddy S Sengupta S K Biswas
1305 Electrophilic Bromination of meta-Substituted Anilines with N-Bromosuccinimide Regioselectivity and Solvent Effect S Bartoli A Cipollone A Squarcia A Madami D Fattori
1309 Cross-Coupling Reactions of Halopurines with Aryl- and Alkyltrifluoroborates The Scope and Limitations in the Synthesis of Modified Purines Z Hasniacutek R Pohl M Hocek
1318 A Convenient Method for Converting Hydroxyacetophenones into Their Ethylene or Trimethylene Acetals F Ono H Takenaka T Fujikawa M Mori T Sato
1323 γ-Chloromagnesio γ-Lactones and δ-Chloromagnesio δ-Lactones Generation Properties and Synthetic Uses H Shimizu S Fukuda S Sugiyama T Satoh
1336 Click Reactions with Nitroxides T Kaacutelai W L Hubbell K Hideg 1341 Synthesis of Novel 14-Benzoquinone-Containing 123-Triazoles An Entry
Into a New Library F Algi M Balci 1348 Efficient Synthesis of Two Sialylated Tetrasaccharides Found in Goat Milk
P K Mandal A K Misra 1355 Dendrimers of Vaccines Consisting of Tumor-Associated Glycopeptide
Antigens and T Cell Epitope Peptides S Keil A Kaiser F Syed H Kunz
1370 IBXTBAB-Mediated Oxidation of Primary Amines to Nitriles F Drouet P Fontaine G Masson J Zhu
1375 Chemoselectivity of Multicomponent Condensations of Barbituric Acids 5-Aminopyrazoles and Aldehydes E A Muravyova S V Shishkina V I Musatov I V Knyazeva O V Shishkin S M Desenko V A Chebanov
1386 Stereoselective Total Syntheses of Leiocarpin A and (ndash)-Galantinic Acid Starting from D-Mannitol K Nagaiah D Sreenu K V Purnima R S Rao J S Yadav
1393 A Facile Mild Deprotection Protocol for 13-Dithianes and 13-Dithiolanes with 30 Hydrogen Peroxide and Iodine Catalyst in Aqueous Micellar System N C Ganguly S K Barik
1400 Rhodium-Catalyzed Gram-Scale Synthesis of Highly Substituted Pyridine Derivatives K Parthasarathy C-H Cheng
1403 Enantioselective Synthesis of (R)-Propylene Carbonate from Ethyl (S)-Lactate J M Whitaker R C Ronald
XIII Forthcoming Articles
no 9 1405 Transition-Metal-Catalyzed Site-Selective Cross-Coupling of Di- and
Polyhalogenated Compounds J-R Wang K Manabe 1428 An Improved Synthesis of (4-4-Hydroxy-3-isopropyl-5-[(4-nitrophenyl)
ethynyl]benzyl-35-dimethylphenoxy)acetic Acid (NH-3) M B Gopinathan K S Rehder
1431 Copper-Catalyzed Tandem CndashN Bond Formation Reaction Selective Synthesis of 2-(Trifluoromethyl)benzimidazoles M-W Chen X-G Zhang P Zhong M-L Hu
1437 Synthesis and Thermochemical Properties of Stereoisomeric Dihydroxy- and Tetrahydroxyalkylammonium Salts M Thomas L Rothman J Hatcher P Agarkar R Ramkirath S Lall-Ramnarine R Engel
1445 Preparation of 5-Substituted 2-(2-Alkylaryl-1H-imidazol-4-yl)oxazoles and 5-Substituted 2-(2-Alkylarylthiazol-4-yl)oxazoles by Utilizing 5-Substituted 2-(2-Bromo-11-diethoxyethyl)oxazole as a Synthon D R St Laurent J L Romine
1459 Novel and Efficient Methods for the Synthesis of Symmetrical Trisulfides A Kertmen S Lach J Rachon D Witt
1463 An Environmentally Benign Electrochemical Process for the Reduction of Carboxylic Acid Hydrazides to Amides M Mentel M J Beier R Breinbauer
1469 Synthesis of 1-Chloroalkynes from Alkynylsilanes Using Trichloroisocyanuric Acid as Chlorinating Agent M H Vilhelmsen A S Andersson M B Nielsen
1473 A Convenient Approach to Enantioenriched Cyclopropanes Bearing Electron-Withdrawing Functionalities H Krawczyń K Wąsek J Kędzia
1477 Synthesis of Cyclopropenes via 12-Elimination of Bromocyclopropanes Catalyzed by Crown Ether W M Sherrill R Kim M Rubin
1485 A Base-Catalysed One-Pot Three-Component Coupling Reaction Leading to Nitrosubstituted Pyrroles I R Baxendale C D Buckle S V Ley L Tamborini
1494 Synthesis of 4-Alkylidene-4H-31-benzoxazine Derivatives by Acid-Catalyzed Cyclization of 2-Isocyanophenyl Ketones in the Presence of a Vinyl Ether K Kobayashi Y Okamura H Konishi
1499 Synthesis of Higher Helicenes via Olefin Metathesis and CndashH Activation J Cocircteacute S K Collins
1506 Azido- and Ethynyl-Substituted 2262-Terpyridines as Suitable Substrates for Click Reactions A Winter A Wild R Hoogenboom M W M Fijten M D Hager R-A Fallahpour U S Schubert
1513 Synthesis of 2-(Arylamino)ethanethiols via Lewis Acid Catalyzed Aminolysis of 22-Dimethylthiirane as Precursors of the 14-Benzothiazine Nucleus R Spogli S Sabatini G Manfroni O Tabarrini V Cecchetti
1520 Iron(III) Chloride A Versatile Catalyst for the Practical Synthesis of 3-Sulfenylindoles J S Yadav B V S Reddy Y J Reddy K Praneeth
1525 Organocatalytic Enantioselective Conjugate Addition of 2-Fluoromalonate to Nitroolefins Direct Synthesis of Chiral Fluorinated γ-Nitro Carboxylic Acid Derivatives H Li L Zu H Xie W Wang
1531 Asymmetric Transfer Hydrogenation of Ketimines with Trichlorosilane Structural Studies Z Zhang P Rooshenas H Hausmann P R Schreiner
1545 Prolinol Sulfinyl Ester Derivatives Organocatalytic Michael Addition of Ketones to Nitroolefins under Neat Conditions X Zeng G Zhong
1551 Asymmetric Oxidations of Electron-Poor Alkenes Promoted by the β-Amino AlcoholTBHP System A Russo A Lattanzi
1557 Enantioselectivity Switch in Direct Asymmetric Aminoxylation Catalyzed by Binaphthyl-Based Chiral Secondary Amines T Kano A Yamamoto F Shirozu K Maruoka
1564 Enantioselective Conjugate Addition of N-Heterocycles to αβ-Unsaturated Ketones Catalyzed by Chiral Primary Amines G Luo S Zhang W Duan W Wang
1573 Sulfonyl Hydrazine as New Functionality in Organocatalysis Camphorsulfonyl Hydrazine Catalyzed Enantioselective Aza-Michael Addition L-Y Chen H He B-J Pei W-H Chan A W M Lee
1578 Conversion of Primary Alcohols and Aldehydes into Methyl Esters by Ruthenium-Catalysed Hydrogen Transfer Reactions N A Owston T D Nixon A J Parker M K Whittlesey J M J Williams
1582 Addendum and Erratum XVII Forthcoming Articles
no 10 1583 Organocatalytic Formation of Quaternary Stereocenters M Bella
T Gasperi 1615 Regioselective Synthesis of 5H-Thiazolo[32-a]pyrimidin-5-ones from
MoritandashBaylisndashHillman Adduct Acetates under Solvent-Free and Base-Free Conditions W Zhong B Guo F Lin Y Liu W Su
1623 First Synthesis of 5-Cyanosalicylates by Formal [3+3] Cyclocondensations of 13-Bis(silyloxy)-13-butadienes A Riahi O Fatunsin M Shkoor R Dede H Reinke C Fischer P Langer
1635 Reaction of Isocyanides Dialkyl Acetylenedicarboxylates and a-Keto Lactones Unexpected Participation of an Ester Carbonyl Group in the Isocyanide-Based Three-Component Reaction A A Esmaeili H Vesalipoor
1639 An Efficient and Chemoselective Synthesis of 16-Naphthyridines and Pyrano[32-c]pyridines under Microwave Irradiation Z-G Han S-J Tu B Jiang S Yan X-H Zhang S-S Wu W-J Hao X-D Cao F Shi G Zhang N Ma
1647 N-Activation of N-Arylimidazoles Facile Syntheses of N-Alkyl-N-arylimidazolium Iodides from Less Expensive Chloro Substrates A M Oertel V Ritleng M J Chetcuti
1651 Synthesis of Polyhalogenated 2-(Phenylamino)pyridines by Thermal Amination Reactions S R Waldvogel A Faust W Barkmann R Froumlhlich O Wolff
1655 Cyanide Ion Promoted Addition of Acylphosphonates to Diethyl Cyanophosphonate Synthesis of Phosphonocyanohydrin O-Phosphates A S Demir A Aybey M Emrullahoglu
1659 Straightforward and Scalable Synthesis of Orthogonally Protected 37-Diazabicyclo[410]heptane H Schramm M Pavlova C Hoenke J Christoffers
1663 Hypervalent Iodine Mediated Oxidation of 12-Diaminobenzimidazole and Its Schiff Bases Efficient Synthesis of 3-Amino-124-benzotriazine and 2-Aryl-124-triazolo[15-a]benzimidazoles A Kumar M Parshad R K Gupta D Kumar
1667 Synthesis of the Reported Protoberberine Gusanlung D P B Wakchaure S Easwar N P Argade
1673 2-(Azidomethyl)arylboronic Acids in the Synthesis of Coumarin-Type Compounds M I Naumov A V Nuchev N S Sitnikov Y B Malysheva A S Shavyrin I P Beletskaya A E Gavryushin S Combes A Y Fedorov
1683 Asymmetric Synthesis of 12-anti-Disubstituted Taurine Derivatives D Enders D Iffland G Raabe
1689 A Novel One-Pot Three-Component Synthesis of 5-Imino-2358-tetrahydropyrazolo[12-a]pyridazin-1-one Derivatives B Qian M-J Fan Y-X Xie L-Y Wu Y Shi Y-M Liang
1694 One-Portion Synthesis of 2-Acetoxy Carbonyl Compounds from Aldehydes by Using an Acetylated Masked Acyl Cyanide H Nemoto T Kawamura K Kitasaki K Yatsuzuka M Kamiya Y Yoshioka
1703 Synthesis of 9-Anthryl Ethers from trans-910-Dihydro-910-dimethoxyanthracene by Acid-Catalyzed Transetherification K S Jang H Y Shin D Y Chi
1708 Efficient Synthesis of Azo Dye Labeled Terpenes Sugars and Steroids Using N-(4-Arylazobenzoyl)-1H-benzotriazoles A R Katritzky S R Tala N E Abo-Dya Z K Abdel-Samii
1715 Tandem CH-ActivationndashImine-Formation Reaction A New Route to Imidazo[21-a]phthalazines A Heim-Riether K R Gipson
1720 A Convenient and Efficient α-Sulfenylation of Carbonyl Compounds E Okragla S Demkowicz J Rachon D Witt
1725 Stereoselective Synthesis of β-Branched Phenylalanine Derivatives via Chelate-Claisen Rearrangement C Quirin U Kazmaier
1732 Catalyst-Free and Base-Free Water-Promoted SNAr Reaction of Heteroaryl Halides with Thiols B Sreedhar P S Reddy M A Reddy
1739 Convenient Methods for Synthesis of C2-Symmetric Diphenyltetrahydrothiophenes M Periasamy G Ramani G P Muthukumaragopal
1744 Highly Diastereoselective Conjugate AdditionndashElimination of Chiral Nickel(II) Glycinate with Activated Allylic Acetates for Asymmetric Synthesis of Glutamic Acid Derivatives J Wang J Shi X Zhang D Lin H Jiang H Liu
1753 Synthesis of 36-Dimethoxybenzene-12-diamine and of 47-Dimethoxy-2-methyl-1H-benzimidazole T Besset C Morin
1757 An Inexpensive Procedure for Reductive Aminations Using Dimethylamineborane on Millimolar and Molar Scale R Ortmann M Schlitzer
1760 Classics in Stereoselective Synthesis Edited by E M Carreira L Kvaerno Reviewed by Rolf Breinbauer
XV Forthcoming Articles
no 11 1761 Transition-Metal-Catalyzed Enantioselective Synthesis of Compounds with
Non-Centrochirality M Ogasawara S Watanabe 1786 One-Pot Synthesis of 3-Acyl-2-(alkylsulfanyl)indoles and 2-(Alkylsulfanyl)-
indole-3-carboxylates from (2-Isocyanophenyl)methyl Ketones or (2-Isocyanophenyl)acetates S Fukamachi H Konishi K Kobayashi
1791 Efficient and Recyclable Phthalocyanine-Based Sensitizers for Photooxygenation Reactions H Xu W-K Chan D K P Ng
1797 A Facile and Practical One-Pot Synthesis of β-Oxo Thioamides from β-Oxo Amides and Isothiocyanates P Huang D Xiang Y Zhou Y Liang T Na D Dong
1801 Microwave-Promoted Solid-Acid-Catalyzed One-Pot Synthesis of Phthalazinones V M Outerbridge S M Landge H Tamaki B Toumlroumlk
1807 Benzylic Brominations with N-Bromosuccinimide in (Trifluoromethyl)-benzene D Suarez G Laval S-M Tu D Jiang C L Robinson R Scott B T Golding
1811 Synthesis of Thioflavanone and Flavanone Derivatives by Cyclization of Chalcones W Konieczny M Konieczny
1815 A New and Expedient Total Synthesis of Ochratoxin A and d5-Ochratoxin A B Gabriele M Attya A Fazio L Di Donna P Plastina G Sindona
1821 Synthesis of Benzopyrrolizidinones by NorrishndashYang Cyclization of 3-(Acylmethyl)-2-alkylisoindol-1-ones J Wu W Zhang C Wang
1829 Reactions of MoritandashBaylisndashHillman Acetates with Huisgen Zwitterions A Novel Strategy for the Synthesis of β-Amino Acid Derivatives A Jose R R Paul R Mohan S C Mathew A T Biju E Suresh V Nair
1834 Peracetylated β-Allyl C-Glycosides of D-Ribofuranose and 2-Deoxy- D-ribofuranose in the Chemical Literature Until Now Mirages in the Literature H Otero Martinez H Reinke D Michalik C Vogel
1841 Core-Tetrasubstituted Naphthalene Diimides by Stille Cross-Coupling Reactions and Characterization of Their Optical and Redox Properties S-L Suraru F Wuumlrthner
1846 A Practical Synthesis of Indole-Based Heterocycles Using an Amidoaluminum-Mediated Strategy R Todd M M Hossain
1851 Synthesis of Fluorinated Pyrrolo[23-b]pyridine and Pyrrolo[23-d]pyrimidine Nucleosides V O Iaroshenko Y Wang D V Sevenard D M Volochnyuk
1858 Recyclization Reactions of 5-Formyl-13-dimethyluracil with Electron-Rich Amino Heterocycles A P Mityuk D M Volochnyuk S V Ryabukhin A S Plaskon A Shivanyuk A A Tolmachev
1865 Facile Synthesis of Fluorinated 1-Desazapurines V O Iaroshenko D V Sevenard D M Volochnyuk Y Wang A Martiloga A O Tolmachev
1876 A Practical Synthesis of 3-Diethoxyphosphoryl-12-pyridazine Derivatives J-C Monbaliu J Marchand-Brynaert
1881 Enantioselective Reduction of Prochiral Ketones Employing Sprouted Pisum sativa as Biocatalyst J S Yadav B V S Reddy C Sreelakshmi A B Rao
1886 Application of Phenolate Ion Mediated Intramolecular Epoxide Ring Opening in the Enantioselective Synthesis of Functionalized 23-Dihydrobenzofurans and 1-Benzopyrans S K Dinda S K Das G Panda
1897 Complementary Synthetic Approaches to Constitutionally Diverse N-Aminoalkylated Isoindolinones Application to the Synthesis of Falipamil and 5-HT1A Receptor Ligand Analogues M Lorion A Couture E Deniau P Grandclaudon
1904 Selective Deprotection of Silyl Ethers with Sodium Periodate J Li D Menche
1909 Micellar Solution of Sodium Dodecyl Sulfate (SDS) Catalyzes KabacknikndashFields Reaction in Aqueous Media S Sobhani A Vafaee
1916 Convenient Methods for the Synthesis of a Library of Hemilabile Phosphines M V Jimeacutenez J J Peacuterez-Torrente M I Bartolomeacute L A Oro
1923 Terminal Aziridines by Addition of Grignard Reagents or Organoceriums to an (α-Chloro)sulfinylimine D M Hodgson J Kloesges B Evans
1933 A Robust Synthesis of Nε-(Carboxymethyl)-L-lysine (CML) R Csuk S Stark A Barthel R Kluge D Stroumlhl
1935 One-Pot Curtius Rearrangement Processes from Carboxylic Acids O Leogane H Lebel
XV Forthcoming Articles
no 12 1941 The Chemistry of Deprotonated α-Aminonitriles T Opatz 1960 An Efficient Synthesis of Tetraalkyl 2345-Thiophenetetracarboxylate
Derivatives A Alizadeh R Hosseinpour 1963 Facile Deprotection of Bulky (Trialkylsilyl)acetylenes with Silver Fluoride
S Kim B Kim J In 1969 Highly Efficient and Reusable Ionic Liquids for the Catalyzed
Hydroamination of Alkenes with Sulfonamides Carbamates and Carboxamides L Yang L-W Xu C-G Xia
1975 Synthesis of 2391016172324-Octasubstituted Phthalocyaninatozinc(II) Complexes Mediated by Reductive Agents G A Gauna A C Monsalvo J Awruch
1979 A Short and Efficient Synthesis of 3-2-[2-(Bromomethyl)thiazol-4-yl]-ethynyl-5-fluorobenzonitrile A Precursor for PET Radioligand [18F]SP203 M B Gopinathan C Jin K S Rehder
1983 Synthesis of a Substituted Benzazepin-2-one Dihydrate S K Boini R K Vaid K P Moder D Mitchell
1987 Synthesis of Novel Trisubstituted Imidazolines F J Lakner M A Parker B Rogovoy A Khvat A Ivachtchenko
1991 A Novel Synthesis of N-But-3-enyl-α- and β-Amino Acids T T Van Nguyen R T C Brownlee A B Hughes
1999 Synthesis of Substituted 5-(3-Hydroxypropyl)pyrrolidin-2-ones and Pyrrolizidinones from Nitroethane via C3 Functionalized 56-Dihydro-4H-12-oxazines A Novel Approach to Some Analogues of the Antidepressant Rolipram A Yu Sukhorukov A V Lesiv Y A Khomutova S L Ioffe V A Tartakovsky
2009 Chiral Cyclobutanols and Cyclopentane Dimers via Samarium(II) Iodide Induced Keto-Olefin Cyclisations of Carbohydrate-Derived Unsaturated Ketones D B G Williams J Caddy K Blann J J C Groveacute C W Holzapfel
2015 Synthesis of Perfluoroalkylthio-Substituted Ferrocenes C Rhode J Lemke M Lieb N Metzler-Nolte
2019 Functionalization of Polyhedral Oligomeric Silsesquioxane (POSS) via Nucleophilic Substitution M Dutkiewicz H Maciejewski B Marciniec
2025 A Novel Synthesis of Aryl Mesylates via One-Pot DemethylationndashMesylation of Aryl Methyl Ethers Using a Mixture of Phosphorus Pentoxide in Methanesulfonic Acid B Kaboudin Y Abedi
2029 Anionic Cyclization of (NN-Dimethylamino)[2-(prop-2-yn-1-yloxy)aryl]-acetonitriles T Zdrojewski J Musielak A Jończyk
2035 Strecker-Type Reaction Catalyzed by Carboxylic Acids in Aqueous Media Z Xie G Li G Zhao J Wang
2040 Synthesis of Novel Structurally Simplified Estrogen Analogues with Electron-Donating Groups in Ring A L F Tietze C A Vock I K Krimmelbein L Nacke
2061 On the Resolution of Secondary Phosphine Oxides via Diastereomeric Complex Formation The Case of tert-Butylphenylphosphine Oxide J Holt A M Maj E P Schudde K M Pietrusiewicz L Sieroń W Wieczorek T Jerphagnon I W C E Arends U Hanefeld A J Minnaard
2066 Enantioselective Copper-Catalyzed Conjugate Addition of Dimethylzinc to 5-(1-Arylalkylidene) Meldrumrsquos Acids A Wilsily T Lou E Fillion
2073 SuzukindashMiyaura Coupling Reactions Using Phosphite Ligands M Jang Y Jo I-K Oh H M Jung S Lee
2076 Synthesis of 2-Methylindoline- and 2-Methyl-1234-tetrahydroquinoline-Derived Phosphoramidites and Their Applications in Iridium-Catalyzed Allylic Alkylation of Indoles W-B Liu H He L-X Dai S-L You
2083 Stereocontrolled Synthesis of 13-Amino Alcohols by Reduction of Substituted 2-1-[(tert-Butylsulfinyl)amino]alkylcyclohexanones J C Gonzaacutelez-Goacutemez F Foubelo M Yus
2089 Tunable Phosphoramidite Ligands for Asymmetric Hydrovinylation Ligands par excellence for Generation of All-Carbon Quaternary Centers C R Smith H J Lim A ZhangT V RajanBabu
2101 Copper-Catalyzed Asymmetric Ring-Opening Reaction of Oxabenzonorbornadienes with Grignard and Aluminum Reagents R Millet L Gremaud T Bernardez L Palais A Alexakis
2113 A Simplified Synthesis of Takemotorsquos Catalyst A Berkessel B Seelig 2116 Pharmaceutical Substances Syntheses Patents and Applications of the
Most Relevant AIPs Edited by Axel Kleeman Juumlrgen Engel Bernhard Kutscher Dietmar Reichert Reviewed by I Agranat
XV Forthcoming Articles
no 13 2117 Recent Advances in the Aza-Claisen Rearrangement K C Majumdar
T Bhattacharyya B Chattopadhyay B Sinha 2143 A Novel and Convenient Synthesis of lsquoReversedrsquo Diamidino 25-Aryl- and
25-Azaheterocycle-Substituted Furans L Hu D W Boykin 2146 Efficient and General Preparation of Pyranostilbenes First Total Synthesis
of Artocarbene and Pawhuskin B B H Park Y R Lee W S Lyoo 2155 Mild Oxidation of Diarylacetylenes to 12-Diketones Using Oxone in
Trifluoroacetic Acid J-H Chu Y-J Chen M-J Wu 2163 One-Pot Microwave-Assisted Selective Azido ReductionTandem Cyclization
in Condensed and Solid Phase with Nickel Boride N Shankaraiah N Markandeya M Espinoza-Moraga C Arancibia A Kamal L Silva Santos
2171 Pyrrolo[321-ij]quinolin-4-one and Pyrrolo[321-ij]quinolin-6-one H McNab D J Nelson E J Rozgowska
2175 Practical Synthesis of 5-Substituted Tetrazoles under Microwave Irradiation J Roh T V Artamonova K Vaacutevrovaacute G I Koldobskii A Hrabaacutelek
2179 A Simple Method for the Synthesis of 3-Arylthieno[23-b]pyridines via Iodine-Mediated Cyclization of 3-(1-Arylalkenyl)-2-[(1-phenylethyl)sulfanyl]pyridines K Kobayashi D Nakamura Y Shiroyama S Fukamachi H Konishi
2184 Synthesis of Four Lysine-Linked Cereulide Analogues Showing Ionophoric Activity Towards Potassium Cations as Lead Compounds for Emetic Toxin-Detection by Immunoassays A Makarasen T Nishikawa M Isobe
2205 Synthesis of α-Aliphatic and β-Aromatic Substituted Taurines via Regioselective Ring Opening of Thiiranes with Ammonia H Yu S Cao L Zhang G Liu J Xu
2210 Stability of 5(6)-Carboxyfluorescein in Microwave-Assisted Synthesis of Fluorescein-Labelled O-Dimannosylated Peptides R Kowalczyk P W R Harris R P Dunbar M A Brimble
2223 Diversity-Oriented Synthesis of Functionalized Diaryl Sulfones by Regioselective [3+3] Cyclizations of 13-Bis(siloxy)buta-13-dienes with 2-(Arylsulfonyl)-3-ethoxy-2-en-1-ones Scope and Limitations M Shkoor A Riahi O Fatunsin H Reinke C Fischer P Langer
2236 Synthesis of Functionalized Salicylates by Formal [3+3] Cyclocondensation of 13-Bis(silyloxy)buta-13-dienes with 3-Alkoxy-2-en-1-ones G Mroszlig S Ladzik H Reinke A Spannenberg C Fischer P Langer
2249 Synthetic Approach to Alkoxy-β-(trifluoromethyl)styrenes and Their Application in the Synthesis of New Trifluoromethylated Heterocycles V M Muzalevskiy V G Nenajdenko A V Shastin E S Balenkova G Haufe
2260 o-Benzenedisulfonimide as a Powerful and Recyclable Organocatalyst for the Nazarov Reaction M Barbero S Cadamuro A Deagostino S Dughera P Larini E G Occhiato C Prandi S Tabasso R Vulcano P Venturello
2267 The Catalytic Potential of 4-Guanidinylpyridines in Acylation Reactions I Held E Larionov C Bozler F Wagner H Zipse
2278 Iron(III) Chloride in EthanolndashWater Highly Efficient Catalytic System for the Synthesis of Garcia Gonzalez Polyhydroxyalkyl- and C-Glycosylfurans L Nagarapu M V Chary A Satyender B Supriya R Bantu
2283 Ruthenium-Catalyzed Addition of Primary Amides to Alkynes A Stereoselective Synthesis of Secondary Enamides L J Gooszligen M Blanchot K S M Salih K Gooszligen
2289 Binaphthyl-Modified Quaternary Phosphonium Salts as Chiral Phase Transfer Catalysts Application to Asymmetric Amination of β-Keto Esters R He K Maruoka
X Table of Contents XI Forthcoming Articles
no 14 2293 Direct Methods for Stereoselective Polypropionate Synthesis A Survey
J Li D Menche 2316 Synthesis of Symmetrical Ketones from Grignard Reagents and
11-Carbonyldiimidazole D Bottalico V Fiandanese G Marchese A Punzi
2319 Synthesis of 45-Substituted Imidazoles by a Fast Condensation of 12-Diketones and Urotropine in Heterogeneous Medium G Bratulescu
2321 (Arylsulfonyl)acetones and -acetonitriles New Activated Methylenic Building Blocks for Synthesis of 123-Triazoles N T Pokhodylo V S Matiychuk M D Obushak
2324 A Safe Convenient and Efficient One-Pot Synthesis of α-Chloroketone Acetals Directly from Ketones Using Iodobenzene Dichloride J Yu C Zhang
2329 An Efficient Oxidative Conversion of Aldehydes into 2-Substituted 2-Oxazolines Using 13-Diiodo-55-dimethylhydantoin S Takahashi H Togo
2333 A Novel Procedure for the Synthesis of Benzo[b][18]naphthyridine-3-carboxylate Derivatives from MoritandashBaylisndashHillman Adduct Acetates W Zhong F Lin R Chen W Su
2341 An Improved Synthesis of 147-Triazacyclononanes (tacns) and 14710-Tetraazacyclododecanes (cyclens) J Huang Z Zhou T H Chan
2345 The Ullmann Coupling between 2-Chlorobenzoic Acids and Amino Acids A Valuable Reaction for Preparing 2-Substituted 1-Acetyl-1H-indol-3-yl Acetates J C Rodriguez Dominguez X Gang G Kirsch
2349 gem-Dibromomethyl Aromatics Efficient Aldehyde Equivalents in the KnoevenagelndashDoebner Reaction J K Augustine Y A Naik S Poojari N Chowdappa B S Sherigara K Areppa
2357 Synthesis of Novel α-Aminophosphonates Containing Adamantyl Fragment M M Kabachnik L I Minaeva I P Beletskaya
2361 Efficient Fluoride-Mediated Synthesis of 5-Amino-Substituted Isothiazoles Y S Zubenko V I Potkin
2365 Phosphine-Catalyzed Reaction of Cyanohydrins with Activated Alkynes A Siby O Loreau F Taran
2371 Sulfanyl-Substituted [3]Cumulenes and Buta-13-dienes from a Tetrakis(pyridinium)-Substituted Butadiene A Schmidt A Rahimi M Gjikaj
2379 Efficient Synthesis of 2-Substituted Pyrido[32-d]pyrimidines Involving SNAr and Palladium-Catalyzed Cross-Coupling Reactions A Tikad S Routier M Akssira J-M Leacuteger C Jarry G Guillaumet
2385 Novel Synthesis of Medium-Sized Heterocycles by Palladium-Catalyzed Intramolecular Heck Reaction via 9-endo-trig Mode of Cyclization K C Majumdar B Chattopadhyay
2393 Facile Synthesis of Fluorinated Benzofuro- and Benzothieno[23-b]pyridines α-Carbolines and Nucleosides Containing the α-Carboline Framework V O Iaroshenko Y Wang B Zhang D Volochnyuk V Ya Sosnovskikh
2403 Synthesis of Functionalized N-Vinyl Nitrogen-Containing Heterocycles S M M Lopes A M Beja M Ramos Silva J A Paixatildeo F Palacios T M V D Pinho e Melo
2408 Kumada Cross-Coupling of Aryl Grignard Reagents with Aryl Halides Catalyzed by an Immobilized Nickel Catalyst X Chen L Wang J Liu
2413 Highly Enantioselective Synthesis of Heteroaromatic Alcohols Catalyzed by Chiral DiaminodiphosphinendashRuthenium(II) Complexes W-Y Shen Y-Y Li Z-R Dong J-X Gao
2418 Concise Total Synthesis of (+)-Disparlure and its trans-Isomer Using Asymmetric Organocatalysis S-G Kim
2423 Rhodium Carbenoid Induced [12]-Migration in an L-Lyxo-Configured α-Diazo β-Keto Ester Synthesis of a New Griseolic Acid Analogue N N Bhujbal K S A Kumar D D Dhavale
2430 Synthesis of 5-Arylthio-3-hydroxyphthalates by the First [4+2] Cycloadditions of 3-Arylthio-1-silyloxy-13-butadienes with Dimethyl Acetylenedicarboxylate I Iqbal M Imran P Langer
2435 Synthesis of Highly Functionalized Proline Derivatives via a One-Pot MichaelSN-AdditionCyclization Approach U Kazmaier C Schmidt
2440 RhodiumGraphite-Catalyzed Hydrogenation of Carbocyclic and Heterocyclic Aromatic Compounds G Falini A Gualandi D Savoia
2447 Potassium [1-(tert-Butoxycarbonyl)-1H-indol-2-yl]trifluoroborate as an Efficient Building Block in Palladium-Catalyzed SuzukindashMiyaura Cross Couplings P Kassis V Beacuteneacuteteau J-Y Meacuterour S Routier
2454 Syntheses of Substituted Furans and Pyrroles by Platinum-Catalyzed Cyclizations of Propargylic Oxiranes and Aziridines in Aqueous Media M Yoshida M Al-Amin K Shishido
2467 Transition-Metal-Free Oxidative Homocoupling of Aryl Alkenyl and Alkynyl Grignard Reagents with TEMPO M S Maji A Studer
XIII Forthcoming Articles
no 15 2471 Advances in Synthetic Approaches for the Preparation of Combretastatin-
Based Anti-Cancer Agents R Singh H Kaur 2492 Synthesis of Unsymmetrical Ureas by Sulfur-Assisted Carbonylation with
Carbon Monoxide and Oxidation with Molecular Oxygen under Mild Conditions T Mizuno T Nakai M Mihara
2497 Ring-OpeningRecyclization Reactions of (Dimethylamino)propenoyl-Substituted Cyclopropanes Facile Synthesis of Halogenated Pyridin-2(1H)-ones R Zhang Y Zhou Y Liang Z Jiang D Dong
2501 Facile and Efficient Total Synthesis of Taspine B Cheng S Zhang L Zhu J Zhang Q Li A Shan L He
2505 Oligomeric Iodosylbenzene Sulfate A Convenient Hypervalent Iodine Reagent for Oxidation of Organic Sulfides and Alkenes M S Yusubov R Y Yusubova T V Funk K-W Chi V V Zhdankin
2509 Pyrrolidine-Based Organocatalysts for Enantioselective Michael Addition of Cyclohexanone to trans-β-Nitrostyrene A P Carley S Dixon J D Kilburn
2517 CundashAl Hydrotalcite An Efficient and Reusable Ligand-Free Catalyst for the Coupling of Aryl Chlorides with Aliphatic Aromatic and N(H)-Heterocyclic Amines B Sreedhar R Arundhathi P L Reddy M A Reddy M L Kantam
2523 Highly Efficient Synthesis of trans-βγ-Unsaturated a-Keto Amides C Allais T Constantieux J Rodriguez
2531 Gas-Phase Synthesis of N-Unsubstituted 3-Hydroxypyrroles and 1H-Pyrrol-3(2H)-ones L Hill G A Hunter S H Imam H McNab W J OrsquoNeill
2535 3-Hydroxy-1H-pyrrole L Hill S H Imam H McNab W J OrsquoNeill 2539 123-Thiadiazoles with Unsaturated Side Chains Synthesis
Polymerization and Photocrosslinking M Al-Smadi N Hanold H Kalbitz H Meier
2547 Synthesis of 1112-Didehydrodibenzo[ae]cycloocten-5(6H)-one A Strained Eight-Membered Alkyne S C Kornmayer F Rominger R Gleiter
2553 Stannous Chloride Dihydrate A Novel and Efficient Catalyst for the Synthesis of gem-Dihydroperoxides from Ketones and Aldehydes D Azarifar K Khosravi F Soleimanei
2557 Synthesis of a Novel Class of Azacrown Macrocycles and Lariat Crown Ethers Containing Two 124-Triazole Rings as Subunits N Foroughifar A Mobinikhaledi S Ebrahimi
2561 Enantioselective Synthesis of the 3C-Protease Inhibitor (ndash)-Thysanone by a StauntonndashWeinreb Annulation Strategy J Sperry T Y Yuen M A Brimble
2570 Stereoselective Synthesis of Unnatural β-Amino Acids from Nitroethane via 56-Dihydro-4H-12-oxazin-3-ylacetates A Yu Sukhorukov A V Lesiv O L Eliseev Y A Khomutova S L Ioffe
2579 A Versatile Unexpected One-Pot Regioselective Synthesis of a New Class of 13-Diazepinoindolones by Reaction of Pyranoindolones with Monosubstituted Ureas D Livadiotou C A Tsoleridis J Stephanidou-Stephanatou
2584 Synthesis of a Trisaccharide and a Tetrasaccharide from the Cell-Wall Lipopolysaccharides of Azospirillum brasilense S17 S Pandey S Ghosh A K Misra
2591 Synthesis of Isoindoline Nitroxides by Electrocyclic Reactions T Kaacutelai J Jekı K Hideg
2596 Glycosylations of Tertiary Alcohols Synthesis of Fully Protected Disaccharides with Sterically Demanding Groups Attached to the Sugar Core A Holkenbrink J B Vicente D B Werz
2605 Copper-Catalyzed [13]-Dipolar Cycloaddition for the Synthesis of Macrocycles Containing Acyclic Aromatic and Steroidal Moieties G V Latyshev M S Baranom A V Kazantsev A D Averin N V Lukashev I P Beletskaya
2616 Aryl Ring Migration Reaction in the Synthesis of 24-Diaryl-4H-31-benzothiazines A V Butin F A Tsiunchik V T Abaev A V Gutnov D A Cheshkov
2627 Hydrogenation of β-N-Substituted and β-NN-Disubstituted Enamino Esters in the Presence of Iridium(I) Catalyst H Hebbache Z Hank C Bruneau J-L Renaud
2634 Stereoselective Olefination Reactions Promoted by Rieke Manganese J M Concelloacuten H Rodriacuteguez-Solla V del Amo P Diacuteaz
2646 Synthesis of Piperidinones through a Radical Cascade E Godineau Y Landais
2650 Asymmetric Organic Synthesis with Enzymes Edited by V Gotor I Alfonso E Garciacutea-Urdiales Reviewed by Steve Collier
XVII Forthcoming Articles
no 16 2651 Synthesis of Spirocyclic Ethers S Rosenberg R Leino 2674 Bimetallic PalladiumndashPlatinum-on-Carbon-Catalyzed HndashD Exchange
Reaction Synergistic Effect on Multiple Deuterium Incorporation T Maegawa N Ito K Oono Y Monguchi H Sajiki
2679 Efficient Copper-Catalyzed Synthesis of 2-Amino-4(3H)-quinazolinone and 2-Aminoquinazoline Derivatives X Huang H Yang H Fu R Qiao Y Zhao
2689 Synthesis and Chemoselective N- and O-Alkylation of Thiadiazolopyrimidine Nucleosides and Uridines A M L Hossion R Islam R K Kandahary T Nagamatsu
2697 Facile and Efficient Synthesis of a New Class of Indole-Substituted Pyridine Derivatives via One-Pot Multicomponent Reactions K Zhao X-P Xu S-L Zhu D-Q Shi Y Zhang S-J Ji
2709 Studies toward a Total Synthesis of Rhizoxin D Stereoselective Preparation of the C11ndashC19 Fragment S Padakanti C K Kumar E Ashok P Das
2715 A Short Synthesis of Enantiomeric Phytoprostanes B1 Type I W Perlikowska M Mikołajczyk
2719 Chemistry of Polyhalogenated Nitrobutadienes Part 7 A Novel Synthetic Access to Chlorinated Nitrile Oxides E Nutz V A Zapolrsquoskii D E Kaufmann
2725 Microwave-Assisted Silver(I)-Mediated Selective O-Alkylation of Aromatic Imidate Systems B K Singh C Cavalluzzo M De Maeyer Z Debyser V S Parmar E Van der Eycken
2729 Iodogen A Novel Reagent for the Oxidation of Urazoles under Heterogeneous Conditions A Khoramabadi A Shiri M A Zolfigol S Mallakpour
2733 An Unprecedented Synthesis of Eight-Membered-Ring Cyclic Thioimidic Esters by a Three-Component Reaction A Alizadeh R Hosseinpour
2737 A Novel Diastereoselective Synthesis of β-Phosphonato Unsaturated Thioimidates A Alizadeh N Zohreh
2741 Synthesis of 21-Benzisoxazoles by Nucleophilic Substitution of Hydrogen in Nitroarenes Activated by the Azole Ring N T Pokhodylo Y O Teslenko V S Matiychuk M D Obushak
2749 A Facile Synthesis of Two Series of Multifunctional Carbon Compounds from αα-Dihalo Ketones Using Allylsamarium Bromide X Liu S Zhang J Di
2756 Stereocontrolled Formation of Protected Aminodeoxyalditols from Simple Carbohydrate Precursors by Debenzylating Cycloetherification Y Jiang Z Fang Q Zheng H Jia J Cheng B Zheng
2761 trans-Stilbene as a Starting Material for the Synthesis of Tamoxifen Based on Palladium-Catalyzed Cross-Coupling Reactions C M Nunes J Limberger S Poersch M Seferin A L Monteiro
2766 Synthesis and Biological Evaluation of 6-Substituted Purinylcarbanucleosides with a Cyclopenta[b]thiophene Pseudosugar P Abeijoacuten J M Blanco O Caamantildeo F Fernaacutendez M D Garciacutea X Garciacutea-Mera J E Rodriacuteguez-Borges J Balzarini E De Clercq
2773 Synthesis and Electrochemical Signature of Novel Norbornyl-ferrocene Hybrids F A Khan S K Upadhyay
2778 A Regioselective TsujindashTrost Pentadienylation of 3-Allyltetronic Acid R Schobert B Barnickel
2785 Copper(I)-Catalyzed CarylndashCalkynyl Bond Formation of Aryl Iodides with Terminal Alkynes K G Thakur G Sekar
2790 Aminolysis of Epoxides Using Iridium Trichloride as an Efficient Catalyst J Agarwal A Duley R Rani R K Peddinti
2797 Preparation of Several Active N-Chloro Compounds from Trichloroisocyanuric Acid A Shiri A Khoramabadi-zad
2802 The First Mineral-Catalyzed One-Pot [3+1+2] Coupling Protocol for Multifunctionalized Fused-Ring Pyrimidines L D S Yadav A Rai
2809 Efficient Synthesis of Tetrahydro-β-carbolin-1-one and Dihydroisoquinolin-1-one Derivatives as Versatile Intermediates K E Judd M F Mahon L Caggiano
2818 A Concise Synthesis of ortho-Iodobenzyl Alcohols via Addition of ortho-Iodophenyl Grignard Reagent to Aldehydes and Ketones J Cvengroš D Stolz A Togni
XIII Forthcoming Articles
no 17 2825 Reactivity of Oxazol-5-(4H)-ones and Their Application toward Natural
Product Synthesis N M Hewlett C D Hupp J J Tepe 2840 Towards the Total Synthesis of 3-Hydroxyvibsanin E B D Schwartz
J R Denton P V Bernhardt H M L Davies C M Williams 2847 Structure Investigations of (ent)-Cladospolide D by De Novo Synthesis and
Kinetic and Thermodynamic Isomerization Y Xing J H Penn G A OrsquoDoherty
2855 New Applications of PhI(OAc)2 in Synthesis Total Synthesis and SAR Development of Potent Antitumor Natural Product PsymberinIrciniastatin A N Shao X Huang A Palani R Aslanian A Buevich J Piwinski R Huryk C Seidel-Dugan
2873 Total Synthesis of Largazole ndash Devolution of a Novel Synthetic Strategy B Wang C J Forsyth
2881 Formal Total Synthesis of Palmerolide A J Jaumlgel M E Maier 2893 Total Synthesis of Bongkrekic Acid via Sequential SuzukindashMiyaura Coupling
Reactions M Kanematsu M Shindo M Yoshida K Shishido 2905 Stereodivergent Approach to Both C28a-syn and C28a-anti Relative
Stereochemical Manifolds in the Lepadin Family via a TiCl4-Promoted G Li L J Carlson I K Sagamanova B W Slafer R P Hsung C Gilardi H M Sklenicka N Sydorenko
2915 Enantioselective Aldol Reaction of Tetrasubstituted Ketene Silyl Acetals with Achiral Aldehydes for the Construction of Asymmetric Tertiary Alcohols An Application for the Divergent Total Syntheses of Buergerinins F and G I Shiina T Iizumi Y-s Yamai Y-i Kawakita K Yokoyama Y-k Yamada
2927 Second-Generation Biomimetic Total Synthesis of Chaetominine A Coste G Karthikeyan F Couty G Evano
2935 Total Synthesis of (+)-Fostriecin and (+)-Phoslactomycin B S Shibahara M Fujino Y Tashiro N Okamoto T Esumi K Takahashi J Ishihara S Hatakeyama
2954 Stereochemical Assignments of the Chlorinated Residues in Victorin C A C Durow C Butts C L Willis
2963 Studies of the Asymmetric Total Synthesis of Clavilactone D by the lsquoLariatrsquo Cyclization Strategy T Yoshimitsu S Nojima M Hashimoto K Tsukamoto T Tanaka
2970 Total Synthesis of the Leucetta-Derived Alkaloid Calcaridine A P B Koswatta R Sivappa H V R Dias C J Lovely
2983 Formal Synthesis of Salinosporamide A Starting from D-Glucose T Momose Y Kaiya J-i Hasegawa T Sato N Chida
2992 Synthesis of Bioactive Natural Products by Asymmetric syn- and anti-Aldol Reactions A K Ghosh Z L Dawson
no 18 3003 Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural
Products B M Trost M K Brennan 3026 One-Pot Synthesis of Furo[34-b]pyridin-5(7H)-ones from 2-
Bromopyridine-3-carboxylic Acid and Carbonyl Compounds K Kobayashi T Kozuki H Konishi
3029 Iodocyclization of N-[2-(Methylthio)phenyl]propiolamides Selective Synthesis of 3-Iodo-15-benzothiazepin-4-ones T-S Jiang X-G Zhang J-H Li
3039 A Facile Synthetic Method for Fluorine-Containing 17-Phenanthrolines Pyridine-Ring Formation Reaction of N-Propargyl-68-bis(trifluoroacetyl)-quinolin-5-amine with Various Nucleophiles D Shibata E Okada M Hinoshita M Meacutedebielle
3047 Enantiotopic Discrimination in Palladium-Mediated Nucleophilic Substitutions on Achiral Substrates Chiral Ligand versus Chiral Nucleophile O Jacquet F Charnay J-C Fiaud J Ollivier
3051 Studies on the Chemistry of 2-[3-(2-Nitrophenyl)-2-oxopropyl]benzaldehydes Novel Syntheses of 5H-Benzo[b]carbazole-611-diones and Indolo[12-b]isoquinoline-611-diones M Fernaacutendez
3061 Studies on the C22ndashC23 Aldol Coupling of Spirangien M Lorenz N Bluhm M Kalesse
3067 One-Pot Synthesis of N-Alkyl Purine Pyrimidine and Azole Derivatives from Alcohols using Ph3PCCl4 A Rapid Route to Carboacyclic Nucleoside Synthesis M N Soltani Rad A Khalafi-Nezhad S Behrouz Z Asrari M Behrouz Z Amini
3077 Synthesis of 2-Amino-34-dihydroquinazolines and Imidazo[21-b]quinazoline-2-ones A Mishra S Batra
3089 Studies on the Reaction of Diimines with Thiourea Synthesis and Solvent-Induced cistrans-Isomerization of 135-Triazinane-2-thiones B Kaboudin T Ghasemi T Yokomatsu
3094 Suzuki Coupling of Heteroaromatic Chlorides Using Highly Electron-Donating ClickPhos Ligands S M Spinella Z-H Guan J Chen X Zhang
3099 Reaction of NN-Dioxyenamines with Anhydrides of Carboxylic and Sulfonic Acids A New Method for the Synthesis of a-Hydroxyoxime Derivatives A A Tabolin A V Lesiv S L Ioffe
3106 Directed ortho Metallation Chemistry and Phosphine Synthesis New Ligands for the SuzukindashMiyaura Reaction D B G Williams S J Evans H de Bod M S Mokhadinyana T Hughes
3113 New Functional Derivatives of 9-Phenylquinine P J Boratyński J SkarŜewski
3120 On the Synthesis of Asymmetric and Dissymmetric Amino Analogues of Troumlgerrsquos Base J Artacho K Waumlrnmark
3127 Synthesis of Polycyclic Sultams by Palladium-Catalyzed Intramolecular Cyclization K C Majumdar S Mondal N De
3136 Synthesis of Functionalized L-Cysteine and L-Methionine by Reaction with Electron-Deficient Acetylenes B A Trofimov A G Malrsquokina O A Shemyakina V V Nosyreva A P Borisova S S Khutsishvili L B Krivdin
3143 A lsquoClickrsquo Approach to the Synthesis of 3-[2-(1-Alkyltriazol-4-yl)ethyl]indoles M Petrini R R Shaikh
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
No 2 165 Selected Synthetic Strategies to Spirocyclics S Kotha A C Deb
K Lahiri E Manivannan 194 Effective Catalytic Activity of the Hydrated Gold Catalyst NaAuCl42H2O To
Construct Highly Fused Cyclopentenones S Karmakar A Kim C H Oh
199 Efficient Synthesis of an Allose-Containing Analogue of the Phytoalexin-Elicitor Glucohexaose and Its Dodecyl Glycoside H Ma D Qiu X Mei J Ning Q Zhao Y Li
205 Synthesis of 14-Benzodiazepine-25-diones Using an Ionic Liquid as a Soluble Support H Xie C Lu G Yang Z Chen
211 A Facile Synthesis of Thioalkyl- and Di(thioalkyl)-Substituted Bipyridines D Chen R De D L Mohler
217 Diastereoselective Synthesis of Dimethyl (4R4aR7aR)-1-Aryl-6-benzoyl-4a-methyl-5-oxo-144a556-hexahydrospiro[pyrazole-47-pyrrolo[34-c]pyridazine]-37a(1H)-dicarboxylates U Uršič U Grošelj A Meden J Svete B Stanovnik
227 Synthesis of 3-Acylpyrroles 3-(Alkoxycarbonyl)pyrroles 1567-Tetrahydro-4H-indol-4-ones and 3-Benzoylpyridines Based on StaudingerndashAza-Wittig Reactions of 13-Dicarbonyl Compounds with 2- and 3-Azido-11-dialkoxyalkanes E Bellur M A Yawer I Hussain A Riahi O Fatunsin C Fischer P Langer
243 Regioselective Synthesis of Functionalized Biaryls Based on the First [3+3] Cyclocondensations of 4-Aryl-13-bis(trimethylsilyloxy)buta-13-dienes M Adeel M A Rashid N Rasool R Ahmad A Villinger H Reinke C Fischer P Langer
251 Synthesis of Functionalized Bicyclic Precursors of Heptulosonic Acid Analogues H Filali S Ballereau F O Chahdi M Baltas
257 Efficient Regio- and Stereoselective Synthesis of 5-Alkyl(aryl)idene- and 5-[Iodoalkyl(aryl)idene]-1H-pyrrol-2(5H)-ones via Electrophilic Cyclization K Cherry A Duchecircne J Thibonnet J-L Parrain E Anselmi M Abarbri
271 PdCu-Catalyzed Oxidative CndashH Alkenylation of Imidazo[12-α]pyridines J Koubachi S Berteina-Raboin A Mouaddib G Guillaumet
277 A Convenient Synthesis of Unsymmetrical Pinacols by Coupling of Structurally Similar Aromatic Aldehydes Mediated by Low-Valent Titanium X-F Duan J-X Feng G-F Zi Z-B Zhang
283 A Method for the Selective Protection of Aromatic Amines in the Presence of Aliphatic Amines V Perron S Abbott N Moreau D Lee C Penney B Zacharie
290 Synthesis and Antiviral Evaluation of (ndash)-3-Methylcarbovir (ndash)-3-Methylabacavir and Modified Purine Analogues P Breacutemond G Audran H Monti E De Clercq C Pannecouque
297 Regioselective Synthesis of 2-(Aryloxythio)benzoates by the First [3+3] Cyclizations of 3-Aryloxythio-1-silyloxybuta-13-dienes with 3-Alkoxy-2-en-1-ones I Iqbal M Imran A Villinger P Langer
306 Molybdenum(VI) Dichloride Dioxide Catalyzed Conversion of b-Hydroxycarbonyls into a-Bromo 13-Dicarbonyls by N-Bromosuccinimide K Jeyakumar D K Chand
311 A Short Route to the Synthesis of Pyrrolocoumarin and Pyrroloquinolone Derivatives by Sonogashira Cross-Coupling and Gold-Catalyzed Cycloisomerization of Acetylenic Amines K C Majumdar B Chattopadhyay S Samanta
318 Aspects of the Synthesis of an Exceptionally Preorganized Self-Immolative SpacerndashPhenolate Unit M Waibel X-B Zhang J Hasserodt
325 Design and Efficient Synthesis of Amino Acid Derived 2-Substituted Imidazoles by Palladium-Catalyzed Cross-Coupling Reactions A Marek J Kulhaacutenek F Bureš
332 A Convenient Preparation of Di-p-chlorobenzyl Azodicarboxylate (DCAD) for Mitsunobu Couplings B R Taft E C Swift B H Lipshutz
335 Enantioselective Rhodium-Catalyzed Alkylative Desymmetrization of 35-Dimethylglutaric Anhydride M J Cook T Rovis
XIII Forthcoming Articles
No 3 339 Intermolecular Addition Reactions of N-Acyliminium Ions (Part I)
A Yazici S G Pyne 369 Desulfurization of Thioamides into Amides with H2O2ZrCl4 Reagent System
K Bahrami M M Khodaei Y Tirandaz 372 Total Synthesis of (plusmn)-1345-Tetragalloylapiitol R M Patel
N P Argade 375 A Convenient Synthesis of 4-Hydroxy-2-oxo-12-dihydro-18-
naphthyridine-3-carboxamide Derivatives K Kobayashi D Iitsuka S Fukamachi H Konishi
379 Intramolecular Ketalization of Functionalized 7-Norbornenols L A Paquette J D Pettigrew
385 Ring Contraction of 12-Dihydronaphthalenes Promoted by Thallium(III) in Acetonitrile A Diastereoselective Approach to Indanes H M C Ferraz V M T Carneiro L F Silva Jr
389 Regio-Controlled Nucleophilic Attack of 3-Thiaisatoic Anhydride by α-Amino Acids One-Pot Synthesis of 3-(2-Thienyl)imidazolidine-24-dione and 34-Substituted Thieno[23-e][14]diazepine-25-dione Analogues Y Brouillette G Sujol J Martinez V Lisowski
395 The Unprecedented Cobalt-Catalysed Oxidative Glaser Coupling under Reductive Conditions G Hilt C Hengst M Arndt
399 Nucleophilic Addition of 4-Hydroxycoumarin to BaylisndashHillman Acetate Adducts C Raji Reddy N Kiranmai K Johny M Pendke P Naresh
403 Palladium-Mediated Heck Reaction to the Synthesis of 3-Substituted Indoles and Indolones K C Majumdar S Chakravorty P K Shyam A Taher
409 Synthesis of Bicyclo[310]hexan-2-ones by Manganese(III) Oxidation in Ethanol K Asahi H Nishino
424 High Regio- and Stereoselective Synthesis of (Z)- or (E)-N-Acryl Butenedioic Monoimide Derivatives by a Multicomponent Reaction F Sha Y Lin X Huang
431 The First Synthesis of Allyl Isonitriles from BaylisndashHillman Adducts and Their Application in the Synthesis of Substituted Imidazo[12-α]pyridines and Tetraazadibenzoazulenes M Nayak S Kanojiya S Batra
438 One-Pot Three-Step Synthesis of Pyrazinothienopyrimidines Using Tandem Aza-WittigElectrocyclic Ring Closure G Blanco A Fernaacutendez-Mato J M Quintela C Peinador
445 Synthesis of Biaryls Fluorenones Cyclopenta[def]phenanthren-4-ones and Benzophenones Based on Formal [3+3] Cyclocondensations of 13-Bis(silyloxy)buta-13-dienes with 3-(Silyloxy)-2-en-1-ones S Reim M Lau M Adeel I Hussain M A Yawer A Riahi Z Ahmed C Fischer H Reinke P Langer
464 Diastereoselective Synthesis of α-Stabilized Phosphorus Ylides via a Four-Component Reaction A Alizadeh N Zohreh L-G Zhu
469 Stereoselective Synthesis of Alkynyl Vinyl Chalcogenides via HornerndashWittig Reaction C C Silveira F Rinaldi R C Guadagnin A L Braga
474 Stereoselective Preparation of C1ndashC10 and C11ndashO14 Fragments of Narbonolide Exploiting the Versatility of Thiazolidinethione Chiral Auxiliary C P Narasimhulu P Das
483 Efficient Catalytic Activity of CopperAluminum Hydrotalcite in Diaryl Ether Synthesis B Sreedhar R Arundhathi M A Reddy M L Kanatm
488 On-Resin Click-Glycoconjugation of Peptoids A S Norgren C Budke Z Majer C Heggemann T Koop N Sewald
495 A Simple and Efficient Preparation of Novel Formaldehyde Derivatives R Hartung G Golz S Schlaf G Silvennoinen K Polborn P Mayer H R Pfaendler
502 2-Oxazol-5-ylethanones by Consecutive Three-Component AmidationndashCouplingndashCycloisomerization (ACCI) Sequence E Merkul O Grotkopp T J J Muumlller
508 SuzukindashMiyaura Cross-Couplings Mediated by trans-PdBr(N-Succ)(PPh3)2 A Convenient Synthetic Method for Diarylmethanes and Aryl(heteroaryl)-methanes I J S Fairlamb P Sehnal R J K Taylor
511 Modern Reduction Methods Edited by P G Andersson and I J Munslow Reviewed by Siegfried R Waldvogel
512 Addendum and Erratum XIII Forthcoming Articles
No 4 513 Intermolecular Addition Reactions of N-Acyliminium Ions (Part II)
A Yazici S G Pyne 542 A Simple Practical Method for the Synthesis of 46-Dimethoxy-135-
triazin-2(1H)-one Using Dimethylamine-Functionalized Solid-Phase Reagents K Hioki K Ohshima Y Sota M Tanaka M Kunishima
545 Conjugation-Amenable Tetrasaccharide of the Side Chain of the Major Glycoprotein of the Bacillus anthracis Exosporium A Large-Scale Preparation S Hou P Kovaacuteč
551 Reductive Amination ndash A Convenient Method for Generating Diverse Mono-Functionalised 5101520-Tetraphenyl Porphyrins C Welch S J Archibald R W Boyle
557 Highly Regioselective Preparation of 13-Dioxolane-4-methanol Derivatives from Glycerol Using Phosphomolybdic Acid N W Fadnavis R Gowrisankar G Ramakrishna M K Mishra G Sheelu
561 Rapid Synthesis of 3-Aminoisoquinoline-5-sulfonamides Using the BuchwaldndashHartwig Reaction N Proisy S Taylor A Nelson I Collins
567 Synthesis of Divalent 22-Linked Mannose Derivatives by Homodimerization F S Ekholm M Polaacutekovaacute A J Pawłowicz R Leino
577 Efficient Synthesis of Substituted Cyclic α-Aminophosphonates I L Odinets O I Artyushin N Shevchenko P V Petrovskii V G Nenajdenko G-V Roumlschenthaler
583 Methylated Imidazolinium-Dithiocarboxylates Two Representatives of a New Class of Ionic Liquids A Blanrue R Wilhelm
587 An Efficient Route to 1-Vinylpyrrole-2-carbaldehydes A I Mikhaleva A V Ivanov E V Skitalrsquotseva I A Ushakov A M Vasilrsquotsov B A Trofimov
591 A Regioselective Route to 5-Substituted Isoxazole- and Isoxazoline-3-phosphonates P Conti A Pinto L Tamborini P Dunkel V Gambaro G L Visconti C De Micheli
597 Solvent-Free One-Pot Conjugate Addition of Benzyl Bromides to β-Nitroalkenes Mediated by Magnesium Powder W Shi J-X Wang
602 Synthesis of 234-Trideoxy-44-difluoro-D-ribo-hexopyranose Adenosines J Xu X Zhang X-L Qiu F-L Qing
609 Synthesis of anti-27-Disubstituted Norbornadienes G C Tsui P Le Marquand A Allen W Tam
620 Novel Peptide Mimetic Inhibitors of Hepatitis C Serine Protease Derived from Isomannide T G Barros S Pinheiro J S Williamson A Tanuri H S Pereira R M Brindeiro J B A Neto O A C Antunes E M F Muri
627 A Practical Synthesis of α-Substituted tert-Butyl Acrylates from Meldrumrsquos Acid and Aldehydes C G Frost S D Penrose R Gleave
636 A New Class of Troumlgerrsquos Base Analogues Bearing Spiro[45] Lactone Straps A B Mahon D C Craig A C Try
643 A New Approach to Di- and Tetrasubstituted 23-Dihydropyridin-4(1H)-ones through Aza-DielsndashAlder Reaction Promoted by Silicon Tetrachloride A Massa V de Sio R Villano M R Acocella L Palombi G Sellitto A Peduto R Filosa P De Capraris A Scettri
650 Palladium-Catalysed Direct Arylation of Sydnones A Rodriguez W J Moran
655 Synthesis of (ndash)-Monomorine I R W Bates P Song 660 Cobalt(II) Chloride HexahydratendashDiisopropylamine Catalyzed Mild and
Chemoselective Reduction of Carboxylic Esters with Sodium Borohydride A R Jagdale A S Paraskar A Sudalai
665 Synthesis of Bi- and Tricyclic αβ-Unsaturated Lactams as Potential Michael Acceptors Starting from Heterocyclic Imines K Schulz M Watzke K Johannes P Ullrich J Martens
674 An Expedient Synthesis of Bis-Fused Benzofuran and a Two-Directional Ring-Closing Metathesis for the Synthesis of Bisbenzoxepines and Bisbenzoxocines K C Majumdar B Chattopadhyay S Chakravorty
681 Palladium-Catalyzed Cross-Couplings of Unsaturated Halides Bearing Relatively Acidic Hydrogen Atoms with Organozinc Reagents Z Dong G Manolikakes J Li P Knochel
687 Synthesis of Enantioenriched aa-Disubstituted Cyclopentenes Catalyzed by N-Heterocyclic Carbenes E M Phillips M Wadamoto K A Scheidt
XVII Forthcoming Articles
No 5 691 Transannulation Reactions in the Synthesis of Natural Products
P A Clarke A T Reeder J Winn 710 Synthesis of DL-erythro-Sphingosine Using a Tethered
Aminohydroxylation Reaction as the Key Step J A Morales-Serna Y Diacuteaz M I Matheu S Castilloacuten
713 Convenient Multigram Synthesis of 4-Chloropyridine-26-dicarbonyl Dichloride K Mitsui J R Parquette
715 A Novel and Efficient Synthesis of Dihydrexidine J P Cueva D E Nichols
721 Synthesis of 57-Dichloro-6-azaindoles and Functionalization via a Highly Selective LithiumndashChlorine Exchange N Lachance L-P Bonhomme-Beaulieu P Joly
731 A Convenient Synthesis of Fluorinated Pyrazolo[34-b]pyridine and Pyrazolo[34-d]pyrimidine Nucleosides V O Iaroshenko D V Sevenard A Kotljarov D M Volochnyuk A O Tolmachev V Y Sosnovskikh
741 Diastereoselective Synthesis of γ-Amino Acids and Their Derivatives from Nitroethane via Intermediacy of 56-Dihydro-4H-12-oxazines Bearing the CH2CH(CO2Me)2 Substituent at C3 A Y Sukhorukov A V Lesiv Y A Khomutova S L Ioffe
755 Synthesis of a New Pyrrolopyridoindole and Its Pyrrolopyridobenzimidazole Regioisomer F Bouchikhi M Sassatelli F Anizon M Prudhomme P Moreau
759 Practical Syntheses of Sphingosine-1-Phosphate and Analogues V Blot U Jacquemard H-U Reissig B Kleuser
767 A Facile Synthetic Route towards Substituted Thieno[32-e]indoles W Van Snick W Nulens S Jambon W Dehaen
775 Microwave-Assisted One-Pot Synthesis of (Aminoalkyl)naphthols and (Aminoalkyl)quinolinols by Using Ammonium Carbamate or Ammonium Hydrogen Carbonate as Solid Ammonia Source I Szatmaacuteri F Fuumlloumlp
779 Enantioselective Synthesis of Flavan-3-ols Using a Mitsunobu Cyclization K Krohn I Ahmed M John 787 Synthesis of a Novel γ-Folic AcidndashNτ-Histidine Conjugate Suitable for
Labeling with 99mTc and 188Re C Sparr U Michel R E Marti C Muumlller R Schibli R Moser V Groehn
793 Palladium-Catalyzed Intramolecular Biaryl Coupling A Highly Efficient Avenue for Benzannulated Pyranoquinolines and Julolidine Derivatives K C Majumdar A Taher P Debnath
801 Preparation of NN-Dimethyl-N-Arylureas Using SS-Dimethyl Dithiocarbonate as a Carbonylating Reagent I Degani R Fochi C Magistris M Migliaccio
809 Versatile Selective α-Carboxylic Acid Esterification of N-Protected Amino Acids and Peptides by Alcalase T Nuijens C Cusan J A W Kruijtzer D T S Rijkers R M J Liskamp P J L M Quaedflieg
815 Efficient Palladium-Catalyzed Amination of Aryl Chlorides Using Dicyclohexylamino[(26-dimethyl)morpholino]phenylphosphine as a PN2 Ligand S-E Park S B Kang K-J Jung J-E Won S-G Lee Y-J Yoon
824 A Clean Facile and Stereospecific Synthesis of α-Oxoketene OS-Acetals in Water Y Li Q Zhang X Cheng Q Liu X Xu
829 Sonogashira Cross-Coupling Reactions and Construction of the Indole Ring System Using a Robust Silica-Supported Palladium Catalyst E Tyrrell L Whiteman N Williams
836 Synthesis of Angular 78-Pyridazinocoumarins via the Transformation of a Hydroxy Group into a Carbonyl Group A Kotali I S Lafazanis P A Harris
841 Synthesis of New Cyclic and Acyclic 5-Halouridine Derivatives as Potential Antiviral Agents M F Elshehry J Balzarini C Meier
848 Dendritic Triphenylmethylium and Tetraphenylmethane Compounds H Meier S Kim A Oehlhof
853 Synthesis of Homoallylic Alcohols via Lewis Acid Assisted Enantioselective Desymmetrization B Yu F Menad N Isono M Lautens
860 Diastereoselective Synthesis of 123-Trisubstituted Indanes via Rhodium(I)-Catalyzed Tandem Conjugate Additions C Navarro A G Csaacutekyuml
864 Bakerrsquos Yeast for Sweet Dough Enables Large-Scale Synthesis of Enantiomerically Pure Bicyclo[331]nonane-26-dione C J Wallentin E Orentas E Butkus K Waumlrnmark
868 Addendum and Erratum XV Forthcoming Articles
No 6 869 Stereoselective Transformations of meso Bicyclic Hydrazines Versatile
Access to Functionalized Aminocyclopentanes C Bournaud F Chung A P Luna M Pasco G Errasti T Lecourt L Micouin
888 Synthesis of Glycoaminoxy Acids as Novel Sugar Building Blocks A Malapelle R Ramozzi J Xie
891 Electrophilic ipso-Halocyclization of N-Arylpropynamides with Polyfluoroalkyl Alcohols Selective Synthesis of 8-(Polyfluoroalkoxy) azaspiro[45]trienes Z-Q Wang B-X Tang H-P Zhang F Wang J-H Li
903 Electrooxidation of Alcohols in N-Oxyl-Immobilized Silica GelWater Disperse System Approach to Totally Closed System M Kuroboshi K Goto H Tanaka
909 Synthetic Routes to Aminotriamantanes Topological Analogues of the Neuroprotector Memantinereg A A Fokin A Merz N A Fokina H Schwertfeger S L Liu J E P Dahl R K M Carlson P R Schreiner
913 Parallel Synthesis of Drug-like 5-Amino-Substituted 124-Thiadiazole Libraries Using Cyclization Reactions of a Carboxamidine Dithiocarbamate Linker J Y Park I A Ryu J H Park D C Ha Y-D Gong
921 Copper-Catalyzed Selective S-Arylation of 12-Bis(o-amino-1H-pyrazolyl) Disulfides with Arylboronic Acids P-S Luo F Wang J-H Li R-Y Tang P Zhong
929 2-Iodoxybenzoic AcidTetraethylammonium BromideWater An Efficient Combination for Oxidative Cleavage of Acetals C Kuhakarn W Panchan S Chiampanichayakul N Samakkanad M Pohmakotr V Reutrakul T Jaipetch
935 Synthesis of Quinonoid Analogues of Diospyrin S Sagar I R Green 941 A One-Pot Method for the Iodination of Aryl Amines via Stable Aryl
Diazonium Silica Sulfates Under Solvent-Free Conditions A Zaroi A R Hajipour L Khazdooz
945 Poly(NN-dichloro-N-ethylbenzene-13-disulfonamide) and NNNN-Tetrachlorobenzene-13-disulfonamide as Novel Reagents for the Synthesis of N-Chloroamines Nitriles and Aldehydes R Ghorbani-Vaghei H Veisi
951 Synthesis of an (R)-Garner-type Aldehyde from L-Serine Useful Building Block for a (+)-Furanomycin Derivative G Bartoli G Di Antonio R Fiocchi S Giuli E Marcantoni M Marcolini
957 An Efficient and Highly Selective Synthesis of (Z)-Fluoroenol Phosphates from Hydroxy Difluorophosphonates P Beier R Pohl A V Alexandrova
963 Iodine-Catalyzed Three-Component Reaction A Rapid Synthesis of α-Alkoxy Azides and Homoallyl Ethers J S Yadav B V S Reddy G M Reddy R Narender
969 Rhodium(I)-Catalyzed Cycloisomerization of 13-Dienes with Alkenes in a Tether Y Oonishi A Saito M Mori Y Sato
980 Synthesis of New Optically Active D-GlucosaminendashPyrrole Derivatives B A Frontana-Uribe M V Escaacutercega-Bobadilla J Juaacuterez-Lagunas R A Toscano G A Garciacutea de la Mora M Salmoacuten
985 Partially Saturated Indeno[12-b]indole Derivatives via Deoxygenation of Heterocyclic α-Hydroxy-NO-hemiaminals H-J Hemmerling G Reiss
1000 Light-Induced Synthesis of Π-Extended Tetrathiafulvalenes Incorporating Ferrocenes An Efficient Route for the Synthesis of Electron-Donor Materials A A O Sarhan C Bolm
1007 Preparation of Nβ-Fmoc-Protected Aza-β3-Amino Acids with Nonproteinogenic Hydrophobic Side Chains for Solid-Phase Syntheses of Pseudopeptides M Laurencin P Bauchat M Baudy-Flocrsquoh
1014 Diastereomeric (η4-diene)Fe(CO)3 Complexes Containing Chiral Amide Groups A Convenient Method for the Resolution of Amino Acids M Schumacher G Coste L Miesch
1021 Palladium-Catalysed Heck Reactions of Alk-1-en-3-ones with Aryl Bromides A Very Simple Access to (E)-1-Arylalk-1-en-3-ones M Lemhadri Y Fall H Doucet M Santelli
1036 An Improved Process for the Synthesis of 4H-Imidazo[15-α][14]benzodiazepines J Yang Y Teng S Ara S Rallapalli J M Cook
1041 Meta- and Para-Difunctionalization of Arenes via an Ortho-Magnesiation and a Subsequent SulfoxidendashMagnesium Exchange L Melzig C B Rauhut P Knochel
XIII Forthcoming Articles
No 7 1049 Catalytic Transformations of Benzylic Carboxylates and Carbonates
R Kuwano 1062 A Simple and Practical Method for the Oxidation of Thebaine to 14-
Hydroxycodeinone by V2O5ndashH2O2 S Das Sharma D Konwar 1065 Umpolung with Sulfur Dioxide CarbonndashCarbon Cross-Coupling of Electron-
Rich 13-Dienes and Alkenes Application to the Enantioselective Synthesis of Long-Chain Polyketide Fragments M Turks C J Exner C Hamel P Vogel
1075 One-Pot Synthesis of 14-Diarylnaphthalenes via a WittigndashHorner Reaction[4+2] CycloadditionDehydrogenation Sequence Z Chen W Shou Y Wang
1081 A Novel and General Method for the Formation of S-Aryl Se-Aryl and Te-Aryl Phosphorochalcogenoates Y-X Gao G Tang Y Cao Y-F Zhao
1087 A Remarkable Access to γ-Fluoroalkylated Propargylamine Derivatives or Fluoroalkylated Dihydroisoxazoles via the Reaction of Fluoroalkylated Acetylides with Various Nitrones T Konno K Moriyasu T Ishihara
1095 Short and Practical Syntheses of (S)-(+)-3-(p-Tolylsulfinyl)furan-2(5H)-one and (S)-(+)-3-(p-Tolylsulfinyl)-56-dihydropyran-2-one D Cruz Cruz A Hernaacutendez Linares F Yuste M R Martiacuten J L Garciacutea Ruano
1099 Decarboxylative Aldol-Type Reaction of 2-(Trifluoroacetyl)-13-diazoles with Activated Acetic Acids P V Khodakovskiy D M Volochnyuk A A Tolmachev
1105 Synthesis of 2-[(Arylmethylene)amino]cyclopropanecarbonitriles via a Two-Step Ring Transformation of 2-(Cyanomethyl)aziridines S Mangelinckx M Drsquohooghe S Peeters N De Kimpe
1113 Synthesis of Dendrimeric Tumor-Associated Mucin-Type Glycopeptide Antigens T Becker A Kaiser H Kunz
1123 A Simple and Efficient Oxidation Procedure for the Synthesis of Acid-Sensitive Epoxides O Bortolini G Fantin M Fogagnolo
1127 Rapid Chemoselective Deprotection of Benzyl Esters by Nickel Boride J M Khurana R Arora
1131 Three-Component Coupling of Isoquinoline Activated Alkyne and Nitromethane A Facile Synthesis of Nitromethyl Derivatives of 12-Dihydroisoquinolines J S Yadav B V S Reddy N N Yadav M K Gupta
1137 Palladium Supported on a Polyionic Resin as an Efficient Ligand-Free and Recyclable Catalyst for Heck SuzukindashMiyaura and Sonogashira Reactions B Basu S Das P Das B Mandal D Banerjee F Almqvist
1147 Oxidation of 25-Dialkylpyrrole Derivatives with Cerium(IV) Ammonium Nitrate R Voloshchuk M Gałęzowski D T Gryko
1153 Practical Syntheses of Enantiomerically Pure Key Intermediates of Opioid Receptor-like 1 (ORL1) Antagonists T Yoshizumi A Ohno T Tsujita H Takahashi O Okamoto I Hayakawa H Kigoshi
1163 An Environmentally Benign TEMPO-Catalyzed Efficient Alcohol Oxidation System with a Recyclable Hypervalent Iodine(III) Reagent and Its Facile Preparation X-Q Li C Zhang
1170 Efficient and Stereoselective Rearrangement of BaylisndashHillman Acetates Catalyzed by Gold(I) ChlorideSilver(I) Trifluoromethanesulfonate Y Liu D Mao J Qian S Lou Z Xu Y Zhang
1175 The First Total Synthesis of Kynapcin-24 by Palladium Catalysis L-Y Yang C-F Chang Y-C Huang Y-J Lee C-C Hu T-H Tseng
1180 Enantioselective Synthesis of N-Protected α-Amino Acid Hydrazides M Bibian S El-Habnouni J Martinez J-A Fehrentz
1185 Synthesis of 11H-Indolo[32-c]quinoline-6-carboxylic Acids by Cascade AutoxidationndashRing Contractions A Becker S Kohfeld T Pies K Wieking L Preu C Kunick
1190 Reaction of N-Nonaflylbenzotriazole with Silyl Enol Ethers M Uhde T Ziegler
1195 2-(Benzoylimino)thiazolidin-4-ones Formation by an Alternative Ring Closure and Analysis of Rotational Barriers H-G Haumlcker P W Elsinghorst S Michels J Daniels G Schnakenburg M Guumltschow
1204 Microwave-Assisted Synthesis and Functionalization of Selenolopyrimidines S Hesse C Chenet D Thomae G Kirsch
1209 12-Disubstituted 4-Quinolones via Copper-Catalyzed Cyclization of 1-(2-Halophenyl)-2-en-3-amin-1-ones R Bernini S Cacchi G Fabrizi A Sferrazza
1220 A New Atom-Economical and Selective Synthesis of Secondary and Tertiary Alkylamines by Means of CpIridium Complex Catalyzed Multiple N-Alkylation of Ammonium Salts with Alcohols without Solvent R Yamaguchi Z Mingwen S Kawagoe C Asai K-i Fujita
1224 Synthesis of Regioisomerically Pure 5-Functionalized 27-Dichlorofluoresceins J C Castro A Malakhov K Burgess
XIII Forthcoming Articles
No 8 1227 Michael Additions to Activated Vinylphosphonates T Janecki J Kędzia
T Wąsek 1255 A Facile and General Synthesis of 2β-Aminosteroids X Ke H Hu
D Zhou W Xu Q Zhu N P Reddy X Hu 1261 Efficacious Preparation of Oppolzerrsquos Glycylsultam via the Deleacutepine
Reaction A Isleyen C Gonsky R C Ronald P Garner 1265 Synthesis of Masked Vicinal Amino Aldehydes of Pyrrolizine and Pyrrolo
[12-c]thiazole Series A V Tverdokhlebov A V Denisenko A A Tolmachev Y M Volovenko S V Shishkina O V Shishkin
1271 Preparation of 9-Substituted Pyridine-Stretched Adenines and Hypoxanthines J A Crawford W Fraser C A Ramsden
1279 A Versatile Synthesis of Heterocyclic Analogues of Neoflavonoids from Enamino Ketones V S Moskvina V P Khilya O V Turov U M Groth
1287 New Stereoselective Synthesis of Paeonilactone B F G Gatti S Serra 1291 The Use of NN-Dialkyltrimethylsilylamines in the Synthesis of
Pentamethinium Salts M Kořiacutenek M Rybaacutečkovaacute Boumlhm 1297 Synthesis of Triazoles via Regioselective Reactions of Aryl Azides with
Cyanoacetyl Pyrroles and Indoles N T Pokhodylo V S Matiychuk M D Obushak
1301 Gallium(III) Chloride Catalyzed Hydroarylation of Arylacetylenes with Naphthols and Phenols A Facile Synthesis of Vinylarenes J S Yadav B V S Reddy S Sengupta S K Biswas
1305 Electrophilic Bromination of meta-Substituted Anilines with N-Bromosuccinimide Regioselectivity and Solvent Effect S Bartoli A Cipollone A Squarcia A Madami D Fattori
1309 Cross-Coupling Reactions of Halopurines with Aryl- and Alkyltrifluoroborates The Scope and Limitations in the Synthesis of Modified Purines Z Hasniacutek R Pohl M Hocek
1318 A Convenient Method for Converting Hydroxyacetophenones into Their Ethylene or Trimethylene Acetals F Ono H Takenaka T Fujikawa M Mori T Sato
1323 γ-Chloromagnesio γ-Lactones and δ-Chloromagnesio δ-Lactones Generation Properties and Synthetic Uses H Shimizu S Fukuda S Sugiyama T Satoh
1336 Click Reactions with Nitroxides T Kaacutelai W L Hubbell K Hideg 1341 Synthesis of Novel 14-Benzoquinone-Containing 123-Triazoles An Entry
Into a New Library F Algi M Balci 1348 Efficient Synthesis of Two Sialylated Tetrasaccharides Found in Goat Milk
P K Mandal A K Misra 1355 Dendrimers of Vaccines Consisting of Tumor-Associated Glycopeptide
Antigens and T Cell Epitope Peptides S Keil A Kaiser F Syed H Kunz
1370 IBXTBAB-Mediated Oxidation of Primary Amines to Nitriles F Drouet P Fontaine G Masson J Zhu
1375 Chemoselectivity of Multicomponent Condensations of Barbituric Acids 5-Aminopyrazoles and Aldehydes E A Muravyova S V Shishkina V I Musatov I V Knyazeva O V Shishkin S M Desenko V A Chebanov
1386 Stereoselective Total Syntheses of Leiocarpin A and (ndash)-Galantinic Acid Starting from D-Mannitol K Nagaiah D Sreenu K V Purnima R S Rao J S Yadav
1393 A Facile Mild Deprotection Protocol for 13-Dithianes and 13-Dithiolanes with 30 Hydrogen Peroxide and Iodine Catalyst in Aqueous Micellar System N C Ganguly S K Barik
1400 Rhodium-Catalyzed Gram-Scale Synthesis of Highly Substituted Pyridine Derivatives K Parthasarathy C-H Cheng
1403 Enantioselective Synthesis of (R)-Propylene Carbonate from Ethyl (S)-Lactate J M Whitaker R C Ronald
XIII Forthcoming Articles
no 9 1405 Transition-Metal-Catalyzed Site-Selective Cross-Coupling of Di- and
Polyhalogenated Compounds J-R Wang K Manabe 1428 An Improved Synthesis of (4-4-Hydroxy-3-isopropyl-5-[(4-nitrophenyl)
ethynyl]benzyl-35-dimethylphenoxy)acetic Acid (NH-3) M B Gopinathan K S Rehder
1431 Copper-Catalyzed Tandem CndashN Bond Formation Reaction Selective Synthesis of 2-(Trifluoromethyl)benzimidazoles M-W Chen X-G Zhang P Zhong M-L Hu
1437 Synthesis and Thermochemical Properties of Stereoisomeric Dihydroxy- and Tetrahydroxyalkylammonium Salts M Thomas L Rothman J Hatcher P Agarkar R Ramkirath S Lall-Ramnarine R Engel
1445 Preparation of 5-Substituted 2-(2-Alkylaryl-1H-imidazol-4-yl)oxazoles and 5-Substituted 2-(2-Alkylarylthiazol-4-yl)oxazoles by Utilizing 5-Substituted 2-(2-Bromo-11-diethoxyethyl)oxazole as a Synthon D R St Laurent J L Romine
1459 Novel and Efficient Methods for the Synthesis of Symmetrical Trisulfides A Kertmen S Lach J Rachon D Witt
1463 An Environmentally Benign Electrochemical Process for the Reduction of Carboxylic Acid Hydrazides to Amides M Mentel M J Beier R Breinbauer
1469 Synthesis of 1-Chloroalkynes from Alkynylsilanes Using Trichloroisocyanuric Acid as Chlorinating Agent M H Vilhelmsen A S Andersson M B Nielsen
1473 A Convenient Approach to Enantioenriched Cyclopropanes Bearing Electron-Withdrawing Functionalities H Krawczyń K Wąsek J Kędzia
1477 Synthesis of Cyclopropenes via 12-Elimination of Bromocyclopropanes Catalyzed by Crown Ether W M Sherrill R Kim M Rubin
1485 A Base-Catalysed One-Pot Three-Component Coupling Reaction Leading to Nitrosubstituted Pyrroles I R Baxendale C D Buckle S V Ley L Tamborini
1494 Synthesis of 4-Alkylidene-4H-31-benzoxazine Derivatives by Acid-Catalyzed Cyclization of 2-Isocyanophenyl Ketones in the Presence of a Vinyl Ether K Kobayashi Y Okamura H Konishi
1499 Synthesis of Higher Helicenes via Olefin Metathesis and CndashH Activation J Cocircteacute S K Collins
1506 Azido- and Ethynyl-Substituted 2262-Terpyridines as Suitable Substrates for Click Reactions A Winter A Wild R Hoogenboom M W M Fijten M D Hager R-A Fallahpour U S Schubert
1513 Synthesis of 2-(Arylamino)ethanethiols via Lewis Acid Catalyzed Aminolysis of 22-Dimethylthiirane as Precursors of the 14-Benzothiazine Nucleus R Spogli S Sabatini G Manfroni O Tabarrini V Cecchetti
1520 Iron(III) Chloride A Versatile Catalyst for the Practical Synthesis of 3-Sulfenylindoles J S Yadav B V S Reddy Y J Reddy K Praneeth
1525 Organocatalytic Enantioselective Conjugate Addition of 2-Fluoromalonate to Nitroolefins Direct Synthesis of Chiral Fluorinated γ-Nitro Carboxylic Acid Derivatives H Li L Zu H Xie W Wang
1531 Asymmetric Transfer Hydrogenation of Ketimines with Trichlorosilane Structural Studies Z Zhang P Rooshenas H Hausmann P R Schreiner
1545 Prolinol Sulfinyl Ester Derivatives Organocatalytic Michael Addition of Ketones to Nitroolefins under Neat Conditions X Zeng G Zhong
1551 Asymmetric Oxidations of Electron-Poor Alkenes Promoted by the β-Amino AlcoholTBHP System A Russo A Lattanzi
1557 Enantioselectivity Switch in Direct Asymmetric Aminoxylation Catalyzed by Binaphthyl-Based Chiral Secondary Amines T Kano A Yamamoto F Shirozu K Maruoka
1564 Enantioselective Conjugate Addition of N-Heterocycles to αβ-Unsaturated Ketones Catalyzed by Chiral Primary Amines G Luo S Zhang W Duan W Wang
1573 Sulfonyl Hydrazine as New Functionality in Organocatalysis Camphorsulfonyl Hydrazine Catalyzed Enantioselective Aza-Michael Addition L-Y Chen H He B-J Pei W-H Chan A W M Lee
1578 Conversion of Primary Alcohols and Aldehydes into Methyl Esters by Ruthenium-Catalysed Hydrogen Transfer Reactions N A Owston T D Nixon A J Parker M K Whittlesey J M J Williams
1582 Addendum and Erratum XVII Forthcoming Articles
no 10 1583 Organocatalytic Formation of Quaternary Stereocenters M Bella
T Gasperi 1615 Regioselective Synthesis of 5H-Thiazolo[32-a]pyrimidin-5-ones from
MoritandashBaylisndashHillman Adduct Acetates under Solvent-Free and Base-Free Conditions W Zhong B Guo F Lin Y Liu W Su
1623 First Synthesis of 5-Cyanosalicylates by Formal [3+3] Cyclocondensations of 13-Bis(silyloxy)-13-butadienes A Riahi O Fatunsin M Shkoor R Dede H Reinke C Fischer P Langer
1635 Reaction of Isocyanides Dialkyl Acetylenedicarboxylates and a-Keto Lactones Unexpected Participation of an Ester Carbonyl Group in the Isocyanide-Based Three-Component Reaction A A Esmaeili H Vesalipoor
1639 An Efficient and Chemoselective Synthesis of 16-Naphthyridines and Pyrano[32-c]pyridines under Microwave Irradiation Z-G Han S-J Tu B Jiang S Yan X-H Zhang S-S Wu W-J Hao X-D Cao F Shi G Zhang N Ma
1647 N-Activation of N-Arylimidazoles Facile Syntheses of N-Alkyl-N-arylimidazolium Iodides from Less Expensive Chloro Substrates A M Oertel V Ritleng M J Chetcuti
1651 Synthesis of Polyhalogenated 2-(Phenylamino)pyridines by Thermal Amination Reactions S R Waldvogel A Faust W Barkmann R Froumlhlich O Wolff
1655 Cyanide Ion Promoted Addition of Acylphosphonates to Diethyl Cyanophosphonate Synthesis of Phosphonocyanohydrin O-Phosphates A S Demir A Aybey M Emrullahoglu
1659 Straightforward and Scalable Synthesis of Orthogonally Protected 37-Diazabicyclo[410]heptane H Schramm M Pavlova C Hoenke J Christoffers
1663 Hypervalent Iodine Mediated Oxidation of 12-Diaminobenzimidazole and Its Schiff Bases Efficient Synthesis of 3-Amino-124-benzotriazine and 2-Aryl-124-triazolo[15-a]benzimidazoles A Kumar M Parshad R K Gupta D Kumar
1667 Synthesis of the Reported Protoberberine Gusanlung D P B Wakchaure S Easwar N P Argade
1673 2-(Azidomethyl)arylboronic Acids in the Synthesis of Coumarin-Type Compounds M I Naumov A V Nuchev N S Sitnikov Y B Malysheva A S Shavyrin I P Beletskaya A E Gavryushin S Combes A Y Fedorov
1683 Asymmetric Synthesis of 12-anti-Disubstituted Taurine Derivatives D Enders D Iffland G Raabe
1689 A Novel One-Pot Three-Component Synthesis of 5-Imino-2358-tetrahydropyrazolo[12-a]pyridazin-1-one Derivatives B Qian M-J Fan Y-X Xie L-Y Wu Y Shi Y-M Liang
1694 One-Portion Synthesis of 2-Acetoxy Carbonyl Compounds from Aldehydes by Using an Acetylated Masked Acyl Cyanide H Nemoto T Kawamura K Kitasaki K Yatsuzuka M Kamiya Y Yoshioka
1703 Synthesis of 9-Anthryl Ethers from trans-910-Dihydro-910-dimethoxyanthracene by Acid-Catalyzed Transetherification K S Jang H Y Shin D Y Chi
1708 Efficient Synthesis of Azo Dye Labeled Terpenes Sugars and Steroids Using N-(4-Arylazobenzoyl)-1H-benzotriazoles A R Katritzky S R Tala N E Abo-Dya Z K Abdel-Samii
1715 Tandem CH-ActivationndashImine-Formation Reaction A New Route to Imidazo[21-a]phthalazines A Heim-Riether K R Gipson
1720 A Convenient and Efficient α-Sulfenylation of Carbonyl Compounds E Okragla S Demkowicz J Rachon D Witt
1725 Stereoselective Synthesis of β-Branched Phenylalanine Derivatives via Chelate-Claisen Rearrangement C Quirin U Kazmaier
1732 Catalyst-Free and Base-Free Water-Promoted SNAr Reaction of Heteroaryl Halides with Thiols B Sreedhar P S Reddy M A Reddy
1739 Convenient Methods for Synthesis of C2-Symmetric Diphenyltetrahydrothiophenes M Periasamy G Ramani G P Muthukumaragopal
1744 Highly Diastereoselective Conjugate AdditionndashElimination of Chiral Nickel(II) Glycinate with Activated Allylic Acetates for Asymmetric Synthesis of Glutamic Acid Derivatives J Wang J Shi X Zhang D Lin H Jiang H Liu
1753 Synthesis of 36-Dimethoxybenzene-12-diamine and of 47-Dimethoxy-2-methyl-1H-benzimidazole T Besset C Morin
1757 An Inexpensive Procedure for Reductive Aminations Using Dimethylamineborane on Millimolar and Molar Scale R Ortmann M Schlitzer
1760 Classics in Stereoselective Synthesis Edited by E M Carreira L Kvaerno Reviewed by Rolf Breinbauer
XV Forthcoming Articles
no 11 1761 Transition-Metal-Catalyzed Enantioselective Synthesis of Compounds with
Non-Centrochirality M Ogasawara S Watanabe 1786 One-Pot Synthesis of 3-Acyl-2-(alkylsulfanyl)indoles and 2-(Alkylsulfanyl)-
indole-3-carboxylates from (2-Isocyanophenyl)methyl Ketones or (2-Isocyanophenyl)acetates S Fukamachi H Konishi K Kobayashi
1791 Efficient and Recyclable Phthalocyanine-Based Sensitizers for Photooxygenation Reactions H Xu W-K Chan D K P Ng
1797 A Facile and Practical One-Pot Synthesis of β-Oxo Thioamides from β-Oxo Amides and Isothiocyanates P Huang D Xiang Y Zhou Y Liang T Na D Dong
1801 Microwave-Promoted Solid-Acid-Catalyzed One-Pot Synthesis of Phthalazinones V M Outerbridge S M Landge H Tamaki B Toumlroumlk
1807 Benzylic Brominations with N-Bromosuccinimide in (Trifluoromethyl)-benzene D Suarez G Laval S-M Tu D Jiang C L Robinson R Scott B T Golding
1811 Synthesis of Thioflavanone and Flavanone Derivatives by Cyclization of Chalcones W Konieczny M Konieczny
1815 A New and Expedient Total Synthesis of Ochratoxin A and d5-Ochratoxin A B Gabriele M Attya A Fazio L Di Donna P Plastina G Sindona
1821 Synthesis of Benzopyrrolizidinones by NorrishndashYang Cyclization of 3-(Acylmethyl)-2-alkylisoindol-1-ones J Wu W Zhang C Wang
1829 Reactions of MoritandashBaylisndashHillman Acetates with Huisgen Zwitterions A Novel Strategy for the Synthesis of β-Amino Acid Derivatives A Jose R R Paul R Mohan S C Mathew A T Biju E Suresh V Nair
1834 Peracetylated β-Allyl C-Glycosides of D-Ribofuranose and 2-Deoxy- D-ribofuranose in the Chemical Literature Until Now Mirages in the Literature H Otero Martinez H Reinke D Michalik C Vogel
1841 Core-Tetrasubstituted Naphthalene Diimides by Stille Cross-Coupling Reactions and Characterization of Their Optical and Redox Properties S-L Suraru F Wuumlrthner
1846 A Practical Synthesis of Indole-Based Heterocycles Using an Amidoaluminum-Mediated Strategy R Todd M M Hossain
1851 Synthesis of Fluorinated Pyrrolo[23-b]pyridine and Pyrrolo[23-d]pyrimidine Nucleosides V O Iaroshenko Y Wang D V Sevenard D M Volochnyuk
1858 Recyclization Reactions of 5-Formyl-13-dimethyluracil with Electron-Rich Amino Heterocycles A P Mityuk D M Volochnyuk S V Ryabukhin A S Plaskon A Shivanyuk A A Tolmachev
1865 Facile Synthesis of Fluorinated 1-Desazapurines V O Iaroshenko D V Sevenard D M Volochnyuk Y Wang A Martiloga A O Tolmachev
1876 A Practical Synthesis of 3-Diethoxyphosphoryl-12-pyridazine Derivatives J-C Monbaliu J Marchand-Brynaert
1881 Enantioselective Reduction of Prochiral Ketones Employing Sprouted Pisum sativa as Biocatalyst J S Yadav B V S Reddy C Sreelakshmi A B Rao
1886 Application of Phenolate Ion Mediated Intramolecular Epoxide Ring Opening in the Enantioselective Synthesis of Functionalized 23-Dihydrobenzofurans and 1-Benzopyrans S K Dinda S K Das G Panda
1897 Complementary Synthetic Approaches to Constitutionally Diverse N-Aminoalkylated Isoindolinones Application to the Synthesis of Falipamil and 5-HT1A Receptor Ligand Analogues M Lorion A Couture E Deniau P Grandclaudon
1904 Selective Deprotection of Silyl Ethers with Sodium Periodate J Li D Menche
1909 Micellar Solution of Sodium Dodecyl Sulfate (SDS) Catalyzes KabacknikndashFields Reaction in Aqueous Media S Sobhani A Vafaee
1916 Convenient Methods for the Synthesis of a Library of Hemilabile Phosphines M V Jimeacutenez J J Peacuterez-Torrente M I Bartolomeacute L A Oro
1923 Terminal Aziridines by Addition of Grignard Reagents or Organoceriums to an (α-Chloro)sulfinylimine D M Hodgson J Kloesges B Evans
1933 A Robust Synthesis of Nε-(Carboxymethyl)-L-lysine (CML) R Csuk S Stark A Barthel R Kluge D Stroumlhl
1935 One-Pot Curtius Rearrangement Processes from Carboxylic Acids O Leogane H Lebel
XV Forthcoming Articles
no 12 1941 The Chemistry of Deprotonated α-Aminonitriles T Opatz 1960 An Efficient Synthesis of Tetraalkyl 2345-Thiophenetetracarboxylate
Derivatives A Alizadeh R Hosseinpour 1963 Facile Deprotection of Bulky (Trialkylsilyl)acetylenes with Silver Fluoride
S Kim B Kim J In 1969 Highly Efficient and Reusable Ionic Liquids for the Catalyzed
Hydroamination of Alkenes with Sulfonamides Carbamates and Carboxamides L Yang L-W Xu C-G Xia
1975 Synthesis of 2391016172324-Octasubstituted Phthalocyaninatozinc(II) Complexes Mediated by Reductive Agents G A Gauna A C Monsalvo J Awruch
1979 A Short and Efficient Synthesis of 3-2-[2-(Bromomethyl)thiazol-4-yl]-ethynyl-5-fluorobenzonitrile A Precursor for PET Radioligand [18F]SP203 M B Gopinathan C Jin K S Rehder
1983 Synthesis of a Substituted Benzazepin-2-one Dihydrate S K Boini R K Vaid K P Moder D Mitchell
1987 Synthesis of Novel Trisubstituted Imidazolines F J Lakner M A Parker B Rogovoy A Khvat A Ivachtchenko
1991 A Novel Synthesis of N-But-3-enyl-α- and β-Amino Acids T T Van Nguyen R T C Brownlee A B Hughes
1999 Synthesis of Substituted 5-(3-Hydroxypropyl)pyrrolidin-2-ones and Pyrrolizidinones from Nitroethane via C3 Functionalized 56-Dihydro-4H-12-oxazines A Novel Approach to Some Analogues of the Antidepressant Rolipram A Yu Sukhorukov A V Lesiv Y A Khomutova S L Ioffe V A Tartakovsky
2009 Chiral Cyclobutanols and Cyclopentane Dimers via Samarium(II) Iodide Induced Keto-Olefin Cyclisations of Carbohydrate-Derived Unsaturated Ketones D B G Williams J Caddy K Blann J J C Groveacute C W Holzapfel
2015 Synthesis of Perfluoroalkylthio-Substituted Ferrocenes C Rhode J Lemke M Lieb N Metzler-Nolte
2019 Functionalization of Polyhedral Oligomeric Silsesquioxane (POSS) via Nucleophilic Substitution M Dutkiewicz H Maciejewski B Marciniec
2025 A Novel Synthesis of Aryl Mesylates via One-Pot DemethylationndashMesylation of Aryl Methyl Ethers Using a Mixture of Phosphorus Pentoxide in Methanesulfonic Acid B Kaboudin Y Abedi
2029 Anionic Cyclization of (NN-Dimethylamino)[2-(prop-2-yn-1-yloxy)aryl]-acetonitriles T Zdrojewski J Musielak A Jończyk
2035 Strecker-Type Reaction Catalyzed by Carboxylic Acids in Aqueous Media Z Xie G Li G Zhao J Wang
2040 Synthesis of Novel Structurally Simplified Estrogen Analogues with Electron-Donating Groups in Ring A L F Tietze C A Vock I K Krimmelbein L Nacke
2061 On the Resolution of Secondary Phosphine Oxides via Diastereomeric Complex Formation The Case of tert-Butylphenylphosphine Oxide J Holt A M Maj E P Schudde K M Pietrusiewicz L Sieroń W Wieczorek T Jerphagnon I W C E Arends U Hanefeld A J Minnaard
2066 Enantioselective Copper-Catalyzed Conjugate Addition of Dimethylzinc to 5-(1-Arylalkylidene) Meldrumrsquos Acids A Wilsily T Lou E Fillion
2073 SuzukindashMiyaura Coupling Reactions Using Phosphite Ligands M Jang Y Jo I-K Oh H M Jung S Lee
2076 Synthesis of 2-Methylindoline- and 2-Methyl-1234-tetrahydroquinoline-Derived Phosphoramidites and Their Applications in Iridium-Catalyzed Allylic Alkylation of Indoles W-B Liu H He L-X Dai S-L You
2083 Stereocontrolled Synthesis of 13-Amino Alcohols by Reduction of Substituted 2-1-[(tert-Butylsulfinyl)amino]alkylcyclohexanones J C Gonzaacutelez-Goacutemez F Foubelo M Yus
2089 Tunable Phosphoramidite Ligands for Asymmetric Hydrovinylation Ligands par excellence for Generation of All-Carbon Quaternary Centers C R Smith H J Lim A ZhangT V RajanBabu
2101 Copper-Catalyzed Asymmetric Ring-Opening Reaction of Oxabenzonorbornadienes with Grignard and Aluminum Reagents R Millet L Gremaud T Bernardez L Palais A Alexakis
2113 A Simplified Synthesis of Takemotorsquos Catalyst A Berkessel B Seelig 2116 Pharmaceutical Substances Syntheses Patents and Applications of the
Most Relevant AIPs Edited by Axel Kleeman Juumlrgen Engel Bernhard Kutscher Dietmar Reichert Reviewed by I Agranat
XV Forthcoming Articles
no 13 2117 Recent Advances in the Aza-Claisen Rearrangement K C Majumdar
T Bhattacharyya B Chattopadhyay B Sinha 2143 A Novel and Convenient Synthesis of lsquoReversedrsquo Diamidino 25-Aryl- and
25-Azaheterocycle-Substituted Furans L Hu D W Boykin 2146 Efficient and General Preparation of Pyranostilbenes First Total Synthesis
of Artocarbene and Pawhuskin B B H Park Y R Lee W S Lyoo 2155 Mild Oxidation of Diarylacetylenes to 12-Diketones Using Oxone in
Trifluoroacetic Acid J-H Chu Y-J Chen M-J Wu 2163 One-Pot Microwave-Assisted Selective Azido ReductionTandem Cyclization
in Condensed and Solid Phase with Nickel Boride N Shankaraiah N Markandeya M Espinoza-Moraga C Arancibia A Kamal L Silva Santos
2171 Pyrrolo[321-ij]quinolin-4-one and Pyrrolo[321-ij]quinolin-6-one H McNab D J Nelson E J Rozgowska
2175 Practical Synthesis of 5-Substituted Tetrazoles under Microwave Irradiation J Roh T V Artamonova K Vaacutevrovaacute G I Koldobskii A Hrabaacutelek
2179 A Simple Method for the Synthesis of 3-Arylthieno[23-b]pyridines via Iodine-Mediated Cyclization of 3-(1-Arylalkenyl)-2-[(1-phenylethyl)sulfanyl]pyridines K Kobayashi D Nakamura Y Shiroyama S Fukamachi H Konishi
2184 Synthesis of Four Lysine-Linked Cereulide Analogues Showing Ionophoric Activity Towards Potassium Cations as Lead Compounds for Emetic Toxin-Detection by Immunoassays A Makarasen T Nishikawa M Isobe
2205 Synthesis of α-Aliphatic and β-Aromatic Substituted Taurines via Regioselective Ring Opening of Thiiranes with Ammonia H Yu S Cao L Zhang G Liu J Xu
2210 Stability of 5(6)-Carboxyfluorescein in Microwave-Assisted Synthesis of Fluorescein-Labelled O-Dimannosylated Peptides R Kowalczyk P W R Harris R P Dunbar M A Brimble
2223 Diversity-Oriented Synthesis of Functionalized Diaryl Sulfones by Regioselective [3+3] Cyclizations of 13-Bis(siloxy)buta-13-dienes with 2-(Arylsulfonyl)-3-ethoxy-2-en-1-ones Scope and Limitations M Shkoor A Riahi O Fatunsin H Reinke C Fischer P Langer
2236 Synthesis of Functionalized Salicylates by Formal [3+3] Cyclocondensation of 13-Bis(silyloxy)buta-13-dienes with 3-Alkoxy-2-en-1-ones G Mroszlig S Ladzik H Reinke A Spannenberg C Fischer P Langer
2249 Synthetic Approach to Alkoxy-β-(trifluoromethyl)styrenes and Their Application in the Synthesis of New Trifluoromethylated Heterocycles V M Muzalevskiy V G Nenajdenko A V Shastin E S Balenkova G Haufe
2260 o-Benzenedisulfonimide as a Powerful and Recyclable Organocatalyst for the Nazarov Reaction M Barbero S Cadamuro A Deagostino S Dughera P Larini E G Occhiato C Prandi S Tabasso R Vulcano P Venturello
2267 The Catalytic Potential of 4-Guanidinylpyridines in Acylation Reactions I Held E Larionov C Bozler F Wagner H Zipse
2278 Iron(III) Chloride in EthanolndashWater Highly Efficient Catalytic System for the Synthesis of Garcia Gonzalez Polyhydroxyalkyl- and C-Glycosylfurans L Nagarapu M V Chary A Satyender B Supriya R Bantu
2283 Ruthenium-Catalyzed Addition of Primary Amides to Alkynes A Stereoselective Synthesis of Secondary Enamides L J Gooszligen M Blanchot K S M Salih K Gooszligen
2289 Binaphthyl-Modified Quaternary Phosphonium Salts as Chiral Phase Transfer Catalysts Application to Asymmetric Amination of β-Keto Esters R He K Maruoka
X Table of Contents XI Forthcoming Articles
no 14 2293 Direct Methods for Stereoselective Polypropionate Synthesis A Survey
J Li D Menche 2316 Synthesis of Symmetrical Ketones from Grignard Reagents and
11-Carbonyldiimidazole D Bottalico V Fiandanese G Marchese A Punzi
2319 Synthesis of 45-Substituted Imidazoles by a Fast Condensation of 12-Diketones and Urotropine in Heterogeneous Medium G Bratulescu
2321 (Arylsulfonyl)acetones and -acetonitriles New Activated Methylenic Building Blocks for Synthesis of 123-Triazoles N T Pokhodylo V S Matiychuk M D Obushak
2324 A Safe Convenient and Efficient One-Pot Synthesis of α-Chloroketone Acetals Directly from Ketones Using Iodobenzene Dichloride J Yu C Zhang
2329 An Efficient Oxidative Conversion of Aldehydes into 2-Substituted 2-Oxazolines Using 13-Diiodo-55-dimethylhydantoin S Takahashi H Togo
2333 A Novel Procedure for the Synthesis of Benzo[b][18]naphthyridine-3-carboxylate Derivatives from MoritandashBaylisndashHillman Adduct Acetates W Zhong F Lin R Chen W Su
2341 An Improved Synthesis of 147-Triazacyclononanes (tacns) and 14710-Tetraazacyclododecanes (cyclens) J Huang Z Zhou T H Chan
2345 The Ullmann Coupling between 2-Chlorobenzoic Acids and Amino Acids A Valuable Reaction for Preparing 2-Substituted 1-Acetyl-1H-indol-3-yl Acetates J C Rodriguez Dominguez X Gang G Kirsch
2349 gem-Dibromomethyl Aromatics Efficient Aldehyde Equivalents in the KnoevenagelndashDoebner Reaction J K Augustine Y A Naik S Poojari N Chowdappa B S Sherigara K Areppa
2357 Synthesis of Novel α-Aminophosphonates Containing Adamantyl Fragment M M Kabachnik L I Minaeva I P Beletskaya
2361 Efficient Fluoride-Mediated Synthesis of 5-Amino-Substituted Isothiazoles Y S Zubenko V I Potkin
2365 Phosphine-Catalyzed Reaction of Cyanohydrins with Activated Alkynes A Siby O Loreau F Taran
2371 Sulfanyl-Substituted [3]Cumulenes and Buta-13-dienes from a Tetrakis(pyridinium)-Substituted Butadiene A Schmidt A Rahimi M Gjikaj
2379 Efficient Synthesis of 2-Substituted Pyrido[32-d]pyrimidines Involving SNAr and Palladium-Catalyzed Cross-Coupling Reactions A Tikad S Routier M Akssira J-M Leacuteger C Jarry G Guillaumet
2385 Novel Synthesis of Medium-Sized Heterocycles by Palladium-Catalyzed Intramolecular Heck Reaction via 9-endo-trig Mode of Cyclization K C Majumdar B Chattopadhyay
2393 Facile Synthesis of Fluorinated Benzofuro- and Benzothieno[23-b]pyridines α-Carbolines and Nucleosides Containing the α-Carboline Framework V O Iaroshenko Y Wang B Zhang D Volochnyuk V Ya Sosnovskikh
2403 Synthesis of Functionalized N-Vinyl Nitrogen-Containing Heterocycles S M M Lopes A M Beja M Ramos Silva J A Paixatildeo F Palacios T M V D Pinho e Melo
2408 Kumada Cross-Coupling of Aryl Grignard Reagents with Aryl Halides Catalyzed by an Immobilized Nickel Catalyst X Chen L Wang J Liu
2413 Highly Enantioselective Synthesis of Heteroaromatic Alcohols Catalyzed by Chiral DiaminodiphosphinendashRuthenium(II) Complexes W-Y Shen Y-Y Li Z-R Dong J-X Gao
2418 Concise Total Synthesis of (+)-Disparlure and its trans-Isomer Using Asymmetric Organocatalysis S-G Kim
2423 Rhodium Carbenoid Induced [12]-Migration in an L-Lyxo-Configured α-Diazo β-Keto Ester Synthesis of a New Griseolic Acid Analogue N N Bhujbal K S A Kumar D D Dhavale
2430 Synthesis of 5-Arylthio-3-hydroxyphthalates by the First [4+2] Cycloadditions of 3-Arylthio-1-silyloxy-13-butadienes with Dimethyl Acetylenedicarboxylate I Iqbal M Imran P Langer
2435 Synthesis of Highly Functionalized Proline Derivatives via a One-Pot MichaelSN-AdditionCyclization Approach U Kazmaier C Schmidt
2440 RhodiumGraphite-Catalyzed Hydrogenation of Carbocyclic and Heterocyclic Aromatic Compounds G Falini A Gualandi D Savoia
2447 Potassium [1-(tert-Butoxycarbonyl)-1H-indol-2-yl]trifluoroborate as an Efficient Building Block in Palladium-Catalyzed SuzukindashMiyaura Cross Couplings P Kassis V Beacuteneacuteteau J-Y Meacuterour S Routier
2454 Syntheses of Substituted Furans and Pyrroles by Platinum-Catalyzed Cyclizations of Propargylic Oxiranes and Aziridines in Aqueous Media M Yoshida M Al-Amin K Shishido
2467 Transition-Metal-Free Oxidative Homocoupling of Aryl Alkenyl and Alkynyl Grignard Reagents with TEMPO M S Maji A Studer
XIII Forthcoming Articles
no 15 2471 Advances in Synthetic Approaches for the Preparation of Combretastatin-
Based Anti-Cancer Agents R Singh H Kaur 2492 Synthesis of Unsymmetrical Ureas by Sulfur-Assisted Carbonylation with
Carbon Monoxide and Oxidation with Molecular Oxygen under Mild Conditions T Mizuno T Nakai M Mihara
2497 Ring-OpeningRecyclization Reactions of (Dimethylamino)propenoyl-Substituted Cyclopropanes Facile Synthesis of Halogenated Pyridin-2(1H)-ones R Zhang Y Zhou Y Liang Z Jiang D Dong
2501 Facile and Efficient Total Synthesis of Taspine B Cheng S Zhang L Zhu J Zhang Q Li A Shan L He
2505 Oligomeric Iodosylbenzene Sulfate A Convenient Hypervalent Iodine Reagent for Oxidation of Organic Sulfides and Alkenes M S Yusubov R Y Yusubova T V Funk K-W Chi V V Zhdankin
2509 Pyrrolidine-Based Organocatalysts for Enantioselective Michael Addition of Cyclohexanone to trans-β-Nitrostyrene A P Carley S Dixon J D Kilburn
2517 CundashAl Hydrotalcite An Efficient and Reusable Ligand-Free Catalyst for the Coupling of Aryl Chlorides with Aliphatic Aromatic and N(H)-Heterocyclic Amines B Sreedhar R Arundhathi P L Reddy M A Reddy M L Kantam
2523 Highly Efficient Synthesis of trans-βγ-Unsaturated a-Keto Amides C Allais T Constantieux J Rodriguez
2531 Gas-Phase Synthesis of N-Unsubstituted 3-Hydroxypyrroles and 1H-Pyrrol-3(2H)-ones L Hill G A Hunter S H Imam H McNab W J OrsquoNeill
2535 3-Hydroxy-1H-pyrrole L Hill S H Imam H McNab W J OrsquoNeill 2539 123-Thiadiazoles with Unsaturated Side Chains Synthesis
Polymerization and Photocrosslinking M Al-Smadi N Hanold H Kalbitz H Meier
2547 Synthesis of 1112-Didehydrodibenzo[ae]cycloocten-5(6H)-one A Strained Eight-Membered Alkyne S C Kornmayer F Rominger R Gleiter
2553 Stannous Chloride Dihydrate A Novel and Efficient Catalyst for the Synthesis of gem-Dihydroperoxides from Ketones and Aldehydes D Azarifar K Khosravi F Soleimanei
2557 Synthesis of a Novel Class of Azacrown Macrocycles and Lariat Crown Ethers Containing Two 124-Triazole Rings as Subunits N Foroughifar A Mobinikhaledi S Ebrahimi
2561 Enantioselective Synthesis of the 3C-Protease Inhibitor (ndash)-Thysanone by a StauntonndashWeinreb Annulation Strategy J Sperry T Y Yuen M A Brimble
2570 Stereoselective Synthesis of Unnatural β-Amino Acids from Nitroethane via 56-Dihydro-4H-12-oxazin-3-ylacetates A Yu Sukhorukov A V Lesiv O L Eliseev Y A Khomutova S L Ioffe
2579 A Versatile Unexpected One-Pot Regioselective Synthesis of a New Class of 13-Diazepinoindolones by Reaction of Pyranoindolones with Monosubstituted Ureas D Livadiotou C A Tsoleridis J Stephanidou-Stephanatou
2584 Synthesis of a Trisaccharide and a Tetrasaccharide from the Cell-Wall Lipopolysaccharides of Azospirillum brasilense S17 S Pandey S Ghosh A K Misra
2591 Synthesis of Isoindoline Nitroxides by Electrocyclic Reactions T Kaacutelai J Jekı K Hideg
2596 Glycosylations of Tertiary Alcohols Synthesis of Fully Protected Disaccharides with Sterically Demanding Groups Attached to the Sugar Core A Holkenbrink J B Vicente D B Werz
2605 Copper-Catalyzed [13]-Dipolar Cycloaddition for the Synthesis of Macrocycles Containing Acyclic Aromatic and Steroidal Moieties G V Latyshev M S Baranom A V Kazantsev A D Averin N V Lukashev I P Beletskaya
2616 Aryl Ring Migration Reaction in the Synthesis of 24-Diaryl-4H-31-benzothiazines A V Butin F A Tsiunchik V T Abaev A V Gutnov D A Cheshkov
2627 Hydrogenation of β-N-Substituted and β-NN-Disubstituted Enamino Esters in the Presence of Iridium(I) Catalyst H Hebbache Z Hank C Bruneau J-L Renaud
2634 Stereoselective Olefination Reactions Promoted by Rieke Manganese J M Concelloacuten H Rodriacuteguez-Solla V del Amo P Diacuteaz
2646 Synthesis of Piperidinones through a Radical Cascade E Godineau Y Landais
2650 Asymmetric Organic Synthesis with Enzymes Edited by V Gotor I Alfonso E Garciacutea-Urdiales Reviewed by Steve Collier
XVII Forthcoming Articles
no 16 2651 Synthesis of Spirocyclic Ethers S Rosenberg R Leino 2674 Bimetallic PalladiumndashPlatinum-on-Carbon-Catalyzed HndashD Exchange
Reaction Synergistic Effect on Multiple Deuterium Incorporation T Maegawa N Ito K Oono Y Monguchi H Sajiki
2679 Efficient Copper-Catalyzed Synthesis of 2-Amino-4(3H)-quinazolinone and 2-Aminoquinazoline Derivatives X Huang H Yang H Fu R Qiao Y Zhao
2689 Synthesis and Chemoselective N- and O-Alkylation of Thiadiazolopyrimidine Nucleosides and Uridines A M L Hossion R Islam R K Kandahary T Nagamatsu
2697 Facile and Efficient Synthesis of a New Class of Indole-Substituted Pyridine Derivatives via One-Pot Multicomponent Reactions K Zhao X-P Xu S-L Zhu D-Q Shi Y Zhang S-J Ji
2709 Studies toward a Total Synthesis of Rhizoxin D Stereoselective Preparation of the C11ndashC19 Fragment S Padakanti C K Kumar E Ashok P Das
2715 A Short Synthesis of Enantiomeric Phytoprostanes B1 Type I W Perlikowska M Mikołajczyk
2719 Chemistry of Polyhalogenated Nitrobutadienes Part 7 A Novel Synthetic Access to Chlorinated Nitrile Oxides E Nutz V A Zapolrsquoskii D E Kaufmann
2725 Microwave-Assisted Silver(I)-Mediated Selective O-Alkylation of Aromatic Imidate Systems B K Singh C Cavalluzzo M De Maeyer Z Debyser V S Parmar E Van der Eycken
2729 Iodogen A Novel Reagent for the Oxidation of Urazoles under Heterogeneous Conditions A Khoramabadi A Shiri M A Zolfigol S Mallakpour
2733 An Unprecedented Synthesis of Eight-Membered-Ring Cyclic Thioimidic Esters by a Three-Component Reaction A Alizadeh R Hosseinpour
2737 A Novel Diastereoselective Synthesis of β-Phosphonato Unsaturated Thioimidates A Alizadeh N Zohreh
2741 Synthesis of 21-Benzisoxazoles by Nucleophilic Substitution of Hydrogen in Nitroarenes Activated by the Azole Ring N T Pokhodylo Y O Teslenko V S Matiychuk M D Obushak
2749 A Facile Synthesis of Two Series of Multifunctional Carbon Compounds from αα-Dihalo Ketones Using Allylsamarium Bromide X Liu S Zhang J Di
2756 Stereocontrolled Formation of Protected Aminodeoxyalditols from Simple Carbohydrate Precursors by Debenzylating Cycloetherification Y Jiang Z Fang Q Zheng H Jia J Cheng B Zheng
2761 trans-Stilbene as a Starting Material for the Synthesis of Tamoxifen Based on Palladium-Catalyzed Cross-Coupling Reactions C M Nunes J Limberger S Poersch M Seferin A L Monteiro
2766 Synthesis and Biological Evaluation of 6-Substituted Purinylcarbanucleosides with a Cyclopenta[b]thiophene Pseudosugar P Abeijoacuten J M Blanco O Caamantildeo F Fernaacutendez M D Garciacutea X Garciacutea-Mera J E Rodriacuteguez-Borges J Balzarini E De Clercq
2773 Synthesis and Electrochemical Signature of Novel Norbornyl-ferrocene Hybrids F A Khan S K Upadhyay
2778 A Regioselective TsujindashTrost Pentadienylation of 3-Allyltetronic Acid R Schobert B Barnickel
2785 Copper(I)-Catalyzed CarylndashCalkynyl Bond Formation of Aryl Iodides with Terminal Alkynes K G Thakur G Sekar
2790 Aminolysis of Epoxides Using Iridium Trichloride as an Efficient Catalyst J Agarwal A Duley R Rani R K Peddinti
2797 Preparation of Several Active N-Chloro Compounds from Trichloroisocyanuric Acid A Shiri A Khoramabadi-zad
2802 The First Mineral-Catalyzed One-Pot [3+1+2] Coupling Protocol for Multifunctionalized Fused-Ring Pyrimidines L D S Yadav A Rai
2809 Efficient Synthesis of Tetrahydro-β-carbolin-1-one and Dihydroisoquinolin-1-one Derivatives as Versatile Intermediates K E Judd M F Mahon L Caggiano
2818 A Concise Synthesis of ortho-Iodobenzyl Alcohols via Addition of ortho-Iodophenyl Grignard Reagent to Aldehydes and Ketones J Cvengroš D Stolz A Togni
XIII Forthcoming Articles
no 17 2825 Reactivity of Oxazol-5-(4H)-ones and Their Application toward Natural
Product Synthesis N M Hewlett C D Hupp J J Tepe 2840 Towards the Total Synthesis of 3-Hydroxyvibsanin E B D Schwartz
J R Denton P V Bernhardt H M L Davies C M Williams 2847 Structure Investigations of (ent)-Cladospolide D by De Novo Synthesis and
Kinetic and Thermodynamic Isomerization Y Xing J H Penn G A OrsquoDoherty
2855 New Applications of PhI(OAc)2 in Synthesis Total Synthesis and SAR Development of Potent Antitumor Natural Product PsymberinIrciniastatin A N Shao X Huang A Palani R Aslanian A Buevich J Piwinski R Huryk C Seidel-Dugan
2873 Total Synthesis of Largazole ndash Devolution of a Novel Synthetic Strategy B Wang C J Forsyth
2881 Formal Total Synthesis of Palmerolide A J Jaumlgel M E Maier 2893 Total Synthesis of Bongkrekic Acid via Sequential SuzukindashMiyaura Coupling
Reactions M Kanematsu M Shindo M Yoshida K Shishido 2905 Stereodivergent Approach to Both C28a-syn and C28a-anti Relative
Stereochemical Manifolds in the Lepadin Family via a TiCl4-Promoted G Li L J Carlson I K Sagamanova B W Slafer R P Hsung C Gilardi H M Sklenicka N Sydorenko
2915 Enantioselective Aldol Reaction of Tetrasubstituted Ketene Silyl Acetals with Achiral Aldehydes for the Construction of Asymmetric Tertiary Alcohols An Application for the Divergent Total Syntheses of Buergerinins F and G I Shiina T Iizumi Y-s Yamai Y-i Kawakita K Yokoyama Y-k Yamada
2927 Second-Generation Biomimetic Total Synthesis of Chaetominine A Coste G Karthikeyan F Couty G Evano
2935 Total Synthesis of (+)-Fostriecin and (+)-Phoslactomycin B S Shibahara M Fujino Y Tashiro N Okamoto T Esumi K Takahashi J Ishihara S Hatakeyama
2954 Stereochemical Assignments of the Chlorinated Residues in Victorin C A C Durow C Butts C L Willis
2963 Studies of the Asymmetric Total Synthesis of Clavilactone D by the lsquoLariatrsquo Cyclization Strategy T Yoshimitsu S Nojima M Hashimoto K Tsukamoto T Tanaka
2970 Total Synthesis of the Leucetta-Derived Alkaloid Calcaridine A P B Koswatta R Sivappa H V R Dias C J Lovely
2983 Formal Synthesis of Salinosporamide A Starting from D-Glucose T Momose Y Kaiya J-i Hasegawa T Sato N Chida
2992 Synthesis of Bioactive Natural Products by Asymmetric syn- and anti-Aldol Reactions A K Ghosh Z L Dawson
no 18 3003 Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural
Products B M Trost M K Brennan 3026 One-Pot Synthesis of Furo[34-b]pyridin-5(7H)-ones from 2-
Bromopyridine-3-carboxylic Acid and Carbonyl Compounds K Kobayashi T Kozuki H Konishi
3029 Iodocyclization of N-[2-(Methylthio)phenyl]propiolamides Selective Synthesis of 3-Iodo-15-benzothiazepin-4-ones T-S Jiang X-G Zhang J-H Li
3039 A Facile Synthetic Method for Fluorine-Containing 17-Phenanthrolines Pyridine-Ring Formation Reaction of N-Propargyl-68-bis(trifluoroacetyl)-quinolin-5-amine with Various Nucleophiles D Shibata E Okada M Hinoshita M Meacutedebielle
3047 Enantiotopic Discrimination in Palladium-Mediated Nucleophilic Substitutions on Achiral Substrates Chiral Ligand versus Chiral Nucleophile O Jacquet F Charnay J-C Fiaud J Ollivier
3051 Studies on the Chemistry of 2-[3-(2-Nitrophenyl)-2-oxopropyl]benzaldehydes Novel Syntheses of 5H-Benzo[b]carbazole-611-diones and Indolo[12-b]isoquinoline-611-diones M Fernaacutendez
3061 Studies on the C22ndashC23 Aldol Coupling of Spirangien M Lorenz N Bluhm M Kalesse
3067 One-Pot Synthesis of N-Alkyl Purine Pyrimidine and Azole Derivatives from Alcohols using Ph3PCCl4 A Rapid Route to Carboacyclic Nucleoside Synthesis M N Soltani Rad A Khalafi-Nezhad S Behrouz Z Asrari M Behrouz Z Amini
3077 Synthesis of 2-Amino-34-dihydroquinazolines and Imidazo[21-b]quinazoline-2-ones A Mishra S Batra
3089 Studies on the Reaction of Diimines with Thiourea Synthesis and Solvent-Induced cistrans-Isomerization of 135-Triazinane-2-thiones B Kaboudin T Ghasemi T Yokomatsu
3094 Suzuki Coupling of Heteroaromatic Chlorides Using Highly Electron-Donating ClickPhos Ligands S M Spinella Z-H Guan J Chen X Zhang
3099 Reaction of NN-Dioxyenamines with Anhydrides of Carboxylic and Sulfonic Acids A New Method for the Synthesis of a-Hydroxyoxime Derivatives A A Tabolin A V Lesiv S L Ioffe
3106 Directed ortho Metallation Chemistry and Phosphine Synthesis New Ligands for the SuzukindashMiyaura Reaction D B G Williams S J Evans H de Bod M S Mokhadinyana T Hughes
3113 New Functional Derivatives of 9-Phenylquinine P J Boratyński J SkarŜewski
3120 On the Synthesis of Asymmetric and Dissymmetric Amino Analogues of Troumlgerrsquos Base J Artacho K Waumlrnmark
3127 Synthesis of Polycyclic Sultams by Palladium-Catalyzed Intramolecular Cyclization K C Majumdar S Mondal N De
3136 Synthesis of Functionalized L-Cysteine and L-Methionine by Reaction with Electron-Deficient Acetylenes B A Trofimov A G Malrsquokina O A Shemyakina V V Nosyreva A P Borisova S S Khutsishvili L B Krivdin
3143 A lsquoClickrsquo Approach to the Synthesis of 3-[2-(1-Alkyltriazol-4-yl)ethyl]indoles M Petrini R R Shaikh
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
311 A Short Route to the Synthesis of Pyrrolocoumarin and Pyrroloquinolone Derivatives by Sonogashira Cross-Coupling and Gold-Catalyzed Cycloisomerization of Acetylenic Amines K C Majumdar B Chattopadhyay S Samanta
318 Aspects of the Synthesis of an Exceptionally Preorganized Self-Immolative SpacerndashPhenolate Unit M Waibel X-B Zhang J Hasserodt
325 Design and Efficient Synthesis of Amino Acid Derived 2-Substituted Imidazoles by Palladium-Catalyzed Cross-Coupling Reactions A Marek J Kulhaacutenek F Bureš
332 A Convenient Preparation of Di-p-chlorobenzyl Azodicarboxylate (DCAD) for Mitsunobu Couplings B R Taft E C Swift B H Lipshutz
335 Enantioselective Rhodium-Catalyzed Alkylative Desymmetrization of 35-Dimethylglutaric Anhydride M J Cook T Rovis
XIII Forthcoming Articles
No 3 339 Intermolecular Addition Reactions of N-Acyliminium Ions (Part I)
A Yazici S G Pyne 369 Desulfurization of Thioamides into Amides with H2O2ZrCl4 Reagent System
K Bahrami M M Khodaei Y Tirandaz 372 Total Synthesis of (plusmn)-1345-Tetragalloylapiitol R M Patel
N P Argade 375 A Convenient Synthesis of 4-Hydroxy-2-oxo-12-dihydro-18-
naphthyridine-3-carboxamide Derivatives K Kobayashi D Iitsuka S Fukamachi H Konishi
379 Intramolecular Ketalization of Functionalized 7-Norbornenols L A Paquette J D Pettigrew
385 Ring Contraction of 12-Dihydronaphthalenes Promoted by Thallium(III) in Acetonitrile A Diastereoselective Approach to Indanes H M C Ferraz V M T Carneiro L F Silva Jr
389 Regio-Controlled Nucleophilic Attack of 3-Thiaisatoic Anhydride by α-Amino Acids One-Pot Synthesis of 3-(2-Thienyl)imidazolidine-24-dione and 34-Substituted Thieno[23-e][14]diazepine-25-dione Analogues Y Brouillette G Sujol J Martinez V Lisowski
395 The Unprecedented Cobalt-Catalysed Oxidative Glaser Coupling under Reductive Conditions G Hilt C Hengst M Arndt
399 Nucleophilic Addition of 4-Hydroxycoumarin to BaylisndashHillman Acetate Adducts C Raji Reddy N Kiranmai K Johny M Pendke P Naresh
403 Palladium-Mediated Heck Reaction to the Synthesis of 3-Substituted Indoles and Indolones K C Majumdar S Chakravorty P K Shyam A Taher
409 Synthesis of Bicyclo[310]hexan-2-ones by Manganese(III) Oxidation in Ethanol K Asahi H Nishino
424 High Regio- and Stereoselective Synthesis of (Z)- or (E)-N-Acryl Butenedioic Monoimide Derivatives by a Multicomponent Reaction F Sha Y Lin X Huang
431 The First Synthesis of Allyl Isonitriles from BaylisndashHillman Adducts and Their Application in the Synthesis of Substituted Imidazo[12-α]pyridines and Tetraazadibenzoazulenes M Nayak S Kanojiya S Batra
438 One-Pot Three-Step Synthesis of Pyrazinothienopyrimidines Using Tandem Aza-WittigElectrocyclic Ring Closure G Blanco A Fernaacutendez-Mato J M Quintela C Peinador
445 Synthesis of Biaryls Fluorenones Cyclopenta[def]phenanthren-4-ones and Benzophenones Based on Formal [3+3] Cyclocondensations of 13-Bis(silyloxy)buta-13-dienes with 3-(Silyloxy)-2-en-1-ones S Reim M Lau M Adeel I Hussain M A Yawer A Riahi Z Ahmed C Fischer H Reinke P Langer
464 Diastereoselective Synthesis of α-Stabilized Phosphorus Ylides via a Four-Component Reaction A Alizadeh N Zohreh L-G Zhu
469 Stereoselective Synthesis of Alkynyl Vinyl Chalcogenides via HornerndashWittig Reaction C C Silveira F Rinaldi R C Guadagnin A L Braga
474 Stereoselective Preparation of C1ndashC10 and C11ndashO14 Fragments of Narbonolide Exploiting the Versatility of Thiazolidinethione Chiral Auxiliary C P Narasimhulu P Das
483 Efficient Catalytic Activity of CopperAluminum Hydrotalcite in Diaryl Ether Synthesis B Sreedhar R Arundhathi M A Reddy M L Kanatm
488 On-Resin Click-Glycoconjugation of Peptoids A S Norgren C Budke Z Majer C Heggemann T Koop N Sewald
495 A Simple and Efficient Preparation of Novel Formaldehyde Derivatives R Hartung G Golz S Schlaf G Silvennoinen K Polborn P Mayer H R Pfaendler
502 2-Oxazol-5-ylethanones by Consecutive Three-Component AmidationndashCouplingndashCycloisomerization (ACCI) Sequence E Merkul O Grotkopp T J J Muumlller
508 SuzukindashMiyaura Cross-Couplings Mediated by trans-PdBr(N-Succ)(PPh3)2 A Convenient Synthetic Method for Diarylmethanes and Aryl(heteroaryl)-methanes I J S Fairlamb P Sehnal R J K Taylor
511 Modern Reduction Methods Edited by P G Andersson and I J Munslow Reviewed by Siegfried R Waldvogel
512 Addendum and Erratum XIII Forthcoming Articles
No 4 513 Intermolecular Addition Reactions of N-Acyliminium Ions (Part II)
A Yazici S G Pyne 542 A Simple Practical Method for the Synthesis of 46-Dimethoxy-135-
triazin-2(1H)-one Using Dimethylamine-Functionalized Solid-Phase Reagents K Hioki K Ohshima Y Sota M Tanaka M Kunishima
545 Conjugation-Amenable Tetrasaccharide of the Side Chain of the Major Glycoprotein of the Bacillus anthracis Exosporium A Large-Scale Preparation S Hou P Kovaacuteč
551 Reductive Amination ndash A Convenient Method for Generating Diverse Mono-Functionalised 5101520-Tetraphenyl Porphyrins C Welch S J Archibald R W Boyle
557 Highly Regioselective Preparation of 13-Dioxolane-4-methanol Derivatives from Glycerol Using Phosphomolybdic Acid N W Fadnavis R Gowrisankar G Ramakrishna M K Mishra G Sheelu
561 Rapid Synthesis of 3-Aminoisoquinoline-5-sulfonamides Using the BuchwaldndashHartwig Reaction N Proisy S Taylor A Nelson I Collins
567 Synthesis of Divalent 22-Linked Mannose Derivatives by Homodimerization F S Ekholm M Polaacutekovaacute A J Pawłowicz R Leino
577 Efficient Synthesis of Substituted Cyclic α-Aminophosphonates I L Odinets O I Artyushin N Shevchenko P V Petrovskii V G Nenajdenko G-V Roumlschenthaler
583 Methylated Imidazolinium-Dithiocarboxylates Two Representatives of a New Class of Ionic Liquids A Blanrue R Wilhelm
587 An Efficient Route to 1-Vinylpyrrole-2-carbaldehydes A I Mikhaleva A V Ivanov E V Skitalrsquotseva I A Ushakov A M Vasilrsquotsov B A Trofimov
591 A Regioselective Route to 5-Substituted Isoxazole- and Isoxazoline-3-phosphonates P Conti A Pinto L Tamborini P Dunkel V Gambaro G L Visconti C De Micheli
597 Solvent-Free One-Pot Conjugate Addition of Benzyl Bromides to β-Nitroalkenes Mediated by Magnesium Powder W Shi J-X Wang
602 Synthesis of 234-Trideoxy-44-difluoro-D-ribo-hexopyranose Adenosines J Xu X Zhang X-L Qiu F-L Qing
609 Synthesis of anti-27-Disubstituted Norbornadienes G C Tsui P Le Marquand A Allen W Tam
620 Novel Peptide Mimetic Inhibitors of Hepatitis C Serine Protease Derived from Isomannide T G Barros S Pinheiro J S Williamson A Tanuri H S Pereira R M Brindeiro J B A Neto O A C Antunes E M F Muri
627 A Practical Synthesis of α-Substituted tert-Butyl Acrylates from Meldrumrsquos Acid and Aldehydes C G Frost S D Penrose R Gleave
636 A New Class of Troumlgerrsquos Base Analogues Bearing Spiro[45] Lactone Straps A B Mahon D C Craig A C Try
643 A New Approach to Di- and Tetrasubstituted 23-Dihydropyridin-4(1H)-ones through Aza-DielsndashAlder Reaction Promoted by Silicon Tetrachloride A Massa V de Sio R Villano M R Acocella L Palombi G Sellitto A Peduto R Filosa P De Capraris A Scettri
650 Palladium-Catalysed Direct Arylation of Sydnones A Rodriguez W J Moran
655 Synthesis of (ndash)-Monomorine I R W Bates P Song 660 Cobalt(II) Chloride HexahydratendashDiisopropylamine Catalyzed Mild and
Chemoselective Reduction of Carboxylic Esters with Sodium Borohydride A R Jagdale A S Paraskar A Sudalai
665 Synthesis of Bi- and Tricyclic αβ-Unsaturated Lactams as Potential Michael Acceptors Starting from Heterocyclic Imines K Schulz M Watzke K Johannes P Ullrich J Martens
674 An Expedient Synthesis of Bis-Fused Benzofuran and a Two-Directional Ring-Closing Metathesis for the Synthesis of Bisbenzoxepines and Bisbenzoxocines K C Majumdar B Chattopadhyay S Chakravorty
681 Palladium-Catalyzed Cross-Couplings of Unsaturated Halides Bearing Relatively Acidic Hydrogen Atoms with Organozinc Reagents Z Dong G Manolikakes J Li P Knochel
687 Synthesis of Enantioenriched aa-Disubstituted Cyclopentenes Catalyzed by N-Heterocyclic Carbenes E M Phillips M Wadamoto K A Scheidt
XVII Forthcoming Articles
No 5 691 Transannulation Reactions in the Synthesis of Natural Products
P A Clarke A T Reeder J Winn 710 Synthesis of DL-erythro-Sphingosine Using a Tethered
Aminohydroxylation Reaction as the Key Step J A Morales-Serna Y Diacuteaz M I Matheu S Castilloacuten
713 Convenient Multigram Synthesis of 4-Chloropyridine-26-dicarbonyl Dichloride K Mitsui J R Parquette
715 A Novel and Efficient Synthesis of Dihydrexidine J P Cueva D E Nichols
721 Synthesis of 57-Dichloro-6-azaindoles and Functionalization via a Highly Selective LithiumndashChlorine Exchange N Lachance L-P Bonhomme-Beaulieu P Joly
731 A Convenient Synthesis of Fluorinated Pyrazolo[34-b]pyridine and Pyrazolo[34-d]pyrimidine Nucleosides V O Iaroshenko D V Sevenard A Kotljarov D M Volochnyuk A O Tolmachev V Y Sosnovskikh
741 Diastereoselective Synthesis of γ-Amino Acids and Their Derivatives from Nitroethane via Intermediacy of 56-Dihydro-4H-12-oxazines Bearing the CH2CH(CO2Me)2 Substituent at C3 A Y Sukhorukov A V Lesiv Y A Khomutova S L Ioffe
755 Synthesis of a New Pyrrolopyridoindole and Its Pyrrolopyridobenzimidazole Regioisomer F Bouchikhi M Sassatelli F Anizon M Prudhomme P Moreau
759 Practical Syntheses of Sphingosine-1-Phosphate and Analogues V Blot U Jacquemard H-U Reissig B Kleuser
767 A Facile Synthetic Route towards Substituted Thieno[32-e]indoles W Van Snick W Nulens S Jambon W Dehaen
775 Microwave-Assisted One-Pot Synthesis of (Aminoalkyl)naphthols and (Aminoalkyl)quinolinols by Using Ammonium Carbamate or Ammonium Hydrogen Carbonate as Solid Ammonia Source I Szatmaacuteri F Fuumlloumlp
779 Enantioselective Synthesis of Flavan-3-ols Using a Mitsunobu Cyclization K Krohn I Ahmed M John 787 Synthesis of a Novel γ-Folic AcidndashNτ-Histidine Conjugate Suitable for
Labeling with 99mTc and 188Re C Sparr U Michel R E Marti C Muumlller R Schibli R Moser V Groehn
793 Palladium-Catalyzed Intramolecular Biaryl Coupling A Highly Efficient Avenue for Benzannulated Pyranoquinolines and Julolidine Derivatives K C Majumdar A Taher P Debnath
801 Preparation of NN-Dimethyl-N-Arylureas Using SS-Dimethyl Dithiocarbonate as a Carbonylating Reagent I Degani R Fochi C Magistris M Migliaccio
809 Versatile Selective α-Carboxylic Acid Esterification of N-Protected Amino Acids and Peptides by Alcalase T Nuijens C Cusan J A W Kruijtzer D T S Rijkers R M J Liskamp P J L M Quaedflieg
815 Efficient Palladium-Catalyzed Amination of Aryl Chlorides Using Dicyclohexylamino[(26-dimethyl)morpholino]phenylphosphine as a PN2 Ligand S-E Park S B Kang K-J Jung J-E Won S-G Lee Y-J Yoon
824 A Clean Facile and Stereospecific Synthesis of α-Oxoketene OS-Acetals in Water Y Li Q Zhang X Cheng Q Liu X Xu
829 Sonogashira Cross-Coupling Reactions and Construction of the Indole Ring System Using a Robust Silica-Supported Palladium Catalyst E Tyrrell L Whiteman N Williams
836 Synthesis of Angular 78-Pyridazinocoumarins via the Transformation of a Hydroxy Group into a Carbonyl Group A Kotali I S Lafazanis P A Harris
841 Synthesis of New Cyclic and Acyclic 5-Halouridine Derivatives as Potential Antiviral Agents M F Elshehry J Balzarini C Meier
848 Dendritic Triphenylmethylium and Tetraphenylmethane Compounds H Meier S Kim A Oehlhof
853 Synthesis of Homoallylic Alcohols via Lewis Acid Assisted Enantioselective Desymmetrization B Yu F Menad N Isono M Lautens
860 Diastereoselective Synthesis of 123-Trisubstituted Indanes via Rhodium(I)-Catalyzed Tandem Conjugate Additions C Navarro A G Csaacutekyuml
864 Bakerrsquos Yeast for Sweet Dough Enables Large-Scale Synthesis of Enantiomerically Pure Bicyclo[331]nonane-26-dione C J Wallentin E Orentas E Butkus K Waumlrnmark
868 Addendum and Erratum XV Forthcoming Articles
No 6 869 Stereoselective Transformations of meso Bicyclic Hydrazines Versatile
Access to Functionalized Aminocyclopentanes C Bournaud F Chung A P Luna M Pasco G Errasti T Lecourt L Micouin
888 Synthesis of Glycoaminoxy Acids as Novel Sugar Building Blocks A Malapelle R Ramozzi J Xie
891 Electrophilic ipso-Halocyclization of N-Arylpropynamides with Polyfluoroalkyl Alcohols Selective Synthesis of 8-(Polyfluoroalkoxy) azaspiro[45]trienes Z-Q Wang B-X Tang H-P Zhang F Wang J-H Li
903 Electrooxidation of Alcohols in N-Oxyl-Immobilized Silica GelWater Disperse System Approach to Totally Closed System M Kuroboshi K Goto H Tanaka
909 Synthetic Routes to Aminotriamantanes Topological Analogues of the Neuroprotector Memantinereg A A Fokin A Merz N A Fokina H Schwertfeger S L Liu J E P Dahl R K M Carlson P R Schreiner
913 Parallel Synthesis of Drug-like 5-Amino-Substituted 124-Thiadiazole Libraries Using Cyclization Reactions of a Carboxamidine Dithiocarbamate Linker J Y Park I A Ryu J H Park D C Ha Y-D Gong
921 Copper-Catalyzed Selective S-Arylation of 12-Bis(o-amino-1H-pyrazolyl) Disulfides with Arylboronic Acids P-S Luo F Wang J-H Li R-Y Tang P Zhong
929 2-Iodoxybenzoic AcidTetraethylammonium BromideWater An Efficient Combination for Oxidative Cleavage of Acetals C Kuhakarn W Panchan S Chiampanichayakul N Samakkanad M Pohmakotr V Reutrakul T Jaipetch
935 Synthesis of Quinonoid Analogues of Diospyrin S Sagar I R Green 941 A One-Pot Method for the Iodination of Aryl Amines via Stable Aryl
Diazonium Silica Sulfates Under Solvent-Free Conditions A Zaroi A R Hajipour L Khazdooz
945 Poly(NN-dichloro-N-ethylbenzene-13-disulfonamide) and NNNN-Tetrachlorobenzene-13-disulfonamide as Novel Reagents for the Synthesis of N-Chloroamines Nitriles and Aldehydes R Ghorbani-Vaghei H Veisi
951 Synthesis of an (R)-Garner-type Aldehyde from L-Serine Useful Building Block for a (+)-Furanomycin Derivative G Bartoli G Di Antonio R Fiocchi S Giuli E Marcantoni M Marcolini
957 An Efficient and Highly Selective Synthesis of (Z)-Fluoroenol Phosphates from Hydroxy Difluorophosphonates P Beier R Pohl A V Alexandrova
963 Iodine-Catalyzed Three-Component Reaction A Rapid Synthesis of α-Alkoxy Azides and Homoallyl Ethers J S Yadav B V S Reddy G M Reddy R Narender
969 Rhodium(I)-Catalyzed Cycloisomerization of 13-Dienes with Alkenes in a Tether Y Oonishi A Saito M Mori Y Sato
980 Synthesis of New Optically Active D-GlucosaminendashPyrrole Derivatives B A Frontana-Uribe M V Escaacutercega-Bobadilla J Juaacuterez-Lagunas R A Toscano G A Garciacutea de la Mora M Salmoacuten
985 Partially Saturated Indeno[12-b]indole Derivatives via Deoxygenation of Heterocyclic α-Hydroxy-NO-hemiaminals H-J Hemmerling G Reiss
1000 Light-Induced Synthesis of Π-Extended Tetrathiafulvalenes Incorporating Ferrocenes An Efficient Route for the Synthesis of Electron-Donor Materials A A O Sarhan C Bolm
1007 Preparation of Nβ-Fmoc-Protected Aza-β3-Amino Acids with Nonproteinogenic Hydrophobic Side Chains for Solid-Phase Syntheses of Pseudopeptides M Laurencin P Bauchat M Baudy-Flocrsquoh
1014 Diastereomeric (η4-diene)Fe(CO)3 Complexes Containing Chiral Amide Groups A Convenient Method for the Resolution of Amino Acids M Schumacher G Coste L Miesch
1021 Palladium-Catalysed Heck Reactions of Alk-1-en-3-ones with Aryl Bromides A Very Simple Access to (E)-1-Arylalk-1-en-3-ones M Lemhadri Y Fall H Doucet M Santelli
1036 An Improved Process for the Synthesis of 4H-Imidazo[15-α][14]benzodiazepines J Yang Y Teng S Ara S Rallapalli J M Cook
1041 Meta- and Para-Difunctionalization of Arenes via an Ortho-Magnesiation and a Subsequent SulfoxidendashMagnesium Exchange L Melzig C B Rauhut P Knochel
XIII Forthcoming Articles
No 7 1049 Catalytic Transformations of Benzylic Carboxylates and Carbonates
R Kuwano 1062 A Simple and Practical Method for the Oxidation of Thebaine to 14-
Hydroxycodeinone by V2O5ndashH2O2 S Das Sharma D Konwar 1065 Umpolung with Sulfur Dioxide CarbonndashCarbon Cross-Coupling of Electron-
Rich 13-Dienes and Alkenes Application to the Enantioselective Synthesis of Long-Chain Polyketide Fragments M Turks C J Exner C Hamel P Vogel
1075 One-Pot Synthesis of 14-Diarylnaphthalenes via a WittigndashHorner Reaction[4+2] CycloadditionDehydrogenation Sequence Z Chen W Shou Y Wang
1081 A Novel and General Method for the Formation of S-Aryl Se-Aryl and Te-Aryl Phosphorochalcogenoates Y-X Gao G Tang Y Cao Y-F Zhao
1087 A Remarkable Access to γ-Fluoroalkylated Propargylamine Derivatives or Fluoroalkylated Dihydroisoxazoles via the Reaction of Fluoroalkylated Acetylides with Various Nitrones T Konno K Moriyasu T Ishihara
1095 Short and Practical Syntheses of (S)-(+)-3-(p-Tolylsulfinyl)furan-2(5H)-one and (S)-(+)-3-(p-Tolylsulfinyl)-56-dihydropyran-2-one D Cruz Cruz A Hernaacutendez Linares F Yuste M R Martiacuten J L Garciacutea Ruano
1099 Decarboxylative Aldol-Type Reaction of 2-(Trifluoroacetyl)-13-diazoles with Activated Acetic Acids P V Khodakovskiy D M Volochnyuk A A Tolmachev
1105 Synthesis of 2-[(Arylmethylene)amino]cyclopropanecarbonitriles via a Two-Step Ring Transformation of 2-(Cyanomethyl)aziridines S Mangelinckx M Drsquohooghe S Peeters N De Kimpe
1113 Synthesis of Dendrimeric Tumor-Associated Mucin-Type Glycopeptide Antigens T Becker A Kaiser H Kunz
1123 A Simple and Efficient Oxidation Procedure for the Synthesis of Acid-Sensitive Epoxides O Bortolini G Fantin M Fogagnolo
1127 Rapid Chemoselective Deprotection of Benzyl Esters by Nickel Boride J M Khurana R Arora
1131 Three-Component Coupling of Isoquinoline Activated Alkyne and Nitromethane A Facile Synthesis of Nitromethyl Derivatives of 12-Dihydroisoquinolines J S Yadav B V S Reddy N N Yadav M K Gupta
1137 Palladium Supported on a Polyionic Resin as an Efficient Ligand-Free and Recyclable Catalyst for Heck SuzukindashMiyaura and Sonogashira Reactions B Basu S Das P Das B Mandal D Banerjee F Almqvist
1147 Oxidation of 25-Dialkylpyrrole Derivatives with Cerium(IV) Ammonium Nitrate R Voloshchuk M Gałęzowski D T Gryko
1153 Practical Syntheses of Enantiomerically Pure Key Intermediates of Opioid Receptor-like 1 (ORL1) Antagonists T Yoshizumi A Ohno T Tsujita H Takahashi O Okamoto I Hayakawa H Kigoshi
1163 An Environmentally Benign TEMPO-Catalyzed Efficient Alcohol Oxidation System with a Recyclable Hypervalent Iodine(III) Reagent and Its Facile Preparation X-Q Li C Zhang
1170 Efficient and Stereoselective Rearrangement of BaylisndashHillman Acetates Catalyzed by Gold(I) ChlorideSilver(I) Trifluoromethanesulfonate Y Liu D Mao J Qian S Lou Z Xu Y Zhang
1175 The First Total Synthesis of Kynapcin-24 by Palladium Catalysis L-Y Yang C-F Chang Y-C Huang Y-J Lee C-C Hu T-H Tseng
1180 Enantioselective Synthesis of N-Protected α-Amino Acid Hydrazides M Bibian S El-Habnouni J Martinez J-A Fehrentz
1185 Synthesis of 11H-Indolo[32-c]quinoline-6-carboxylic Acids by Cascade AutoxidationndashRing Contractions A Becker S Kohfeld T Pies K Wieking L Preu C Kunick
1190 Reaction of N-Nonaflylbenzotriazole with Silyl Enol Ethers M Uhde T Ziegler
1195 2-(Benzoylimino)thiazolidin-4-ones Formation by an Alternative Ring Closure and Analysis of Rotational Barriers H-G Haumlcker P W Elsinghorst S Michels J Daniels G Schnakenburg M Guumltschow
1204 Microwave-Assisted Synthesis and Functionalization of Selenolopyrimidines S Hesse C Chenet D Thomae G Kirsch
1209 12-Disubstituted 4-Quinolones via Copper-Catalyzed Cyclization of 1-(2-Halophenyl)-2-en-3-amin-1-ones R Bernini S Cacchi G Fabrizi A Sferrazza
1220 A New Atom-Economical and Selective Synthesis of Secondary and Tertiary Alkylamines by Means of CpIridium Complex Catalyzed Multiple N-Alkylation of Ammonium Salts with Alcohols without Solvent R Yamaguchi Z Mingwen S Kawagoe C Asai K-i Fujita
1224 Synthesis of Regioisomerically Pure 5-Functionalized 27-Dichlorofluoresceins J C Castro A Malakhov K Burgess
XIII Forthcoming Articles
No 8 1227 Michael Additions to Activated Vinylphosphonates T Janecki J Kędzia
T Wąsek 1255 A Facile and General Synthesis of 2β-Aminosteroids X Ke H Hu
D Zhou W Xu Q Zhu N P Reddy X Hu 1261 Efficacious Preparation of Oppolzerrsquos Glycylsultam via the Deleacutepine
Reaction A Isleyen C Gonsky R C Ronald P Garner 1265 Synthesis of Masked Vicinal Amino Aldehydes of Pyrrolizine and Pyrrolo
[12-c]thiazole Series A V Tverdokhlebov A V Denisenko A A Tolmachev Y M Volovenko S V Shishkina O V Shishkin
1271 Preparation of 9-Substituted Pyridine-Stretched Adenines and Hypoxanthines J A Crawford W Fraser C A Ramsden
1279 A Versatile Synthesis of Heterocyclic Analogues of Neoflavonoids from Enamino Ketones V S Moskvina V P Khilya O V Turov U M Groth
1287 New Stereoselective Synthesis of Paeonilactone B F G Gatti S Serra 1291 The Use of NN-Dialkyltrimethylsilylamines in the Synthesis of
Pentamethinium Salts M Kořiacutenek M Rybaacutečkovaacute Boumlhm 1297 Synthesis of Triazoles via Regioselective Reactions of Aryl Azides with
Cyanoacetyl Pyrroles and Indoles N T Pokhodylo V S Matiychuk M D Obushak
1301 Gallium(III) Chloride Catalyzed Hydroarylation of Arylacetylenes with Naphthols and Phenols A Facile Synthesis of Vinylarenes J S Yadav B V S Reddy S Sengupta S K Biswas
1305 Electrophilic Bromination of meta-Substituted Anilines with N-Bromosuccinimide Regioselectivity and Solvent Effect S Bartoli A Cipollone A Squarcia A Madami D Fattori
1309 Cross-Coupling Reactions of Halopurines with Aryl- and Alkyltrifluoroborates The Scope and Limitations in the Synthesis of Modified Purines Z Hasniacutek R Pohl M Hocek
1318 A Convenient Method for Converting Hydroxyacetophenones into Their Ethylene or Trimethylene Acetals F Ono H Takenaka T Fujikawa M Mori T Sato
1323 γ-Chloromagnesio γ-Lactones and δ-Chloromagnesio δ-Lactones Generation Properties and Synthetic Uses H Shimizu S Fukuda S Sugiyama T Satoh
1336 Click Reactions with Nitroxides T Kaacutelai W L Hubbell K Hideg 1341 Synthesis of Novel 14-Benzoquinone-Containing 123-Triazoles An Entry
Into a New Library F Algi M Balci 1348 Efficient Synthesis of Two Sialylated Tetrasaccharides Found in Goat Milk
P K Mandal A K Misra 1355 Dendrimers of Vaccines Consisting of Tumor-Associated Glycopeptide
Antigens and T Cell Epitope Peptides S Keil A Kaiser F Syed H Kunz
1370 IBXTBAB-Mediated Oxidation of Primary Amines to Nitriles F Drouet P Fontaine G Masson J Zhu
1375 Chemoselectivity of Multicomponent Condensations of Barbituric Acids 5-Aminopyrazoles and Aldehydes E A Muravyova S V Shishkina V I Musatov I V Knyazeva O V Shishkin S M Desenko V A Chebanov
1386 Stereoselective Total Syntheses of Leiocarpin A and (ndash)-Galantinic Acid Starting from D-Mannitol K Nagaiah D Sreenu K V Purnima R S Rao J S Yadav
1393 A Facile Mild Deprotection Protocol for 13-Dithianes and 13-Dithiolanes with 30 Hydrogen Peroxide and Iodine Catalyst in Aqueous Micellar System N C Ganguly S K Barik
1400 Rhodium-Catalyzed Gram-Scale Synthesis of Highly Substituted Pyridine Derivatives K Parthasarathy C-H Cheng
1403 Enantioselective Synthesis of (R)-Propylene Carbonate from Ethyl (S)-Lactate J M Whitaker R C Ronald
XIII Forthcoming Articles
no 9 1405 Transition-Metal-Catalyzed Site-Selective Cross-Coupling of Di- and
Polyhalogenated Compounds J-R Wang K Manabe 1428 An Improved Synthesis of (4-4-Hydroxy-3-isopropyl-5-[(4-nitrophenyl)
ethynyl]benzyl-35-dimethylphenoxy)acetic Acid (NH-3) M B Gopinathan K S Rehder
1431 Copper-Catalyzed Tandem CndashN Bond Formation Reaction Selective Synthesis of 2-(Trifluoromethyl)benzimidazoles M-W Chen X-G Zhang P Zhong M-L Hu
1437 Synthesis and Thermochemical Properties of Stereoisomeric Dihydroxy- and Tetrahydroxyalkylammonium Salts M Thomas L Rothman J Hatcher P Agarkar R Ramkirath S Lall-Ramnarine R Engel
1445 Preparation of 5-Substituted 2-(2-Alkylaryl-1H-imidazol-4-yl)oxazoles and 5-Substituted 2-(2-Alkylarylthiazol-4-yl)oxazoles by Utilizing 5-Substituted 2-(2-Bromo-11-diethoxyethyl)oxazole as a Synthon D R St Laurent J L Romine
1459 Novel and Efficient Methods for the Synthesis of Symmetrical Trisulfides A Kertmen S Lach J Rachon D Witt
1463 An Environmentally Benign Electrochemical Process for the Reduction of Carboxylic Acid Hydrazides to Amides M Mentel M J Beier R Breinbauer
1469 Synthesis of 1-Chloroalkynes from Alkynylsilanes Using Trichloroisocyanuric Acid as Chlorinating Agent M H Vilhelmsen A S Andersson M B Nielsen
1473 A Convenient Approach to Enantioenriched Cyclopropanes Bearing Electron-Withdrawing Functionalities H Krawczyń K Wąsek J Kędzia
1477 Synthesis of Cyclopropenes via 12-Elimination of Bromocyclopropanes Catalyzed by Crown Ether W M Sherrill R Kim M Rubin
1485 A Base-Catalysed One-Pot Three-Component Coupling Reaction Leading to Nitrosubstituted Pyrroles I R Baxendale C D Buckle S V Ley L Tamborini
1494 Synthesis of 4-Alkylidene-4H-31-benzoxazine Derivatives by Acid-Catalyzed Cyclization of 2-Isocyanophenyl Ketones in the Presence of a Vinyl Ether K Kobayashi Y Okamura H Konishi
1499 Synthesis of Higher Helicenes via Olefin Metathesis and CndashH Activation J Cocircteacute S K Collins
1506 Azido- and Ethynyl-Substituted 2262-Terpyridines as Suitable Substrates for Click Reactions A Winter A Wild R Hoogenboom M W M Fijten M D Hager R-A Fallahpour U S Schubert
1513 Synthesis of 2-(Arylamino)ethanethiols via Lewis Acid Catalyzed Aminolysis of 22-Dimethylthiirane as Precursors of the 14-Benzothiazine Nucleus R Spogli S Sabatini G Manfroni O Tabarrini V Cecchetti
1520 Iron(III) Chloride A Versatile Catalyst for the Practical Synthesis of 3-Sulfenylindoles J S Yadav B V S Reddy Y J Reddy K Praneeth
1525 Organocatalytic Enantioselective Conjugate Addition of 2-Fluoromalonate to Nitroolefins Direct Synthesis of Chiral Fluorinated γ-Nitro Carboxylic Acid Derivatives H Li L Zu H Xie W Wang
1531 Asymmetric Transfer Hydrogenation of Ketimines with Trichlorosilane Structural Studies Z Zhang P Rooshenas H Hausmann P R Schreiner
1545 Prolinol Sulfinyl Ester Derivatives Organocatalytic Michael Addition of Ketones to Nitroolefins under Neat Conditions X Zeng G Zhong
1551 Asymmetric Oxidations of Electron-Poor Alkenes Promoted by the β-Amino AlcoholTBHP System A Russo A Lattanzi
1557 Enantioselectivity Switch in Direct Asymmetric Aminoxylation Catalyzed by Binaphthyl-Based Chiral Secondary Amines T Kano A Yamamoto F Shirozu K Maruoka
1564 Enantioselective Conjugate Addition of N-Heterocycles to αβ-Unsaturated Ketones Catalyzed by Chiral Primary Amines G Luo S Zhang W Duan W Wang
1573 Sulfonyl Hydrazine as New Functionality in Organocatalysis Camphorsulfonyl Hydrazine Catalyzed Enantioselective Aza-Michael Addition L-Y Chen H He B-J Pei W-H Chan A W M Lee
1578 Conversion of Primary Alcohols and Aldehydes into Methyl Esters by Ruthenium-Catalysed Hydrogen Transfer Reactions N A Owston T D Nixon A J Parker M K Whittlesey J M J Williams
1582 Addendum and Erratum XVII Forthcoming Articles
no 10 1583 Organocatalytic Formation of Quaternary Stereocenters M Bella
T Gasperi 1615 Regioselective Synthesis of 5H-Thiazolo[32-a]pyrimidin-5-ones from
MoritandashBaylisndashHillman Adduct Acetates under Solvent-Free and Base-Free Conditions W Zhong B Guo F Lin Y Liu W Su
1623 First Synthesis of 5-Cyanosalicylates by Formal [3+3] Cyclocondensations of 13-Bis(silyloxy)-13-butadienes A Riahi O Fatunsin M Shkoor R Dede H Reinke C Fischer P Langer
1635 Reaction of Isocyanides Dialkyl Acetylenedicarboxylates and a-Keto Lactones Unexpected Participation of an Ester Carbonyl Group in the Isocyanide-Based Three-Component Reaction A A Esmaeili H Vesalipoor
1639 An Efficient and Chemoselective Synthesis of 16-Naphthyridines and Pyrano[32-c]pyridines under Microwave Irradiation Z-G Han S-J Tu B Jiang S Yan X-H Zhang S-S Wu W-J Hao X-D Cao F Shi G Zhang N Ma
1647 N-Activation of N-Arylimidazoles Facile Syntheses of N-Alkyl-N-arylimidazolium Iodides from Less Expensive Chloro Substrates A M Oertel V Ritleng M J Chetcuti
1651 Synthesis of Polyhalogenated 2-(Phenylamino)pyridines by Thermal Amination Reactions S R Waldvogel A Faust W Barkmann R Froumlhlich O Wolff
1655 Cyanide Ion Promoted Addition of Acylphosphonates to Diethyl Cyanophosphonate Synthesis of Phosphonocyanohydrin O-Phosphates A S Demir A Aybey M Emrullahoglu
1659 Straightforward and Scalable Synthesis of Orthogonally Protected 37-Diazabicyclo[410]heptane H Schramm M Pavlova C Hoenke J Christoffers
1663 Hypervalent Iodine Mediated Oxidation of 12-Diaminobenzimidazole and Its Schiff Bases Efficient Synthesis of 3-Amino-124-benzotriazine and 2-Aryl-124-triazolo[15-a]benzimidazoles A Kumar M Parshad R K Gupta D Kumar
1667 Synthesis of the Reported Protoberberine Gusanlung D P B Wakchaure S Easwar N P Argade
1673 2-(Azidomethyl)arylboronic Acids in the Synthesis of Coumarin-Type Compounds M I Naumov A V Nuchev N S Sitnikov Y B Malysheva A S Shavyrin I P Beletskaya A E Gavryushin S Combes A Y Fedorov
1683 Asymmetric Synthesis of 12-anti-Disubstituted Taurine Derivatives D Enders D Iffland G Raabe
1689 A Novel One-Pot Three-Component Synthesis of 5-Imino-2358-tetrahydropyrazolo[12-a]pyridazin-1-one Derivatives B Qian M-J Fan Y-X Xie L-Y Wu Y Shi Y-M Liang
1694 One-Portion Synthesis of 2-Acetoxy Carbonyl Compounds from Aldehydes by Using an Acetylated Masked Acyl Cyanide H Nemoto T Kawamura K Kitasaki K Yatsuzuka M Kamiya Y Yoshioka
1703 Synthesis of 9-Anthryl Ethers from trans-910-Dihydro-910-dimethoxyanthracene by Acid-Catalyzed Transetherification K S Jang H Y Shin D Y Chi
1708 Efficient Synthesis of Azo Dye Labeled Terpenes Sugars and Steroids Using N-(4-Arylazobenzoyl)-1H-benzotriazoles A R Katritzky S R Tala N E Abo-Dya Z K Abdel-Samii
1715 Tandem CH-ActivationndashImine-Formation Reaction A New Route to Imidazo[21-a]phthalazines A Heim-Riether K R Gipson
1720 A Convenient and Efficient α-Sulfenylation of Carbonyl Compounds E Okragla S Demkowicz J Rachon D Witt
1725 Stereoselective Synthesis of β-Branched Phenylalanine Derivatives via Chelate-Claisen Rearrangement C Quirin U Kazmaier
1732 Catalyst-Free and Base-Free Water-Promoted SNAr Reaction of Heteroaryl Halides with Thiols B Sreedhar P S Reddy M A Reddy
1739 Convenient Methods for Synthesis of C2-Symmetric Diphenyltetrahydrothiophenes M Periasamy G Ramani G P Muthukumaragopal
1744 Highly Diastereoselective Conjugate AdditionndashElimination of Chiral Nickel(II) Glycinate with Activated Allylic Acetates for Asymmetric Synthesis of Glutamic Acid Derivatives J Wang J Shi X Zhang D Lin H Jiang H Liu
1753 Synthesis of 36-Dimethoxybenzene-12-diamine and of 47-Dimethoxy-2-methyl-1H-benzimidazole T Besset C Morin
1757 An Inexpensive Procedure for Reductive Aminations Using Dimethylamineborane on Millimolar and Molar Scale R Ortmann M Schlitzer
1760 Classics in Stereoselective Synthesis Edited by E M Carreira L Kvaerno Reviewed by Rolf Breinbauer
XV Forthcoming Articles
no 11 1761 Transition-Metal-Catalyzed Enantioselective Synthesis of Compounds with
Non-Centrochirality M Ogasawara S Watanabe 1786 One-Pot Synthesis of 3-Acyl-2-(alkylsulfanyl)indoles and 2-(Alkylsulfanyl)-
indole-3-carboxylates from (2-Isocyanophenyl)methyl Ketones or (2-Isocyanophenyl)acetates S Fukamachi H Konishi K Kobayashi
1791 Efficient and Recyclable Phthalocyanine-Based Sensitizers for Photooxygenation Reactions H Xu W-K Chan D K P Ng
1797 A Facile and Practical One-Pot Synthesis of β-Oxo Thioamides from β-Oxo Amides and Isothiocyanates P Huang D Xiang Y Zhou Y Liang T Na D Dong
1801 Microwave-Promoted Solid-Acid-Catalyzed One-Pot Synthesis of Phthalazinones V M Outerbridge S M Landge H Tamaki B Toumlroumlk
1807 Benzylic Brominations with N-Bromosuccinimide in (Trifluoromethyl)-benzene D Suarez G Laval S-M Tu D Jiang C L Robinson R Scott B T Golding
1811 Synthesis of Thioflavanone and Flavanone Derivatives by Cyclization of Chalcones W Konieczny M Konieczny
1815 A New and Expedient Total Synthesis of Ochratoxin A and d5-Ochratoxin A B Gabriele M Attya A Fazio L Di Donna P Plastina G Sindona
1821 Synthesis of Benzopyrrolizidinones by NorrishndashYang Cyclization of 3-(Acylmethyl)-2-alkylisoindol-1-ones J Wu W Zhang C Wang
1829 Reactions of MoritandashBaylisndashHillman Acetates with Huisgen Zwitterions A Novel Strategy for the Synthesis of β-Amino Acid Derivatives A Jose R R Paul R Mohan S C Mathew A T Biju E Suresh V Nair
1834 Peracetylated β-Allyl C-Glycosides of D-Ribofuranose and 2-Deoxy- D-ribofuranose in the Chemical Literature Until Now Mirages in the Literature H Otero Martinez H Reinke D Michalik C Vogel
1841 Core-Tetrasubstituted Naphthalene Diimides by Stille Cross-Coupling Reactions and Characterization of Their Optical and Redox Properties S-L Suraru F Wuumlrthner
1846 A Practical Synthesis of Indole-Based Heterocycles Using an Amidoaluminum-Mediated Strategy R Todd M M Hossain
1851 Synthesis of Fluorinated Pyrrolo[23-b]pyridine and Pyrrolo[23-d]pyrimidine Nucleosides V O Iaroshenko Y Wang D V Sevenard D M Volochnyuk
1858 Recyclization Reactions of 5-Formyl-13-dimethyluracil with Electron-Rich Amino Heterocycles A P Mityuk D M Volochnyuk S V Ryabukhin A S Plaskon A Shivanyuk A A Tolmachev
1865 Facile Synthesis of Fluorinated 1-Desazapurines V O Iaroshenko D V Sevenard D M Volochnyuk Y Wang A Martiloga A O Tolmachev
1876 A Practical Synthesis of 3-Diethoxyphosphoryl-12-pyridazine Derivatives J-C Monbaliu J Marchand-Brynaert
1881 Enantioselective Reduction of Prochiral Ketones Employing Sprouted Pisum sativa as Biocatalyst J S Yadav B V S Reddy C Sreelakshmi A B Rao
1886 Application of Phenolate Ion Mediated Intramolecular Epoxide Ring Opening in the Enantioselective Synthesis of Functionalized 23-Dihydrobenzofurans and 1-Benzopyrans S K Dinda S K Das G Panda
1897 Complementary Synthetic Approaches to Constitutionally Diverse N-Aminoalkylated Isoindolinones Application to the Synthesis of Falipamil and 5-HT1A Receptor Ligand Analogues M Lorion A Couture E Deniau P Grandclaudon
1904 Selective Deprotection of Silyl Ethers with Sodium Periodate J Li D Menche
1909 Micellar Solution of Sodium Dodecyl Sulfate (SDS) Catalyzes KabacknikndashFields Reaction in Aqueous Media S Sobhani A Vafaee
1916 Convenient Methods for the Synthesis of a Library of Hemilabile Phosphines M V Jimeacutenez J J Peacuterez-Torrente M I Bartolomeacute L A Oro
1923 Terminal Aziridines by Addition of Grignard Reagents or Organoceriums to an (α-Chloro)sulfinylimine D M Hodgson J Kloesges B Evans
1933 A Robust Synthesis of Nε-(Carboxymethyl)-L-lysine (CML) R Csuk S Stark A Barthel R Kluge D Stroumlhl
1935 One-Pot Curtius Rearrangement Processes from Carboxylic Acids O Leogane H Lebel
XV Forthcoming Articles
no 12 1941 The Chemistry of Deprotonated α-Aminonitriles T Opatz 1960 An Efficient Synthesis of Tetraalkyl 2345-Thiophenetetracarboxylate
Derivatives A Alizadeh R Hosseinpour 1963 Facile Deprotection of Bulky (Trialkylsilyl)acetylenes with Silver Fluoride
S Kim B Kim J In 1969 Highly Efficient and Reusable Ionic Liquids for the Catalyzed
Hydroamination of Alkenes with Sulfonamides Carbamates and Carboxamides L Yang L-W Xu C-G Xia
1975 Synthesis of 2391016172324-Octasubstituted Phthalocyaninatozinc(II) Complexes Mediated by Reductive Agents G A Gauna A C Monsalvo J Awruch
1979 A Short and Efficient Synthesis of 3-2-[2-(Bromomethyl)thiazol-4-yl]-ethynyl-5-fluorobenzonitrile A Precursor for PET Radioligand [18F]SP203 M B Gopinathan C Jin K S Rehder
1983 Synthesis of a Substituted Benzazepin-2-one Dihydrate S K Boini R K Vaid K P Moder D Mitchell
1987 Synthesis of Novel Trisubstituted Imidazolines F J Lakner M A Parker B Rogovoy A Khvat A Ivachtchenko
1991 A Novel Synthesis of N-But-3-enyl-α- and β-Amino Acids T T Van Nguyen R T C Brownlee A B Hughes
1999 Synthesis of Substituted 5-(3-Hydroxypropyl)pyrrolidin-2-ones and Pyrrolizidinones from Nitroethane via C3 Functionalized 56-Dihydro-4H-12-oxazines A Novel Approach to Some Analogues of the Antidepressant Rolipram A Yu Sukhorukov A V Lesiv Y A Khomutova S L Ioffe V A Tartakovsky
2009 Chiral Cyclobutanols and Cyclopentane Dimers via Samarium(II) Iodide Induced Keto-Olefin Cyclisations of Carbohydrate-Derived Unsaturated Ketones D B G Williams J Caddy K Blann J J C Groveacute C W Holzapfel
2015 Synthesis of Perfluoroalkylthio-Substituted Ferrocenes C Rhode J Lemke M Lieb N Metzler-Nolte
2019 Functionalization of Polyhedral Oligomeric Silsesquioxane (POSS) via Nucleophilic Substitution M Dutkiewicz H Maciejewski B Marciniec
2025 A Novel Synthesis of Aryl Mesylates via One-Pot DemethylationndashMesylation of Aryl Methyl Ethers Using a Mixture of Phosphorus Pentoxide in Methanesulfonic Acid B Kaboudin Y Abedi
2029 Anionic Cyclization of (NN-Dimethylamino)[2-(prop-2-yn-1-yloxy)aryl]-acetonitriles T Zdrojewski J Musielak A Jończyk
2035 Strecker-Type Reaction Catalyzed by Carboxylic Acids in Aqueous Media Z Xie G Li G Zhao J Wang
2040 Synthesis of Novel Structurally Simplified Estrogen Analogues with Electron-Donating Groups in Ring A L F Tietze C A Vock I K Krimmelbein L Nacke
2061 On the Resolution of Secondary Phosphine Oxides via Diastereomeric Complex Formation The Case of tert-Butylphenylphosphine Oxide J Holt A M Maj E P Schudde K M Pietrusiewicz L Sieroń W Wieczorek T Jerphagnon I W C E Arends U Hanefeld A J Minnaard
2066 Enantioselective Copper-Catalyzed Conjugate Addition of Dimethylzinc to 5-(1-Arylalkylidene) Meldrumrsquos Acids A Wilsily T Lou E Fillion
2073 SuzukindashMiyaura Coupling Reactions Using Phosphite Ligands M Jang Y Jo I-K Oh H M Jung S Lee
2076 Synthesis of 2-Methylindoline- and 2-Methyl-1234-tetrahydroquinoline-Derived Phosphoramidites and Their Applications in Iridium-Catalyzed Allylic Alkylation of Indoles W-B Liu H He L-X Dai S-L You
2083 Stereocontrolled Synthesis of 13-Amino Alcohols by Reduction of Substituted 2-1-[(tert-Butylsulfinyl)amino]alkylcyclohexanones J C Gonzaacutelez-Goacutemez F Foubelo M Yus
2089 Tunable Phosphoramidite Ligands for Asymmetric Hydrovinylation Ligands par excellence for Generation of All-Carbon Quaternary Centers C R Smith H J Lim A ZhangT V RajanBabu
2101 Copper-Catalyzed Asymmetric Ring-Opening Reaction of Oxabenzonorbornadienes with Grignard and Aluminum Reagents R Millet L Gremaud T Bernardez L Palais A Alexakis
2113 A Simplified Synthesis of Takemotorsquos Catalyst A Berkessel B Seelig 2116 Pharmaceutical Substances Syntheses Patents and Applications of the
Most Relevant AIPs Edited by Axel Kleeman Juumlrgen Engel Bernhard Kutscher Dietmar Reichert Reviewed by I Agranat
XV Forthcoming Articles
no 13 2117 Recent Advances in the Aza-Claisen Rearrangement K C Majumdar
T Bhattacharyya B Chattopadhyay B Sinha 2143 A Novel and Convenient Synthesis of lsquoReversedrsquo Diamidino 25-Aryl- and
25-Azaheterocycle-Substituted Furans L Hu D W Boykin 2146 Efficient and General Preparation of Pyranostilbenes First Total Synthesis
of Artocarbene and Pawhuskin B B H Park Y R Lee W S Lyoo 2155 Mild Oxidation of Diarylacetylenes to 12-Diketones Using Oxone in
Trifluoroacetic Acid J-H Chu Y-J Chen M-J Wu 2163 One-Pot Microwave-Assisted Selective Azido ReductionTandem Cyclization
in Condensed and Solid Phase with Nickel Boride N Shankaraiah N Markandeya M Espinoza-Moraga C Arancibia A Kamal L Silva Santos
2171 Pyrrolo[321-ij]quinolin-4-one and Pyrrolo[321-ij]quinolin-6-one H McNab D J Nelson E J Rozgowska
2175 Practical Synthesis of 5-Substituted Tetrazoles under Microwave Irradiation J Roh T V Artamonova K Vaacutevrovaacute G I Koldobskii A Hrabaacutelek
2179 A Simple Method for the Synthesis of 3-Arylthieno[23-b]pyridines via Iodine-Mediated Cyclization of 3-(1-Arylalkenyl)-2-[(1-phenylethyl)sulfanyl]pyridines K Kobayashi D Nakamura Y Shiroyama S Fukamachi H Konishi
2184 Synthesis of Four Lysine-Linked Cereulide Analogues Showing Ionophoric Activity Towards Potassium Cations as Lead Compounds for Emetic Toxin-Detection by Immunoassays A Makarasen T Nishikawa M Isobe
2205 Synthesis of α-Aliphatic and β-Aromatic Substituted Taurines via Regioselective Ring Opening of Thiiranes with Ammonia H Yu S Cao L Zhang G Liu J Xu
2210 Stability of 5(6)-Carboxyfluorescein in Microwave-Assisted Synthesis of Fluorescein-Labelled O-Dimannosylated Peptides R Kowalczyk P W R Harris R P Dunbar M A Brimble
2223 Diversity-Oriented Synthesis of Functionalized Diaryl Sulfones by Regioselective [3+3] Cyclizations of 13-Bis(siloxy)buta-13-dienes with 2-(Arylsulfonyl)-3-ethoxy-2-en-1-ones Scope and Limitations M Shkoor A Riahi O Fatunsin H Reinke C Fischer P Langer
2236 Synthesis of Functionalized Salicylates by Formal [3+3] Cyclocondensation of 13-Bis(silyloxy)buta-13-dienes with 3-Alkoxy-2-en-1-ones G Mroszlig S Ladzik H Reinke A Spannenberg C Fischer P Langer
2249 Synthetic Approach to Alkoxy-β-(trifluoromethyl)styrenes and Their Application in the Synthesis of New Trifluoromethylated Heterocycles V M Muzalevskiy V G Nenajdenko A V Shastin E S Balenkova G Haufe
2260 o-Benzenedisulfonimide as a Powerful and Recyclable Organocatalyst for the Nazarov Reaction M Barbero S Cadamuro A Deagostino S Dughera P Larini E G Occhiato C Prandi S Tabasso R Vulcano P Venturello
2267 The Catalytic Potential of 4-Guanidinylpyridines in Acylation Reactions I Held E Larionov C Bozler F Wagner H Zipse
2278 Iron(III) Chloride in EthanolndashWater Highly Efficient Catalytic System for the Synthesis of Garcia Gonzalez Polyhydroxyalkyl- and C-Glycosylfurans L Nagarapu M V Chary A Satyender B Supriya R Bantu
2283 Ruthenium-Catalyzed Addition of Primary Amides to Alkynes A Stereoselective Synthesis of Secondary Enamides L J Gooszligen M Blanchot K S M Salih K Gooszligen
2289 Binaphthyl-Modified Quaternary Phosphonium Salts as Chiral Phase Transfer Catalysts Application to Asymmetric Amination of β-Keto Esters R He K Maruoka
X Table of Contents XI Forthcoming Articles
no 14 2293 Direct Methods for Stereoselective Polypropionate Synthesis A Survey
J Li D Menche 2316 Synthesis of Symmetrical Ketones from Grignard Reagents and
11-Carbonyldiimidazole D Bottalico V Fiandanese G Marchese A Punzi
2319 Synthesis of 45-Substituted Imidazoles by a Fast Condensation of 12-Diketones and Urotropine in Heterogeneous Medium G Bratulescu
2321 (Arylsulfonyl)acetones and -acetonitriles New Activated Methylenic Building Blocks for Synthesis of 123-Triazoles N T Pokhodylo V S Matiychuk M D Obushak
2324 A Safe Convenient and Efficient One-Pot Synthesis of α-Chloroketone Acetals Directly from Ketones Using Iodobenzene Dichloride J Yu C Zhang
2329 An Efficient Oxidative Conversion of Aldehydes into 2-Substituted 2-Oxazolines Using 13-Diiodo-55-dimethylhydantoin S Takahashi H Togo
2333 A Novel Procedure for the Synthesis of Benzo[b][18]naphthyridine-3-carboxylate Derivatives from MoritandashBaylisndashHillman Adduct Acetates W Zhong F Lin R Chen W Su
2341 An Improved Synthesis of 147-Triazacyclononanes (tacns) and 14710-Tetraazacyclododecanes (cyclens) J Huang Z Zhou T H Chan
2345 The Ullmann Coupling between 2-Chlorobenzoic Acids and Amino Acids A Valuable Reaction for Preparing 2-Substituted 1-Acetyl-1H-indol-3-yl Acetates J C Rodriguez Dominguez X Gang G Kirsch
2349 gem-Dibromomethyl Aromatics Efficient Aldehyde Equivalents in the KnoevenagelndashDoebner Reaction J K Augustine Y A Naik S Poojari N Chowdappa B S Sherigara K Areppa
2357 Synthesis of Novel α-Aminophosphonates Containing Adamantyl Fragment M M Kabachnik L I Minaeva I P Beletskaya
2361 Efficient Fluoride-Mediated Synthesis of 5-Amino-Substituted Isothiazoles Y S Zubenko V I Potkin
2365 Phosphine-Catalyzed Reaction of Cyanohydrins with Activated Alkynes A Siby O Loreau F Taran
2371 Sulfanyl-Substituted [3]Cumulenes and Buta-13-dienes from a Tetrakis(pyridinium)-Substituted Butadiene A Schmidt A Rahimi M Gjikaj
2379 Efficient Synthesis of 2-Substituted Pyrido[32-d]pyrimidines Involving SNAr and Palladium-Catalyzed Cross-Coupling Reactions A Tikad S Routier M Akssira J-M Leacuteger C Jarry G Guillaumet
2385 Novel Synthesis of Medium-Sized Heterocycles by Palladium-Catalyzed Intramolecular Heck Reaction via 9-endo-trig Mode of Cyclization K C Majumdar B Chattopadhyay
2393 Facile Synthesis of Fluorinated Benzofuro- and Benzothieno[23-b]pyridines α-Carbolines and Nucleosides Containing the α-Carboline Framework V O Iaroshenko Y Wang B Zhang D Volochnyuk V Ya Sosnovskikh
2403 Synthesis of Functionalized N-Vinyl Nitrogen-Containing Heterocycles S M M Lopes A M Beja M Ramos Silva J A Paixatildeo F Palacios T M V D Pinho e Melo
2408 Kumada Cross-Coupling of Aryl Grignard Reagents with Aryl Halides Catalyzed by an Immobilized Nickel Catalyst X Chen L Wang J Liu
2413 Highly Enantioselective Synthesis of Heteroaromatic Alcohols Catalyzed by Chiral DiaminodiphosphinendashRuthenium(II) Complexes W-Y Shen Y-Y Li Z-R Dong J-X Gao
2418 Concise Total Synthesis of (+)-Disparlure and its trans-Isomer Using Asymmetric Organocatalysis S-G Kim
2423 Rhodium Carbenoid Induced [12]-Migration in an L-Lyxo-Configured α-Diazo β-Keto Ester Synthesis of a New Griseolic Acid Analogue N N Bhujbal K S A Kumar D D Dhavale
2430 Synthesis of 5-Arylthio-3-hydroxyphthalates by the First [4+2] Cycloadditions of 3-Arylthio-1-silyloxy-13-butadienes with Dimethyl Acetylenedicarboxylate I Iqbal M Imran P Langer
2435 Synthesis of Highly Functionalized Proline Derivatives via a One-Pot MichaelSN-AdditionCyclization Approach U Kazmaier C Schmidt
2440 RhodiumGraphite-Catalyzed Hydrogenation of Carbocyclic and Heterocyclic Aromatic Compounds G Falini A Gualandi D Savoia
2447 Potassium [1-(tert-Butoxycarbonyl)-1H-indol-2-yl]trifluoroborate as an Efficient Building Block in Palladium-Catalyzed SuzukindashMiyaura Cross Couplings P Kassis V Beacuteneacuteteau J-Y Meacuterour S Routier
2454 Syntheses of Substituted Furans and Pyrroles by Platinum-Catalyzed Cyclizations of Propargylic Oxiranes and Aziridines in Aqueous Media M Yoshida M Al-Amin K Shishido
2467 Transition-Metal-Free Oxidative Homocoupling of Aryl Alkenyl and Alkynyl Grignard Reagents with TEMPO M S Maji A Studer
XIII Forthcoming Articles
no 15 2471 Advances in Synthetic Approaches for the Preparation of Combretastatin-
Based Anti-Cancer Agents R Singh H Kaur 2492 Synthesis of Unsymmetrical Ureas by Sulfur-Assisted Carbonylation with
Carbon Monoxide and Oxidation with Molecular Oxygen under Mild Conditions T Mizuno T Nakai M Mihara
2497 Ring-OpeningRecyclization Reactions of (Dimethylamino)propenoyl-Substituted Cyclopropanes Facile Synthesis of Halogenated Pyridin-2(1H)-ones R Zhang Y Zhou Y Liang Z Jiang D Dong
2501 Facile and Efficient Total Synthesis of Taspine B Cheng S Zhang L Zhu J Zhang Q Li A Shan L He
2505 Oligomeric Iodosylbenzene Sulfate A Convenient Hypervalent Iodine Reagent for Oxidation of Organic Sulfides and Alkenes M S Yusubov R Y Yusubova T V Funk K-W Chi V V Zhdankin
2509 Pyrrolidine-Based Organocatalysts for Enantioselective Michael Addition of Cyclohexanone to trans-β-Nitrostyrene A P Carley S Dixon J D Kilburn
2517 CundashAl Hydrotalcite An Efficient and Reusable Ligand-Free Catalyst for the Coupling of Aryl Chlorides with Aliphatic Aromatic and N(H)-Heterocyclic Amines B Sreedhar R Arundhathi P L Reddy M A Reddy M L Kantam
2523 Highly Efficient Synthesis of trans-βγ-Unsaturated a-Keto Amides C Allais T Constantieux J Rodriguez
2531 Gas-Phase Synthesis of N-Unsubstituted 3-Hydroxypyrroles and 1H-Pyrrol-3(2H)-ones L Hill G A Hunter S H Imam H McNab W J OrsquoNeill
2535 3-Hydroxy-1H-pyrrole L Hill S H Imam H McNab W J OrsquoNeill 2539 123-Thiadiazoles with Unsaturated Side Chains Synthesis
Polymerization and Photocrosslinking M Al-Smadi N Hanold H Kalbitz H Meier
2547 Synthesis of 1112-Didehydrodibenzo[ae]cycloocten-5(6H)-one A Strained Eight-Membered Alkyne S C Kornmayer F Rominger R Gleiter
2553 Stannous Chloride Dihydrate A Novel and Efficient Catalyst for the Synthesis of gem-Dihydroperoxides from Ketones and Aldehydes D Azarifar K Khosravi F Soleimanei
2557 Synthesis of a Novel Class of Azacrown Macrocycles and Lariat Crown Ethers Containing Two 124-Triazole Rings as Subunits N Foroughifar A Mobinikhaledi S Ebrahimi
2561 Enantioselective Synthesis of the 3C-Protease Inhibitor (ndash)-Thysanone by a StauntonndashWeinreb Annulation Strategy J Sperry T Y Yuen M A Brimble
2570 Stereoselective Synthesis of Unnatural β-Amino Acids from Nitroethane via 56-Dihydro-4H-12-oxazin-3-ylacetates A Yu Sukhorukov A V Lesiv O L Eliseev Y A Khomutova S L Ioffe
2579 A Versatile Unexpected One-Pot Regioselective Synthesis of a New Class of 13-Diazepinoindolones by Reaction of Pyranoindolones with Monosubstituted Ureas D Livadiotou C A Tsoleridis J Stephanidou-Stephanatou
2584 Synthesis of a Trisaccharide and a Tetrasaccharide from the Cell-Wall Lipopolysaccharides of Azospirillum brasilense S17 S Pandey S Ghosh A K Misra
2591 Synthesis of Isoindoline Nitroxides by Electrocyclic Reactions T Kaacutelai J Jekı K Hideg
2596 Glycosylations of Tertiary Alcohols Synthesis of Fully Protected Disaccharides with Sterically Demanding Groups Attached to the Sugar Core A Holkenbrink J B Vicente D B Werz
2605 Copper-Catalyzed [13]-Dipolar Cycloaddition for the Synthesis of Macrocycles Containing Acyclic Aromatic and Steroidal Moieties G V Latyshev M S Baranom A V Kazantsev A D Averin N V Lukashev I P Beletskaya
2616 Aryl Ring Migration Reaction in the Synthesis of 24-Diaryl-4H-31-benzothiazines A V Butin F A Tsiunchik V T Abaev A V Gutnov D A Cheshkov
2627 Hydrogenation of β-N-Substituted and β-NN-Disubstituted Enamino Esters in the Presence of Iridium(I) Catalyst H Hebbache Z Hank C Bruneau J-L Renaud
2634 Stereoselective Olefination Reactions Promoted by Rieke Manganese J M Concelloacuten H Rodriacuteguez-Solla V del Amo P Diacuteaz
2646 Synthesis of Piperidinones through a Radical Cascade E Godineau Y Landais
2650 Asymmetric Organic Synthesis with Enzymes Edited by V Gotor I Alfonso E Garciacutea-Urdiales Reviewed by Steve Collier
XVII Forthcoming Articles
no 16 2651 Synthesis of Spirocyclic Ethers S Rosenberg R Leino 2674 Bimetallic PalladiumndashPlatinum-on-Carbon-Catalyzed HndashD Exchange
Reaction Synergistic Effect on Multiple Deuterium Incorporation T Maegawa N Ito K Oono Y Monguchi H Sajiki
2679 Efficient Copper-Catalyzed Synthesis of 2-Amino-4(3H)-quinazolinone and 2-Aminoquinazoline Derivatives X Huang H Yang H Fu R Qiao Y Zhao
2689 Synthesis and Chemoselective N- and O-Alkylation of Thiadiazolopyrimidine Nucleosides and Uridines A M L Hossion R Islam R K Kandahary T Nagamatsu
2697 Facile and Efficient Synthesis of a New Class of Indole-Substituted Pyridine Derivatives via One-Pot Multicomponent Reactions K Zhao X-P Xu S-L Zhu D-Q Shi Y Zhang S-J Ji
2709 Studies toward a Total Synthesis of Rhizoxin D Stereoselective Preparation of the C11ndashC19 Fragment S Padakanti C K Kumar E Ashok P Das
2715 A Short Synthesis of Enantiomeric Phytoprostanes B1 Type I W Perlikowska M Mikołajczyk
2719 Chemistry of Polyhalogenated Nitrobutadienes Part 7 A Novel Synthetic Access to Chlorinated Nitrile Oxides E Nutz V A Zapolrsquoskii D E Kaufmann
2725 Microwave-Assisted Silver(I)-Mediated Selective O-Alkylation of Aromatic Imidate Systems B K Singh C Cavalluzzo M De Maeyer Z Debyser V S Parmar E Van der Eycken
2729 Iodogen A Novel Reagent for the Oxidation of Urazoles under Heterogeneous Conditions A Khoramabadi A Shiri M A Zolfigol S Mallakpour
2733 An Unprecedented Synthesis of Eight-Membered-Ring Cyclic Thioimidic Esters by a Three-Component Reaction A Alizadeh R Hosseinpour
2737 A Novel Diastereoselective Synthesis of β-Phosphonato Unsaturated Thioimidates A Alizadeh N Zohreh
2741 Synthesis of 21-Benzisoxazoles by Nucleophilic Substitution of Hydrogen in Nitroarenes Activated by the Azole Ring N T Pokhodylo Y O Teslenko V S Matiychuk M D Obushak
2749 A Facile Synthesis of Two Series of Multifunctional Carbon Compounds from αα-Dihalo Ketones Using Allylsamarium Bromide X Liu S Zhang J Di
2756 Stereocontrolled Formation of Protected Aminodeoxyalditols from Simple Carbohydrate Precursors by Debenzylating Cycloetherification Y Jiang Z Fang Q Zheng H Jia J Cheng B Zheng
2761 trans-Stilbene as a Starting Material for the Synthesis of Tamoxifen Based on Palladium-Catalyzed Cross-Coupling Reactions C M Nunes J Limberger S Poersch M Seferin A L Monteiro
2766 Synthesis and Biological Evaluation of 6-Substituted Purinylcarbanucleosides with a Cyclopenta[b]thiophene Pseudosugar P Abeijoacuten J M Blanco O Caamantildeo F Fernaacutendez M D Garciacutea X Garciacutea-Mera J E Rodriacuteguez-Borges J Balzarini E De Clercq
2773 Synthesis and Electrochemical Signature of Novel Norbornyl-ferrocene Hybrids F A Khan S K Upadhyay
2778 A Regioselective TsujindashTrost Pentadienylation of 3-Allyltetronic Acid R Schobert B Barnickel
2785 Copper(I)-Catalyzed CarylndashCalkynyl Bond Formation of Aryl Iodides with Terminal Alkynes K G Thakur G Sekar
2790 Aminolysis of Epoxides Using Iridium Trichloride as an Efficient Catalyst J Agarwal A Duley R Rani R K Peddinti
2797 Preparation of Several Active N-Chloro Compounds from Trichloroisocyanuric Acid A Shiri A Khoramabadi-zad
2802 The First Mineral-Catalyzed One-Pot [3+1+2] Coupling Protocol for Multifunctionalized Fused-Ring Pyrimidines L D S Yadav A Rai
2809 Efficient Synthesis of Tetrahydro-β-carbolin-1-one and Dihydroisoquinolin-1-one Derivatives as Versatile Intermediates K E Judd M F Mahon L Caggiano
2818 A Concise Synthesis of ortho-Iodobenzyl Alcohols via Addition of ortho-Iodophenyl Grignard Reagent to Aldehydes and Ketones J Cvengroš D Stolz A Togni
XIII Forthcoming Articles
no 17 2825 Reactivity of Oxazol-5-(4H)-ones and Their Application toward Natural
Product Synthesis N M Hewlett C D Hupp J J Tepe 2840 Towards the Total Synthesis of 3-Hydroxyvibsanin E B D Schwartz
J R Denton P V Bernhardt H M L Davies C M Williams 2847 Structure Investigations of (ent)-Cladospolide D by De Novo Synthesis and
Kinetic and Thermodynamic Isomerization Y Xing J H Penn G A OrsquoDoherty
2855 New Applications of PhI(OAc)2 in Synthesis Total Synthesis and SAR Development of Potent Antitumor Natural Product PsymberinIrciniastatin A N Shao X Huang A Palani R Aslanian A Buevich J Piwinski R Huryk C Seidel-Dugan
2873 Total Synthesis of Largazole ndash Devolution of a Novel Synthetic Strategy B Wang C J Forsyth
2881 Formal Total Synthesis of Palmerolide A J Jaumlgel M E Maier 2893 Total Synthesis of Bongkrekic Acid via Sequential SuzukindashMiyaura Coupling
Reactions M Kanematsu M Shindo M Yoshida K Shishido 2905 Stereodivergent Approach to Both C28a-syn and C28a-anti Relative
Stereochemical Manifolds in the Lepadin Family via a TiCl4-Promoted G Li L J Carlson I K Sagamanova B W Slafer R P Hsung C Gilardi H M Sklenicka N Sydorenko
2915 Enantioselective Aldol Reaction of Tetrasubstituted Ketene Silyl Acetals with Achiral Aldehydes for the Construction of Asymmetric Tertiary Alcohols An Application for the Divergent Total Syntheses of Buergerinins F and G I Shiina T Iizumi Y-s Yamai Y-i Kawakita K Yokoyama Y-k Yamada
2927 Second-Generation Biomimetic Total Synthesis of Chaetominine A Coste G Karthikeyan F Couty G Evano
2935 Total Synthesis of (+)-Fostriecin and (+)-Phoslactomycin B S Shibahara M Fujino Y Tashiro N Okamoto T Esumi K Takahashi J Ishihara S Hatakeyama
2954 Stereochemical Assignments of the Chlorinated Residues in Victorin C A C Durow C Butts C L Willis
2963 Studies of the Asymmetric Total Synthesis of Clavilactone D by the lsquoLariatrsquo Cyclization Strategy T Yoshimitsu S Nojima M Hashimoto K Tsukamoto T Tanaka
2970 Total Synthesis of the Leucetta-Derived Alkaloid Calcaridine A P B Koswatta R Sivappa H V R Dias C J Lovely
2983 Formal Synthesis of Salinosporamide A Starting from D-Glucose T Momose Y Kaiya J-i Hasegawa T Sato N Chida
2992 Synthesis of Bioactive Natural Products by Asymmetric syn- and anti-Aldol Reactions A K Ghosh Z L Dawson
no 18 3003 Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural
Products B M Trost M K Brennan 3026 One-Pot Synthesis of Furo[34-b]pyridin-5(7H)-ones from 2-
Bromopyridine-3-carboxylic Acid and Carbonyl Compounds K Kobayashi T Kozuki H Konishi
3029 Iodocyclization of N-[2-(Methylthio)phenyl]propiolamides Selective Synthesis of 3-Iodo-15-benzothiazepin-4-ones T-S Jiang X-G Zhang J-H Li
3039 A Facile Synthetic Method for Fluorine-Containing 17-Phenanthrolines Pyridine-Ring Formation Reaction of N-Propargyl-68-bis(trifluoroacetyl)-quinolin-5-amine with Various Nucleophiles D Shibata E Okada M Hinoshita M Meacutedebielle
3047 Enantiotopic Discrimination in Palladium-Mediated Nucleophilic Substitutions on Achiral Substrates Chiral Ligand versus Chiral Nucleophile O Jacquet F Charnay J-C Fiaud J Ollivier
3051 Studies on the Chemistry of 2-[3-(2-Nitrophenyl)-2-oxopropyl]benzaldehydes Novel Syntheses of 5H-Benzo[b]carbazole-611-diones and Indolo[12-b]isoquinoline-611-diones M Fernaacutendez
3061 Studies on the C22ndashC23 Aldol Coupling of Spirangien M Lorenz N Bluhm M Kalesse
3067 One-Pot Synthesis of N-Alkyl Purine Pyrimidine and Azole Derivatives from Alcohols using Ph3PCCl4 A Rapid Route to Carboacyclic Nucleoside Synthesis M N Soltani Rad A Khalafi-Nezhad S Behrouz Z Asrari M Behrouz Z Amini
3077 Synthesis of 2-Amino-34-dihydroquinazolines and Imidazo[21-b]quinazoline-2-ones A Mishra S Batra
3089 Studies on the Reaction of Diimines with Thiourea Synthesis and Solvent-Induced cistrans-Isomerization of 135-Triazinane-2-thiones B Kaboudin T Ghasemi T Yokomatsu
3094 Suzuki Coupling of Heteroaromatic Chlorides Using Highly Electron-Donating ClickPhos Ligands S M Spinella Z-H Guan J Chen X Zhang
3099 Reaction of NN-Dioxyenamines with Anhydrides of Carboxylic and Sulfonic Acids A New Method for the Synthesis of a-Hydroxyoxime Derivatives A A Tabolin A V Lesiv S L Ioffe
3106 Directed ortho Metallation Chemistry and Phosphine Synthesis New Ligands for the SuzukindashMiyaura Reaction D B G Williams S J Evans H de Bod M S Mokhadinyana T Hughes
3113 New Functional Derivatives of 9-Phenylquinine P J Boratyński J SkarŜewski
3120 On the Synthesis of Asymmetric and Dissymmetric Amino Analogues of Troumlgerrsquos Base J Artacho K Waumlrnmark
3127 Synthesis of Polycyclic Sultams by Palladium-Catalyzed Intramolecular Cyclization K C Majumdar S Mondal N De
3136 Synthesis of Functionalized L-Cysteine and L-Methionine by Reaction with Electron-Deficient Acetylenes B A Trofimov A G Malrsquokina O A Shemyakina V V Nosyreva A P Borisova S S Khutsishvili L B Krivdin
3143 A lsquoClickrsquo Approach to the Synthesis of 3-[2-(1-Alkyltriazol-4-yl)ethyl]indoles M Petrini R R Shaikh
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
No 3 339 Intermolecular Addition Reactions of N-Acyliminium Ions (Part I)
A Yazici S G Pyne 369 Desulfurization of Thioamides into Amides with H2O2ZrCl4 Reagent System
K Bahrami M M Khodaei Y Tirandaz 372 Total Synthesis of (plusmn)-1345-Tetragalloylapiitol R M Patel
N P Argade 375 A Convenient Synthesis of 4-Hydroxy-2-oxo-12-dihydro-18-
naphthyridine-3-carboxamide Derivatives K Kobayashi D Iitsuka S Fukamachi H Konishi
379 Intramolecular Ketalization of Functionalized 7-Norbornenols L A Paquette J D Pettigrew
385 Ring Contraction of 12-Dihydronaphthalenes Promoted by Thallium(III) in Acetonitrile A Diastereoselective Approach to Indanes H M C Ferraz V M T Carneiro L F Silva Jr
389 Regio-Controlled Nucleophilic Attack of 3-Thiaisatoic Anhydride by α-Amino Acids One-Pot Synthesis of 3-(2-Thienyl)imidazolidine-24-dione and 34-Substituted Thieno[23-e][14]diazepine-25-dione Analogues Y Brouillette G Sujol J Martinez V Lisowski
395 The Unprecedented Cobalt-Catalysed Oxidative Glaser Coupling under Reductive Conditions G Hilt C Hengst M Arndt
399 Nucleophilic Addition of 4-Hydroxycoumarin to BaylisndashHillman Acetate Adducts C Raji Reddy N Kiranmai K Johny M Pendke P Naresh
403 Palladium-Mediated Heck Reaction to the Synthesis of 3-Substituted Indoles and Indolones K C Majumdar S Chakravorty P K Shyam A Taher
409 Synthesis of Bicyclo[310]hexan-2-ones by Manganese(III) Oxidation in Ethanol K Asahi H Nishino
424 High Regio- and Stereoselective Synthesis of (Z)- or (E)-N-Acryl Butenedioic Monoimide Derivatives by a Multicomponent Reaction F Sha Y Lin X Huang
431 The First Synthesis of Allyl Isonitriles from BaylisndashHillman Adducts and Their Application in the Synthesis of Substituted Imidazo[12-α]pyridines and Tetraazadibenzoazulenes M Nayak S Kanojiya S Batra
438 One-Pot Three-Step Synthesis of Pyrazinothienopyrimidines Using Tandem Aza-WittigElectrocyclic Ring Closure G Blanco A Fernaacutendez-Mato J M Quintela C Peinador
445 Synthesis of Biaryls Fluorenones Cyclopenta[def]phenanthren-4-ones and Benzophenones Based on Formal [3+3] Cyclocondensations of 13-Bis(silyloxy)buta-13-dienes with 3-(Silyloxy)-2-en-1-ones S Reim M Lau M Adeel I Hussain M A Yawer A Riahi Z Ahmed C Fischer H Reinke P Langer
464 Diastereoselective Synthesis of α-Stabilized Phosphorus Ylides via a Four-Component Reaction A Alizadeh N Zohreh L-G Zhu
469 Stereoselective Synthesis of Alkynyl Vinyl Chalcogenides via HornerndashWittig Reaction C C Silveira F Rinaldi R C Guadagnin A L Braga
474 Stereoselective Preparation of C1ndashC10 and C11ndashO14 Fragments of Narbonolide Exploiting the Versatility of Thiazolidinethione Chiral Auxiliary C P Narasimhulu P Das
483 Efficient Catalytic Activity of CopperAluminum Hydrotalcite in Diaryl Ether Synthesis B Sreedhar R Arundhathi M A Reddy M L Kanatm
488 On-Resin Click-Glycoconjugation of Peptoids A S Norgren C Budke Z Majer C Heggemann T Koop N Sewald
495 A Simple and Efficient Preparation of Novel Formaldehyde Derivatives R Hartung G Golz S Schlaf G Silvennoinen K Polborn P Mayer H R Pfaendler
502 2-Oxazol-5-ylethanones by Consecutive Three-Component AmidationndashCouplingndashCycloisomerization (ACCI) Sequence E Merkul O Grotkopp T J J Muumlller
508 SuzukindashMiyaura Cross-Couplings Mediated by trans-PdBr(N-Succ)(PPh3)2 A Convenient Synthetic Method for Diarylmethanes and Aryl(heteroaryl)-methanes I J S Fairlamb P Sehnal R J K Taylor
511 Modern Reduction Methods Edited by P G Andersson and I J Munslow Reviewed by Siegfried R Waldvogel
512 Addendum and Erratum XIII Forthcoming Articles
No 4 513 Intermolecular Addition Reactions of N-Acyliminium Ions (Part II)
A Yazici S G Pyne 542 A Simple Practical Method for the Synthesis of 46-Dimethoxy-135-
triazin-2(1H)-one Using Dimethylamine-Functionalized Solid-Phase Reagents K Hioki K Ohshima Y Sota M Tanaka M Kunishima
545 Conjugation-Amenable Tetrasaccharide of the Side Chain of the Major Glycoprotein of the Bacillus anthracis Exosporium A Large-Scale Preparation S Hou P Kovaacuteč
551 Reductive Amination ndash A Convenient Method for Generating Diverse Mono-Functionalised 5101520-Tetraphenyl Porphyrins C Welch S J Archibald R W Boyle
557 Highly Regioselective Preparation of 13-Dioxolane-4-methanol Derivatives from Glycerol Using Phosphomolybdic Acid N W Fadnavis R Gowrisankar G Ramakrishna M K Mishra G Sheelu
561 Rapid Synthesis of 3-Aminoisoquinoline-5-sulfonamides Using the BuchwaldndashHartwig Reaction N Proisy S Taylor A Nelson I Collins
567 Synthesis of Divalent 22-Linked Mannose Derivatives by Homodimerization F S Ekholm M Polaacutekovaacute A J Pawłowicz R Leino
577 Efficient Synthesis of Substituted Cyclic α-Aminophosphonates I L Odinets O I Artyushin N Shevchenko P V Petrovskii V G Nenajdenko G-V Roumlschenthaler
583 Methylated Imidazolinium-Dithiocarboxylates Two Representatives of a New Class of Ionic Liquids A Blanrue R Wilhelm
587 An Efficient Route to 1-Vinylpyrrole-2-carbaldehydes A I Mikhaleva A V Ivanov E V Skitalrsquotseva I A Ushakov A M Vasilrsquotsov B A Trofimov
591 A Regioselective Route to 5-Substituted Isoxazole- and Isoxazoline-3-phosphonates P Conti A Pinto L Tamborini P Dunkel V Gambaro G L Visconti C De Micheli
597 Solvent-Free One-Pot Conjugate Addition of Benzyl Bromides to β-Nitroalkenes Mediated by Magnesium Powder W Shi J-X Wang
602 Synthesis of 234-Trideoxy-44-difluoro-D-ribo-hexopyranose Adenosines J Xu X Zhang X-L Qiu F-L Qing
609 Synthesis of anti-27-Disubstituted Norbornadienes G C Tsui P Le Marquand A Allen W Tam
620 Novel Peptide Mimetic Inhibitors of Hepatitis C Serine Protease Derived from Isomannide T G Barros S Pinheiro J S Williamson A Tanuri H S Pereira R M Brindeiro J B A Neto O A C Antunes E M F Muri
627 A Practical Synthesis of α-Substituted tert-Butyl Acrylates from Meldrumrsquos Acid and Aldehydes C G Frost S D Penrose R Gleave
636 A New Class of Troumlgerrsquos Base Analogues Bearing Spiro[45] Lactone Straps A B Mahon D C Craig A C Try
643 A New Approach to Di- and Tetrasubstituted 23-Dihydropyridin-4(1H)-ones through Aza-DielsndashAlder Reaction Promoted by Silicon Tetrachloride A Massa V de Sio R Villano M R Acocella L Palombi G Sellitto A Peduto R Filosa P De Capraris A Scettri
650 Palladium-Catalysed Direct Arylation of Sydnones A Rodriguez W J Moran
655 Synthesis of (ndash)-Monomorine I R W Bates P Song 660 Cobalt(II) Chloride HexahydratendashDiisopropylamine Catalyzed Mild and
Chemoselective Reduction of Carboxylic Esters with Sodium Borohydride A R Jagdale A S Paraskar A Sudalai
665 Synthesis of Bi- and Tricyclic αβ-Unsaturated Lactams as Potential Michael Acceptors Starting from Heterocyclic Imines K Schulz M Watzke K Johannes P Ullrich J Martens
674 An Expedient Synthesis of Bis-Fused Benzofuran and a Two-Directional Ring-Closing Metathesis for the Synthesis of Bisbenzoxepines and Bisbenzoxocines K C Majumdar B Chattopadhyay S Chakravorty
681 Palladium-Catalyzed Cross-Couplings of Unsaturated Halides Bearing Relatively Acidic Hydrogen Atoms with Organozinc Reagents Z Dong G Manolikakes J Li P Knochel
687 Synthesis of Enantioenriched aa-Disubstituted Cyclopentenes Catalyzed by N-Heterocyclic Carbenes E M Phillips M Wadamoto K A Scheidt
XVII Forthcoming Articles
No 5 691 Transannulation Reactions in the Synthesis of Natural Products
P A Clarke A T Reeder J Winn 710 Synthesis of DL-erythro-Sphingosine Using a Tethered
Aminohydroxylation Reaction as the Key Step J A Morales-Serna Y Diacuteaz M I Matheu S Castilloacuten
713 Convenient Multigram Synthesis of 4-Chloropyridine-26-dicarbonyl Dichloride K Mitsui J R Parquette
715 A Novel and Efficient Synthesis of Dihydrexidine J P Cueva D E Nichols
721 Synthesis of 57-Dichloro-6-azaindoles and Functionalization via a Highly Selective LithiumndashChlorine Exchange N Lachance L-P Bonhomme-Beaulieu P Joly
731 A Convenient Synthesis of Fluorinated Pyrazolo[34-b]pyridine and Pyrazolo[34-d]pyrimidine Nucleosides V O Iaroshenko D V Sevenard A Kotljarov D M Volochnyuk A O Tolmachev V Y Sosnovskikh
741 Diastereoselective Synthesis of γ-Amino Acids and Their Derivatives from Nitroethane via Intermediacy of 56-Dihydro-4H-12-oxazines Bearing the CH2CH(CO2Me)2 Substituent at C3 A Y Sukhorukov A V Lesiv Y A Khomutova S L Ioffe
755 Synthesis of a New Pyrrolopyridoindole and Its Pyrrolopyridobenzimidazole Regioisomer F Bouchikhi M Sassatelli F Anizon M Prudhomme P Moreau
759 Practical Syntheses of Sphingosine-1-Phosphate and Analogues V Blot U Jacquemard H-U Reissig B Kleuser
767 A Facile Synthetic Route towards Substituted Thieno[32-e]indoles W Van Snick W Nulens S Jambon W Dehaen
775 Microwave-Assisted One-Pot Synthesis of (Aminoalkyl)naphthols and (Aminoalkyl)quinolinols by Using Ammonium Carbamate or Ammonium Hydrogen Carbonate as Solid Ammonia Source I Szatmaacuteri F Fuumlloumlp
779 Enantioselective Synthesis of Flavan-3-ols Using a Mitsunobu Cyclization K Krohn I Ahmed M John 787 Synthesis of a Novel γ-Folic AcidndashNτ-Histidine Conjugate Suitable for
Labeling with 99mTc and 188Re C Sparr U Michel R E Marti C Muumlller R Schibli R Moser V Groehn
793 Palladium-Catalyzed Intramolecular Biaryl Coupling A Highly Efficient Avenue for Benzannulated Pyranoquinolines and Julolidine Derivatives K C Majumdar A Taher P Debnath
801 Preparation of NN-Dimethyl-N-Arylureas Using SS-Dimethyl Dithiocarbonate as a Carbonylating Reagent I Degani R Fochi C Magistris M Migliaccio
809 Versatile Selective α-Carboxylic Acid Esterification of N-Protected Amino Acids and Peptides by Alcalase T Nuijens C Cusan J A W Kruijtzer D T S Rijkers R M J Liskamp P J L M Quaedflieg
815 Efficient Palladium-Catalyzed Amination of Aryl Chlorides Using Dicyclohexylamino[(26-dimethyl)morpholino]phenylphosphine as a PN2 Ligand S-E Park S B Kang K-J Jung J-E Won S-G Lee Y-J Yoon
824 A Clean Facile and Stereospecific Synthesis of α-Oxoketene OS-Acetals in Water Y Li Q Zhang X Cheng Q Liu X Xu
829 Sonogashira Cross-Coupling Reactions and Construction of the Indole Ring System Using a Robust Silica-Supported Palladium Catalyst E Tyrrell L Whiteman N Williams
836 Synthesis of Angular 78-Pyridazinocoumarins via the Transformation of a Hydroxy Group into a Carbonyl Group A Kotali I S Lafazanis P A Harris
841 Synthesis of New Cyclic and Acyclic 5-Halouridine Derivatives as Potential Antiviral Agents M F Elshehry J Balzarini C Meier
848 Dendritic Triphenylmethylium and Tetraphenylmethane Compounds H Meier S Kim A Oehlhof
853 Synthesis of Homoallylic Alcohols via Lewis Acid Assisted Enantioselective Desymmetrization B Yu F Menad N Isono M Lautens
860 Diastereoselective Synthesis of 123-Trisubstituted Indanes via Rhodium(I)-Catalyzed Tandem Conjugate Additions C Navarro A G Csaacutekyuml
864 Bakerrsquos Yeast for Sweet Dough Enables Large-Scale Synthesis of Enantiomerically Pure Bicyclo[331]nonane-26-dione C J Wallentin E Orentas E Butkus K Waumlrnmark
868 Addendum and Erratum XV Forthcoming Articles
No 6 869 Stereoselective Transformations of meso Bicyclic Hydrazines Versatile
Access to Functionalized Aminocyclopentanes C Bournaud F Chung A P Luna M Pasco G Errasti T Lecourt L Micouin
888 Synthesis of Glycoaminoxy Acids as Novel Sugar Building Blocks A Malapelle R Ramozzi J Xie
891 Electrophilic ipso-Halocyclization of N-Arylpropynamides with Polyfluoroalkyl Alcohols Selective Synthesis of 8-(Polyfluoroalkoxy) azaspiro[45]trienes Z-Q Wang B-X Tang H-P Zhang F Wang J-H Li
903 Electrooxidation of Alcohols in N-Oxyl-Immobilized Silica GelWater Disperse System Approach to Totally Closed System M Kuroboshi K Goto H Tanaka
909 Synthetic Routes to Aminotriamantanes Topological Analogues of the Neuroprotector Memantinereg A A Fokin A Merz N A Fokina H Schwertfeger S L Liu J E P Dahl R K M Carlson P R Schreiner
913 Parallel Synthesis of Drug-like 5-Amino-Substituted 124-Thiadiazole Libraries Using Cyclization Reactions of a Carboxamidine Dithiocarbamate Linker J Y Park I A Ryu J H Park D C Ha Y-D Gong
921 Copper-Catalyzed Selective S-Arylation of 12-Bis(o-amino-1H-pyrazolyl) Disulfides with Arylboronic Acids P-S Luo F Wang J-H Li R-Y Tang P Zhong
929 2-Iodoxybenzoic AcidTetraethylammonium BromideWater An Efficient Combination for Oxidative Cleavage of Acetals C Kuhakarn W Panchan S Chiampanichayakul N Samakkanad M Pohmakotr V Reutrakul T Jaipetch
935 Synthesis of Quinonoid Analogues of Diospyrin S Sagar I R Green 941 A One-Pot Method for the Iodination of Aryl Amines via Stable Aryl
Diazonium Silica Sulfates Under Solvent-Free Conditions A Zaroi A R Hajipour L Khazdooz
945 Poly(NN-dichloro-N-ethylbenzene-13-disulfonamide) and NNNN-Tetrachlorobenzene-13-disulfonamide as Novel Reagents for the Synthesis of N-Chloroamines Nitriles and Aldehydes R Ghorbani-Vaghei H Veisi
951 Synthesis of an (R)-Garner-type Aldehyde from L-Serine Useful Building Block for a (+)-Furanomycin Derivative G Bartoli G Di Antonio R Fiocchi S Giuli E Marcantoni M Marcolini
957 An Efficient and Highly Selective Synthesis of (Z)-Fluoroenol Phosphates from Hydroxy Difluorophosphonates P Beier R Pohl A V Alexandrova
963 Iodine-Catalyzed Three-Component Reaction A Rapid Synthesis of α-Alkoxy Azides and Homoallyl Ethers J S Yadav B V S Reddy G M Reddy R Narender
969 Rhodium(I)-Catalyzed Cycloisomerization of 13-Dienes with Alkenes in a Tether Y Oonishi A Saito M Mori Y Sato
980 Synthesis of New Optically Active D-GlucosaminendashPyrrole Derivatives B A Frontana-Uribe M V Escaacutercega-Bobadilla J Juaacuterez-Lagunas R A Toscano G A Garciacutea de la Mora M Salmoacuten
985 Partially Saturated Indeno[12-b]indole Derivatives via Deoxygenation of Heterocyclic α-Hydroxy-NO-hemiaminals H-J Hemmerling G Reiss
1000 Light-Induced Synthesis of Π-Extended Tetrathiafulvalenes Incorporating Ferrocenes An Efficient Route for the Synthesis of Electron-Donor Materials A A O Sarhan C Bolm
1007 Preparation of Nβ-Fmoc-Protected Aza-β3-Amino Acids with Nonproteinogenic Hydrophobic Side Chains for Solid-Phase Syntheses of Pseudopeptides M Laurencin P Bauchat M Baudy-Flocrsquoh
1014 Diastereomeric (η4-diene)Fe(CO)3 Complexes Containing Chiral Amide Groups A Convenient Method for the Resolution of Amino Acids M Schumacher G Coste L Miesch
1021 Palladium-Catalysed Heck Reactions of Alk-1-en-3-ones with Aryl Bromides A Very Simple Access to (E)-1-Arylalk-1-en-3-ones M Lemhadri Y Fall H Doucet M Santelli
1036 An Improved Process for the Synthesis of 4H-Imidazo[15-α][14]benzodiazepines J Yang Y Teng S Ara S Rallapalli J M Cook
1041 Meta- and Para-Difunctionalization of Arenes via an Ortho-Magnesiation and a Subsequent SulfoxidendashMagnesium Exchange L Melzig C B Rauhut P Knochel
XIII Forthcoming Articles
No 7 1049 Catalytic Transformations of Benzylic Carboxylates and Carbonates
R Kuwano 1062 A Simple and Practical Method for the Oxidation of Thebaine to 14-
Hydroxycodeinone by V2O5ndashH2O2 S Das Sharma D Konwar 1065 Umpolung with Sulfur Dioxide CarbonndashCarbon Cross-Coupling of Electron-
Rich 13-Dienes and Alkenes Application to the Enantioselective Synthesis of Long-Chain Polyketide Fragments M Turks C J Exner C Hamel P Vogel
1075 One-Pot Synthesis of 14-Diarylnaphthalenes via a WittigndashHorner Reaction[4+2] CycloadditionDehydrogenation Sequence Z Chen W Shou Y Wang
1081 A Novel and General Method for the Formation of S-Aryl Se-Aryl and Te-Aryl Phosphorochalcogenoates Y-X Gao G Tang Y Cao Y-F Zhao
1087 A Remarkable Access to γ-Fluoroalkylated Propargylamine Derivatives or Fluoroalkylated Dihydroisoxazoles via the Reaction of Fluoroalkylated Acetylides with Various Nitrones T Konno K Moriyasu T Ishihara
1095 Short and Practical Syntheses of (S)-(+)-3-(p-Tolylsulfinyl)furan-2(5H)-one and (S)-(+)-3-(p-Tolylsulfinyl)-56-dihydropyran-2-one D Cruz Cruz A Hernaacutendez Linares F Yuste M R Martiacuten J L Garciacutea Ruano
1099 Decarboxylative Aldol-Type Reaction of 2-(Trifluoroacetyl)-13-diazoles with Activated Acetic Acids P V Khodakovskiy D M Volochnyuk A A Tolmachev
1105 Synthesis of 2-[(Arylmethylene)amino]cyclopropanecarbonitriles via a Two-Step Ring Transformation of 2-(Cyanomethyl)aziridines S Mangelinckx M Drsquohooghe S Peeters N De Kimpe
1113 Synthesis of Dendrimeric Tumor-Associated Mucin-Type Glycopeptide Antigens T Becker A Kaiser H Kunz
1123 A Simple and Efficient Oxidation Procedure for the Synthesis of Acid-Sensitive Epoxides O Bortolini G Fantin M Fogagnolo
1127 Rapid Chemoselective Deprotection of Benzyl Esters by Nickel Boride J M Khurana R Arora
1131 Three-Component Coupling of Isoquinoline Activated Alkyne and Nitromethane A Facile Synthesis of Nitromethyl Derivatives of 12-Dihydroisoquinolines J S Yadav B V S Reddy N N Yadav M K Gupta
1137 Palladium Supported on a Polyionic Resin as an Efficient Ligand-Free and Recyclable Catalyst for Heck SuzukindashMiyaura and Sonogashira Reactions B Basu S Das P Das B Mandal D Banerjee F Almqvist
1147 Oxidation of 25-Dialkylpyrrole Derivatives with Cerium(IV) Ammonium Nitrate R Voloshchuk M Gałęzowski D T Gryko
1153 Practical Syntheses of Enantiomerically Pure Key Intermediates of Opioid Receptor-like 1 (ORL1) Antagonists T Yoshizumi A Ohno T Tsujita H Takahashi O Okamoto I Hayakawa H Kigoshi
1163 An Environmentally Benign TEMPO-Catalyzed Efficient Alcohol Oxidation System with a Recyclable Hypervalent Iodine(III) Reagent and Its Facile Preparation X-Q Li C Zhang
1170 Efficient and Stereoselective Rearrangement of BaylisndashHillman Acetates Catalyzed by Gold(I) ChlorideSilver(I) Trifluoromethanesulfonate Y Liu D Mao J Qian S Lou Z Xu Y Zhang
1175 The First Total Synthesis of Kynapcin-24 by Palladium Catalysis L-Y Yang C-F Chang Y-C Huang Y-J Lee C-C Hu T-H Tseng
1180 Enantioselective Synthesis of N-Protected α-Amino Acid Hydrazides M Bibian S El-Habnouni J Martinez J-A Fehrentz
1185 Synthesis of 11H-Indolo[32-c]quinoline-6-carboxylic Acids by Cascade AutoxidationndashRing Contractions A Becker S Kohfeld T Pies K Wieking L Preu C Kunick
1190 Reaction of N-Nonaflylbenzotriazole with Silyl Enol Ethers M Uhde T Ziegler
1195 2-(Benzoylimino)thiazolidin-4-ones Formation by an Alternative Ring Closure and Analysis of Rotational Barriers H-G Haumlcker P W Elsinghorst S Michels J Daniels G Schnakenburg M Guumltschow
1204 Microwave-Assisted Synthesis and Functionalization of Selenolopyrimidines S Hesse C Chenet D Thomae G Kirsch
1209 12-Disubstituted 4-Quinolones via Copper-Catalyzed Cyclization of 1-(2-Halophenyl)-2-en-3-amin-1-ones R Bernini S Cacchi G Fabrizi A Sferrazza
1220 A New Atom-Economical and Selective Synthesis of Secondary and Tertiary Alkylamines by Means of CpIridium Complex Catalyzed Multiple N-Alkylation of Ammonium Salts with Alcohols without Solvent R Yamaguchi Z Mingwen S Kawagoe C Asai K-i Fujita
1224 Synthesis of Regioisomerically Pure 5-Functionalized 27-Dichlorofluoresceins J C Castro A Malakhov K Burgess
XIII Forthcoming Articles
No 8 1227 Michael Additions to Activated Vinylphosphonates T Janecki J Kędzia
T Wąsek 1255 A Facile and General Synthesis of 2β-Aminosteroids X Ke H Hu
D Zhou W Xu Q Zhu N P Reddy X Hu 1261 Efficacious Preparation of Oppolzerrsquos Glycylsultam via the Deleacutepine
Reaction A Isleyen C Gonsky R C Ronald P Garner 1265 Synthesis of Masked Vicinal Amino Aldehydes of Pyrrolizine and Pyrrolo
[12-c]thiazole Series A V Tverdokhlebov A V Denisenko A A Tolmachev Y M Volovenko S V Shishkina O V Shishkin
1271 Preparation of 9-Substituted Pyridine-Stretched Adenines and Hypoxanthines J A Crawford W Fraser C A Ramsden
1279 A Versatile Synthesis of Heterocyclic Analogues of Neoflavonoids from Enamino Ketones V S Moskvina V P Khilya O V Turov U M Groth
1287 New Stereoselective Synthesis of Paeonilactone B F G Gatti S Serra 1291 The Use of NN-Dialkyltrimethylsilylamines in the Synthesis of
Pentamethinium Salts M Kořiacutenek M Rybaacutečkovaacute Boumlhm 1297 Synthesis of Triazoles via Regioselective Reactions of Aryl Azides with
Cyanoacetyl Pyrroles and Indoles N T Pokhodylo V S Matiychuk M D Obushak
1301 Gallium(III) Chloride Catalyzed Hydroarylation of Arylacetylenes with Naphthols and Phenols A Facile Synthesis of Vinylarenes J S Yadav B V S Reddy S Sengupta S K Biswas
1305 Electrophilic Bromination of meta-Substituted Anilines with N-Bromosuccinimide Regioselectivity and Solvent Effect S Bartoli A Cipollone A Squarcia A Madami D Fattori
1309 Cross-Coupling Reactions of Halopurines with Aryl- and Alkyltrifluoroborates The Scope and Limitations in the Synthesis of Modified Purines Z Hasniacutek R Pohl M Hocek
1318 A Convenient Method for Converting Hydroxyacetophenones into Their Ethylene or Trimethylene Acetals F Ono H Takenaka T Fujikawa M Mori T Sato
1323 γ-Chloromagnesio γ-Lactones and δ-Chloromagnesio δ-Lactones Generation Properties and Synthetic Uses H Shimizu S Fukuda S Sugiyama T Satoh
1336 Click Reactions with Nitroxides T Kaacutelai W L Hubbell K Hideg 1341 Synthesis of Novel 14-Benzoquinone-Containing 123-Triazoles An Entry
Into a New Library F Algi M Balci 1348 Efficient Synthesis of Two Sialylated Tetrasaccharides Found in Goat Milk
P K Mandal A K Misra 1355 Dendrimers of Vaccines Consisting of Tumor-Associated Glycopeptide
Antigens and T Cell Epitope Peptides S Keil A Kaiser F Syed H Kunz
1370 IBXTBAB-Mediated Oxidation of Primary Amines to Nitriles F Drouet P Fontaine G Masson J Zhu
1375 Chemoselectivity of Multicomponent Condensations of Barbituric Acids 5-Aminopyrazoles and Aldehydes E A Muravyova S V Shishkina V I Musatov I V Knyazeva O V Shishkin S M Desenko V A Chebanov
1386 Stereoselective Total Syntheses of Leiocarpin A and (ndash)-Galantinic Acid Starting from D-Mannitol K Nagaiah D Sreenu K V Purnima R S Rao J S Yadav
1393 A Facile Mild Deprotection Protocol for 13-Dithianes and 13-Dithiolanes with 30 Hydrogen Peroxide and Iodine Catalyst in Aqueous Micellar System N C Ganguly S K Barik
1400 Rhodium-Catalyzed Gram-Scale Synthesis of Highly Substituted Pyridine Derivatives K Parthasarathy C-H Cheng
1403 Enantioselective Synthesis of (R)-Propylene Carbonate from Ethyl (S)-Lactate J M Whitaker R C Ronald
XIII Forthcoming Articles
no 9 1405 Transition-Metal-Catalyzed Site-Selective Cross-Coupling of Di- and
Polyhalogenated Compounds J-R Wang K Manabe 1428 An Improved Synthesis of (4-4-Hydroxy-3-isopropyl-5-[(4-nitrophenyl)
ethynyl]benzyl-35-dimethylphenoxy)acetic Acid (NH-3) M B Gopinathan K S Rehder
1431 Copper-Catalyzed Tandem CndashN Bond Formation Reaction Selective Synthesis of 2-(Trifluoromethyl)benzimidazoles M-W Chen X-G Zhang P Zhong M-L Hu
1437 Synthesis and Thermochemical Properties of Stereoisomeric Dihydroxy- and Tetrahydroxyalkylammonium Salts M Thomas L Rothman J Hatcher P Agarkar R Ramkirath S Lall-Ramnarine R Engel
1445 Preparation of 5-Substituted 2-(2-Alkylaryl-1H-imidazol-4-yl)oxazoles and 5-Substituted 2-(2-Alkylarylthiazol-4-yl)oxazoles by Utilizing 5-Substituted 2-(2-Bromo-11-diethoxyethyl)oxazole as a Synthon D R St Laurent J L Romine
1459 Novel and Efficient Methods for the Synthesis of Symmetrical Trisulfides A Kertmen S Lach J Rachon D Witt
1463 An Environmentally Benign Electrochemical Process for the Reduction of Carboxylic Acid Hydrazides to Amides M Mentel M J Beier R Breinbauer
1469 Synthesis of 1-Chloroalkynes from Alkynylsilanes Using Trichloroisocyanuric Acid as Chlorinating Agent M H Vilhelmsen A S Andersson M B Nielsen
1473 A Convenient Approach to Enantioenriched Cyclopropanes Bearing Electron-Withdrawing Functionalities H Krawczyń K Wąsek J Kędzia
1477 Synthesis of Cyclopropenes via 12-Elimination of Bromocyclopropanes Catalyzed by Crown Ether W M Sherrill R Kim M Rubin
1485 A Base-Catalysed One-Pot Three-Component Coupling Reaction Leading to Nitrosubstituted Pyrroles I R Baxendale C D Buckle S V Ley L Tamborini
1494 Synthesis of 4-Alkylidene-4H-31-benzoxazine Derivatives by Acid-Catalyzed Cyclization of 2-Isocyanophenyl Ketones in the Presence of a Vinyl Ether K Kobayashi Y Okamura H Konishi
1499 Synthesis of Higher Helicenes via Olefin Metathesis and CndashH Activation J Cocircteacute S K Collins
1506 Azido- and Ethynyl-Substituted 2262-Terpyridines as Suitable Substrates for Click Reactions A Winter A Wild R Hoogenboom M W M Fijten M D Hager R-A Fallahpour U S Schubert
1513 Synthesis of 2-(Arylamino)ethanethiols via Lewis Acid Catalyzed Aminolysis of 22-Dimethylthiirane as Precursors of the 14-Benzothiazine Nucleus R Spogli S Sabatini G Manfroni O Tabarrini V Cecchetti
1520 Iron(III) Chloride A Versatile Catalyst for the Practical Synthesis of 3-Sulfenylindoles J S Yadav B V S Reddy Y J Reddy K Praneeth
1525 Organocatalytic Enantioselective Conjugate Addition of 2-Fluoromalonate to Nitroolefins Direct Synthesis of Chiral Fluorinated γ-Nitro Carboxylic Acid Derivatives H Li L Zu H Xie W Wang
1531 Asymmetric Transfer Hydrogenation of Ketimines with Trichlorosilane Structural Studies Z Zhang P Rooshenas H Hausmann P R Schreiner
1545 Prolinol Sulfinyl Ester Derivatives Organocatalytic Michael Addition of Ketones to Nitroolefins under Neat Conditions X Zeng G Zhong
1551 Asymmetric Oxidations of Electron-Poor Alkenes Promoted by the β-Amino AlcoholTBHP System A Russo A Lattanzi
1557 Enantioselectivity Switch in Direct Asymmetric Aminoxylation Catalyzed by Binaphthyl-Based Chiral Secondary Amines T Kano A Yamamoto F Shirozu K Maruoka
1564 Enantioselective Conjugate Addition of N-Heterocycles to αβ-Unsaturated Ketones Catalyzed by Chiral Primary Amines G Luo S Zhang W Duan W Wang
1573 Sulfonyl Hydrazine as New Functionality in Organocatalysis Camphorsulfonyl Hydrazine Catalyzed Enantioselective Aza-Michael Addition L-Y Chen H He B-J Pei W-H Chan A W M Lee
1578 Conversion of Primary Alcohols and Aldehydes into Methyl Esters by Ruthenium-Catalysed Hydrogen Transfer Reactions N A Owston T D Nixon A J Parker M K Whittlesey J M J Williams
1582 Addendum and Erratum XVII Forthcoming Articles
no 10 1583 Organocatalytic Formation of Quaternary Stereocenters M Bella
T Gasperi 1615 Regioselective Synthesis of 5H-Thiazolo[32-a]pyrimidin-5-ones from
MoritandashBaylisndashHillman Adduct Acetates under Solvent-Free and Base-Free Conditions W Zhong B Guo F Lin Y Liu W Su
1623 First Synthesis of 5-Cyanosalicylates by Formal [3+3] Cyclocondensations of 13-Bis(silyloxy)-13-butadienes A Riahi O Fatunsin M Shkoor R Dede H Reinke C Fischer P Langer
1635 Reaction of Isocyanides Dialkyl Acetylenedicarboxylates and a-Keto Lactones Unexpected Participation of an Ester Carbonyl Group in the Isocyanide-Based Three-Component Reaction A A Esmaeili H Vesalipoor
1639 An Efficient and Chemoselective Synthesis of 16-Naphthyridines and Pyrano[32-c]pyridines under Microwave Irradiation Z-G Han S-J Tu B Jiang S Yan X-H Zhang S-S Wu W-J Hao X-D Cao F Shi G Zhang N Ma
1647 N-Activation of N-Arylimidazoles Facile Syntheses of N-Alkyl-N-arylimidazolium Iodides from Less Expensive Chloro Substrates A M Oertel V Ritleng M J Chetcuti
1651 Synthesis of Polyhalogenated 2-(Phenylamino)pyridines by Thermal Amination Reactions S R Waldvogel A Faust W Barkmann R Froumlhlich O Wolff
1655 Cyanide Ion Promoted Addition of Acylphosphonates to Diethyl Cyanophosphonate Synthesis of Phosphonocyanohydrin O-Phosphates A S Demir A Aybey M Emrullahoglu
1659 Straightforward and Scalable Synthesis of Orthogonally Protected 37-Diazabicyclo[410]heptane H Schramm M Pavlova C Hoenke J Christoffers
1663 Hypervalent Iodine Mediated Oxidation of 12-Diaminobenzimidazole and Its Schiff Bases Efficient Synthesis of 3-Amino-124-benzotriazine and 2-Aryl-124-triazolo[15-a]benzimidazoles A Kumar M Parshad R K Gupta D Kumar
1667 Synthesis of the Reported Protoberberine Gusanlung D P B Wakchaure S Easwar N P Argade
1673 2-(Azidomethyl)arylboronic Acids in the Synthesis of Coumarin-Type Compounds M I Naumov A V Nuchev N S Sitnikov Y B Malysheva A S Shavyrin I P Beletskaya A E Gavryushin S Combes A Y Fedorov
1683 Asymmetric Synthesis of 12-anti-Disubstituted Taurine Derivatives D Enders D Iffland G Raabe
1689 A Novel One-Pot Three-Component Synthesis of 5-Imino-2358-tetrahydropyrazolo[12-a]pyridazin-1-one Derivatives B Qian M-J Fan Y-X Xie L-Y Wu Y Shi Y-M Liang
1694 One-Portion Synthesis of 2-Acetoxy Carbonyl Compounds from Aldehydes by Using an Acetylated Masked Acyl Cyanide H Nemoto T Kawamura K Kitasaki K Yatsuzuka M Kamiya Y Yoshioka
1703 Synthesis of 9-Anthryl Ethers from trans-910-Dihydro-910-dimethoxyanthracene by Acid-Catalyzed Transetherification K S Jang H Y Shin D Y Chi
1708 Efficient Synthesis of Azo Dye Labeled Terpenes Sugars and Steroids Using N-(4-Arylazobenzoyl)-1H-benzotriazoles A R Katritzky S R Tala N E Abo-Dya Z K Abdel-Samii
1715 Tandem CH-ActivationndashImine-Formation Reaction A New Route to Imidazo[21-a]phthalazines A Heim-Riether K R Gipson
1720 A Convenient and Efficient α-Sulfenylation of Carbonyl Compounds E Okragla S Demkowicz J Rachon D Witt
1725 Stereoselective Synthesis of β-Branched Phenylalanine Derivatives via Chelate-Claisen Rearrangement C Quirin U Kazmaier
1732 Catalyst-Free and Base-Free Water-Promoted SNAr Reaction of Heteroaryl Halides with Thiols B Sreedhar P S Reddy M A Reddy
1739 Convenient Methods for Synthesis of C2-Symmetric Diphenyltetrahydrothiophenes M Periasamy G Ramani G P Muthukumaragopal
1744 Highly Diastereoselective Conjugate AdditionndashElimination of Chiral Nickel(II) Glycinate with Activated Allylic Acetates for Asymmetric Synthesis of Glutamic Acid Derivatives J Wang J Shi X Zhang D Lin H Jiang H Liu
1753 Synthesis of 36-Dimethoxybenzene-12-diamine and of 47-Dimethoxy-2-methyl-1H-benzimidazole T Besset C Morin
1757 An Inexpensive Procedure for Reductive Aminations Using Dimethylamineborane on Millimolar and Molar Scale R Ortmann M Schlitzer
1760 Classics in Stereoselective Synthesis Edited by E M Carreira L Kvaerno Reviewed by Rolf Breinbauer
XV Forthcoming Articles
no 11 1761 Transition-Metal-Catalyzed Enantioselective Synthesis of Compounds with
Non-Centrochirality M Ogasawara S Watanabe 1786 One-Pot Synthesis of 3-Acyl-2-(alkylsulfanyl)indoles and 2-(Alkylsulfanyl)-
indole-3-carboxylates from (2-Isocyanophenyl)methyl Ketones or (2-Isocyanophenyl)acetates S Fukamachi H Konishi K Kobayashi
1791 Efficient and Recyclable Phthalocyanine-Based Sensitizers for Photooxygenation Reactions H Xu W-K Chan D K P Ng
1797 A Facile and Practical One-Pot Synthesis of β-Oxo Thioamides from β-Oxo Amides and Isothiocyanates P Huang D Xiang Y Zhou Y Liang T Na D Dong
1801 Microwave-Promoted Solid-Acid-Catalyzed One-Pot Synthesis of Phthalazinones V M Outerbridge S M Landge H Tamaki B Toumlroumlk
1807 Benzylic Brominations with N-Bromosuccinimide in (Trifluoromethyl)-benzene D Suarez G Laval S-M Tu D Jiang C L Robinson R Scott B T Golding
1811 Synthesis of Thioflavanone and Flavanone Derivatives by Cyclization of Chalcones W Konieczny M Konieczny
1815 A New and Expedient Total Synthesis of Ochratoxin A and d5-Ochratoxin A B Gabriele M Attya A Fazio L Di Donna P Plastina G Sindona
1821 Synthesis of Benzopyrrolizidinones by NorrishndashYang Cyclization of 3-(Acylmethyl)-2-alkylisoindol-1-ones J Wu W Zhang C Wang
1829 Reactions of MoritandashBaylisndashHillman Acetates with Huisgen Zwitterions A Novel Strategy for the Synthesis of β-Amino Acid Derivatives A Jose R R Paul R Mohan S C Mathew A T Biju E Suresh V Nair
1834 Peracetylated β-Allyl C-Glycosides of D-Ribofuranose and 2-Deoxy- D-ribofuranose in the Chemical Literature Until Now Mirages in the Literature H Otero Martinez H Reinke D Michalik C Vogel
1841 Core-Tetrasubstituted Naphthalene Diimides by Stille Cross-Coupling Reactions and Characterization of Their Optical and Redox Properties S-L Suraru F Wuumlrthner
1846 A Practical Synthesis of Indole-Based Heterocycles Using an Amidoaluminum-Mediated Strategy R Todd M M Hossain
1851 Synthesis of Fluorinated Pyrrolo[23-b]pyridine and Pyrrolo[23-d]pyrimidine Nucleosides V O Iaroshenko Y Wang D V Sevenard D M Volochnyuk
1858 Recyclization Reactions of 5-Formyl-13-dimethyluracil with Electron-Rich Amino Heterocycles A P Mityuk D M Volochnyuk S V Ryabukhin A S Plaskon A Shivanyuk A A Tolmachev
1865 Facile Synthesis of Fluorinated 1-Desazapurines V O Iaroshenko D V Sevenard D M Volochnyuk Y Wang A Martiloga A O Tolmachev
1876 A Practical Synthesis of 3-Diethoxyphosphoryl-12-pyridazine Derivatives J-C Monbaliu J Marchand-Brynaert
1881 Enantioselective Reduction of Prochiral Ketones Employing Sprouted Pisum sativa as Biocatalyst J S Yadav B V S Reddy C Sreelakshmi A B Rao
1886 Application of Phenolate Ion Mediated Intramolecular Epoxide Ring Opening in the Enantioselective Synthesis of Functionalized 23-Dihydrobenzofurans and 1-Benzopyrans S K Dinda S K Das G Panda
1897 Complementary Synthetic Approaches to Constitutionally Diverse N-Aminoalkylated Isoindolinones Application to the Synthesis of Falipamil and 5-HT1A Receptor Ligand Analogues M Lorion A Couture E Deniau P Grandclaudon
1904 Selective Deprotection of Silyl Ethers with Sodium Periodate J Li D Menche
1909 Micellar Solution of Sodium Dodecyl Sulfate (SDS) Catalyzes KabacknikndashFields Reaction in Aqueous Media S Sobhani A Vafaee
1916 Convenient Methods for the Synthesis of a Library of Hemilabile Phosphines M V Jimeacutenez J J Peacuterez-Torrente M I Bartolomeacute L A Oro
1923 Terminal Aziridines by Addition of Grignard Reagents or Organoceriums to an (α-Chloro)sulfinylimine D M Hodgson J Kloesges B Evans
1933 A Robust Synthesis of Nε-(Carboxymethyl)-L-lysine (CML) R Csuk S Stark A Barthel R Kluge D Stroumlhl
1935 One-Pot Curtius Rearrangement Processes from Carboxylic Acids O Leogane H Lebel
XV Forthcoming Articles
no 12 1941 The Chemistry of Deprotonated α-Aminonitriles T Opatz 1960 An Efficient Synthesis of Tetraalkyl 2345-Thiophenetetracarboxylate
Derivatives A Alizadeh R Hosseinpour 1963 Facile Deprotection of Bulky (Trialkylsilyl)acetylenes with Silver Fluoride
S Kim B Kim J In 1969 Highly Efficient and Reusable Ionic Liquids for the Catalyzed
Hydroamination of Alkenes with Sulfonamides Carbamates and Carboxamides L Yang L-W Xu C-G Xia
1975 Synthesis of 2391016172324-Octasubstituted Phthalocyaninatozinc(II) Complexes Mediated by Reductive Agents G A Gauna A C Monsalvo J Awruch
1979 A Short and Efficient Synthesis of 3-2-[2-(Bromomethyl)thiazol-4-yl]-ethynyl-5-fluorobenzonitrile A Precursor for PET Radioligand [18F]SP203 M B Gopinathan C Jin K S Rehder
1983 Synthesis of a Substituted Benzazepin-2-one Dihydrate S K Boini R K Vaid K P Moder D Mitchell
1987 Synthesis of Novel Trisubstituted Imidazolines F J Lakner M A Parker B Rogovoy A Khvat A Ivachtchenko
1991 A Novel Synthesis of N-But-3-enyl-α- and β-Amino Acids T T Van Nguyen R T C Brownlee A B Hughes
1999 Synthesis of Substituted 5-(3-Hydroxypropyl)pyrrolidin-2-ones and Pyrrolizidinones from Nitroethane via C3 Functionalized 56-Dihydro-4H-12-oxazines A Novel Approach to Some Analogues of the Antidepressant Rolipram A Yu Sukhorukov A V Lesiv Y A Khomutova S L Ioffe V A Tartakovsky
2009 Chiral Cyclobutanols and Cyclopentane Dimers via Samarium(II) Iodide Induced Keto-Olefin Cyclisations of Carbohydrate-Derived Unsaturated Ketones D B G Williams J Caddy K Blann J J C Groveacute C W Holzapfel
2015 Synthesis of Perfluoroalkylthio-Substituted Ferrocenes C Rhode J Lemke M Lieb N Metzler-Nolte
2019 Functionalization of Polyhedral Oligomeric Silsesquioxane (POSS) via Nucleophilic Substitution M Dutkiewicz H Maciejewski B Marciniec
2025 A Novel Synthesis of Aryl Mesylates via One-Pot DemethylationndashMesylation of Aryl Methyl Ethers Using a Mixture of Phosphorus Pentoxide in Methanesulfonic Acid B Kaboudin Y Abedi
2029 Anionic Cyclization of (NN-Dimethylamino)[2-(prop-2-yn-1-yloxy)aryl]-acetonitriles T Zdrojewski J Musielak A Jończyk
2035 Strecker-Type Reaction Catalyzed by Carboxylic Acids in Aqueous Media Z Xie G Li G Zhao J Wang
2040 Synthesis of Novel Structurally Simplified Estrogen Analogues with Electron-Donating Groups in Ring A L F Tietze C A Vock I K Krimmelbein L Nacke
2061 On the Resolution of Secondary Phosphine Oxides via Diastereomeric Complex Formation The Case of tert-Butylphenylphosphine Oxide J Holt A M Maj E P Schudde K M Pietrusiewicz L Sieroń W Wieczorek T Jerphagnon I W C E Arends U Hanefeld A J Minnaard
2066 Enantioselective Copper-Catalyzed Conjugate Addition of Dimethylzinc to 5-(1-Arylalkylidene) Meldrumrsquos Acids A Wilsily T Lou E Fillion
2073 SuzukindashMiyaura Coupling Reactions Using Phosphite Ligands M Jang Y Jo I-K Oh H M Jung S Lee
2076 Synthesis of 2-Methylindoline- and 2-Methyl-1234-tetrahydroquinoline-Derived Phosphoramidites and Their Applications in Iridium-Catalyzed Allylic Alkylation of Indoles W-B Liu H He L-X Dai S-L You
2083 Stereocontrolled Synthesis of 13-Amino Alcohols by Reduction of Substituted 2-1-[(tert-Butylsulfinyl)amino]alkylcyclohexanones J C Gonzaacutelez-Goacutemez F Foubelo M Yus
2089 Tunable Phosphoramidite Ligands for Asymmetric Hydrovinylation Ligands par excellence for Generation of All-Carbon Quaternary Centers C R Smith H J Lim A ZhangT V RajanBabu
2101 Copper-Catalyzed Asymmetric Ring-Opening Reaction of Oxabenzonorbornadienes with Grignard and Aluminum Reagents R Millet L Gremaud T Bernardez L Palais A Alexakis
2113 A Simplified Synthesis of Takemotorsquos Catalyst A Berkessel B Seelig 2116 Pharmaceutical Substances Syntheses Patents and Applications of the
Most Relevant AIPs Edited by Axel Kleeman Juumlrgen Engel Bernhard Kutscher Dietmar Reichert Reviewed by I Agranat
XV Forthcoming Articles
no 13 2117 Recent Advances in the Aza-Claisen Rearrangement K C Majumdar
T Bhattacharyya B Chattopadhyay B Sinha 2143 A Novel and Convenient Synthesis of lsquoReversedrsquo Diamidino 25-Aryl- and
25-Azaheterocycle-Substituted Furans L Hu D W Boykin 2146 Efficient and General Preparation of Pyranostilbenes First Total Synthesis
of Artocarbene and Pawhuskin B B H Park Y R Lee W S Lyoo 2155 Mild Oxidation of Diarylacetylenes to 12-Diketones Using Oxone in
Trifluoroacetic Acid J-H Chu Y-J Chen M-J Wu 2163 One-Pot Microwave-Assisted Selective Azido ReductionTandem Cyclization
in Condensed and Solid Phase with Nickel Boride N Shankaraiah N Markandeya M Espinoza-Moraga C Arancibia A Kamal L Silva Santos
2171 Pyrrolo[321-ij]quinolin-4-one and Pyrrolo[321-ij]quinolin-6-one H McNab D J Nelson E J Rozgowska
2175 Practical Synthesis of 5-Substituted Tetrazoles under Microwave Irradiation J Roh T V Artamonova K Vaacutevrovaacute G I Koldobskii A Hrabaacutelek
2179 A Simple Method for the Synthesis of 3-Arylthieno[23-b]pyridines via Iodine-Mediated Cyclization of 3-(1-Arylalkenyl)-2-[(1-phenylethyl)sulfanyl]pyridines K Kobayashi D Nakamura Y Shiroyama S Fukamachi H Konishi
2184 Synthesis of Four Lysine-Linked Cereulide Analogues Showing Ionophoric Activity Towards Potassium Cations as Lead Compounds for Emetic Toxin-Detection by Immunoassays A Makarasen T Nishikawa M Isobe
2205 Synthesis of α-Aliphatic and β-Aromatic Substituted Taurines via Regioselective Ring Opening of Thiiranes with Ammonia H Yu S Cao L Zhang G Liu J Xu
2210 Stability of 5(6)-Carboxyfluorescein in Microwave-Assisted Synthesis of Fluorescein-Labelled O-Dimannosylated Peptides R Kowalczyk P W R Harris R P Dunbar M A Brimble
2223 Diversity-Oriented Synthesis of Functionalized Diaryl Sulfones by Regioselective [3+3] Cyclizations of 13-Bis(siloxy)buta-13-dienes with 2-(Arylsulfonyl)-3-ethoxy-2-en-1-ones Scope and Limitations M Shkoor A Riahi O Fatunsin H Reinke C Fischer P Langer
2236 Synthesis of Functionalized Salicylates by Formal [3+3] Cyclocondensation of 13-Bis(silyloxy)buta-13-dienes with 3-Alkoxy-2-en-1-ones G Mroszlig S Ladzik H Reinke A Spannenberg C Fischer P Langer
2249 Synthetic Approach to Alkoxy-β-(trifluoromethyl)styrenes and Their Application in the Synthesis of New Trifluoromethylated Heterocycles V M Muzalevskiy V G Nenajdenko A V Shastin E S Balenkova G Haufe
2260 o-Benzenedisulfonimide as a Powerful and Recyclable Organocatalyst for the Nazarov Reaction M Barbero S Cadamuro A Deagostino S Dughera P Larini E G Occhiato C Prandi S Tabasso R Vulcano P Venturello
2267 The Catalytic Potential of 4-Guanidinylpyridines in Acylation Reactions I Held E Larionov C Bozler F Wagner H Zipse
2278 Iron(III) Chloride in EthanolndashWater Highly Efficient Catalytic System for the Synthesis of Garcia Gonzalez Polyhydroxyalkyl- and C-Glycosylfurans L Nagarapu M V Chary A Satyender B Supriya R Bantu
2283 Ruthenium-Catalyzed Addition of Primary Amides to Alkynes A Stereoselective Synthesis of Secondary Enamides L J Gooszligen M Blanchot K S M Salih K Gooszligen
2289 Binaphthyl-Modified Quaternary Phosphonium Salts as Chiral Phase Transfer Catalysts Application to Asymmetric Amination of β-Keto Esters R He K Maruoka
X Table of Contents XI Forthcoming Articles
no 14 2293 Direct Methods for Stereoselective Polypropionate Synthesis A Survey
J Li D Menche 2316 Synthesis of Symmetrical Ketones from Grignard Reagents and
11-Carbonyldiimidazole D Bottalico V Fiandanese G Marchese A Punzi
2319 Synthesis of 45-Substituted Imidazoles by a Fast Condensation of 12-Diketones and Urotropine in Heterogeneous Medium G Bratulescu
2321 (Arylsulfonyl)acetones and -acetonitriles New Activated Methylenic Building Blocks for Synthesis of 123-Triazoles N T Pokhodylo V S Matiychuk M D Obushak
2324 A Safe Convenient and Efficient One-Pot Synthesis of α-Chloroketone Acetals Directly from Ketones Using Iodobenzene Dichloride J Yu C Zhang
2329 An Efficient Oxidative Conversion of Aldehydes into 2-Substituted 2-Oxazolines Using 13-Diiodo-55-dimethylhydantoin S Takahashi H Togo
2333 A Novel Procedure for the Synthesis of Benzo[b][18]naphthyridine-3-carboxylate Derivatives from MoritandashBaylisndashHillman Adduct Acetates W Zhong F Lin R Chen W Su
2341 An Improved Synthesis of 147-Triazacyclononanes (tacns) and 14710-Tetraazacyclododecanes (cyclens) J Huang Z Zhou T H Chan
2345 The Ullmann Coupling between 2-Chlorobenzoic Acids and Amino Acids A Valuable Reaction for Preparing 2-Substituted 1-Acetyl-1H-indol-3-yl Acetates J C Rodriguez Dominguez X Gang G Kirsch
2349 gem-Dibromomethyl Aromatics Efficient Aldehyde Equivalents in the KnoevenagelndashDoebner Reaction J K Augustine Y A Naik S Poojari N Chowdappa B S Sherigara K Areppa
2357 Synthesis of Novel α-Aminophosphonates Containing Adamantyl Fragment M M Kabachnik L I Minaeva I P Beletskaya
2361 Efficient Fluoride-Mediated Synthesis of 5-Amino-Substituted Isothiazoles Y S Zubenko V I Potkin
2365 Phosphine-Catalyzed Reaction of Cyanohydrins with Activated Alkynes A Siby O Loreau F Taran
2371 Sulfanyl-Substituted [3]Cumulenes and Buta-13-dienes from a Tetrakis(pyridinium)-Substituted Butadiene A Schmidt A Rahimi M Gjikaj
2379 Efficient Synthesis of 2-Substituted Pyrido[32-d]pyrimidines Involving SNAr and Palladium-Catalyzed Cross-Coupling Reactions A Tikad S Routier M Akssira J-M Leacuteger C Jarry G Guillaumet
2385 Novel Synthesis of Medium-Sized Heterocycles by Palladium-Catalyzed Intramolecular Heck Reaction via 9-endo-trig Mode of Cyclization K C Majumdar B Chattopadhyay
2393 Facile Synthesis of Fluorinated Benzofuro- and Benzothieno[23-b]pyridines α-Carbolines and Nucleosides Containing the α-Carboline Framework V O Iaroshenko Y Wang B Zhang D Volochnyuk V Ya Sosnovskikh
2403 Synthesis of Functionalized N-Vinyl Nitrogen-Containing Heterocycles S M M Lopes A M Beja M Ramos Silva J A Paixatildeo F Palacios T M V D Pinho e Melo
2408 Kumada Cross-Coupling of Aryl Grignard Reagents with Aryl Halides Catalyzed by an Immobilized Nickel Catalyst X Chen L Wang J Liu
2413 Highly Enantioselective Synthesis of Heteroaromatic Alcohols Catalyzed by Chiral DiaminodiphosphinendashRuthenium(II) Complexes W-Y Shen Y-Y Li Z-R Dong J-X Gao
2418 Concise Total Synthesis of (+)-Disparlure and its trans-Isomer Using Asymmetric Organocatalysis S-G Kim
2423 Rhodium Carbenoid Induced [12]-Migration in an L-Lyxo-Configured α-Diazo β-Keto Ester Synthesis of a New Griseolic Acid Analogue N N Bhujbal K S A Kumar D D Dhavale
2430 Synthesis of 5-Arylthio-3-hydroxyphthalates by the First [4+2] Cycloadditions of 3-Arylthio-1-silyloxy-13-butadienes with Dimethyl Acetylenedicarboxylate I Iqbal M Imran P Langer
2435 Synthesis of Highly Functionalized Proline Derivatives via a One-Pot MichaelSN-AdditionCyclization Approach U Kazmaier C Schmidt
2440 RhodiumGraphite-Catalyzed Hydrogenation of Carbocyclic and Heterocyclic Aromatic Compounds G Falini A Gualandi D Savoia
2447 Potassium [1-(tert-Butoxycarbonyl)-1H-indol-2-yl]trifluoroborate as an Efficient Building Block in Palladium-Catalyzed SuzukindashMiyaura Cross Couplings P Kassis V Beacuteneacuteteau J-Y Meacuterour S Routier
2454 Syntheses of Substituted Furans and Pyrroles by Platinum-Catalyzed Cyclizations of Propargylic Oxiranes and Aziridines in Aqueous Media M Yoshida M Al-Amin K Shishido
2467 Transition-Metal-Free Oxidative Homocoupling of Aryl Alkenyl and Alkynyl Grignard Reagents with TEMPO M S Maji A Studer
XIII Forthcoming Articles
no 15 2471 Advances in Synthetic Approaches for the Preparation of Combretastatin-
Based Anti-Cancer Agents R Singh H Kaur 2492 Synthesis of Unsymmetrical Ureas by Sulfur-Assisted Carbonylation with
Carbon Monoxide and Oxidation with Molecular Oxygen under Mild Conditions T Mizuno T Nakai M Mihara
2497 Ring-OpeningRecyclization Reactions of (Dimethylamino)propenoyl-Substituted Cyclopropanes Facile Synthesis of Halogenated Pyridin-2(1H)-ones R Zhang Y Zhou Y Liang Z Jiang D Dong
2501 Facile and Efficient Total Synthesis of Taspine B Cheng S Zhang L Zhu J Zhang Q Li A Shan L He
2505 Oligomeric Iodosylbenzene Sulfate A Convenient Hypervalent Iodine Reagent for Oxidation of Organic Sulfides and Alkenes M S Yusubov R Y Yusubova T V Funk K-W Chi V V Zhdankin
2509 Pyrrolidine-Based Organocatalysts for Enantioselective Michael Addition of Cyclohexanone to trans-β-Nitrostyrene A P Carley S Dixon J D Kilburn
2517 CundashAl Hydrotalcite An Efficient and Reusable Ligand-Free Catalyst for the Coupling of Aryl Chlorides with Aliphatic Aromatic and N(H)-Heterocyclic Amines B Sreedhar R Arundhathi P L Reddy M A Reddy M L Kantam
2523 Highly Efficient Synthesis of trans-βγ-Unsaturated a-Keto Amides C Allais T Constantieux J Rodriguez
2531 Gas-Phase Synthesis of N-Unsubstituted 3-Hydroxypyrroles and 1H-Pyrrol-3(2H)-ones L Hill G A Hunter S H Imam H McNab W J OrsquoNeill
2535 3-Hydroxy-1H-pyrrole L Hill S H Imam H McNab W J OrsquoNeill 2539 123-Thiadiazoles with Unsaturated Side Chains Synthesis
Polymerization and Photocrosslinking M Al-Smadi N Hanold H Kalbitz H Meier
2547 Synthesis of 1112-Didehydrodibenzo[ae]cycloocten-5(6H)-one A Strained Eight-Membered Alkyne S C Kornmayer F Rominger R Gleiter
2553 Stannous Chloride Dihydrate A Novel and Efficient Catalyst for the Synthesis of gem-Dihydroperoxides from Ketones and Aldehydes D Azarifar K Khosravi F Soleimanei
2557 Synthesis of a Novel Class of Azacrown Macrocycles and Lariat Crown Ethers Containing Two 124-Triazole Rings as Subunits N Foroughifar A Mobinikhaledi S Ebrahimi
2561 Enantioselective Synthesis of the 3C-Protease Inhibitor (ndash)-Thysanone by a StauntonndashWeinreb Annulation Strategy J Sperry T Y Yuen M A Brimble
2570 Stereoselective Synthesis of Unnatural β-Amino Acids from Nitroethane via 56-Dihydro-4H-12-oxazin-3-ylacetates A Yu Sukhorukov A V Lesiv O L Eliseev Y A Khomutova S L Ioffe
2579 A Versatile Unexpected One-Pot Regioselective Synthesis of a New Class of 13-Diazepinoindolones by Reaction of Pyranoindolones with Monosubstituted Ureas D Livadiotou C A Tsoleridis J Stephanidou-Stephanatou
2584 Synthesis of a Trisaccharide and a Tetrasaccharide from the Cell-Wall Lipopolysaccharides of Azospirillum brasilense S17 S Pandey S Ghosh A K Misra
2591 Synthesis of Isoindoline Nitroxides by Electrocyclic Reactions T Kaacutelai J Jekı K Hideg
2596 Glycosylations of Tertiary Alcohols Synthesis of Fully Protected Disaccharides with Sterically Demanding Groups Attached to the Sugar Core A Holkenbrink J B Vicente D B Werz
2605 Copper-Catalyzed [13]-Dipolar Cycloaddition for the Synthesis of Macrocycles Containing Acyclic Aromatic and Steroidal Moieties G V Latyshev M S Baranom A V Kazantsev A D Averin N V Lukashev I P Beletskaya
2616 Aryl Ring Migration Reaction in the Synthesis of 24-Diaryl-4H-31-benzothiazines A V Butin F A Tsiunchik V T Abaev A V Gutnov D A Cheshkov
2627 Hydrogenation of β-N-Substituted and β-NN-Disubstituted Enamino Esters in the Presence of Iridium(I) Catalyst H Hebbache Z Hank C Bruneau J-L Renaud
2634 Stereoselective Olefination Reactions Promoted by Rieke Manganese J M Concelloacuten H Rodriacuteguez-Solla V del Amo P Diacuteaz
2646 Synthesis of Piperidinones through a Radical Cascade E Godineau Y Landais
2650 Asymmetric Organic Synthesis with Enzymes Edited by V Gotor I Alfonso E Garciacutea-Urdiales Reviewed by Steve Collier
XVII Forthcoming Articles
no 16 2651 Synthesis of Spirocyclic Ethers S Rosenberg R Leino 2674 Bimetallic PalladiumndashPlatinum-on-Carbon-Catalyzed HndashD Exchange
Reaction Synergistic Effect on Multiple Deuterium Incorporation T Maegawa N Ito K Oono Y Monguchi H Sajiki
2679 Efficient Copper-Catalyzed Synthesis of 2-Amino-4(3H)-quinazolinone and 2-Aminoquinazoline Derivatives X Huang H Yang H Fu R Qiao Y Zhao
2689 Synthesis and Chemoselective N- and O-Alkylation of Thiadiazolopyrimidine Nucleosides and Uridines A M L Hossion R Islam R K Kandahary T Nagamatsu
2697 Facile and Efficient Synthesis of a New Class of Indole-Substituted Pyridine Derivatives via One-Pot Multicomponent Reactions K Zhao X-P Xu S-L Zhu D-Q Shi Y Zhang S-J Ji
2709 Studies toward a Total Synthesis of Rhizoxin D Stereoselective Preparation of the C11ndashC19 Fragment S Padakanti C K Kumar E Ashok P Das
2715 A Short Synthesis of Enantiomeric Phytoprostanes B1 Type I W Perlikowska M Mikołajczyk
2719 Chemistry of Polyhalogenated Nitrobutadienes Part 7 A Novel Synthetic Access to Chlorinated Nitrile Oxides E Nutz V A Zapolrsquoskii D E Kaufmann
2725 Microwave-Assisted Silver(I)-Mediated Selective O-Alkylation of Aromatic Imidate Systems B K Singh C Cavalluzzo M De Maeyer Z Debyser V S Parmar E Van der Eycken
2729 Iodogen A Novel Reagent for the Oxidation of Urazoles under Heterogeneous Conditions A Khoramabadi A Shiri M A Zolfigol S Mallakpour
2733 An Unprecedented Synthesis of Eight-Membered-Ring Cyclic Thioimidic Esters by a Three-Component Reaction A Alizadeh R Hosseinpour
2737 A Novel Diastereoselective Synthesis of β-Phosphonato Unsaturated Thioimidates A Alizadeh N Zohreh
2741 Synthesis of 21-Benzisoxazoles by Nucleophilic Substitution of Hydrogen in Nitroarenes Activated by the Azole Ring N T Pokhodylo Y O Teslenko V S Matiychuk M D Obushak
2749 A Facile Synthesis of Two Series of Multifunctional Carbon Compounds from αα-Dihalo Ketones Using Allylsamarium Bromide X Liu S Zhang J Di
2756 Stereocontrolled Formation of Protected Aminodeoxyalditols from Simple Carbohydrate Precursors by Debenzylating Cycloetherification Y Jiang Z Fang Q Zheng H Jia J Cheng B Zheng
2761 trans-Stilbene as a Starting Material for the Synthesis of Tamoxifen Based on Palladium-Catalyzed Cross-Coupling Reactions C M Nunes J Limberger S Poersch M Seferin A L Monteiro
2766 Synthesis and Biological Evaluation of 6-Substituted Purinylcarbanucleosides with a Cyclopenta[b]thiophene Pseudosugar P Abeijoacuten J M Blanco O Caamantildeo F Fernaacutendez M D Garciacutea X Garciacutea-Mera J E Rodriacuteguez-Borges J Balzarini E De Clercq
2773 Synthesis and Electrochemical Signature of Novel Norbornyl-ferrocene Hybrids F A Khan S K Upadhyay
2778 A Regioselective TsujindashTrost Pentadienylation of 3-Allyltetronic Acid R Schobert B Barnickel
2785 Copper(I)-Catalyzed CarylndashCalkynyl Bond Formation of Aryl Iodides with Terminal Alkynes K G Thakur G Sekar
2790 Aminolysis of Epoxides Using Iridium Trichloride as an Efficient Catalyst J Agarwal A Duley R Rani R K Peddinti
2797 Preparation of Several Active N-Chloro Compounds from Trichloroisocyanuric Acid A Shiri A Khoramabadi-zad
2802 The First Mineral-Catalyzed One-Pot [3+1+2] Coupling Protocol for Multifunctionalized Fused-Ring Pyrimidines L D S Yadav A Rai
2809 Efficient Synthesis of Tetrahydro-β-carbolin-1-one and Dihydroisoquinolin-1-one Derivatives as Versatile Intermediates K E Judd M F Mahon L Caggiano
2818 A Concise Synthesis of ortho-Iodobenzyl Alcohols via Addition of ortho-Iodophenyl Grignard Reagent to Aldehydes and Ketones J Cvengroš D Stolz A Togni
XIII Forthcoming Articles
no 17 2825 Reactivity of Oxazol-5-(4H)-ones and Their Application toward Natural
Product Synthesis N M Hewlett C D Hupp J J Tepe 2840 Towards the Total Synthesis of 3-Hydroxyvibsanin E B D Schwartz
J R Denton P V Bernhardt H M L Davies C M Williams 2847 Structure Investigations of (ent)-Cladospolide D by De Novo Synthesis and
Kinetic and Thermodynamic Isomerization Y Xing J H Penn G A OrsquoDoherty
2855 New Applications of PhI(OAc)2 in Synthesis Total Synthesis and SAR Development of Potent Antitumor Natural Product PsymberinIrciniastatin A N Shao X Huang A Palani R Aslanian A Buevich J Piwinski R Huryk C Seidel-Dugan
2873 Total Synthesis of Largazole ndash Devolution of a Novel Synthetic Strategy B Wang C J Forsyth
2881 Formal Total Synthesis of Palmerolide A J Jaumlgel M E Maier 2893 Total Synthesis of Bongkrekic Acid via Sequential SuzukindashMiyaura Coupling
Reactions M Kanematsu M Shindo M Yoshida K Shishido 2905 Stereodivergent Approach to Both C28a-syn and C28a-anti Relative
Stereochemical Manifolds in the Lepadin Family via a TiCl4-Promoted G Li L J Carlson I K Sagamanova B W Slafer R P Hsung C Gilardi H M Sklenicka N Sydorenko
2915 Enantioselective Aldol Reaction of Tetrasubstituted Ketene Silyl Acetals with Achiral Aldehydes for the Construction of Asymmetric Tertiary Alcohols An Application for the Divergent Total Syntheses of Buergerinins F and G I Shiina T Iizumi Y-s Yamai Y-i Kawakita K Yokoyama Y-k Yamada
2927 Second-Generation Biomimetic Total Synthesis of Chaetominine A Coste G Karthikeyan F Couty G Evano
2935 Total Synthesis of (+)-Fostriecin and (+)-Phoslactomycin B S Shibahara M Fujino Y Tashiro N Okamoto T Esumi K Takahashi J Ishihara S Hatakeyama
2954 Stereochemical Assignments of the Chlorinated Residues in Victorin C A C Durow C Butts C L Willis
2963 Studies of the Asymmetric Total Synthesis of Clavilactone D by the lsquoLariatrsquo Cyclization Strategy T Yoshimitsu S Nojima M Hashimoto K Tsukamoto T Tanaka
2970 Total Synthesis of the Leucetta-Derived Alkaloid Calcaridine A P B Koswatta R Sivappa H V R Dias C J Lovely
2983 Formal Synthesis of Salinosporamide A Starting from D-Glucose T Momose Y Kaiya J-i Hasegawa T Sato N Chida
2992 Synthesis of Bioactive Natural Products by Asymmetric syn- and anti-Aldol Reactions A K Ghosh Z L Dawson
no 18 3003 Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural
Products B M Trost M K Brennan 3026 One-Pot Synthesis of Furo[34-b]pyridin-5(7H)-ones from 2-
Bromopyridine-3-carboxylic Acid and Carbonyl Compounds K Kobayashi T Kozuki H Konishi
3029 Iodocyclization of N-[2-(Methylthio)phenyl]propiolamides Selective Synthesis of 3-Iodo-15-benzothiazepin-4-ones T-S Jiang X-G Zhang J-H Li
3039 A Facile Synthetic Method for Fluorine-Containing 17-Phenanthrolines Pyridine-Ring Formation Reaction of N-Propargyl-68-bis(trifluoroacetyl)-quinolin-5-amine with Various Nucleophiles D Shibata E Okada M Hinoshita M Meacutedebielle
3047 Enantiotopic Discrimination in Palladium-Mediated Nucleophilic Substitutions on Achiral Substrates Chiral Ligand versus Chiral Nucleophile O Jacquet F Charnay J-C Fiaud J Ollivier
3051 Studies on the Chemistry of 2-[3-(2-Nitrophenyl)-2-oxopropyl]benzaldehydes Novel Syntheses of 5H-Benzo[b]carbazole-611-diones and Indolo[12-b]isoquinoline-611-diones M Fernaacutendez
3061 Studies on the C22ndashC23 Aldol Coupling of Spirangien M Lorenz N Bluhm M Kalesse
3067 One-Pot Synthesis of N-Alkyl Purine Pyrimidine and Azole Derivatives from Alcohols using Ph3PCCl4 A Rapid Route to Carboacyclic Nucleoside Synthesis M N Soltani Rad A Khalafi-Nezhad S Behrouz Z Asrari M Behrouz Z Amini
3077 Synthesis of 2-Amino-34-dihydroquinazolines and Imidazo[21-b]quinazoline-2-ones A Mishra S Batra
3089 Studies on the Reaction of Diimines with Thiourea Synthesis and Solvent-Induced cistrans-Isomerization of 135-Triazinane-2-thiones B Kaboudin T Ghasemi T Yokomatsu
3094 Suzuki Coupling of Heteroaromatic Chlorides Using Highly Electron-Donating ClickPhos Ligands S M Spinella Z-H Guan J Chen X Zhang
3099 Reaction of NN-Dioxyenamines with Anhydrides of Carboxylic and Sulfonic Acids A New Method for the Synthesis of a-Hydroxyoxime Derivatives A A Tabolin A V Lesiv S L Ioffe
3106 Directed ortho Metallation Chemistry and Phosphine Synthesis New Ligands for the SuzukindashMiyaura Reaction D B G Williams S J Evans H de Bod M S Mokhadinyana T Hughes
3113 New Functional Derivatives of 9-Phenylquinine P J Boratyński J SkarŜewski
3120 On the Synthesis of Asymmetric and Dissymmetric Amino Analogues of Troumlgerrsquos Base J Artacho K Waumlrnmark
3127 Synthesis of Polycyclic Sultams by Palladium-Catalyzed Intramolecular Cyclization K C Majumdar S Mondal N De
3136 Synthesis of Functionalized L-Cysteine and L-Methionine by Reaction with Electron-Deficient Acetylenes B A Trofimov A G Malrsquokina O A Shemyakina V V Nosyreva A P Borisova S S Khutsishvili L B Krivdin
3143 A lsquoClickrsquo Approach to the Synthesis of 3-[2-(1-Alkyltriazol-4-yl)ethyl]indoles M Petrini R R Shaikh
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
483 Efficient Catalytic Activity of CopperAluminum Hydrotalcite in Diaryl Ether Synthesis B Sreedhar R Arundhathi M A Reddy M L Kanatm
488 On-Resin Click-Glycoconjugation of Peptoids A S Norgren C Budke Z Majer C Heggemann T Koop N Sewald
495 A Simple and Efficient Preparation of Novel Formaldehyde Derivatives R Hartung G Golz S Schlaf G Silvennoinen K Polborn P Mayer H R Pfaendler
502 2-Oxazol-5-ylethanones by Consecutive Three-Component AmidationndashCouplingndashCycloisomerization (ACCI) Sequence E Merkul O Grotkopp T J J Muumlller
508 SuzukindashMiyaura Cross-Couplings Mediated by trans-PdBr(N-Succ)(PPh3)2 A Convenient Synthetic Method for Diarylmethanes and Aryl(heteroaryl)-methanes I J S Fairlamb P Sehnal R J K Taylor
511 Modern Reduction Methods Edited by P G Andersson and I J Munslow Reviewed by Siegfried R Waldvogel
512 Addendum and Erratum XIII Forthcoming Articles
No 4 513 Intermolecular Addition Reactions of N-Acyliminium Ions (Part II)
A Yazici S G Pyne 542 A Simple Practical Method for the Synthesis of 46-Dimethoxy-135-
triazin-2(1H)-one Using Dimethylamine-Functionalized Solid-Phase Reagents K Hioki K Ohshima Y Sota M Tanaka M Kunishima
545 Conjugation-Amenable Tetrasaccharide of the Side Chain of the Major Glycoprotein of the Bacillus anthracis Exosporium A Large-Scale Preparation S Hou P Kovaacuteč
551 Reductive Amination ndash A Convenient Method for Generating Diverse Mono-Functionalised 5101520-Tetraphenyl Porphyrins C Welch S J Archibald R W Boyle
557 Highly Regioselective Preparation of 13-Dioxolane-4-methanol Derivatives from Glycerol Using Phosphomolybdic Acid N W Fadnavis R Gowrisankar G Ramakrishna M K Mishra G Sheelu
561 Rapid Synthesis of 3-Aminoisoquinoline-5-sulfonamides Using the BuchwaldndashHartwig Reaction N Proisy S Taylor A Nelson I Collins
567 Synthesis of Divalent 22-Linked Mannose Derivatives by Homodimerization F S Ekholm M Polaacutekovaacute A J Pawłowicz R Leino
577 Efficient Synthesis of Substituted Cyclic α-Aminophosphonates I L Odinets O I Artyushin N Shevchenko P V Petrovskii V G Nenajdenko G-V Roumlschenthaler
583 Methylated Imidazolinium-Dithiocarboxylates Two Representatives of a New Class of Ionic Liquids A Blanrue R Wilhelm
587 An Efficient Route to 1-Vinylpyrrole-2-carbaldehydes A I Mikhaleva A V Ivanov E V Skitalrsquotseva I A Ushakov A M Vasilrsquotsov B A Trofimov
591 A Regioselective Route to 5-Substituted Isoxazole- and Isoxazoline-3-phosphonates P Conti A Pinto L Tamborini P Dunkel V Gambaro G L Visconti C De Micheli
597 Solvent-Free One-Pot Conjugate Addition of Benzyl Bromides to β-Nitroalkenes Mediated by Magnesium Powder W Shi J-X Wang
602 Synthesis of 234-Trideoxy-44-difluoro-D-ribo-hexopyranose Adenosines J Xu X Zhang X-L Qiu F-L Qing
609 Synthesis of anti-27-Disubstituted Norbornadienes G C Tsui P Le Marquand A Allen W Tam
620 Novel Peptide Mimetic Inhibitors of Hepatitis C Serine Protease Derived from Isomannide T G Barros S Pinheiro J S Williamson A Tanuri H S Pereira R M Brindeiro J B A Neto O A C Antunes E M F Muri
627 A Practical Synthesis of α-Substituted tert-Butyl Acrylates from Meldrumrsquos Acid and Aldehydes C G Frost S D Penrose R Gleave
636 A New Class of Troumlgerrsquos Base Analogues Bearing Spiro[45] Lactone Straps A B Mahon D C Craig A C Try
643 A New Approach to Di- and Tetrasubstituted 23-Dihydropyridin-4(1H)-ones through Aza-DielsndashAlder Reaction Promoted by Silicon Tetrachloride A Massa V de Sio R Villano M R Acocella L Palombi G Sellitto A Peduto R Filosa P De Capraris A Scettri
650 Palladium-Catalysed Direct Arylation of Sydnones A Rodriguez W J Moran
655 Synthesis of (ndash)-Monomorine I R W Bates P Song 660 Cobalt(II) Chloride HexahydratendashDiisopropylamine Catalyzed Mild and
Chemoselective Reduction of Carboxylic Esters with Sodium Borohydride A R Jagdale A S Paraskar A Sudalai
665 Synthesis of Bi- and Tricyclic αβ-Unsaturated Lactams as Potential Michael Acceptors Starting from Heterocyclic Imines K Schulz M Watzke K Johannes P Ullrich J Martens
674 An Expedient Synthesis of Bis-Fused Benzofuran and a Two-Directional Ring-Closing Metathesis for the Synthesis of Bisbenzoxepines and Bisbenzoxocines K C Majumdar B Chattopadhyay S Chakravorty
681 Palladium-Catalyzed Cross-Couplings of Unsaturated Halides Bearing Relatively Acidic Hydrogen Atoms with Organozinc Reagents Z Dong G Manolikakes J Li P Knochel
687 Synthesis of Enantioenriched aa-Disubstituted Cyclopentenes Catalyzed by N-Heterocyclic Carbenes E M Phillips M Wadamoto K A Scheidt
XVII Forthcoming Articles
No 5 691 Transannulation Reactions in the Synthesis of Natural Products
P A Clarke A T Reeder J Winn 710 Synthesis of DL-erythro-Sphingosine Using a Tethered
Aminohydroxylation Reaction as the Key Step J A Morales-Serna Y Diacuteaz M I Matheu S Castilloacuten
713 Convenient Multigram Synthesis of 4-Chloropyridine-26-dicarbonyl Dichloride K Mitsui J R Parquette
715 A Novel and Efficient Synthesis of Dihydrexidine J P Cueva D E Nichols
721 Synthesis of 57-Dichloro-6-azaindoles and Functionalization via a Highly Selective LithiumndashChlorine Exchange N Lachance L-P Bonhomme-Beaulieu P Joly
731 A Convenient Synthesis of Fluorinated Pyrazolo[34-b]pyridine and Pyrazolo[34-d]pyrimidine Nucleosides V O Iaroshenko D V Sevenard A Kotljarov D M Volochnyuk A O Tolmachev V Y Sosnovskikh
741 Diastereoselective Synthesis of γ-Amino Acids and Their Derivatives from Nitroethane via Intermediacy of 56-Dihydro-4H-12-oxazines Bearing the CH2CH(CO2Me)2 Substituent at C3 A Y Sukhorukov A V Lesiv Y A Khomutova S L Ioffe
755 Synthesis of a New Pyrrolopyridoindole and Its Pyrrolopyridobenzimidazole Regioisomer F Bouchikhi M Sassatelli F Anizon M Prudhomme P Moreau
759 Practical Syntheses of Sphingosine-1-Phosphate and Analogues V Blot U Jacquemard H-U Reissig B Kleuser
767 A Facile Synthetic Route towards Substituted Thieno[32-e]indoles W Van Snick W Nulens S Jambon W Dehaen
775 Microwave-Assisted One-Pot Synthesis of (Aminoalkyl)naphthols and (Aminoalkyl)quinolinols by Using Ammonium Carbamate or Ammonium Hydrogen Carbonate as Solid Ammonia Source I Szatmaacuteri F Fuumlloumlp
779 Enantioselective Synthesis of Flavan-3-ols Using a Mitsunobu Cyclization K Krohn I Ahmed M John 787 Synthesis of a Novel γ-Folic AcidndashNτ-Histidine Conjugate Suitable for
Labeling with 99mTc and 188Re C Sparr U Michel R E Marti C Muumlller R Schibli R Moser V Groehn
793 Palladium-Catalyzed Intramolecular Biaryl Coupling A Highly Efficient Avenue for Benzannulated Pyranoquinolines and Julolidine Derivatives K C Majumdar A Taher P Debnath
801 Preparation of NN-Dimethyl-N-Arylureas Using SS-Dimethyl Dithiocarbonate as a Carbonylating Reagent I Degani R Fochi C Magistris M Migliaccio
809 Versatile Selective α-Carboxylic Acid Esterification of N-Protected Amino Acids and Peptides by Alcalase T Nuijens C Cusan J A W Kruijtzer D T S Rijkers R M J Liskamp P J L M Quaedflieg
815 Efficient Palladium-Catalyzed Amination of Aryl Chlorides Using Dicyclohexylamino[(26-dimethyl)morpholino]phenylphosphine as a PN2 Ligand S-E Park S B Kang K-J Jung J-E Won S-G Lee Y-J Yoon
824 A Clean Facile and Stereospecific Synthesis of α-Oxoketene OS-Acetals in Water Y Li Q Zhang X Cheng Q Liu X Xu
829 Sonogashira Cross-Coupling Reactions and Construction of the Indole Ring System Using a Robust Silica-Supported Palladium Catalyst E Tyrrell L Whiteman N Williams
836 Synthesis of Angular 78-Pyridazinocoumarins via the Transformation of a Hydroxy Group into a Carbonyl Group A Kotali I S Lafazanis P A Harris
841 Synthesis of New Cyclic and Acyclic 5-Halouridine Derivatives as Potential Antiviral Agents M F Elshehry J Balzarini C Meier
848 Dendritic Triphenylmethylium and Tetraphenylmethane Compounds H Meier S Kim A Oehlhof
853 Synthesis of Homoallylic Alcohols via Lewis Acid Assisted Enantioselective Desymmetrization B Yu F Menad N Isono M Lautens
860 Diastereoselective Synthesis of 123-Trisubstituted Indanes via Rhodium(I)-Catalyzed Tandem Conjugate Additions C Navarro A G Csaacutekyuml
864 Bakerrsquos Yeast for Sweet Dough Enables Large-Scale Synthesis of Enantiomerically Pure Bicyclo[331]nonane-26-dione C J Wallentin E Orentas E Butkus K Waumlrnmark
868 Addendum and Erratum XV Forthcoming Articles
No 6 869 Stereoselective Transformations of meso Bicyclic Hydrazines Versatile
Access to Functionalized Aminocyclopentanes C Bournaud F Chung A P Luna M Pasco G Errasti T Lecourt L Micouin
888 Synthesis of Glycoaminoxy Acids as Novel Sugar Building Blocks A Malapelle R Ramozzi J Xie
891 Electrophilic ipso-Halocyclization of N-Arylpropynamides with Polyfluoroalkyl Alcohols Selective Synthesis of 8-(Polyfluoroalkoxy) azaspiro[45]trienes Z-Q Wang B-X Tang H-P Zhang F Wang J-H Li
903 Electrooxidation of Alcohols in N-Oxyl-Immobilized Silica GelWater Disperse System Approach to Totally Closed System M Kuroboshi K Goto H Tanaka
909 Synthetic Routes to Aminotriamantanes Topological Analogues of the Neuroprotector Memantinereg A A Fokin A Merz N A Fokina H Schwertfeger S L Liu J E P Dahl R K M Carlson P R Schreiner
913 Parallel Synthesis of Drug-like 5-Amino-Substituted 124-Thiadiazole Libraries Using Cyclization Reactions of a Carboxamidine Dithiocarbamate Linker J Y Park I A Ryu J H Park D C Ha Y-D Gong
921 Copper-Catalyzed Selective S-Arylation of 12-Bis(o-amino-1H-pyrazolyl) Disulfides with Arylboronic Acids P-S Luo F Wang J-H Li R-Y Tang P Zhong
929 2-Iodoxybenzoic AcidTetraethylammonium BromideWater An Efficient Combination for Oxidative Cleavage of Acetals C Kuhakarn W Panchan S Chiampanichayakul N Samakkanad M Pohmakotr V Reutrakul T Jaipetch
935 Synthesis of Quinonoid Analogues of Diospyrin S Sagar I R Green 941 A One-Pot Method for the Iodination of Aryl Amines via Stable Aryl
Diazonium Silica Sulfates Under Solvent-Free Conditions A Zaroi A R Hajipour L Khazdooz
945 Poly(NN-dichloro-N-ethylbenzene-13-disulfonamide) and NNNN-Tetrachlorobenzene-13-disulfonamide as Novel Reagents for the Synthesis of N-Chloroamines Nitriles and Aldehydes R Ghorbani-Vaghei H Veisi
951 Synthesis of an (R)-Garner-type Aldehyde from L-Serine Useful Building Block for a (+)-Furanomycin Derivative G Bartoli G Di Antonio R Fiocchi S Giuli E Marcantoni M Marcolini
957 An Efficient and Highly Selective Synthesis of (Z)-Fluoroenol Phosphates from Hydroxy Difluorophosphonates P Beier R Pohl A V Alexandrova
963 Iodine-Catalyzed Three-Component Reaction A Rapid Synthesis of α-Alkoxy Azides and Homoallyl Ethers J S Yadav B V S Reddy G M Reddy R Narender
969 Rhodium(I)-Catalyzed Cycloisomerization of 13-Dienes with Alkenes in a Tether Y Oonishi A Saito M Mori Y Sato
980 Synthesis of New Optically Active D-GlucosaminendashPyrrole Derivatives B A Frontana-Uribe M V Escaacutercega-Bobadilla J Juaacuterez-Lagunas R A Toscano G A Garciacutea de la Mora M Salmoacuten
985 Partially Saturated Indeno[12-b]indole Derivatives via Deoxygenation of Heterocyclic α-Hydroxy-NO-hemiaminals H-J Hemmerling G Reiss
1000 Light-Induced Synthesis of Π-Extended Tetrathiafulvalenes Incorporating Ferrocenes An Efficient Route for the Synthesis of Electron-Donor Materials A A O Sarhan C Bolm
1007 Preparation of Nβ-Fmoc-Protected Aza-β3-Amino Acids with Nonproteinogenic Hydrophobic Side Chains for Solid-Phase Syntheses of Pseudopeptides M Laurencin P Bauchat M Baudy-Flocrsquoh
1014 Diastereomeric (η4-diene)Fe(CO)3 Complexes Containing Chiral Amide Groups A Convenient Method for the Resolution of Amino Acids M Schumacher G Coste L Miesch
1021 Palladium-Catalysed Heck Reactions of Alk-1-en-3-ones with Aryl Bromides A Very Simple Access to (E)-1-Arylalk-1-en-3-ones M Lemhadri Y Fall H Doucet M Santelli
1036 An Improved Process for the Synthesis of 4H-Imidazo[15-α][14]benzodiazepines J Yang Y Teng S Ara S Rallapalli J M Cook
1041 Meta- and Para-Difunctionalization of Arenes via an Ortho-Magnesiation and a Subsequent SulfoxidendashMagnesium Exchange L Melzig C B Rauhut P Knochel
XIII Forthcoming Articles
No 7 1049 Catalytic Transformations of Benzylic Carboxylates and Carbonates
R Kuwano 1062 A Simple and Practical Method for the Oxidation of Thebaine to 14-
Hydroxycodeinone by V2O5ndashH2O2 S Das Sharma D Konwar 1065 Umpolung with Sulfur Dioxide CarbonndashCarbon Cross-Coupling of Electron-
Rich 13-Dienes and Alkenes Application to the Enantioselective Synthesis of Long-Chain Polyketide Fragments M Turks C J Exner C Hamel P Vogel
1075 One-Pot Synthesis of 14-Diarylnaphthalenes via a WittigndashHorner Reaction[4+2] CycloadditionDehydrogenation Sequence Z Chen W Shou Y Wang
1081 A Novel and General Method for the Formation of S-Aryl Se-Aryl and Te-Aryl Phosphorochalcogenoates Y-X Gao G Tang Y Cao Y-F Zhao
1087 A Remarkable Access to γ-Fluoroalkylated Propargylamine Derivatives or Fluoroalkylated Dihydroisoxazoles via the Reaction of Fluoroalkylated Acetylides with Various Nitrones T Konno K Moriyasu T Ishihara
1095 Short and Practical Syntheses of (S)-(+)-3-(p-Tolylsulfinyl)furan-2(5H)-one and (S)-(+)-3-(p-Tolylsulfinyl)-56-dihydropyran-2-one D Cruz Cruz A Hernaacutendez Linares F Yuste M R Martiacuten J L Garciacutea Ruano
1099 Decarboxylative Aldol-Type Reaction of 2-(Trifluoroacetyl)-13-diazoles with Activated Acetic Acids P V Khodakovskiy D M Volochnyuk A A Tolmachev
1105 Synthesis of 2-[(Arylmethylene)amino]cyclopropanecarbonitriles via a Two-Step Ring Transformation of 2-(Cyanomethyl)aziridines S Mangelinckx M Drsquohooghe S Peeters N De Kimpe
1113 Synthesis of Dendrimeric Tumor-Associated Mucin-Type Glycopeptide Antigens T Becker A Kaiser H Kunz
1123 A Simple and Efficient Oxidation Procedure for the Synthesis of Acid-Sensitive Epoxides O Bortolini G Fantin M Fogagnolo
1127 Rapid Chemoselective Deprotection of Benzyl Esters by Nickel Boride J M Khurana R Arora
1131 Three-Component Coupling of Isoquinoline Activated Alkyne and Nitromethane A Facile Synthesis of Nitromethyl Derivatives of 12-Dihydroisoquinolines J S Yadav B V S Reddy N N Yadav M K Gupta
1137 Palladium Supported on a Polyionic Resin as an Efficient Ligand-Free and Recyclable Catalyst for Heck SuzukindashMiyaura and Sonogashira Reactions B Basu S Das P Das B Mandal D Banerjee F Almqvist
1147 Oxidation of 25-Dialkylpyrrole Derivatives with Cerium(IV) Ammonium Nitrate R Voloshchuk M Gałęzowski D T Gryko
1153 Practical Syntheses of Enantiomerically Pure Key Intermediates of Opioid Receptor-like 1 (ORL1) Antagonists T Yoshizumi A Ohno T Tsujita H Takahashi O Okamoto I Hayakawa H Kigoshi
1163 An Environmentally Benign TEMPO-Catalyzed Efficient Alcohol Oxidation System with a Recyclable Hypervalent Iodine(III) Reagent and Its Facile Preparation X-Q Li C Zhang
1170 Efficient and Stereoselective Rearrangement of BaylisndashHillman Acetates Catalyzed by Gold(I) ChlorideSilver(I) Trifluoromethanesulfonate Y Liu D Mao J Qian S Lou Z Xu Y Zhang
1175 The First Total Synthesis of Kynapcin-24 by Palladium Catalysis L-Y Yang C-F Chang Y-C Huang Y-J Lee C-C Hu T-H Tseng
1180 Enantioselective Synthesis of N-Protected α-Amino Acid Hydrazides M Bibian S El-Habnouni J Martinez J-A Fehrentz
1185 Synthesis of 11H-Indolo[32-c]quinoline-6-carboxylic Acids by Cascade AutoxidationndashRing Contractions A Becker S Kohfeld T Pies K Wieking L Preu C Kunick
1190 Reaction of N-Nonaflylbenzotriazole with Silyl Enol Ethers M Uhde T Ziegler
1195 2-(Benzoylimino)thiazolidin-4-ones Formation by an Alternative Ring Closure and Analysis of Rotational Barriers H-G Haumlcker P W Elsinghorst S Michels J Daniels G Schnakenburg M Guumltschow
1204 Microwave-Assisted Synthesis and Functionalization of Selenolopyrimidines S Hesse C Chenet D Thomae G Kirsch
1209 12-Disubstituted 4-Quinolones via Copper-Catalyzed Cyclization of 1-(2-Halophenyl)-2-en-3-amin-1-ones R Bernini S Cacchi G Fabrizi A Sferrazza
1220 A New Atom-Economical and Selective Synthesis of Secondary and Tertiary Alkylamines by Means of CpIridium Complex Catalyzed Multiple N-Alkylation of Ammonium Salts with Alcohols without Solvent R Yamaguchi Z Mingwen S Kawagoe C Asai K-i Fujita
1224 Synthesis of Regioisomerically Pure 5-Functionalized 27-Dichlorofluoresceins J C Castro A Malakhov K Burgess
XIII Forthcoming Articles
No 8 1227 Michael Additions to Activated Vinylphosphonates T Janecki J Kędzia
T Wąsek 1255 A Facile and General Synthesis of 2β-Aminosteroids X Ke H Hu
D Zhou W Xu Q Zhu N P Reddy X Hu 1261 Efficacious Preparation of Oppolzerrsquos Glycylsultam via the Deleacutepine
Reaction A Isleyen C Gonsky R C Ronald P Garner 1265 Synthesis of Masked Vicinal Amino Aldehydes of Pyrrolizine and Pyrrolo
[12-c]thiazole Series A V Tverdokhlebov A V Denisenko A A Tolmachev Y M Volovenko S V Shishkina O V Shishkin
1271 Preparation of 9-Substituted Pyridine-Stretched Adenines and Hypoxanthines J A Crawford W Fraser C A Ramsden
1279 A Versatile Synthesis of Heterocyclic Analogues of Neoflavonoids from Enamino Ketones V S Moskvina V P Khilya O V Turov U M Groth
1287 New Stereoselective Synthesis of Paeonilactone B F G Gatti S Serra 1291 The Use of NN-Dialkyltrimethylsilylamines in the Synthesis of
Pentamethinium Salts M Kořiacutenek M Rybaacutečkovaacute Boumlhm 1297 Synthesis of Triazoles via Regioselective Reactions of Aryl Azides with
Cyanoacetyl Pyrroles and Indoles N T Pokhodylo V S Matiychuk M D Obushak
1301 Gallium(III) Chloride Catalyzed Hydroarylation of Arylacetylenes with Naphthols and Phenols A Facile Synthesis of Vinylarenes J S Yadav B V S Reddy S Sengupta S K Biswas
1305 Electrophilic Bromination of meta-Substituted Anilines with N-Bromosuccinimide Regioselectivity and Solvent Effect S Bartoli A Cipollone A Squarcia A Madami D Fattori
1309 Cross-Coupling Reactions of Halopurines with Aryl- and Alkyltrifluoroborates The Scope and Limitations in the Synthesis of Modified Purines Z Hasniacutek R Pohl M Hocek
1318 A Convenient Method for Converting Hydroxyacetophenones into Their Ethylene or Trimethylene Acetals F Ono H Takenaka T Fujikawa M Mori T Sato
1323 γ-Chloromagnesio γ-Lactones and δ-Chloromagnesio δ-Lactones Generation Properties and Synthetic Uses H Shimizu S Fukuda S Sugiyama T Satoh
1336 Click Reactions with Nitroxides T Kaacutelai W L Hubbell K Hideg 1341 Synthesis of Novel 14-Benzoquinone-Containing 123-Triazoles An Entry
Into a New Library F Algi M Balci 1348 Efficient Synthesis of Two Sialylated Tetrasaccharides Found in Goat Milk
P K Mandal A K Misra 1355 Dendrimers of Vaccines Consisting of Tumor-Associated Glycopeptide
Antigens and T Cell Epitope Peptides S Keil A Kaiser F Syed H Kunz
1370 IBXTBAB-Mediated Oxidation of Primary Amines to Nitriles F Drouet P Fontaine G Masson J Zhu
1375 Chemoselectivity of Multicomponent Condensations of Barbituric Acids 5-Aminopyrazoles and Aldehydes E A Muravyova S V Shishkina V I Musatov I V Knyazeva O V Shishkin S M Desenko V A Chebanov
1386 Stereoselective Total Syntheses of Leiocarpin A and (ndash)-Galantinic Acid Starting from D-Mannitol K Nagaiah D Sreenu K V Purnima R S Rao J S Yadav
1393 A Facile Mild Deprotection Protocol for 13-Dithianes and 13-Dithiolanes with 30 Hydrogen Peroxide and Iodine Catalyst in Aqueous Micellar System N C Ganguly S K Barik
1400 Rhodium-Catalyzed Gram-Scale Synthesis of Highly Substituted Pyridine Derivatives K Parthasarathy C-H Cheng
1403 Enantioselective Synthesis of (R)-Propylene Carbonate from Ethyl (S)-Lactate J M Whitaker R C Ronald
XIII Forthcoming Articles
no 9 1405 Transition-Metal-Catalyzed Site-Selective Cross-Coupling of Di- and
Polyhalogenated Compounds J-R Wang K Manabe 1428 An Improved Synthesis of (4-4-Hydroxy-3-isopropyl-5-[(4-nitrophenyl)
ethynyl]benzyl-35-dimethylphenoxy)acetic Acid (NH-3) M B Gopinathan K S Rehder
1431 Copper-Catalyzed Tandem CndashN Bond Formation Reaction Selective Synthesis of 2-(Trifluoromethyl)benzimidazoles M-W Chen X-G Zhang P Zhong M-L Hu
1437 Synthesis and Thermochemical Properties of Stereoisomeric Dihydroxy- and Tetrahydroxyalkylammonium Salts M Thomas L Rothman J Hatcher P Agarkar R Ramkirath S Lall-Ramnarine R Engel
1445 Preparation of 5-Substituted 2-(2-Alkylaryl-1H-imidazol-4-yl)oxazoles and 5-Substituted 2-(2-Alkylarylthiazol-4-yl)oxazoles by Utilizing 5-Substituted 2-(2-Bromo-11-diethoxyethyl)oxazole as a Synthon D R St Laurent J L Romine
1459 Novel and Efficient Methods for the Synthesis of Symmetrical Trisulfides A Kertmen S Lach J Rachon D Witt
1463 An Environmentally Benign Electrochemical Process for the Reduction of Carboxylic Acid Hydrazides to Amides M Mentel M J Beier R Breinbauer
1469 Synthesis of 1-Chloroalkynes from Alkynylsilanes Using Trichloroisocyanuric Acid as Chlorinating Agent M H Vilhelmsen A S Andersson M B Nielsen
1473 A Convenient Approach to Enantioenriched Cyclopropanes Bearing Electron-Withdrawing Functionalities H Krawczyń K Wąsek J Kędzia
1477 Synthesis of Cyclopropenes via 12-Elimination of Bromocyclopropanes Catalyzed by Crown Ether W M Sherrill R Kim M Rubin
1485 A Base-Catalysed One-Pot Three-Component Coupling Reaction Leading to Nitrosubstituted Pyrroles I R Baxendale C D Buckle S V Ley L Tamborini
1494 Synthesis of 4-Alkylidene-4H-31-benzoxazine Derivatives by Acid-Catalyzed Cyclization of 2-Isocyanophenyl Ketones in the Presence of a Vinyl Ether K Kobayashi Y Okamura H Konishi
1499 Synthesis of Higher Helicenes via Olefin Metathesis and CndashH Activation J Cocircteacute S K Collins
1506 Azido- and Ethynyl-Substituted 2262-Terpyridines as Suitable Substrates for Click Reactions A Winter A Wild R Hoogenboom M W M Fijten M D Hager R-A Fallahpour U S Schubert
1513 Synthesis of 2-(Arylamino)ethanethiols via Lewis Acid Catalyzed Aminolysis of 22-Dimethylthiirane as Precursors of the 14-Benzothiazine Nucleus R Spogli S Sabatini G Manfroni O Tabarrini V Cecchetti
1520 Iron(III) Chloride A Versatile Catalyst for the Practical Synthesis of 3-Sulfenylindoles J S Yadav B V S Reddy Y J Reddy K Praneeth
1525 Organocatalytic Enantioselective Conjugate Addition of 2-Fluoromalonate to Nitroolefins Direct Synthesis of Chiral Fluorinated γ-Nitro Carboxylic Acid Derivatives H Li L Zu H Xie W Wang
1531 Asymmetric Transfer Hydrogenation of Ketimines with Trichlorosilane Structural Studies Z Zhang P Rooshenas H Hausmann P R Schreiner
1545 Prolinol Sulfinyl Ester Derivatives Organocatalytic Michael Addition of Ketones to Nitroolefins under Neat Conditions X Zeng G Zhong
1551 Asymmetric Oxidations of Electron-Poor Alkenes Promoted by the β-Amino AlcoholTBHP System A Russo A Lattanzi
1557 Enantioselectivity Switch in Direct Asymmetric Aminoxylation Catalyzed by Binaphthyl-Based Chiral Secondary Amines T Kano A Yamamoto F Shirozu K Maruoka
1564 Enantioselective Conjugate Addition of N-Heterocycles to αβ-Unsaturated Ketones Catalyzed by Chiral Primary Amines G Luo S Zhang W Duan W Wang
1573 Sulfonyl Hydrazine as New Functionality in Organocatalysis Camphorsulfonyl Hydrazine Catalyzed Enantioselective Aza-Michael Addition L-Y Chen H He B-J Pei W-H Chan A W M Lee
1578 Conversion of Primary Alcohols and Aldehydes into Methyl Esters by Ruthenium-Catalysed Hydrogen Transfer Reactions N A Owston T D Nixon A J Parker M K Whittlesey J M J Williams
1582 Addendum and Erratum XVII Forthcoming Articles
no 10 1583 Organocatalytic Formation of Quaternary Stereocenters M Bella
T Gasperi 1615 Regioselective Synthesis of 5H-Thiazolo[32-a]pyrimidin-5-ones from
MoritandashBaylisndashHillman Adduct Acetates under Solvent-Free and Base-Free Conditions W Zhong B Guo F Lin Y Liu W Su
1623 First Synthesis of 5-Cyanosalicylates by Formal [3+3] Cyclocondensations of 13-Bis(silyloxy)-13-butadienes A Riahi O Fatunsin M Shkoor R Dede H Reinke C Fischer P Langer
1635 Reaction of Isocyanides Dialkyl Acetylenedicarboxylates and a-Keto Lactones Unexpected Participation of an Ester Carbonyl Group in the Isocyanide-Based Three-Component Reaction A A Esmaeili H Vesalipoor
1639 An Efficient and Chemoselective Synthesis of 16-Naphthyridines and Pyrano[32-c]pyridines under Microwave Irradiation Z-G Han S-J Tu B Jiang S Yan X-H Zhang S-S Wu W-J Hao X-D Cao F Shi G Zhang N Ma
1647 N-Activation of N-Arylimidazoles Facile Syntheses of N-Alkyl-N-arylimidazolium Iodides from Less Expensive Chloro Substrates A M Oertel V Ritleng M J Chetcuti
1651 Synthesis of Polyhalogenated 2-(Phenylamino)pyridines by Thermal Amination Reactions S R Waldvogel A Faust W Barkmann R Froumlhlich O Wolff
1655 Cyanide Ion Promoted Addition of Acylphosphonates to Diethyl Cyanophosphonate Synthesis of Phosphonocyanohydrin O-Phosphates A S Demir A Aybey M Emrullahoglu
1659 Straightforward and Scalable Synthesis of Orthogonally Protected 37-Diazabicyclo[410]heptane H Schramm M Pavlova C Hoenke J Christoffers
1663 Hypervalent Iodine Mediated Oxidation of 12-Diaminobenzimidazole and Its Schiff Bases Efficient Synthesis of 3-Amino-124-benzotriazine and 2-Aryl-124-triazolo[15-a]benzimidazoles A Kumar M Parshad R K Gupta D Kumar
1667 Synthesis of the Reported Protoberberine Gusanlung D P B Wakchaure S Easwar N P Argade
1673 2-(Azidomethyl)arylboronic Acids in the Synthesis of Coumarin-Type Compounds M I Naumov A V Nuchev N S Sitnikov Y B Malysheva A S Shavyrin I P Beletskaya A E Gavryushin S Combes A Y Fedorov
1683 Asymmetric Synthesis of 12-anti-Disubstituted Taurine Derivatives D Enders D Iffland G Raabe
1689 A Novel One-Pot Three-Component Synthesis of 5-Imino-2358-tetrahydropyrazolo[12-a]pyridazin-1-one Derivatives B Qian M-J Fan Y-X Xie L-Y Wu Y Shi Y-M Liang
1694 One-Portion Synthesis of 2-Acetoxy Carbonyl Compounds from Aldehydes by Using an Acetylated Masked Acyl Cyanide H Nemoto T Kawamura K Kitasaki K Yatsuzuka M Kamiya Y Yoshioka
1703 Synthesis of 9-Anthryl Ethers from trans-910-Dihydro-910-dimethoxyanthracene by Acid-Catalyzed Transetherification K S Jang H Y Shin D Y Chi
1708 Efficient Synthesis of Azo Dye Labeled Terpenes Sugars and Steroids Using N-(4-Arylazobenzoyl)-1H-benzotriazoles A R Katritzky S R Tala N E Abo-Dya Z K Abdel-Samii
1715 Tandem CH-ActivationndashImine-Formation Reaction A New Route to Imidazo[21-a]phthalazines A Heim-Riether K R Gipson
1720 A Convenient and Efficient α-Sulfenylation of Carbonyl Compounds E Okragla S Demkowicz J Rachon D Witt
1725 Stereoselective Synthesis of β-Branched Phenylalanine Derivatives via Chelate-Claisen Rearrangement C Quirin U Kazmaier
1732 Catalyst-Free and Base-Free Water-Promoted SNAr Reaction of Heteroaryl Halides with Thiols B Sreedhar P S Reddy M A Reddy
1739 Convenient Methods for Synthesis of C2-Symmetric Diphenyltetrahydrothiophenes M Periasamy G Ramani G P Muthukumaragopal
1744 Highly Diastereoselective Conjugate AdditionndashElimination of Chiral Nickel(II) Glycinate with Activated Allylic Acetates for Asymmetric Synthesis of Glutamic Acid Derivatives J Wang J Shi X Zhang D Lin H Jiang H Liu
1753 Synthesis of 36-Dimethoxybenzene-12-diamine and of 47-Dimethoxy-2-methyl-1H-benzimidazole T Besset C Morin
1757 An Inexpensive Procedure for Reductive Aminations Using Dimethylamineborane on Millimolar and Molar Scale R Ortmann M Schlitzer
1760 Classics in Stereoselective Synthesis Edited by E M Carreira L Kvaerno Reviewed by Rolf Breinbauer
XV Forthcoming Articles
no 11 1761 Transition-Metal-Catalyzed Enantioselective Synthesis of Compounds with
Non-Centrochirality M Ogasawara S Watanabe 1786 One-Pot Synthesis of 3-Acyl-2-(alkylsulfanyl)indoles and 2-(Alkylsulfanyl)-
indole-3-carboxylates from (2-Isocyanophenyl)methyl Ketones or (2-Isocyanophenyl)acetates S Fukamachi H Konishi K Kobayashi
1791 Efficient and Recyclable Phthalocyanine-Based Sensitizers for Photooxygenation Reactions H Xu W-K Chan D K P Ng
1797 A Facile and Practical One-Pot Synthesis of β-Oxo Thioamides from β-Oxo Amides and Isothiocyanates P Huang D Xiang Y Zhou Y Liang T Na D Dong
1801 Microwave-Promoted Solid-Acid-Catalyzed One-Pot Synthesis of Phthalazinones V M Outerbridge S M Landge H Tamaki B Toumlroumlk
1807 Benzylic Brominations with N-Bromosuccinimide in (Trifluoromethyl)-benzene D Suarez G Laval S-M Tu D Jiang C L Robinson R Scott B T Golding
1811 Synthesis of Thioflavanone and Flavanone Derivatives by Cyclization of Chalcones W Konieczny M Konieczny
1815 A New and Expedient Total Synthesis of Ochratoxin A and d5-Ochratoxin A B Gabriele M Attya A Fazio L Di Donna P Plastina G Sindona
1821 Synthesis of Benzopyrrolizidinones by NorrishndashYang Cyclization of 3-(Acylmethyl)-2-alkylisoindol-1-ones J Wu W Zhang C Wang
1829 Reactions of MoritandashBaylisndashHillman Acetates with Huisgen Zwitterions A Novel Strategy for the Synthesis of β-Amino Acid Derivatives A Jose R R Paul R Mohan S C Mathew A T Biju E Suresh V Nair
1834 Peracetylated β-Allyl C-Glycosides of D-Ribofuranose and 2-Deoxy- D-ribofuranose in the Chemical Literature Until Now Mirages in the Literature H Otero Martinez H Reinke D Michalik C Vogel
1841 Core-Tetrasubstituted Naphthalene Diimides by Stille Cross-Coupling Reactions and Characterization of Their Optical and Redox Properties S-L Suraru F Wuumlrthner
1846 A Practical Synthesis of Indole-Based Heterocycles Using an Amidoaluminum-Mediated Strategy R Todd M M Hossain
1851 Synthesis of Fluorinated Pyrrolo[23-b]pyridine and Pyrrolo[23-d]pyrimidine Nucleosides V O Iaroshenko Y Wang D V Sevenard D M Volochnyuk
1858 Recyclization Reactions of 5-Formyl-13-dimethyluracil with Electron-Rich Amino Heterocycles A P Mityuk D M Volochnyuk S V Ryabukhin A S Plaskon A Shivanyuk A A Tolmachev
1865 Facile Synthesis of Fluorinated 1-Desazapurines V O Iaroshenko D V Sevenard D M Volochnyuk Y Wang A Martiloga A O Tolmachev
1876 A Practical Synthesis of 3-Diethoxyphosphoryl-12-pyridazine Derivatives J-C Monbaliu J Marchand-Brynaert
1881 Enantioselective Reduction of Prochiral Ketones Employing Sprouted Pisum sativa as Biocatalyst J S Yadav B V S Reddy C Sreelakshmi A B Rao
1886 Application of Phenolate Ion Mediated Intramolecular Epoxide Ring Opening in the Enantioselective Synthesis of Functionalized 23-Dihydrobenzofurans and 1-Benzopyrans S K Dinda S K Das G Panda
1897 Complementary Synthetic Approaches to Constitutionally Diverse N-Aminoalkylated Isoindolinones Application to the Synthesis of Falipamil and 5-HT1A Receptor Ligand Analogues M Lorion A Couture E Deniau P Grandclaudon
1904 Selective Deprotection of Silyl Ethers with Sodium Periodate J Li D Menche
1909 Micellar Solution of Sodium Dodecyl Sulfate (SDS) Catalyzes KabacknikndashFields Reaction in Aqueous Media S Sobhani A Vafaee
1916 Convenient Methods for the Synthesis of a Library of Hemilabile Phosphines M V Jimeacutenez J J Peacuterez-Torrente M I Bartolomeacute L A Oro
1923 Terminal Aziridines by Addition of Grignard Reagents or Organoceriums to an (α-Chloro)sulfinylimine D M Hodgson J Kloesges B Evans
1933 A Robust Synthesis of Nε-(Carboxymethyl)-L-lysine (CML) R Csuk S Stark A Barthel R Kluge D Stroumlhl
1935 One-Pot Curtius Rearrangement Processes from Carboxylic Acids O Leogane H Lebel
XV Forthcoming Articles
no 12 1941 The Chemistry of Deprotonated α-Aminonitriles T Opatz 1960 An Efficient Synthesis of Tetraalkyl 2345-Thiophenetetracarboxylate
Derivatives A Alizadeh R Hosseinpour 1963 Facile Deprotection of Bulky (Trialkylsilyl)acetylenes with Silver Fluoride
S Kim B Kim J In 1969 Highly Efficient and Reusable Ionic Liquids for the Catalyzed
Hydroamination of Alkenes with Sulfonamides Carbamates and Carboxamides L Yang L-W Xu C-G Xia
1975 Synthesis of 2391016172324-Octasubstituted Phthalocyaninatozinc(II) Complexes Mediated by Reductive Agents G A Gauna A C Monsalvo J Awruch
1979 A Short and Efficient Synthesis of 3-2-[2-(Bromomethyl)thiazol-4-yl]-ethynyl-5-fluorobenzonitrile A Precursor for PET Radioligand [18F]SP203 M B Gopinathan C Jin K S Rehder
1983 Synthesis of a Substituted Benzazepin-2-one Dihydrate S K Boini R K Vaid K P Moder D Mitchell
1987 Synthesis of Novel Trisubstituted Imidazolines F J Lakner M A Parker B Rogovoy A Khvat A Ivachtchenko
1991 A Novel Synthesis of N-But-3-enyl-α- and β-Amino Acids T T Van Nguyen R T C Brownlee A B Hughes
1999 Synthesis of Substituted 5-(3-Hydroxypropyl)pyrrolidin-2-ones and Pyrrolizidinones from Nitroethane via C3 Functionalized 56-Dihydro-4H-12-oxazines A Novel Approach to Some Analogues of the Antidepressant Rolipram A Yu Sukhorukov A V Lesiv Y A Khomutova S L Ioffe V A Tartakovsky
2009 Chiral Cyclobutanols and Cyclopentane Dimers via Samarium(II) Iodide Induced Keto-Olefin Cyclisations of Carbohydrate-Derived Unsaturated Ketones D B G Williams J Caddy K Blann J J C Groveacute C W Holzapfel
2015 Synthesis of Perfluoroalkylthio-Substituted Ferrocenes C Rhode J Lemke M Lieb N Metzler-Nolte
2019 Functionalization of Polyhedral Oligomeric Silsesquioxane (POSS) via Nucleophilic Substitution M Dutkiewicz H Maciejewski B Marciniec
2025 A Novel Synthesis of Aryl Mesylates via One-Pot DemethylationndashMesylation of Aryl Methyl Ethers Using a Mixture of Phosphorus Pentoxide in Methanesulfonic Acid B Kaboudin Y Abedi
2029 Anionic Cyclization of (NN-Dimethylamino)[2-(prop-2-yn-1-yloxy)aryl]-acetonitriles T Zdrojewski J Musielak A Jończyk
2035 Strecker-Type Reaction Catalyzed by Carboxylic Acids in Aqueous Media Z Xie G Li G Zhao J Wang
2040 Synthesis of Novel Structurally Simplified Estrogen Analogues with Electron-Donating Groups in Ring A L F Tietze C A Vock I K Krimmelbein L Nacke
2061 On the Resolution of Secondary Phosphine Oxides via Diastereomeric Complex Formation The Case of tert-Butylphenylphosphine Oxide J Holt A M Maj E P Schudde K M Pietrusiewicz L Sieroń W Wieczorek T Jerphagnon I W C E Arends U Hanefeld A J Minnaard
2066 Enantioselective Copper-Catalyzed Conjugate Addition of Dimethylzinc to 5-(1-Arylalkylidene) Meldrumrsquos Acids A Wilsily T Lou E Fillion
2073 SuzukindashMiyaura Coupling Reactions Using Phosphite Ligands M Jang Y Jo I-K Oh H M Jung S Lee
2076 Synthesis of 2-Methylindoline- and 2-Methyl-1234-tetrahydroquinoline-Derived Phosphoramidites and Their Applications in Iridium-Catalyzed Allylic Alkylation of Indoles W-B Liu H He L-X Dai S-L You
2083 Stereocontrolled Synthesis of 13-Amino Alcohols by Reduction of Substituted 2-1-[(tert-Butylsulfinyl)amino]alkylcyclohexanones J C Gonzaacutelez-Goacutemez F Foubelo M Yus
2089 Tunable Phosphoramidite Ligands for Asymmetric Hydrovinylation Ligands par excellence for Generation of All-Carbon Quaternary Centers C R Smith H J Lim A ZhangT V RajanBabu
2101 Copper-Catalyzed Asymmetric Ring-Opening Reaction of Oxabenzonorbornadienes with Grignard and Aluminum Reagents R Millet L Gremaud T Bernardez L Palais A Alexakis
2113 A Simplified Synthesis of Takemotorsquos Catalyst A Berkessel B Seelig 2116 Pharmaceutical Substances Syntheses Patents and Applications of the
Most Relevant AIPs Edited by Axel Kleeman Juumlrgen Engel Bernhard Kutscher Dietmar Reichert Reviewed by I Agranat
XV Forthcoming Articles
no 13 2117 Recent Advances in the Aza-Claisen Rearrangement K C Majumdar
T Bhattacharyya B Chattopadhyay B Sinha 2143 A Novel and Convenient Synthesis of lsquoReversedrsquo Diamidino 25-Aryl- and
25-Azaheterocycle-Substituted Furans L Hu D W Boykin 2146 Efficient and General Preparation of Pyranostilbenes First Total Synthesis
of Artocarbene and Pawhuskin B B H Park Y R Lee W S Lyoo 2155 Mild Oxidation of Diarylacetylenes to 12-Diketones Using Oxone in
Trifluoroacetic Acid J-H Chu Y-J Chen M-J Wu 2163 One-Pot Microwave-Assisted Selective Azido ReductionTandem Cyclization
in Condensed and Solid Phase with Nickel Boride N Shankaraiah N Markandeya M Espinoza-Moraga C Arancibia A Kamal L Silva Santos
2171 Pyrrolo[321-ij]quinolin-4-one and Pyrrolo[321-ij]quinolin-6-one H McNab D J Nelson E J Rozgowska
2175 Practical Synthesis of 5-Substituted Tetrazoles under Microwave Irradiation J Roh T V Artamonova K Vaacutevrovaacute G I Koldobskii A Hrabaacutelek
2179 A Simple Method for the Synthesis of 3-Arylthieno[23-b]pyridines via Iodine-Mediated Cyclization of 3-(1-Arylalkenyl)-2-[(1-phenylethyl)sulfanyl]pyridines K Kobayashi D Nakamura Y Shiroyama S Fukamachi H Konishi
2184 Synthesis of Four Lysine-Linked Cereulide Analogues Showing Ionophoric Activity Towards Potassium Cations as Lead Compounds for Emetic Toxin-Detection by Immunoassays A Makarasen T Nishikawa M Isobe
2205 Synthesis of α-Aliphatic and β-Aromatic Substituted Taurines via Regioselective Ring Opening of Thiiranes with Ammonia H Yu S Cao L Zhang G Liu J Xu
2210 Stability of 5(6)-Carboxyfluorescein in Microwave-Assisted Synthesis of Fluorescein-Labelled O-Dimannosylated Peptides R Kowalczyk P W R Harris R P Dunbar M A Brimble
2223 Diversity-Oriented Synthesis of Functionalized Diaryl Sulfones by Regioselective [3+3] Cyclizations of 13-Bis(siloxy)buta-13-dienes with 2-(Arylsulfonyl)-3-ethoxy-2-en-1-ones Scope and Limitations M Shkoor A Riahi O Fatunsin H Reinke C Fischer P Langer
2236 Synthesis of Functionalized Salicylates by Formal [3+3] Cyclocondensation of 13-Bis(silyloxy)buta-13-dienes with 3-Alkoxy-2-en-1-ones G Mroszlig S Ladzik H Reinke A Spannenberg C Fischer P Langer
2249 Synthetic Approach to Alkoxy-β-(trifluoromethyl)styrenes and Their Application in the Synthesis of New Trifluoromethylated Heterocycles V M Muzalevskiy V G Nenajdenko A V Shastin E S Balenkova G Haufe
2260 o-Benzenedisulfonimide as a Powerful and Recyclable Organocatalyst for the Nazarov Reaction M Barbero S Cadamuro A Deagostino S Dughera P Larini E G Occhiato C Prandi S Tabasso R Vulcano P Venturello
2267 The Catalytic Potential of 4-Guanidinylpyridines in Acylation Reactions I Held E Larionov C Bozler F Wagner H Zipse
2278 Iron(III) Chloride in EthanolndashWater Highly Efficient Catalytic System for the Synthesis of Garcia Gonzalez Polyhydroxyalkyl- and C-Glycosylfurans L Nagarapu M V Chary A Satyender B Supriya R Bantu
2283 Ruthenium-Catalyzed Addition of Primary Amides to Alkynes A Stereoselective Synthesis of Secondary Enamides L J Gooszligen M Blanchot K S M Salih K Gooszligen
2289 Binaphthyl-Modified Quaternary Phosphonium Salts as Chiral Phase Transfer Catalysts Application to Asymmetric Amination of β-Keto Esters R He K Maruoka
X Table of Contents XI Forthcoming Articles
no 14 2293 Direct Methods for Stereoselective Polypropionate Synthesis A Survey
J Li D Menche 2316 Synthesis of Symmetrical Ketones from Grignard Reagents and
11-Carbonyldiimidazole D Bottalico V Fiandanese G Marchese A Punzi
2319 Synthesis of 45-Substituted Imidazoles by a Fast Condensation of 12-Diketones and Urotropine in Heterogeneous Medium G Bratulescu
2321 (Arylsulfonyl)acetones and -acetonitriles New Activated Methylenic Building Blocks for Synthesis of 123-Triazoles N T Pokhodylo V S Matiychuk M D Obushak
2324 A Safe Convenient and Efficient One-Pot Synthesis of α-Chloroketone Acetals Directly from Ketones Using Iodobenzene Dichloride J Yu C Zhang
2329 An Efficient Oxidative Conversion of Aldehydes into 2-Substituted 2-Oxazolines Using 13-Diiodo-55-dimethylhydantoin S Takahashi H Togo
2333 A Novel Procedure for the Synthesis of Benzo[b][18]naphthyridine-3-carboxylate Derivatives from MoritandashBaylisndashHillman Adduct Acetates W Zhong F Lin R Chen W Su
2341 An Improved Synthesis of 147-Triazacyclononanes (tacns) and 14710-Tetraazacyclododecanes (cyclens) J Huang Z Zhou T H Chan
2345 The Ullmann Coupling between 2-Chlorobenzoic Acids and Amino Acids A Valuable Reaction for Preparing 2-Substituted 1-Acetyl-1H-indol-3-yl Acetates J C Rodriguez Dominguez X Gang G Kirsch
2349 gem-Dibromomethyl Aromatics Efficient Aldehyde Equivalents in the KnoevenagelndashDoebner Reaction J K Augustine Y A Naik S Poojari N Chowdappa B S Sherigara K Areppa
2357 Synthesis of Novel α-Aminophosphonates Containing Adamantyl Fragment M M Kabachnik L I Minaeva I P Beletskaya
2361 Efficient Fluoride-Mediated Synthesis of 5-Amino-Substituted Isothiazoles Y S Zubenko V I Potkin
2365 Phosphine-Catalyzed Reaction of Cyanohydrins with Activated Alkynes A Siby O Loreau F Taran
2371 Sulfanyl-Substituted [3]Cumulenes and Buta-13-dienes from a Tetrakis(pyridinium)-Substituted Butadiene A Schmidt A Rahimi M Gjikaj
2379 Efficient Synthesis of 2-Substituted Pyrido[32-d]pyrimidines Involving SNAr and Palladium-Catalyzed Cross-Coupling Reactions A Tikad S Routier M Akssira J-M Leacuteger C Jarry G Guillaumet
2385 Novel Synthesis of Medium-Sized Heterocycles by Palladium-Catalyzed Intramolecular Heck Reaction via 9-endo-trig Mode of Cyclization K C Majumdar B Chattopadhyay
2393 Facile Synthesis of Fluorinated Benzofuro- and Benzothieno[23-b]pyridines α-Carbolines and Nucleosides Containing the α-Carboline Framework V O Iaroshenko Y Wang B Zhang D Volochnyuk V Ya Sosnovskikh
2403 Synthesis of Functionalized N-Vinyl Nitrogen-Containing Heterocycles S M M Lopes A M Beja M Ramos Silva J A Paixatildeo F Palacios T M V D Pinho e Melo
2408 Kumada Cross-Coupling of Aryl Grignard Reagents with Aryl Halides Catalyzed by an Immobilized Nickel Catalyst X Chen L Wang J Liu
2413 Highly Enantioselective Synthesis of Heteroaromatic Alcohols Catalyzed by Chiral DiaminodiphosphinendashRuthenium(II) Complexes W-Y Shen Y-Y Li Z-R Dong J-X Gao
2418 Concise Total Synthesis of (+)-Disparlure and its trans-Isomer Using Asymmetric Organocatalysis S-G Kim
2423 Rhodium Carbenoid Induced [12]-Migration in an L-Lyxo-Configured α-Diazo β-Keto Ester Synthesis of a New Griseolic Acid Analogue N N Bhujbal K S A Kumar D D Dhavale
2430 Synthesis of 5-Arylthio-3-hydroxyphthalates by the First [4+2] Cycloadditions of 3-Arylthio-1-silyloxy-13-butadienes with Dimethyl Acetylenedicarboxylate I Iqbal M Imran P Langer
2435 Synthesis of Highly Functionalized Proline Derivatives via a One-Pot MichaelSN-AdditionCyclization Approach U Kazmaier C Schmidt
2440 RhodiumGraphite-Catalyzed Hydrogenation of Carbocyclic and Heterocyclic Aromatic Compounds G Falini A Gualandi D Savoia
2447 Potassium [1-(tert-Butoxycarbonyl)-1H-indol-2-yl]trifluoroborate as an Efficient Building Block in Palladium-Catalyzed SuzukindashMiyaura Cross Couplings P Kassis V Beacuteneacuteteau J-Y Meacuterour S Routier
2454 Syntheses of Substituted Furans and Pyrroles by Platinum-Catalyzed Cyclizations of Propargylic Oxiranes and Aziridines in Aqueous Media M Yoshida M Al-Amin K Shishido
2467 Transition-Metal-Free Oxidative Homocoupling of Aryl Alkenyl and Alkynyl Grignard Reagents with TEMPO M S Maji A Studer
XIII Forthcoming Articles
no 15 2471 Advances in Synthetic Approaches for the Preparation of Combretastatin-
Based Anti-Cancer Agents R Singh H Kaur 2492 Synthesis of Unsymmetrical Ureas by Sulfur-Assisted Carbonylation with
Carbon Monoxide and Oxidation with Molecular Oxygen under Mild Conditions T Mizuno T Nakai M Mihara
2497 Ring-OpeningRecyclization Reactions of (Dimethylamino)propenoyl-Substituted Cyclopropanes Facile Synthesis of Halogenated Pyridin-2(1H)-ones R Zhang Y Zhou Y Liang Z Jiang D Dong
2501 Facile and Efficient Total Synthesis of Taspine B Cheng S Zhang L Zhu J Zhang Q Li A Shan L He
2505 Oligomeric Iodosylbenzene Sulfate A Convenient Hypervalent Iodine Reagent for Oxidation of Organic Sulfides and Alkenes M S Yusubov R Y Yusubova T V Funk K-W Chi V V Zhdankin
2509 Pyrrolidine-Based Organocatalysts for Enantioselective Michael Addition of Cyclohexanone to trans-β-Nitrostyrene A P Carley S Dixon J D Kilburn
2517 CundashAl Hydrotalcite An Efficient and Reusable Ligand-Free Catalyst for the Coupling of Aryl Chlorides with Aliphatic Aromatic and N(H)-Heterocyclic Amines B Sreedhar R Arundhathi P L Reddy M A Reddy M L Kantam
2523 Highly Efficient Synthesis of trans-βγ-Unsaturated a-Keto Amides C Allais T Constantieux J Rodriguez
2531 Gas-Phase Synthesis of N-Unsubstituted 3-Hydroxypyrroles and 1H-Pyrrol-3(2H)-ones L Hill G A Hunter S H Imam H McNab W J OrsquoNeill
2535 3-Hydroxy-1H-pyrrole L Hill S H Imam H McNab W J OrsquoNeill 2539 123-Thiadiazoles with Unsaturated Side Chains Synthesis
Polymerization and Photocrosslinking M Al-Smadi N Hanold H Kalbitz H Meier
2547 Synthesis of 1112-Didehydrodibenzo[ae]cycloocten-5(6H)-one A Strained Eight-Membered Alkyne S C Kornmayer F Rominger R Gleiter
2553 Stannous Chloride Dihydrate A Novel and Efficient Catalyst for the Synthesis of gem-Dihydroperoxides from Ketones and Aldehydes D Azarifar K Khosravi F Soleimanei
2557 Synthesis of a Novel Class of Azacrown Macrocycles and Lariat Crown Ethers Containing Two 124-Triazole Rings as Subunits N Foroughifar A Mobinikhaledi S Ebrahimi
2561 Enantioselective Synthesis of the 3C-Protease Inhibitor (ndash)-Thysanone by a StauntonndashWeinreb Annulation Strategy J Sperry T Y Yuen M A Brimble
2570 Stereoselective Synthesis of Unnatural β-Amino Acids from Nitroethane via 56-Dihydro-4H-12-oxazin-3-ylacetates A Yu Sukhorukov A V Lesiv O L Eliseev Y A Khomutova S L Ioffe
2579 A Versatile Unexpected One-Pot Regioselective Synthesis of a New Class of 13-Diazepinoindolones by Reaction of Pyranoindolones with Monosubstituted Ureas D Livadiotou C A Tsoleridis J Stephanidou-Stephanatou
2584 Synthesis of a Trisaccharide and a Tetrasaccharide from the Cell-Wall Lipopolysaccharides of Azospirillum brasilense S17 S Pandey S Ghosh A K Misra
2591 Synthesis of Isoindoline Nitroxides by Electrocyclic Reactions T Kaacutelai J Jekı K Hideg
2596 Glycosylations of Tertiary Alcohols Synthesis of Fully Protected Disaccharides with Sterically Demanding Groups Attached to the Sugar Core A Holkenbrink J B Vicente D B Werz
2605 Copper-Catalyzed [13]-Dipolar Cycloaddition for the Synthesis of Macrocycles Containing Acyclic Aromatic and Steroidal Moieties G V Latyshev M S Baranom A V Kazantsev A D Averin N V Lukashev I P Beletskaya
2616 Aryl Ring Migration Reaction in the Synthesis of 24-Diaryl-4H-31-benzothiazines A V Butin F A Tsiunchik V T Abaev A V Gutnov D A Cheshkov
2627 Hydrogenation of β-N-Substituted and β-NN-Disubstituted Enamino Esters in the Presence of Iridium(I) Catalyst H Hebbache Z Hank C Bruneau J-L Renaud
2634 Stereoselective Olefination Reactions Promoted by Rieke Manganese J M Concelloacuten H Rodriacuteguez-Solla V del Amo P Diacuteaz
2646 Synthesis of Piperidinones through a Radical Cascade E Godineau Y Landais
2650 Asymmetric Organic Synthesis with Enzymes Edited by V Gotor I Alfonso E Garciacutea-Urdiales Reviewed by Steve Collier
XVII Forthcoming Articles
no 16 2651 Synthesis of Spirocyclic Ethers S Rosenberg R Leino 2674 Bimetallic PalladiumndashPlatinum-on-Carbon-Catalyzed HndashD Exchange
Reaction Synergistic Effect on Multiple Deuterium Incorporation T Maegawa N Ito K Oono Y Monguchi H Sajiki
2679 Efficient Copper-Catalyzed Synthesis of 2-Amino-4(3H)-quinazolinone and 2-Aminoquinazoline Derivatives X Huang H Yang H Fu R Qiao Y Zhao
2689 Synthesis and Chemoselective N- and O-Alkylation of Thiadiazolopyrimidine Nucleosides and Uridines A M L Hossion R Islam R K Kandahary T Nagamatsu
2697 Facile and Efficient Synthesis of a New Class of Indole-Substituted Pyridine Derivatives via One-Pot Multicomponent Reactions K Zhao X-P Xu S-L Zhu D-Q Shi Y Zhang S-J Ji
2709 Studies toward a Total Synthesis of Rhizoxin D Stereoselective Preparation of the C11ndashC19 Fragment S Padakanti C K Kumar E Ashok P Das
2715 A Short Synthesis of Enantiomeric Phytoprostanes B1 Type I W Perlikowska M Mikołajczyk
2719 Chemistry of Polyhalogenated Nitrobutadienes Part 7 A Novel Synthetic Access to Chlorinated Nitrile Oxides E Nutz V A Zapolrsquoskii D E Kaufmann
2725 Microwave-Assisted Silver(I)-Mediated Selective O-Alkylation of Aromatic Imidate Systems B K Singh C Cavalluzzo M De Maeyer Z Debyser V S Parmar E Van der Eycken
2729 Iodogen A Novel Reagent for the Oxidation of Urazoles under Heterogeneous Conditions A Khoramabadi A Shiri M A Zolfigol S Mallakpour
2733 An Unprecedented Synthesis of Eight-Membered-Ring Cyclic Thioimidic Esters by a Three-Component Reaction A Alizadeh R Hosseinpour
2737 A Novel Diastereoselective Synthesis of β-Phosphonato Unsaturated Thioimidates A Alizadeh N Zohreh
2741 Synthesis of 21-Benzisoxazoles by Nucleophilic Substitution of Hydrogen in Nitroarenes Activated by the Azole Ring N T Pokhodylo Y O Teslenko V S Matiychuk M D Obushak
2749 A Facile Synthesis of Two Series of Multifunctional Carbon Compounds from αα-Dihalo Ketones Using Allylsamarium Bromide X Liu S Zhang J Di
2756 Stereocontrolled Formation of Protected Aminodeoxyalditols from Simple Carbohydrate Precursors by Debenzylating Cycloetherification Y Jiang Z Fang Q Zheng H Jia J Cheng B Zheng
2761 trans-Stilbene as a Starting Material for the Synthesis of Tamoxifen Based on Palladium-Catalyzed Cross-Coupling Reactions C M Nunes J Limberger S Poersch M Seferin A L Monteiro
2766 Synthesis and Biological Evaluation of 6-Substituted Purinylcarbanucleosides with a Cyclopenta[b]thiophene Pseudosugar P Abeijoacuten J M Blanco O Caamantildeo F Fernaacutendez M D Garciacutea X Garciacutea-Mera J E Rodriacuteguez-Borges J Balzarini E De Clercq
2773 Synthesis and Electrochemical Signature of Novel Norbornyl-ferrocene Hybrids F A Khan S K Upadhyay
2778 A Regioselective TsujindashTrost Pentadienylation of 3-Allyltetronic Acid R Schobert B Barnickel
2785 Copper(I)-Catalyzed CarylndashCalkynyl Bond Formation of Aryl Iodides with Terminal Alkynes K G Thakur G Sekar
2790 Aminolysis of Epoxides Using Iridium Trichloride as an Efficient Catalyst J Agarwal A Duley R Rani R K Peddinti
2797 Preparation of Several Active N-Chloro Compounds from Trichloroisocyanuric Acid A Shiri A Khoramabadi-zad
2802 The First Mineral-Catalyzed One-Pot [3+1+2] Coupling Protocol for Multifunctionalized Fused-Ring Pyrimidines L D S Yadav A Rai
2809 Efficient Synthesis of Tetrahydro-β-carbolin-1-one and Dihydroisoquinolin-1-one Derivatives as Versatile Intermediates K E Judd M F Mahon L Caggiano
2818 A Concise Synthesis of ortho-Iodobenzyl Alcohols via Addition of ortho-Iodophenyl Grignard Reagent to Aldehydes and Ketones J Cvengroš D Stolz A Togni
XIII Forthcoming Articles
no 17 2825 Reactivity of Oxazol-5-(4H)-ones and Their Application toward Natural
Product Synthesis N M Hewlett C D Hupp J J Tepe 2840 Towards the Total Synthesis of 3-Hydroxyvibsanin E B D Schwartz
J R Denton P V Bernhardt H M L Davies C M Williams 2847 Structure Investigations of (ent)-Cladospolide D by De Novo Synthesis and
Kinetic and Thermodynamic Isomerization Y Xing J H Penn G A OrsquoDoherty
2855 New Applications of PhI(OAc)2 in Synthesis Total Synthesis and SAR Development of Potent Antitumor Natural Product PsymberinIrciniastatin A N Shao X Huang A Palani R Aslanian A Buevich J Piwinski R Huryk C Seidel-Dugan
2873 Total Synthesis of Largazole ndash Devolution of a Novel Synthetic Strategy B Wang C J Forsyth
2881 Formal Total Synthesis of Palmerolide A J Jaumlgel M E Maier 2893 Total Synthesis of Bongkrekic Acid via Sequential SuzukindashMiyaura Coupling
Reactions M Kanematsu M Shindo M Yoshida K Shishido 2905 Stereodivergent Approach to Both C28a-syn and C28a-anti Relative
Stereochemical Manifolds in the Lepadin Family via a TiCl4-Promoted G Li L J Carlson I K Sagamanova B W Slafer R P Hsung C Gilardi H M Sklenicka N Sydorenko
2915 Enantioselective Aldol Reaction of Tetrasubstituted Ketene Silyl Acetals with Achiral Aldehydes for the Construction of Asymmetric Tertiary Alcohols An Application for the Divergent Total Syntheses of Buergerinins F and G I Shiina T Iizumi Y-s Yamai Y-i Kawakita K Yokoyama Y-k Yamada
2927 Second-Generation Biomimetic Total Synthesis of Chaetominine A Coste G Karthikeyan F Couty G Evano
2935 Total Synthesis of (+)-Fostriecin and (+)-Phoslactomycin B S Shibahara M Fujino Y Tashiro N Okamoto T Esumi K Takahashi J Ishihara S Hatakeyama
2954 Stereochemical Assignments of the Chlorinated Residues in Victorin C A C Durow C Butts C L Willis
2963 Studies of the Asymmetric Total Synthesis of Clavilactone D by the lsquoLariatrsquo Cyclization Strategy T Yoshimitsu S Nojima M Hashimoto K Tsukamoto T Tanaka
2970 Total Synthesis of the Leucetta-Derived Alkaloid Calcaridine A P B Koswatta R Sivappa H V R Dias C J Lovely
2983 Formal Synthesis of Salinosporamide A Starting from D-Glucose T Momose Y Kaiya J-i Hasegawa T Sato N Chida
2992 Synthesis of Bioactive Natural Products by Asymmetric syn- and anti-Aldol Reactions A K Ghosh Z L Dawson
no 18 3003 Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural
Products B M Trost M K Brennan 3026 One-Pot Synthesis of Furo[34-b]pyridin-5(7H)-ones from 2-
Bromopyridine-3-carboxylic Acid and Carbonyl Compounds K Kobayashi T Kozuki H Konishi
3029 Iodocyclization of N-[2-(Methylthio)phenyl]propiolamides Selective Synthesis of 3-Iodo-15-benzothiazepin-4-ones T-S Jiang X-G Zhang J-H Li
3039 A Facile Synthetic Method for Fluorine-Containing 17-Phenanthrolines Pyridine-Ring Formation Reaction of N-Propargyl-68-bis(trifluoroacetyl)-quinolin-5-amine with Various Nucleophiles D Shibata E Okada M Hinoshita M Meacutedebielle
3047 Enantiotopic Discrimination in Palladium-Mediated Nucleophilic Substitutions on Achiral Substrates Chiral Ligand versus Chiral Nucleophile O Jacquet F Charnay J-C Fiaud J Ollivier
3051 Studies on the Chemistry of 2-[3-(2-Nitrophenyl)-2-oxopropyl]benzaldehydes Novel Syntheses of 5H-Benzo[b]carbazole-611-diones and Indolo[12-b]isoquinoline-611-diones M Fernaacutendez
3061 Studies on the C22ndashC23 Aldol Coupling of Spirangien M Lorenz N Bluhm M Kalesse
3067 One-Pot Synthesis of N-Alkyl Purine Pyrimidine and Azole Derivatives from Alcohols using Ph3PCCl4 A Rapid Route to Carboacyclic Nucleoside Synthesis M N Soltani Rad A Khalafi-Nezhad S Behrouz Z Asrari M Behrouz Z Amini
3077 Synthesis of 2-Amino-34-dihydroquinazolines and Imidazo[21-b]quinazoline-2-ones A Mishra S Batra
3089 Studies on the Reaction of Diimines with Thiourea Synthesis and Solvent-Induced cistrans-Isomerization of 135-Triazinane-2-thiones B Kaboudin T Ghasemi T Yokomatsu
3094 Suzuki Coupling of Heteroaromatic Chlorides Using Highly Electron-Donating ClickPhos Ligands S M Spinella Z-H Guan J Chen X Zhang
3099 Reaction of NN-Dioxyenamines with Anhydrides of Carboxylic and Sulfonic Acids A New Method for the Synthesis of a-Hydroxyoxime Derivatives A A Tabolin A V Lesiv S L Ioffe
3106 Directed ortho Metallation Chemistry and Phosphine Synthesis New Ligands for the SuzukindashMiyaura Reaction D B G Williams S J Evans H de Bod M S Mokhadinyana T Hughes
3113 New Functional Derivatives of 9-Phenylquinine P J Boratyński J SkarŜewski
3120 On the Synthesis of Asymmetric and Dissymmetric Amino Analogues of Troumlgerrsquos Base J Artacho K Waumlrnmark
3127 Synthesis of Polycyclic Sultams by Palladium-Catalyzed Intramolecular Cyclization K C Majumdar S Mondal N De
3136 Synthesis of Functionalized L-Cysteine and L-Methionine by Reaction with Electron-Deficient Acetylenes B A Trofimov A G Malrsquokina O A Shemyakina V V Nosyreva A P Borisova S S Khutsishvili L B Krivdin
3143 A lsquoClickrsquo Approach to the Synthesis of 3-[2-(1-Alkyltriazol-4-yl)ethyl]indoles M Petrini R R Shaikh
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
No 4 513 Intermolecular Addition Reactions of N-Acyliminium Ions (Part II)
A Yazici S G Pyne 542 A Simple Practical Method for the Synthesis of 46-Dimethoxy-135-
triazin-2(1H)-one Using Dimethylamine-Functionalized Solid-Phase Reagents K Hioki K Ohshima Y Sota M Tanaka M Kunishima
545 Conjugation-Amenable Tetrasaccharide of the Side Chain of the Major Glycoprotein of the Bacillus anthracis Exosporium A Large-Scale Preparation S Hou P Kovaacuteč
551 Reductive Amination ndash A Convenient Method for Generating Diverse Mono-Functionalised 5101520-Tetraphenyl Porphyrins C Welch S J Archibald R W Boyle
557 Highly Regioselective Preparation of 13-Dioxolane-4-methanol Derivatives from Glycerol Using Phosphomolybdic Acid N W Fadnavis R Gowrisankar G Ramakrishna M K Mishra G Sheelu
561 Rapid Synthesis of 3-Aminoisoquinoline-5-sulfonamides Using the BuchwaldndashHartwig Reaction N Proisy S Taylor A Nelson I Collins
567 Synthesis of Divalent 22-Linked Mannose Derivatives by Homodimerization F S Ekholm M Polaacutekovaacute A J Pawłowicz R Leino
577 Efficient Synthesis of Substituted Cyclic α-Aminophosphonates I L Odinets O I Artyushin N Shevchenko P V Petrovskii V G Nenajdenko G-V Roumlschenthaler
583 Methylated Imidazolinium-Dithiocarboxylates Two Representatives of a New Class of Ionic Liquids A Blanrue R Wilhelm
587 An Efficient Route to 1-Vinylpyrrole-2-carbaldehydes A I Mikhaleva A V Ivanov E V Skitalrsquotseva I A Ushakov A M Vasilrsquotsov B A Trofimov
591 A Regioselective Route to 5-Substituted Isoxazole- and Isoxazoline-3-phosphonates P Conti A Pinto L Tamborini P Dunkel V Gambaro G L Visconti C De Micheli
597 Solvent-Free One-Pot Conjugate Addition of Benzyl Bromides to β-Nitroalkenes Mediated by Magnesium Powder W Shi J-X Wang
602 Synthesis of 234-Trideoxy-44-difluoro-D-ribo-hexopyranose Adenosines J Xu X Zhang X-L Qiu F-L Qing
609 Synthesis of anti-27-Disubstituted Norbornadienes G C Tsui P Le Marquand A Allen W Tam
620 Novel Peptide Mimetic Inhibitors of Hepatitis C Serine Protease Derived from Isomannide T G Barros S Pinheiro J S Williamson A Tanuri H S Pereira R M Brindeiro J B A Neto O A C Antunes E M F Muri
627 A Practical Synthesis of α-Substituted tert-Butyl Acrylates from Meldrumrsquos Acid and Aldehydes C G Frost S D Penrose R Gleave
636 A New Class of Troumlgerrsquos Base Analogues Bearing Spiro[45] Lactone Straps A B Mahon D C Craig A C Try
643 A New Approach to Di- and Tetrasubstituted 23-Dihydropyridin-4(1H)-ones through Aza-DielsndashAlder Reaction Promoted by Silicon Tetrachloride A Massa V de Sio R Villano M R Acocella L Palombi G Sellitto A Peduto R Filosa P De Capraris A Scettri
650 Palladium-Catalysed Direct Arylation of Sydnones A Rodriguez W J Moran
655 Synthesis of (ndash)-Monomorine I R W Bates P Song 660 Cobalt(II) Chloride HexahydratendashDiisopropylamine Catalyzed Mild and
Chemoselective Reduction of Carboxylic Esters with Sodium Borohydride A R Jagdale A S Paraskar A Sudalai
665 Synthesis of Bi- and Tricyclic αβ-Unsaturated Lactams as Potential Michael Acceptors Starting from Heterocyclic Imines K Schulz M Watzke K Johannes P Ullrich J Martens
674 An Expedient Synthesis of Bis-Fused Benzofuran and a Two-Directional Ring-Closing Metathesis for the Synthesis of Bisbenzoxepines and Bisbenzoxocines K C Majumdar B Chattopadhyay S Chakravorty
681 Palladium-Catalyzed Cross-Couplings of Unsaturated Halides Bearing Relatively Acidic Hydrogen Atoms with Organozinc Reagents Z Dong G Manolikakes J Li P Knochel
687 Synthesis of Enantioenriched aa-Disubstituted Cyclopentenes Catalyzed by N-Heterocyclic Carbenes E M Phillips M Wadamoto K A Scheidt
XVII Forthcoming Articles
No 5 691 Transannulation Reactions in the Synthesis of Natural Products
P A Clarke A T Reeder J Winn 710 Synthesis of DL-erythro-Sphingosine Using a Tethered
Aminohydroxylation Reaction as the Key Step J A Morales-Serna Y Diacuteaz M I Matheu S Castilloacuten
713 Convenient Multigram Synthesis of 4-Chloropyridine-26-dicarbonyl Dichloride K Mitsui J R Parquette
715 A Novel and Efficient Synthesis of Dihydrexidine J P Cueva D E Nichols
721 Synthesis of 57-Dichloro-6-azaindoles and Functionalization via a Highly Selective LithiumndashChlorine Exchange N Lachance L-P Bonhomme-Beaulieu P Joly
731 A Convenient Synthesis of Fluorinated Pyrazolo[34-b]pyridine and Pyrazolo[34-d]pyrimidine Nucleosides V O Iaroshenko D V Sevenard A Kotljarov D M Volochnyuk A O Tolmachev V Y Sosnovskikh
741 Diastereoselective Synthesis of γ-Amino Acids and Their Derivatives from Nitroethane via Intermediacy of 56-Dihydro-4H-12-oxazines Bearing the CH2CH(CO2Me)2 Substituent at C3 A Y Sukhorukov A V Lesiv Y A Khomutova S L Ioffe
755 Synthesis of a New Pyrrolopyridoindole and Its Pyrrolopyridobenzimidazole Regioisomer F Bouchikhi M Sassatelli F Anizon M Prudhomme P Moreau
759 Practical Syntheses of Sphingosine-1-Phosphate and Analogues V Blot U Jacquemard H-U Reissig B Kleuser
767 A Facile Synthetic Route towards Substituted Thieno[32-e]indoles W Van Snick W Nulens S Jambon W Dehaen
775 Microwave-Assisted One-Pot Synthesis of (Aminoalkyl)naphthols and (Aminoalkyl)quinolinols by Using Ammonium Carbamate or Ammonium Hydrogen Carbonate as Solid Ammonia Source I Szatmaacuteri F Fuumlloumlp
779 Enantioselective Synthesis of Flavan-3-ols Using a Mitsunobu Cyclization K Krohn I Ahmed M John 787 Synthesis of a Novel γ-Folic AcidndashNτ-Histidine Conjugate Suitable for
Labeling with 99mTc and 188Re C Sparr U Michel R E Marti C Muumlller R Schibli R Moser V Groehn
793 Palladium-Catalyzed Intramolecular Biaryl Coupling A Highly Efficient Avenue for Benzannulated Pyranoquinolines and Julolidine Derivatives K C Majumdar A Taher P Debnath
801 Preparation of NN-Dimethyl-N-Arylureas Using SS-Dimethyl Dithiocarbonate as a Carbonylating Reagent I Degani R Fochi C Magistris M Migliaccio
809 Versatile Selective α-Carboxylic Acid Esterification of N-Protected Amino Acids and Peptides by Alcalase T Nuijens C Cusan J A W Kruijtzer D T S Rijkers R M J Liskamp P J L M Quaedflieg
815 Efficient Palladium-Catalyzed Amination of Aryl Chlorides Using Dicyclohexylamino[(26-dimethyl)morpholino]phenylphosphine as a PN2 Ligand S-E Park S B Kang K-J Jung J-E Won S-G Lee Y-J Yoon
824 A Clean Facile and Stereospecific Synthesis of α-Oxoketene OS-Acetals in Water Y Li Q Zhang X Cheng Q Liu X Xu
829 Sonogashira Cross-Coupling Reactions and Construction of the Indole Ring System Using a Robust Silica-Supported Palladium Catalyst E Tyrrell L Whiteman N Williams
836 Synthesis of Angular 78-Pyridazinocoumarins via the Transformation of a Hydroxy Group into a Carbonyl Group A Kotali I S Lafazanis P A Harris
841 Synthesis of New Cyclic and Acyclic 5-Halouridine Derivatives as Potential Antiviral Agents M F Elshehry J Balzarini C Meier
848 Dendritic Triphenylmethylium and Tetraphenylmethane Compounds H Meier S Kim A Oehlhof
853 Synthesis of Homoallylic Alcohols via Lewis Acid Assisted Enantioselective Desymmetrization B Yu F Menad N Isono M Lautens
860 Diastereoselective Synthesis of 123-Trisubstituted Indanes via Rhodium(I)-Catalyzed Tandem Conjugate Additions C Navarro A G Csaacutekyuml
864 Bakerrsquos Yeast for Sweet Dough Enables Large-Scale Synthesis of Enantiomerically Pure Bicyclo[331]nonane-26-dione C J Wallentin E Orentas E Butkus K Waumlrnmark
868 Addendum and Erratum XV Forthcoming Articles
No 6 869 Stereoselective Transformations of meso Bicyclic Hydrazines Versatile
Access to Functionalized Aminocyclopentanes C Bournaud F Chung A P Luna M Pasco G Errasti T Lecourt L Micouin
888 Synthesis of Glycoaminoxy Acids as Novel Sugar Building Blocks A Malapelle R Ramozzi J Xie
891 Electrophilic ipso-Halocyclization of N-Arylpropynamides with Polyfluoroalkyl Alcohols Selective Synthesis of 8-(Polyfluoroalkoxy) azaspiro[45]trienes Z-Q Wang B-X Tang H-P Zhang F Wang J-H Li
903 Electrooxidation of Alcohols in N-Oxyl-Immobilized Silica GelWater Disperse System Approach to Totally Closed System M Kuroboshi K Goto H Tanaka
909 Synthetic Routes to Aminotriamantanes Topological Analogues of the Neuroprotector Memantinereg A A Fokin A Merz N A Fokina H Schwertfeger S L Liu J E P Dahl R K M Carlson P R Schreiner
913 Parallel Synthesis of Drug-like 5-Amino-Substituted 124-Thiadiazole Libraries Using Cyclization Reactions of a Carboxamidine Dithiocarbamate Linker J Y Park I A Ryu J H Park D C Ha Y-D Gong
921 Copper-Catalyzed Selective S-Arylation of 12-Bis(o-amino-1H-pyrazolyl) Disulfides with Arylboronic Acids P-S Luo F Wang J-H Li R-Y Tang P Zhong
929 2-Iodoxybenzoic AcidTetraethylammonium BromideWater An Efficient Combination for Oxidative Cleavage of Acetals C Kuhakarn W Panchan S Chiampanichayakul N Samakkanad M Pohmakotr V Reutrakul T Jaipetch
935 Synthesis of Quinonoid Analogues of Diospyrin S Sagar I R Green 941 A One-Pot Method for the Iodination of Aryl Amines via Stable Aryl
Diazonium Silica Sulfates Under Solvent-Free Conditions A Zaroi A R Hajipour L Khazdooz
945 Poly(NN-dichloro-N-ethylbenzene-13-disulfonamide) and NNNN-Tetrachlorobenzene-13-disulfonamide as Novel Reagents for the Synthesis of N-Chloroamines Nitriles and Aldehydes R Ghorbani-Vaghei H Veisi
951 Synthesis of an (R)-Garner-type Aldehyde from L-Serine Useful Building Block for a (+)-Furanomycin Derivative G Bartoli G Di Antonio R Fiocchi S Giuli E Marcantoni M Marcolini
957 An Efficient and Highly Selective Synthesis of (Z)-Fluoroenol Phosphates from Hydroxy Difluorophosphonates P Beier R Pohl A V Alexandrova
963 Iodine-Catalyzed Three-Component Reaction A Rapid Synthesis of α-Alkoxy Azides and Homoallyl Ethers J S Yadav B V S Reddy G M Reddy R Narender
969 Rhodium(I)-Catalyzed Cycloisomerization of 13-Dienes with Alkenes in a Tether Y Oonishi A Saito M Mori Y Sato
980 Synthesis of New Optically Active D-GlucosaminendashPyrrole Derivatives B A Frontana-Uribe M V Escaacutercega-Bobadilla J Juaacuterez-Lagunas R A Toscano G A Garciacutea de la Mora M Salmoacuten
985 Partially Saturated Indeno[12-b]indole Derivatives via Deoxygenation of Heterocyclic α-Hydroxy-NO-hemiaminals H-J Hemmerling G Reiss
1000 Light-Induced Synthesis of Π-Extended Tetrathiafulvalenes Incorporating Ferrocenes An Efficient Route for the Synthesis of Electron-Donor Materials A A O Sarhan C Bolm
1007 Preparation of Nβ-Fmoc-Protected Aza-β3-Amino Acids with Nonproteinogenic Hydrophobic Side Chains for Solid-Phase Syntheses of Pseudopeptides M Laurencin P Bauchat M Baudy-Flocrsquoh
1014 Diastereomeric (η4-diene)Fe(CO)3 Complexes Containing Chiral Amide Groups A Convenient Method for the Resolution of Amino Acids M Schumacher G Coste L Miesch
1021 Palladium-Catalysed Heck Reactions of Alk-1-en-3-ones with Aryl Bromides A Very Simple Access to (E)-1-Arylalk-1-en-3-ones M Lemhadri Y Fall H Doucet M Santelli
1036 An Improved Process for the Synthesis of 4H-Imidazo[15-α][14]benzodiazepines J Yang Y Teng S Ara S Rallapalli J M Cook
1041 Meta- and Para-Difunctionalization of Arenes via an Ortho-Magnesiation and a Subsequent SulfoxidendashMagnesium Exchange L Melzig C B Rauhut P Knochel
XIII Forthcoming Articles
No 7 1049 Catalytic Transformations of Benzylic Carboxylates and Carbonates
R Kuwano 1062 A Simple and Practical Method for the Oxidation of Thebaine to 14-
Hydroxycodeinone by V2O5ndashH2O2 S Das Sharma D Konwar 1065 Umpolung with Sulfur Dioxide CarbonndashCarbon Cross-Coupling of Electron-
Rich 13-Dienes and Alkenes Application to the Enantioselective Synthesis of Long-Chain Polyketide Fragments M Turks C J Exner C Hamel P Vogel
1075 One-Pot Synthesis of 14-Diarylnaphthalenes via a WittigndashHorner Reaction[4+2] CycloadditionDehydrogenation Sequence Z Chen W Shou Y Wang
1081 A Novel and General Method for the Formation of S-Aryl Se-Aryl and Te-Aryl Phosphorochalcogenoates Y-X Gao G Tang Y Cao Y-F Zhao
1087 A Remarkable Access to γ-Fluoroalkylated Propargylamine Derivatives or Fluoroalkylated Dihydroisoxazoles via the Reaction of Fluoroalkylated Acetylides with Various Nitrones T Konno K Moriyasu T Ishihara
1095 Short and Practical Syntheses of (S)-(+)-3-(p-Tolylsulfinyl)furan-2(5H)-one and (S)-(+)-3-(p-Tolylsulfinyl)-56-dihydropyran-2-one D Cruz Cruz A Hernaacutendez Linares F Yuste M R Martiacuten J L Garciacutea Ruano
1099 Decarboxylative Aldol-Type Reaction of 2-(Trifluoroacetyl)-13-diazoles with Activated Acetic Acids P V Khodakovskiy D M Volochnyuk A A Tolmachev
1105 Synthesis of 2-[(Arylmethylene)amino]cyclopropanecarbonitriles via a Two-Step Ring Transformation of 2-(Cyanomethyl)aziridines S Mangelinckx M Drsquohooghe S Peeters N De Kimpe
1113 Synthesis of Dendrimeric Tumor-Associated Mucin-Type Glycopeptide Antigens T Becker A Kaiser H Kunz
1123 A Simple and Efficient Oxidation Procedure for the Synthesis of Acid-Sensitive Epoxides O Bortolini G Fantin M Fogagnolo
1127 Rapid Chemoselective Deprotection of Benzyl Esters by Nickel Boride J M Khurana R Arora
1131 Three-Component Coupling of Isoquinoline Activated Alkyne and Nitromethane A Facile Synthesis of Nitromethyl Derivatives of 12-Dihydroisoquinolines J S Yadav B V S Reddy N N Yadav M K Gupta
1137 Palladium Supported on a Polyionic Resin as an Efficient Ligand-Free and Recyclable Catalyst for Heck SuzukindashMiyaura and Sonogashira Reactions B Basu S Das P Das B Mandal D Banerjee F Almqvist
1147 Oxidation of 25-Dialkylpyrrole Derivatives with Cerium(IV) Ammonium Nitrate R Voloshchuk M Gałęzowski D T Gryko
1153 Practical Syntheses of Enantiomerically Pure Key Intermediates of Opioid Receptor-like 1 (ORL1) Antagonists T Yoshizumi A Ohno T Tsujita H Takahashi O Okamoto I Hayakawa H Kigoshi
1163 An Environmentally Benign TEMPO-Catalyzed Efficient Alcohol Oxidation System with a Recyclable Hypervalent Iodine(III) Reagent and Its Facile Preparation X-Q Li C Zhang
1170 Efficient and Stereoselective Rearrangement of BaylisndashHillman Acetates Catalyzed by Gold(I) ChlorideSilver(I) Trifluoromethanesulfonate Y Liu D Mao J Qian S Lou Z Xu Y Zhang
1175 The First Total Synthesis of Kynapcin-24 by Palladium Catalysis L-Y Yang C-F Chang Y-C Huang Y-J Lee C-C Hu T-H Tseng
1180 Enantioselective Synthesis of N-Protected α-Amino Acid Hydrazides M Bibian S El-Habnouni J Martinez J-A Fehrentz
1185 Synthesis of 11H-Indolo[32-c]quinoline-6-carboxylic Acids by Cascade AutoxidationndashRing Contractions A Becker S Kohfeld T Pies K Wieking L Preu C Kunick
1190 Reaction of N-Nonaflylbenzotriazole with Silyl Enol Ethers M Uhde T Ziegler
1195 2-(Benzoylimino)thiazolidin-4-ones Formation by an Alternative Ring Closure and Analysis of Rotational Barriers H-G Haumlcker P W Elsinghorst S Michels J Daniels G Schnakenburg M Guumltschow
1204 Microwave-Assisted Synthesis and Functionalization of Selenolopyrimidines S Hesse C Chenet D Thomae G Kirsch
1209 12-Disubstituted 4-Quinolones via Copper-Catalyzed Cyclization of 1-(2-Halophenyl)-2-en-3-amin-1-ones R Bernini S Cacchi G Fabrizi A Sferrazza
1220 A New Atom-Economical and Selective Synthesis of Secondary and Tertiary Alkylamines by Means of CpIridium Complex Catalyzed Multiple N-Alkylation of Ammonium Salts with Alcohols without Solvent R Yamaguchi Z Mingwen S Kawagoe C Asai K-i Fujita
1224 Synthesis of Regioisomerically Pure 5-Functionalized 27-Dichlorofluoresceins J C Castro A Malakhov K Burgess
XIII Forthcoming Articles
No 8 1227 Michael Additions to Activated Vinylphosphonates T Janecki J Kędzia
T Wąsek 1255 A Facile and General Synthesis of 2β-Aminosteroids X Ke H Hu
D Zhou W Xu Q Zhu N P Reddy X Hu 1261 Efficacious Preparation of Oppolzerrsquos Glycylsultam via the Deleacutepine
Reaction A Isleyen C Gonsky R C Ronald P Garner 1265 Synthesis of Masked Vicinal Amino Aldehydes of Pyrrolizine and Pyrrolo
[12-c]thiazole Series A V Tverdokhlebov A V Denisenko A A Tolmachev Y M Volovenko S V Shishkina O V Shishkin
1271 Preparation of 9-Substituted Pyridine-Stretched Adenines and Hypoxanthines J A Crawford W Fraser C A Ramsden
1279 A Versatile Synthesis of Heterocyclic Analogues of Neoflavonoids from Enamino Ketones V S Moskvina V P Khilya O V Turov U M Groth
1287 New Stereoselective Synthesis of Paeonilactone B F G Gatti S Serra 1291 The Use of NN-Dialkyltrimethylsilylamines in the Synthesis of
Pentamethinium Salts M Kořiacutenek M Rybaacutečkovaacute Boumlhm 1297 Synthesis of Triazoles via Regioselective Reactions of Aryl Azides with
Cyanoacetyl Pyrroles and Indoles N T Pokhodylo V S Matiychuk M D Obushak
1301 Gallium(III) Chloride Catalyzed Hydroarylation of Arylacetylenes with Naphthols and Phenols A Facile Synthesis of Vinylarenes J S Yadav B V S Reddy S Sengupta S K Biswas
1305 Electrophilic Bromination of meta-Substituted Anilines with N-Bromosuccinimide Regioselectivity and Solvent Effect S Bartoli A Cipollone A Squarcia A Madami D Fattori
1309 Cross-Coupling Reactions of Halopurines with Aryl- and Alkyltrifluoroborates The Scope and Limitations in the Synthesis of Modified Purines Z Hasniacutek R Pohl M Hocek
1318 A Convenient Method for Converting Hydroxyacetophenones into Their Ethylene or Trimethylene Acetals F Ono H Takenaka T Fujikawa M Mori T Sato
1323 γ-Chloromagnesio γ-Lactones and δ-Chloromagnesio δ-Lactones Generation Properties and Synthetic Uses H Shimizu S Fukuda S Sugiyama T Satoh
1336 Click Reactions with Nitroxides T Kaacutelai W L Hubbell K Hideg 1341 Synthesis of Novel 14-Benzoquinone-Containing 123-Triazoles An Entry
Into a New Library F Algi M Balci 1348 Efficient Synthesis of Two Sialylated Tetrasaccharides Found in Goat Milk
P K Mandal A K Misra 1355 Dendrimers of Vaccines Consisting of Tumor-Associated Glycopeptide
Antigens and T Cell Epitope Peptides S Keil A Kaiser F Syed H Kunz
1370 IBXTBAB-Mediated Oxidation of Primary Amines to Nitriles F Drouet P Fontaine G Masson J Zhu
1375 Chemoselectivity of Multicomponent Condensations of Barbituric Acids 5-Aminopyrazoles and Aldehydes E A Muravyova S V Shishkina V I Musatov I V Knyazeva O V Shishkin S M Desenko V A Chebanov
1386 Stereoselective Total Syntheses of Leiocarpin A and (ndash)-Galantinic Acid Starting from D-Mannitol K Nagaiah D Sreenu K V Purnima R S Rao J S Yadav
1393 A Facile Mild Deprotection Protocol for 13-Dithianes and 13-Dithiolanes with 30 Hydrogen Peroxide and Iodine Catalyst in Aqueous Micellar System N C Ganguly S K Barik
1400 Rhodium-Catalyzed Gram-Scale Synthesis of Highly Substituted Pyridine Derivatives K Parthasarathy C-H Cheng
1403 Enantioselective Synthesis of (R)-Propylene Carbonate from Ethyl (S)-Lactate J M Whitaker R C Ronald
XIII Forthcoming Articles
no 9 1405 Transition-Metal-Catalyzed Site-Selective Cross-Coupling of Di- and
Polyhalogenated Compounds J-R Wang K Manabe 1428 An Improved Synthesis of (4-4-Hydroxy-3-isopropyl-5-[(4-nitrophenyl)
ethynyl]benzyl-35-dimethylphenoxy)acetic Acid (NH-3) M B Gopinathan K S Rehder
1431 Copper-Catalyzed Tandem CndashN Bond Formation Reaction Selective Synthesis of 2-(Trifluoromethyl)benzimidazoles M-W Chen X-G Zhang P Zhong M-L Hu
1437 Synthesis and Thermochemical Properties of Stereoisomeric Dihydroxy- and Tetrahydroxyalkylammonium Salts M Thomas L Rothman J Hatcher P Agarkar R Ramkirath S Lall-Ramnarine R Engel
1445 Preparation of 5-Substituted 2-(2-Alkylaryl-1H-imidazol-4-yl)oxazoles and 5-Substituted 2-(2-Alkylarylthiazol-4-yl)oxazoles by Utilizing 5-Substituted 2-(2-Bromo-11-diethoxyethyl)oxazole as a Synthon D R St Laurent J L Romine
1459 Novel and Efficient Methods for the Synthesis of Symmetrical Trisulfides A Kertmen S Lach J Rachon D Witt
1463 An Environmentally Benign Electrochemical Process for the Reduction of Carboxylic Acid Hydrazides to Amides M Mentel M J Beier R Breinbauer
1469 Synthesis of 1-Chloroalkynes from Alkynylsilanes Using Trichloroisocyanuric Acid as Chlorinating Agent M H Vilhelmsen A S Andersson M B Nielsen
1473 A Convenient Approach to Enantioenriched Cyclopropanes Bearing Electron-Withdrawing Functionalities H Krawczyń K Wąsek J Kędzia
1477 Synthesis of Cyclopropenes via 12-Elimination of Bromocyclopropanes Catalyzed by Crown Ether W M Sherrill R Kim M Rubin
1485 A Base-Catalysed One-Pot Three-Component Coupling Reaction Leading to Nitrosubstituted Pyrroles I R Baxendale C D Buckle S V Ley L Tamborini
1494 Synthesis of 4-Alkylidene-4H-31-benzoxazine Derivatives by Acid-Catalyzed Cyclization of 2-Isocyanophenyl Ketones in the Presence of a Vinyl Ether K Kobayashi Y Okamura H Konishi
1499 Synthesis of Higher Helicenes via Olefin Metathesis and CndashH Activation J Cocircteacute S K Collins
1506 Azido- and Ethynyl-Substituted 2262-Terpyridines as Suitable Substrates for Click Reactions A Winter A Wild R Hoogenboom M W M Fijten M D Hager R-A Fallahpour U S Schubert
1513 Synthesis of 2-(Arylamino)ethanethiols via Lewis Acid Catalyzed Aminolysis of 22-Dimethylthiirane as Precursors of the 14-Benzothiazine Nucleus R Spogli S Sabatini G Manfroni O Tabarrini V Cecchetti
1520 Iron(III) Chloride A Versatile Catalyst for the Practical Synthesis of 3-Sulfenylindoles J S Yadav B V S Reddy Y J Reddy K Praneeth
1525 Organocatalytic Enantioselective Conjugate Addition of 2-Fluoromalonate to Nitroolefins Direct Synthesis of Chiral Fluorinated γ-Nitro Carboxylic Acid Derivatives H Li L Zu H Xie W Wang
1531 Asymmetric Transfer Hydrogenation of Ketimines with Trichlorosilane Structural Studies Z Zhang P Rooshenas H Hausmann P R Schreiner
1545 Prolinol Sulfinyl Ester Derivatives Organocatalytic Michael Addition of Ketones to Nitroolefins under Neat Conditions X Zeng G Zhong
1551 Asymmetric Oxidations of Electron-Poor Alkenes Promoted by the β-Amino AlcoholTBHP System A Russo A Lattanzi
1557 Enantioselectivity Switch in Direct Asymmetric Aminoxylation Catalyzed by Binaphthyl-Based Chiral Secondary Amines T Kano A Yamamoto F Shirozu K Maruoka
1564 Enantioselective Conjugate Addition of N-Heterocycles to αβ-Unsaturated Ketones Catalyzed by Chiral Primary Amines G Luo S Zhang W Duan W Wang
1573 Sulfonyl Hydrazine as New Functionality in Organocatalysis Camphorsulfonyl Hydrazine Catalyzed Enantioselective Aza-Michael Addition L-Y Chen H He B-J Pei W-H Chan A W M Lee
1578 Conversion of Primary Alcohols and Aldehydes into Methyl Esters by Ruthenium-Catalysed Hydrogen Transfer Reactions N A Owston T D Nixon A J Parker M K Whittlesey J M J Williams
1582 Addendum and Erratum XVII Forthcoming Articles
no 10 1583 Organocatalytic Formation of Quaternary Stereocenters M Bella
T Gasperi 1615 Regioselective Synthesis of 5H-Thiazolo[32-a]pyrimidin-5-ones from
MoritandashBaylisndashHillman Adduct Acetates under Solvent-Free and Base-Free Conditions W Zhong B Guo F Lin Y Liu W Su
1623 First Synthesis of 5-Cyanosalicylates by Formal [3+3] Cyclocondensations of 13-Bis(silyloxy)-13-butadienes A Riahi O Fatunsin M Shkoor R Dede H Reinke C Fischer P Langer
1635 Reaction of Isocyanides Dialkyl Acetylenedicarboxylates and a-Keto Lactones Unexpected Participation of an Ester Carbonyl Group in the Isocyanide-Based Three-Component Reaction A A Esmaeili H Vesalipoor
1639 An Efficient and Chemoselective Synthesis of 16-Naphthyridines and Pyrano[32-c]pyridines under Microwave Irradiation Z-G Han S-J Tu B Jiang S Yan X-H Zhang S-S Wu W-J Hao X-D Cao F Shi G Zhang N Ma
1647 N-Activation of N-Arylimidazoles Facile Syntheses of N-Alkyl-N-arylimidazolium Iodides from Less Expensive Chloro Substrates A M Oertel V Ritleng M J Chetcuti
1651 Synthesis of Polyhalogenated 2-(Phenylamino)pyridines by Thermal Amination Reactions S R Waldvogel A Faust W Barkmann R Froumlhlich O Wolff
1655 Cyanide Ion Promoted Addition of Acylphosphonates to Diethyl Cyanophosphonate Synthesis of Phosphonocyanohydrin O-Phosphates A S Demir A Aybey M Emrullahoglu
1659 Straightforward and Scalable Synthesis of Orthogonally Protected 37-Diazabicyclo[410]heptane H Schramm M Pavlova C Hoenke J Christoffers
1663 Hypervalent Iodine Mediated Oxidation of 12-Diaminobenzimidazole and Its Schiff Bases Efficient Synthesis of 3-Amino-124-benzotriazine and 2-Aryl-124-triazolo[15-a]benzimidazoles A Kumar M Parshad R K Gupta D Kumar
1667 Synthesis of the Reported Protoberberine Gusanlung D P B Wakchaure S Easwar N P Argade
1673 2-(Azidomethyl)arylboronic Acids in the Synthesis of Coumarin-Type Compounds M I Naumov A V Nuchev N S Sitnikov Y B Malysheva A S Shavyrin I P Beletskaya A E Gavryushin S Combes A Y Fedorov
1683 Asymmetric Synthesis of 12-anti-Disubstituted Taurine Derivatives D Enders D Iffland G Raabe
1689 A Novel One-Pot Three-Component Synthesis of 5-Imino-2358-tetrahydropyrazolo[12-a]pyridazin-1-one Derivatives B Qian M-J Fan Y-X Xie L-Y Wu Y Shi Y-M Liang
1694 One-Portion Synthesis of 2-Acetoxy Carbonyl Compounds from Aldehydes by Using an Acetylated Masked Acyl Cyanide H Nemoto T Kawamura K Kitasaki K Yatsuzuka M Kamiya Y Yoshioka
1703 Synthesis of 9-Anthryl Ethers from trans-910-Dihydro-910-dimethoxyanthracene by Acid-Catalyzed Transetherification K S Jang H Y Shin D Y Chi
1708 Efficient Synthesis of Azo Dye Labeled Terpenes Sugars and Steroids Using N-(4-Arylazobenzoyl)-1H-benzotriazoles A R Katritzky S R Tala N E Abo-Dya Z K Abdel-Samii
1715 Tandem CH-ActivationndashImine-Formation Reaction A New Route to Imidazo[21-a]phthalazines A Heim-Riether K R Gipson
1720 A Convenient and Efficient α-Sulfenylation of Carbonyl Compounds E Okragla S Demkowicz J Rachon D Witt
1725 Stereoselective Synthesis of β-Branched Phenylalanine Derivatives via Chelate-Claisen Rearrangement C Quirin U Kazmaier
1732 Catalyst-Free and Base-Free Water-Promoted SNAr Reaction of Heteroaryl Halides with Thiols B Sreedhar P S Reddy M A Reddy
1739 Convenient Methods for Synthesis of C2-Symmetric Diphenyltetrahydrothiophenes M Periasamy G Ramani G P Muthukumaragopal
1744 Highly Diastereoselective Conjugate AdditionndashElimination of Chiral Nickel(II) Glycinate with Activated Allylic Acetates for Asymmetric Synthesis of Glutamic Acid Derivatives J Wang J Shi X Zhang D Lin H Jiang H Liu
1753 Synthesis of 36-Dimethoxybenzene-12-diamine and of 47-Dimethoxy-2-methyl-1H-benzimidazole T Besset C Morin
1757 An Inexpensive Procedure for Reductive Aminations Using Dimethylamineborane on Millimolar and Molar Scale R Ortmann M Schlitzer
1760 Classics in Stereoselective Synthesis Edited by E M Carreira L Kvaerno Reviewed by Rolf Breinbauer
XV Forthcoming Articles
no 11 1761 Transition-Metal-Catalyzed Enantioselective Synthesis of Compounds with
Non-Centrochirality M Ogasawara S Watanabe 1786 One-Pot Synthesis of 3-Acyl-2-(alkylsulfanyl)indoles and 2-(Alkylsulfanyl)-
indole-3-carboxylates from (2-Isocyanophenyl)methyl Ketones or (2-Isocyanophenyl)acetates S Fukamachi H Konishi K Kobayashi
1791 Efficient and Recyclable Phthalocyanine-Based Sensitizers for Photooxygenation Reactions H Xu W-K Chan D K P Ng
1797 A Facile and Practical One-Pot Synthesis of β-Oxo Thioamides from β-Oxo Amides and Isothiocyanates P Huang D Xiang Y Zhou Y Liang T Na D Dong
1801 Microwave-Promoted Solid-Acid-Catalyzed One-Pot Synthesis of Phthalazinones V M Outerbridge S M Landge H Tamaki B Toumlroumlk
1807 Benzylic Brominations with N-Bromosuccinimide in (Trifluoromethyl)-benzene D Suarez G Laval S-M Tu D Jiang C L Robinson R Scott B T Golding
1811 Synthesis of Thioflavanone and Flavanone Derivatives by Cyclization of Chalcones W Konieczny M Konieczny
1815 A New and Expedient Total Synthesis of Ochratoxin A and d5-Ochratoxin A B Gabriele M Attya A Fazio L Di Donna P Plastina G Sindona
1821 Synthesis of Benzopyrrolizidinones by NorrishndashYang Cyclization of 3-(Acylmethyl)-2-alkylisoindol-1-ones J Wu W Zhang C Wang
1829 Reactions of MoritandashBaylisndashHillman Acetates with Huisgen Zwitterions A Novel Strategy for the Synthesis of β-Amino Acid Derivatives A Jose R R Paul R Mohan S C Mathew A T Biju E Suresh V Nair
1834 Peracetylated β-Allyl C-Glycosides of D-Ribofuranose and 2-Deoxy- D-ribofuranose in the Chemical Literature Until Now Mirages in the Literature H Otero Martinez H Reinke D Michalik C Vogel
1841 Core-Tetrasubstituted Naphthalene Diimides by Stille Cross-Coupling Reactions and Characterization of Their Optical and Redox Properties S-L Suraru F Wuumlrthner
1846 A Practical Synthesis of Indole-Based Heterocycles Using an Amidoaluminum-Mediated Strategy R Todd M M Hossain
1851 Synthesis of Fluorinated Pyrrolo[23-b]pyridine and Pyrrolo[23-d]pyrimidine Nucleosides V O Iaroshenko Y Wang D V Sevenard D M Volochnyuk
1858 Recyclization Reactions of 5-Formyl-13-dimethyluracil with Electron-Rich Amino Heterocycles A P Mityuk D M Volochnyuk S V Ryabukhin A S Plaskon A Shivanyuk A A Tolmachev
1865 Facile Synthesis of Fluorinated 1-Desazapurines V O Iaroshenko D V Sevenard D M Volochnyuk Y Wang A Martiloga A O Tolmachev
1876 A Practical Synthesis of 3-Diethoxyphosphoryl-12-pyridazine Derivatives J-C Monbaliu J Marchand-Brynaert
1881 Enantioselective Reduction of Prochiral Ketones Employing Sprouted Pisum sativa as Biocatalyst J S Yadav B V S Reddy C Sreelakshmi A B Rao
1886 Application of Phenolate Ion Mediated Intramolecular Epoxide Ring Opening in the Enantioselective Synthesis of Functionalized 23-Dihydrobenzofurans and 1-Benzopyrans S K Dinda S K Das G Panda
1897 Complementary Synthetic Approaches to Constitutionally Diverse N-Aminoalkylated Isoindolinones Application to the Synthesis of Falipamil and 5-HT1A Receptor Ligand Analogues M Lorion A Couture E Deniau P Grandclaudon
1904 Selective Deprotection of Silyl Ethers with Sodium Periodate J Li D Menche
1909 Micellar Solution of Sodium Dodecyl Sulfate (SDS) Catalyzes KabacknikndashFields Reaction in Aqueous Media S Sobhani A Vafaee
1916 Convenient Methods for the Synthesis of a Library of Hemilabile Phosphines M V Jimeacutenez J J Peacuterez-Torrente M I Bartolomeacute L A Oro
1923 Terminal Aziridines by Addition of Grignard Reagents or Organoceriums to an (α-Chloro)sulfinylimine D M Hodgson J Kloesges B Evans
1933 A Robust Synthesis of Nε-(Carboxymethyl)-L-lysine (CML) R Csuk S Stark A Barthel R Kluge D Stroumlhl
1935 One-Pot Curtius Rearrangement Processes from Carboxylic Acids O Leogane H Lebel
XV Forthcoming Articles
no 12 1941 The Chemistry of Deprotonated α-Aminonitriles T Opatz 1960 An Efficient Synthesis of Tetraalkyl 2345-Thiophenetetracarboxylate
Derivatives A Alizadeh R Hosseinpour 1963 Facile Deprotection of Bulky (Trialkylsilyl)acetylenes with Silver Fluoride
S Kim B Kim J In 1969 Highly Efficient and Reusable Ionic Liquids for the Catalyzed
Hydroamination of Alkenes with Sulfonamides Carbamates and Carboxamides L Yang L-W Xu C-G Xia
1975 Synthesis of 2391016172324-Octasubstituted Phthalocyaninatozinc(II) Complexes Mediated by Reductive Agents G A Gauna A C Monsalvo J Awruch
1979 A Short and Efficient Synthesis of 3-2-[2-(Bromomethyl)thiazol-4-yl]-ethynyl-5-fluorobenzonitrile A Precursor for PET Radioligand [18F]SP203 M B Gopinathan C Jin K S Rehder
1983 Synthesis of a Substituted Benzazepin-2-one Dihydrate S K Boini R K Vaid K P Moder D Mitchell
1987 Synthesis of Novel Trisubstituted Imidazolines F J Lakner M A Parker B Rogovoy A Khvat A Ivachtchenko
1991 A Novel Synthesis of N-But-3-enyl-α- and β-Amino Acids T T Van Nguyen R T C Brownlee A B Hughes
1999 Synthesis of Substituted 5-(3-Hydroxypropyl)pyrrolidin-2-ones and Pyrrolizidinones from Nitroethane via C3 Functionalized 56-Dihydro-4H-12-oxazines A Novel Approach to Some Analogues of the Antidepressant Rolipram A Yu Sukhorukov A V Lesiv Y A Khomutova S L Ioffe V A Tartakovsky
2009 Chiral Cyclobutanols and Cyclopentane Dimers via Samarium(II) Iodide Induced Keto-Olefin Cyclisations of Carbohydrate-Derived Unsaturated Ketones D B G Williams J Caddy K Blann J J C Groveacute C W Holzapfel
2015 Synthesis of Perfluoroalkylthio-Substituted Ferrocenes C Rhode J Lemke M Lieb N Metzler-Nolte
2019 Functionalization of Polyhedral Oligomeric Silsesquioxane (POSS) via Nucleophilic Substitution M Dutkiewicz H Maciejewski B Marciniec
2025 A Novel Synthesis of Aryl Mesylates via One-Pot DemethylationndashMesylation of Aryl Methyl Ethers Using a Mixture of Phosphorus Pentoxide in Methanesulfonic Acid B Kaboudin Y Abedi
2029 Anionic Cyclization of (NN-Dimethylamino)[2-(prop-2-yn-1-yloxy)aryl]-acetonitriles T Zdrojewski J Musielak A Jończyk
2035 Strecker-Type Reaction Catalyzed by Carboxylic Acids in Aqueous Media Z Xie G Li G Zhao J Wang
2040 Synthesis of Novel Structurally Simplified Estrogen Analogues with Electron-Donating Groups in Ring A L F Tietze C A Vock I K Krimmelbein L Nacke
2061 On the Resolution of Secondary Phosphine Oxides via Diastereomeric Complex Formation The Case of tert-Butylphenylphosphine Oxide J Holt A M Maj E P Schudde K M Pietrusiewicz L Sieroń W Wieczorek T Jerphagnon I W C E Arends U Hanefeld A J Minnaard
2066 Enantioselective Copper-Catalyzed Conjugate Addition of Dimethylzinc to 5-(1-Arylalkylidene) Meldrumrsquos Acids A Wilsily T Lou E Fillion
2073 SuzukindashMiyaura Coupling Reactions Using Phosphite Ligands M Jang Y Jo I-K Oh H M Jung S Lee
2076 Synthesis of 2-Methylindoline- and 2-Methyl-1234-tetrahydroquinoline-Derived Phosphoramidites and Their Applications in Iridium-Catalyzed Allylic Alkylation of Indoles W-B Liu H He L-X Dai S-L You
2083 Stereocontrolled Synthesis of 13-Amino Alcohols by Reduction of Substituted 2-1-[(tert-Butylsulfinyl)amino]alkylcyclohexanones J C Gonzaacutelez-Goacutemez F Foubelo M Yus
2089 Tunable Phosphoramidite Ligands for Asymmetric Hydrovinylation Ligands par excellence for Generation of All-Carbon Quaternary Centers C R Smith H J Lim A ZhangT V RajanBabu
2101 Copper-Catalyzed Asymmetric Ring-Opening Reaction of Oxabenzonorbornadienes with Grignard and Aluminum Reagents R Millet L Gremaud T Bernardez L Palais A Alexakis
2113 A Simplified Synthesis of Takemotorsquos Catalyst A Berkessel B Seelig 2116 Pharmaceutical Substances Syntheses Patents and Applications of the
Most Relevant AIPs Edited by Axel Kleeman Juumlrgen Engel Bernhard Kutscher Dietmar Reichert Reviewed by I Agranat
XV Forthcoming Articles
no 13 2117 Recent Advances in the Aza-Claisen Rearrangement K C Majumdar
T Bhattacharyya B Chattopadhyay B Sinha 2143 A Novel and Convenient Synthesis of lsquoReversedrsquo Diamidino 25-Aryl- and
25-Azaheterocycle-Substituted Furans L Hu D W Boykin 2146 Efficient and General Preparation of Pyranostilbenes First Total Synthesis
of Artocarbene and Pawhuskin B B H Park Y R Lee W S Lyoo 2155 Mild Oxidation of Diarylacetylenes to 12-Diketones Using Oxone in
Trifluoroacetic Acid J-H Chu Y-J Chen M-J Wu 2163 One-Pot Microwave-Assisted Selective Azido ReductionTandem Cyclization
in Condensed and Solid Phase with Nickel Boride N Shankaraiah N Markandeya M Espinoza-Moraga C Arancibia A Kamal L Silva Santos
2171 Pyrrolo[321-ij]quinolin-4-one and Pyrrolo[321-ij]quinolin-6-one H McNab D J Nelson E J Rozgowska
2175 Practical Synthesis of 5-Substituted Tetrazoles under Microwave Irradiation J Roh T V Artamonova K Vaacutevrovaacute G I Koldobskii A Hrabaacutelek
2179 A Simple Method for the Synthesis of 3-Arylthieno[23-b]pyridines via Iodine-Mediated Cyclization of 3-(1-Arylalkenyl)-2-[(1-phenylethyl)sulfanyl]pyridines K Kobayashi D Nakamura Y Shiroyama S Fukamachi H Konishi
2184 Synthesis of Four Lysine-Linked Cereulide Analogues Showing Ionophoric Activity Towards Potassium Cations as Lead Compounds for Emetic Toxin-Detection by Immunoassays A Makarasen T Nishikawa M Isobe
2205 Synthesis of α-Aliphatic and β-Aromatic Substituted Taurines via Regioselective Ring Opening of Thiiranes with Ammonia H Yu S Cao L Zhang G Liu J Xu
2210 Stability of 5(6)-Carboxyfluorescein in Microwave-Assisted Synthesis of Fluorescein-Labelled O-Dimannosylated Peptides R Kowalczyk P W R Harris R P Dunbar M A Brimble
2223 Diversity-Oriented Synthesis of Functionalized Diaryl Sulfones by Regioselective [3+3] Cyclizations of 13-Bis(siloxy)buta-13-dienes with 2-(Arylsulfonyl)-3-ethoxy-2-en-1-ones Scope and Limitations M Shkoor A Riahi O Fatunsin H Reinke C Fischer P Langer
2236 Synthesis of Functionalized Salicylates by Formal [3+3] Cyclocondensation of 13-Bis(silyloxy)buta-13-dienes with 3-Alkoxy-2-en-1-ones G Mroszlig S Ladzik H Reinke A Spannenberg C Fischer P Langer
2249 Synthetic Approach to Alkoxy-β-(trifluoromethyl)styrenes and Their Application in the Synthesis of New Trifluoromethylated Heterocycles V M Muzalevskiy V G Nenajdenko A V Shastin E S Balenkova G Haufe
2260 o-Benzenedisulfonimide as a Powerful and Recyclable Organocatalyst for the Nazarov Reaction M Barbero S Cadamuro A Deagostino S Dughera P Larini E G Occhiato C Prandi S Tabasso R Vulcano P Venturello
2267 The Catalytic Potential of 4-Guanidinylpyridines in Acylation Reactions I Held E Larionov C Bozler F Wagner H Zipse
2278 Iron(III) Chloride in EthanolndashWater Highly Efficient Catalytic System for the Synthesis of Garcia Gonzalez Polyhydroxyalkyl- and C-Glycosylfurans L Nagarapu M V Chary A Satyender B Supriya R Bantu
2283 Ruthenium-Catalyzed Addition of Primary Amides to Alkynes A Stereoselective Synthesis of Secondary Enamides L J Gooszligen M Blanchot K S M Salih K Gooszligen
2289 Binaphthyl-Modified Quaternary Phosphonium Salts as Chiral Phase Transfer Catalysts Application to Asymmetric Amination of β-Keto Esters R He K Maruoka
X Table of Contents XI Forthcoming Articles
no 14 2293 Direct Methods for Stereoselective Polypropionate Synthesis A Survey
J Li D Menche 2316 Synthesis of Symmetrical Ketones from Grignard Reagents and
11-Carbonyldiimidazole D Bottalico V Fiandanese G Marchese A Punzi
2319 Synthesis of 45-Substituted Imidazoles by a Fast Condensation of 12-Diketones and Urotropine in Heterogeneous Medium G Bratulescu
2321 (Arylsulfonyl)acetones and -acetonitriles New Activated Methylenic Building Blocks for Synthesis of 123-Triazoles N T Pokhodylo V S Matiychuk M D Obushak
2324 A Safe Convenient and Efficient One-Pot Synthesis of α-Chloroketone Acetals Directly from Ketones Using Iodobenzene Dichloride J Yu C Zhang
2329 An Efficient Oxidative Conversion of Aldehydes into 2-Substituted 2-Oxazolines Using 13-Diiodo-55-dimethylhydantoin S Takahashi H Togo
2333 A Novel Procedure for the Synthesis of Benzo[b][18]naphthyridine-3-carboxylate Derivatives from MoritandashBaylisndashHillman Adduct Acetates W Zhong F Lin R Chen W Su
2341 An Improved Synthesis of 147-Triazacyclononanes (tacns) and 14710-Tetraazacyclododecanes (cyclens) J Huang Z Zhou T H Chan
2345 The Ullmann Coupling between 2-Chlorobenzoic Acids and Amino Acids A Valuable Reaction for Preparing 2-Substituted 1-Acetyl-1H-indol-3-yl Acetates J C Rodriguez Dominguez X Gang G Kirsch
2349 gem-Dibromomethyl Aromatics Efficient Aldehyde Equivalents in the KnoevenagelndashDoebner Reaction J K Augustine Y A Naik S Poojari N Chowdappa B S Sherigara K Areppa
2357 Synthesis of Novel α-Aminophosphonates Containing Adamantyl Fragment M M Kabachnik L I Minaeva I P Beletskaya
2361 Efficient Fluoride-Mediated Synthesis of 5-Amino-Substituted Isothiazoles Y S Zubenko V I Potkin
2365 Phosphine-Catalyzed Reaction of Cyanohydrins with Activated Alkynes A Siby O Loreau F Taran
2371 Sulfanyl-Substituted [3]Cumulenes and Buta-13-dienes from a Tetrakis(pyridinium)-Substituted Butadiene A Schmidt A Rahimi M Gjikaj
2379 Efficient Synthesis of 2-Substituted Pyrido[32-d]pyrimidines Involving SNAr and Palladium-Catalyzed Cross-Coupling Reactions A Tikad S Routier M Akssira J-M Leacuteger C Jarry G Guillaumet
2385 Novel Synthesis of Medium-Sized Heterocycles by Palladium-Catalyzed Intramolecular Heck Reaction via 9-endo-trig Mode of Cyclization K C Majumdar B Chattopadhyay
2393 Facile Synthesis of Fluorinated Benzofuro- and Benzothieno[23-b]pyridines α-Carbolines and Nucleosides Containing the α-Carboline Framework V O Iaroshenko Y Wang B Zhang D Volochnyuk V Ya Sosnovskikh
2403 Synthesis of Functionalized N-Vinyl Nitrogen-Containing Heterocycles S M M Lopes A M Beja M Ramos Silva J A Paixatildeo F Palacios T M V D Pinho e Melo
2408 Kumada Cross-Coupling of Aryl Grignard Reagents with Aryl Halides Catalyzed by an Immobilized Nickel Catalyst X Chen L Wang J Liu
2413 Highly Enantioselective Synthesis of Heteroaromatic Alcohols Catalyzed by Chiral DiaminodiphosphinendashRuthenium(II) Complexes W-Y Shen Y-Y Li Z-R Dong J-X Gao
2418 Concise Total Synthesis of (+)-Disparlure and its trans-Isomer Using Asymmetric Organocatalysis S-G Kim
2423 Rhodium Carbenoid Induced [12]-Migration in an L-Lyxo-Configured α-Diazo β-Keto Ester Synthesis of a New Griseolic Acid Analogue N N Bhujbal K S A Kumar D D Dhavale
2430 Synthesis of 5-Arylthio-3-hydroxyphthalates by the First [4+2] Cycloadditions of 3-Arylthio-1-silyloxy-13-butadienes with Dimethyl Acetylenedicarboxylate I Iqbal M Imran P Langer
2435 Synthesis of Highly Functionalized Proline Derivatives via a One-Pot MichaelSN-AdditionCyclization Approach U Kazmaier C Schmidt
2440 RhodiumGraphite-Catalyzed Hydrogenation of Carbocyclic and Heterocyclic Aromatic Compounds G Falini A Gualandi D Savoia
2447 Potassium [1-(tert-Butoxycarbonyl)-1H-indol-2-yl]trifluoroborate as an Efficient Building Block in Palladium-Catalyzed SuzukindashMiyaura Cross Couplings P Kassis V Beacuteneacuteteau J-Y Meacuterour S Routier
2454 Syntheses of Substituted Furans and Pyrroles by Platinum-Catalyzed Cyclizations of Propargylic Oxiranes and Aziridines in Aqueous Media M Yoshida M Al-Amin K Shishido
2467 Transition-Metal-Free Oxidative Homocoupling of Aryl Alkenyl and Alkynyl Grignard Reagents with TEMPO M S Maji A Studer
XIII Forthcoming Articles
no 15 2471 Advances in Synthetic Approaches for the Preparation of Combretastatin-
Based Anti-Cancer Agents R Singh H Kaur 2492 Synthesis of Unsymmetrical Ureas by Sulfur-Assisted Carbonylation with
Carbon Monoxide and Oxidation with Molecular Oxygen under Mild Conditions T Mizuno T Nakai M Mihara
2497 Ring-OpeningRecyclization Reactions of (Dimethylamino)propenoyl-Substituted Cyclopropanes Facile Synthesis of Halogenated Pyridin-2(1H)-ones R Zhang Y Zhou Y Liang Z Jiang D Dong
2501 Facile and Efficient Total Synthesis of Taspine B Cheng S Zhang L Zhu J Zhang Q Li A Shan L He
2505 Oligomeric Iodosylbenzene Sulfate A Convenient Hypervalent Iodine Reagent for Oxidation of Organic Sulfides and Alkenes M S Yusubov R Y Yusubova T V Funk K-W Chi V V Zhdankin
2509 Pyrrolidine-Based Organocatalysts for Enantioselective Michael Addition of Cyclohexanone to trans-β-Nitrostyrene A P Carley S Dixon J D Kilburn
2517 CundashAl Hydrotalcite An Efficient and Reusable Ligand-Free Catalyst for the Coupling of Aryl Chlorides with Aliphatic Aromatic and N(H)-Heterocyclic Amines B Sreedhar R Arundhathi P L Reddy M A Reddy M L Kantam
2523 Highly Efficient Synthesis of trans-βγ-Unsaturated a-Keto Amides C Allais T Constantieux J Rodriguez
2531 Gas-Phase Synthesis of N-Unsubstituted 3-Hydroxypyrroles and 1H-Pyrrol-3(2H)-ones L Hill G A Hunter S H Imam H McNab W J OrsquoNeill
2535 3-Hydroxy-1H-pyrrole L Hill S H Imam H McNab W J OrsquoNeill 2539 123-Thiadiazoles with Unsaturated Side Chains Synthesis
Polymerization and Photocrosslinking M Al-Smadi N Hanold H Kalbitz H Meier
2547 Synthesis of 1112-Didehydrodibenzo[ae]cycloocten-5(6H)-one A Strained Eight-Membered Alkyne S C Kornmayer F Rominger R Gleiter
2553 Stannous Chloride Dihydrate A Novel and Efficient Catalyst for the Synthesis of gem-Dihydroperoxides from Ketones and Aldehydes D Azarifar K Khosravi F Soleimanei
2557 Synthesis of a Novel Class of Azacrown Macrocycles and Lariat Crown Ethers Containing Two 124-Triazole Rings as Subunits N Foroughifar A Mobinikhaledi S Ebrahimi
2561 Enantioselective Synthesis of the 3C-Protease Inhibitor (ndash)-Thysanone by a StauntonndashWeinreb Annulation Strategy J Sperry T Y Yuen M A Brimble
2570 Stereoselective Synthesis of Unnatural β-Amino Acids from Nitroethane via 56-Dihydro-4H-12-oxazin-3-ylacetates A Yu Sukhorukov A V Lesiv O L Eliseev Y A Khomutova S L Ioffe
2579 A Versatile Unexpected One-Pot Regioselective Synthesis of a New Class of 13-Diazepinoindolones by Reaction of Pyranoindolones with Monosubstituted Ureas D Livadiotou C A Tsoleridis J Stephanidou-Stephanatou
2584 Synthesis of a Trisaccharide and a Tetrasaccharide from the Cell-Wall Lipopolysaccharides of Azospirillum brasilense S17 S Pandey S Ghosh A K Misra
2591 Synthesis of Isoindoline Nitroxides by Electrocyclic Reactions T Kaacutelai J Jekı K Hideg
2596 Glycosylations of Tertiary Alcohols Synthesis of Fully Protected Disaccharides with Sterically Demanding Groups Attached to the Sugar Core A Holkenbrink J B Vicente D B Werz
2605 Copper-Catalyzed [13]-Dipolar Cycloaddition for the Synthesis of Macrocycles Containing Acyclic Aromatic and Steroidal Moieties G V Latyshev M S Baranom A V Kazantsev A D Averin N V Lukashev I P Beletskaya
2616 Aryl Ring Migration Reaction in the Synthesis of 24-Diaryl-4H-31-benzothiazines A V Butin F A Tsiunchik V T Abaev A V Gutnov D A Cheshkov
2627 Hydrogenation of β-N-Substituted and β-NN-Disubstituted Enamino Esters in the Presence of Iridium(I) Catalyst H Hebbache Z Hank C Bruneau J-L Renaud
2634 Stereoselective Olefination Reactions Promoted by Rieke Manganese J M Concelloacuten H Rodriacuteguez-Solla V del Amo P Diacuteaz
2646 Synthesis of Piperidinones through a Radical Cascade E Godineau Y Landais
2650 Asymmetric Organic Synthesis with Enzymes Edited by V Gotor I Alfonso E Garciacutea-Urdiales Reviewed by Steve Collier
XVII Forthcoming Articles
no 16 2651 Synthesis of Spirocyclic Ethers S Rosenberg R Leino 2674 Bimetallic PalladiumndashPlatinum-on-Carbon-Catalyzed HndashD Exchange
Reaction Synergistic Effect on Multiple Deuterium Incorporation T Maegawa N Ito K Oono Y Monguchi H Sajiki
2679 Efficient Copper-Catalyzed Synthesis of 2-Amino-4(3H)-quinazolinone and 2-Aminoquinazoline Derivatives X Huang H Yang H Fu R Qiao Y Zhao
2689 Synthesis and Chemoselective N- and O-Alkylation of Thiadiazolopyrimidine Nucleosides and Uridines A M L Hossion R Islam R K Kandahary T Nagamatsu
2697 Facile and Efficient Synthesis of a New Class of Indole-Substituted Pyridine Derivatives via One-Pot Multicomponent Reactions K Zhao X-P Xu S-L Zhu D-Q Shi Y Zhang S-J Ji
2709 Studies toward a Total Synthesis of Rhizoxin D Stereoselective Preparation of the C11ndashC19 Fragment S Padakanti C K Kumar E Ashok P Das
2715 A Short Synthesis of Enantiomeric Phytoprostanes B1 Type I W Perlikowska M Mikołajczyk
2719 Chemistry of Polyhalogenated Nitrobutadienes Part 7 A Novel Synthetic Access to Chlorinated Nitrile Oxides E Nutz V A Zapolrsquoskii D E Kaufmann
2725 Microwave-Assisted Silver(I)-Mediated Selective O-Alkylation of Aromatic Imidate Systems B K Singh C Cavalluzzo M De Maeyer Z Debyser V S Parmar E Van der Eycken
2729 Iodogen A Novel Reagent for the Oxidation of Urazoles under Heterogeneous Conditions A Khoramabadi A Shiri M A Zolfigol S Mallakpour
2733 An Unprecedented Synthesis of Eight-Membered-Ring Cyclic Thioimidic Esters by a Three-Component Reaction A Alizadeh R Hosseinpour
2737 A Novel Diastereoselective Synthesis of β-Phosphonato Unsaturated Thioimidates A Alizadeh N Zohreh
2741 Synthesis of 21-Benzisoxazoles by Nucleophilic Substitution of Hydrogen in Nitroarenes Activated by the Azole Ring N T Pokhodylo Y O Teslenko V S Matiychuk M D Obushak
2749 A Facile Synthesis of Two Series of Multifunctional Carbon Compounds from αα-Dihalo Ketones Using Allylsamarium Bromide X Liu S Zhang J Di
2756 Stereocontrolled Formation of Protected Aminodeoxyalditols from Simple Carbohydrate Precursors by Debenzylating Cycloetherification Y Jiang Z Fang Q Zheng H Jia J Cheng B Zheng
2761 trans-Stilbene as a Starting Material for the Synthesis of Tamoxifen Based on Palladium-Catalyzed Cross-Coupling Reactions C M Nunes J Limberger S Poersch M Seferin A L Monteiro
2766 Synthesis and Biological Evaluation of 6-Substituted Purinylcarbanucleosides with a Cyclopenta[b]thiophene Pseudosugar P Abeijoacuten J M Blanco O Caamantildeo F Fernaacutendez M D Garciacutea X Garciacutea-Mera J E Rodriacuteguez-Borges J Balzarini E De Clercq
2773 Synthesis and Electrochemical Signature of Novel Norbornyl-ferrocene Hybrids F A Khan S K Upadhyay
2778 A Regioselective TsujindashTrost Pentadienylation of 3-Allyltetronic Acid R Schobert B Barnickel
2785 Copper(I)-Catalyzed CarylndashCalkynyl Bond Formation of Aryl Iodides with Terminal Alkynes K G Thakur G Sekar
2790 Aminolysis of Epoxides Using Iridium Trichloride as an Efficient Catalyst J Agarwal A Duley R Rani R K Peddinti
2797 Preparation of Several Active N-Chloro Compounds from Trichloroisocyanuric Acid A Shiri A Khoramabadi-zad
2802 The First Mineral-Catalyzed One-Pot [3+1+2] Coupling Protocol for Multifunctionalized Fused-Ring Pyrimidines L D S Yadav A Rai
2809 Efficient Synthesis of Tetrahydro-β-carbolin-1-one and Dihydroisoquinolin-1-one Derivatives as Versatile Intermediates K E Judd M F Mahon L Caggiano
2818 A Concise Synthesis of ortho-Iodobenzyl Alcohols via Addition of ortho-Iodophenyl Grignard Reagent to Aldehydes and Ketones J Cvengroš D Stolz A Togni
XIII Forthcoming Articles
no 17 2825 Reactivity of Oxazol-5-(4H)-ones and Their Application toward Natural
Product Synthesis N M Hewlett C D Hupp J J Tepe 2840 Towards the Total Synthesis of 3-Hydroxyvibsanin E B D Schwartz
J R Denton P V Bernhardt H M L Davies C M Williams 2847 Structure Investigations of (ent)-Cladospolide D by De Novo Synthesis and
Kinetic and Thermodynamic Isomerization Y Xing J H Penn G A OrsquoDoherty
2855 New Applications of PhI(OAc)2 in Synthesis Total Synthesis and SAR Development of Potent Antitumor Natural Product PsymberinIrciniastatin A N Shao X Huang A Palani R Aslanian A Buevich J Piwinski R Huryk C Seidel-Dugan
2873 Total Synthesis of Largazole ndash Devolution of a Novel Synthetic Strategy B Wang C J Forsyth
2881 Formal Total Synthesis of Palmerolide A J Jaumlgel M E Maier 2893 Total Synthesis of Bongkrekic Acid via Sequential SuzukindashMiyaura Coupling
Reactions M Kanematsu M Shindo M Yoshida K Shishido 2905 Stereodivergent Approach to Both C28a-syn and C28a-anti Relative
Stereochemical Manifolds in the Lepadin Family via a TiCl4-Promoted G Li L J Carlson I K Sagamanova B W Slafer R P Hsung C Gilardi H M Sklenicka N Sydorenko
2915 Enantioselective Aldol Reaction of Tetrasubstituted Ketene Silyl Acetals with Achiral Aldehydes for the Construction of Asymmetric Tertiary Alcohols An Application for the Divergent Total Syntheses of Buergerinins F and G I Shiina T Iizumi Y-s Yamai Y-i Kawakita K Yokoyama Y-k Yamada
2927 Second-Generation Biomimetic Total Synthesis of Chaetominine A Coste G Karthikeyan F Couty G Evano
2935 Total Synthesis of (+)-Fostriecin and (+)-Phoslactomycin B S Shibahara M Fujino Y Tashiro N Okamoto T Esumi K Takahashi J Ishihara S Hatakeyama
2954 Stereochemical Assignments of the Chlorinated Residues in Victorin C A C Durow C Butts C L Willis
2963 Studies of the Asymmetric Total Synthesis of Clavilactone D by the lsquoLariatrsquo Cyclization Strategy T Yoshimitsu S Nojima M Hashimoto K Tsukamoto T Tanaka
2970 Total Synthesis of the Leucetta-Derived Alkaloid Calcaridine A P B Koswatta R Sivappa H V R Dias C J Lovely
2983 Formal Synthesis of Salinosporamide A Starting from D-Glucose T Momose Y Kaiya J-i Hasegawa T Sato N Chida
2992 Synthesis of Bioactive Natural Products by Asymmetric syn- and anti-Aldol Reactions A K Ghosh Z L Dawson
no 18 3003 Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural
Products B M Trost M K Brennan 3026 One-Pot Synthesis of Furo[34-b]pyridin-5(7H)-ones from 2-
Bromopyridine-3-carboxylic Acid and Carbonyl Compounds K Kobayashi T Kozuki H Konishi
3029 Iodocyclization of N-[2-(Methylthio)phenyl]propiolamides Selective Synthesis of 3-Iodo-15-benzothiazepin-4-ones T-S Jiang X-G Zhang J-H Li
3039 A Facile Synthetic Method for Fluorine-Containing 17-Phenanthrolines Pyridine-Ring Formation Reaction of N-Propargyl-68-bis(trifluoroacetyl)-quinolin-5-amine with Various Nucleophiles D Shibata E Okada M Hinoshita M Meacutedebielle
3047 Enantiotopic Discrimination in Palladium-Mediated Nucleophilic Substitutions on Achiral Substrates Chiral Ligand versus Chiral Nucleophile O Jacquet F Charnay J-C Fiaud J Ollivier
3051 Studies on the Chemistry of 2-[3-(2-Nitrophenyl)-2-oxopropyl]benzaldehydes Novel Syntheses of 5H-Benzo[b]carbazole-611-diones and Indolo[12-b]isoquinoline-611-diones M Fernaacutendez
3061 Studies on the C22ndashC23 Aldol Coupling of Spirangien M Lorenz N Bluhm M Kalesse
3067 One-Pot Synthesis of N-Alkyl Purine Pyrimidine and Azole Derivatives from Alcohols using Ph3PCCl4 A Rapid Route to Carboacyclic Nucleoside Synthesis M N Soltani Rad A Khalafi-Nezhad S Behrouz Z Asrari M Behrouz Z Amini
3077 Synthesis of 2-Amino-34-dihydroquinazolines and Imidazo[21-b]quinazoline-2-ones A Mishra S Batra
3089 Studies on the Reaction of Diimines with Thiourea Synthesis and Solvent-Induced cistrans-Isomerization of 135-Triazinane-2-thiones B Kaboudin T Ghasemi T Yokomatsu
3094 Suzuki Coupling of Heteroaromatic Chlorides Using Highly Electron-Donating ClickPhos Ligands S M Spinella Z-H Guan J Chen X Zhang
3099 Reaction of NN-Dioxyenamines with Anhydrides of Carboxylic and Sulfonic Acids A New Method for the Synthesis of a-Hydroxyoxime Derivatives A A Tabolin A V Lesiv S L Ioffe
3106 Directed ortho Metallation Chemistry and Phosphine Synthesis New Ligands for the SuzukindashMiyaura Reaction D B G Williams S J Evans H de Bod M S Mokhadinyana T Hughes
3113 New Functional Derivatives of 9-Phenylquinine P J Boratyński J SkarŜewski
3120 On the Synthesis of Asymmetric and Dissymmetric Amino Analogues of Troumlgerrsquos Base J Artacho K Waumlrnmark
3127 Synthesis of Polycyclic Sultams by Palladium-Catalyzed Intramolecular Cyclization K C Majumdar S Mondal N De
3136 Synthesis of Functionalized L-Cysteine and L-Methionine by Reaction with Electron-Deficient Acetylenes B A Trofimov A G Malrsquokina O A Shemyakina V V Nosyreva A P Borisova S S Khutsishvili L B Krivdin
3143 A lsquoClickrsquo Approach to the Synthesis of 3-[2-(1-Alkyltriazol-4-yl)ethyl]indoles M Petrini R R Shaikh
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
655 Synthesis of (ndash)-Monomorine I R W Bates P Song 660 Cobalt(II) Chloride HexahydratendashDiisopropylamine Catalyzed Mild and
Chemoselective Reduction of Carboxylic Esters with Sodium Borohydride A R Jagdale A S Paraskar A Sudalai
665 Synthesis of Bi- and Tricyclic αβ-Unsaturated Lactams as Potential Michael Acceptors Starting from Heterocyclic Imines K Schulz M Watzke K Johannes P Ullrich J Martens
674 An Expedient Synthesis of Bis-Fused Benzofuran and a Two-Directional Ring-Closing Metathesis for the Synthesis of Bisbenzoxepines and Bisbenzoxocines K C Majumdar B Chattopadhyay S Chakravorty
681 Palladium-Catalyzed Cross-Couplings of Unsaturated Halides Bearing Relatively Acidic Hydrogen Atoms with Organozinc Reagents Z Dong G Manolikakes J Li P Knochel
687 Synthesis of Enantioenriched aa-Disubstituted Cyclopentenes Catalyzed by N-Heterocyclic Carbenes E M Phillips M Wadamoto K A Scheidt
XVII Forthcoming Articles
No 5 691 Transannulation Reactions in the Synthesis of Natural Products
P A Clarke A T Reeder J Winn 710 Synthesis of DL-erythro-Sphingosine Using a Tethered
Aminohydroxylation Reaction as the Key Step J A Morales-Serna Y Diacuteaz M I Matheu S Castilloacuten
713 Convenient Multigram Synthesis of 4-Chloropyridine-26-dicarbonyl Dichloride K Mitsui J R Parquette
715 A Novel and Efficient Synthesis of Dihydrexidine J P Cueva D E Nichols
721 Synthesis of 57-Dichloro-6-azaindoles and Functionalization via a Highly Selective LithiumndashChlorine Exchange N Lachance L-P Bonhomme-Beaulieu P Joly
731 A Convenient Synthesis of Fluorinated Pyrazolo[34-b]pyridine and Pyrazolo[34-d]pyrimidine Nucleosides V O Iaroshenko D V Sevenard A Kotljarov D M Volochnyuk A O Tolmachev V Y Sosnovskikh
741 Diastereoselective Synthesis of γ-Amino Acids and Their Derivatives from Nitroethane via Intermediacy of 56-Dihydro-4H-12-oxazines Bearing the CH2CH(CO2Me)2 Substituent at C3 A Y Sukhorukov A V Lesiv Y A Khomutova S L Ioffe
755 Synthesis of a New Pyrrolopyridoindole and Its Pyrrolopyridobenzimidazole Regioisomer F Bouchikhi M Sassatelli F Anizon M Prudhomme P Moreau
759 Practical Syntheses of Sphingosine-1-Phosphate and Analogues V Blot U Jacquemard H-U Reissig B Kleuser
767 A Facile Synthetic Route towards Substituted Thieno[32-e]indoles W Van Snick W Nulens S Jambon W Dehaen
775 Microwave-Assisted One-Pot Synthesis of (Aminoalkyl)naphthols and (Aminoalkyl)quinolinols by Using Ammonium Carbamate or Ammonium Hydrogen Carbonate as Solid Ammonia Source I Szatmaacuteri F Fuumlloumlp
779 Enantioselective Synthesis of Flavan-3-ols Using a Mitsunobu Cyclization K Krohn I Ahmed M John 787 Synthesis of a Novel γ-Folic AcidndashNτ-Histidine Conjugate Suitable for
Labeling with 99mTc and 188Re C Sparr U Michel R E Marti C Muumlller R Schibli R Moser V Groehn
793 Palladium-Catalyzed Intramolecular Biaryl Coupling A Highly Efficient Avenue for Benzannulated Pyranoquinolines and Julolidine Derivatives K C Majumdar A Taher P Debnath
801 Preparation of NN-Dimethyl-N-Arylureas Using SS-Dimethyl Dithiocarbonate as a Carbonylating Reagent I Degani R Fochi C Magistris M Migliaccio
809 Versatile Selective α-Carboxylic Acid Esterification of N-Protected Amino Acids and Peptides by Alcalase T Nuijens C Cusan J A W Kruijtzer D T S Rijkers R M J Liskamp P J L M Quaedflieg
815 Efficient Palladium-Catalyzed Amination of Aryl Chlorides Using Dicyclohexylamino[(26-dimethyl)morpholino]phenylphosphine as a PN2 Ligand S-E Park S B Kang K-J Jung J-E Won S-G Lee Y-J Yoon
824 A Clean Facile and Stereospecific Synthesis of α-Oxoketene OS-Acetals in Water Y Li Q Zhang X Cheng Q Liu X Xu
829 Sonogashira Cross-Coupling Reactions and Construction of the Indole Ring System Using a Robust Silica-Supported Palladium Catalyst E Tyrrell L Whiteman N Williams
836 Synthesis of Angular 78-Pyridazinocoumarins via the Transformation of a Hydroxy Group into a Carbonyl Group A Kotali I S Lafazanis P A Harris
841 Synthesis of New Cyclic and Acyclic 5-Halouridine Derivatives as Potential Antiviral Agents M F Elshehry J Balzarini C Meier
848 Dendritic Triphenylmethylium and Tetraphenylmethane Compounds H Meier S Kim A Oehlhof
853 Synthesis of Homoallylic Alcohols via Lewis Acid Assisted Enantioselective Desymmetrization B Yu F Menad N Isono M Lautens
860 Diastereoselective Synthesis of 123-Trisubstituted Indanes via Rhodium(I)-Catalyzed Tandem Conjugate Additions C Navarro A G Csaacutekyuml
864 Bakerrsquos Yeast for Sweet Dough Enables Large-Scale Synthesis of Enantiomerically Pure Bicyclo[331]nonane-26-dione C J Wallentin E Orentas E Butkus K Waumlrnmark
868 Addendum and Erratum XV Forthcoming Articles
No 6 869 Stereoselective Transformations of meso Bicyclic Hydrazines Versatile
Access to Functionalized Aminocyclopentanes C Bournaud F Chung A P Luna M Pasco G Errasti T Lecourt L Micouin
888 Synthesis of Glycoaminoxy Acids as Novel Sugar Building Blocks A Malapelle R Ramozzi J Xie
891 Electrophilic ipso-Halocyclization of N-Arylpropynamides with Polyfluoroalkyl Alcohols Selective Synthesis of 8-(Polyfluoroalkoxy) azaspiro[45]trienes Z-Q Wang B-X Tang H-P Zhang F Wang J-H Li
903 Electrooxidation of Alcohols in N-Oxyl-Immobilized Silica GelWater Disperse System Approach to Totally Closed System M Kuroboshi K Goto H Tanaka
909 Synthetic Routes to Aminotriamantanes Topological Analogues of the Neuroprotector Memantinereg A A Fokin A Merz N A Fokina H Schwertfeger S L Liu J E P Dahl R K M Carlson P R Schreiner
913 Parallel Synthesis of Drug-like 5-Amino-Substituted 124-Thiadiazole Libraries Using Cyclization Reactions of a Carboxamidine Dithiocarbamate Linker J Y Park I A Ryu J H Park D C Ha Y-D Gong
921 Copper-Catalyzed Selective S-Arylation of 12-Bis(o-amino-1H-pyrazolyl) Disulfides with Arylboronic Acids P-S Luo F Wang J-H Li R-Y Tang P Zhong
929 2-Iodoxybenzoic AcidTetraethylammonium BromideWater An Efficient Combination for Oxidative Cleavage of Acetals C Kuhakarn W Panchan S Chiampanichayakul N Samakkanad M Pohmakotr V Reutrakul T Jaipetch
935 Synthesis of Quinonoid Analogues of Diospyrin S Sagar I R Green 941 A One-Pot Method for the Iodination of Aryl Amines via Stable Aryl
Diazonium Silica Sulfates Under Solvent-Free Conditions A Zaroi A R Hajipour L Khazdooz
945 Poly(NN-dichloro-N-ethylbenzene-13-disulfonamide) and NNNN-Tetrachlorobenzene-13-disulfonamide as Novel Reagents for the Synthesis of N-Chloroamines Nitriles and Aldehydes R Ghorbani-Vaghei H Veisi
951 Synthesis of an (R)-Garner-type Aldehyde from L-Serine Useful Building Block for a (+)-Furanomycin Derivative G Bartoli G Di Antonio R Fiocchi S Giuli E Marcantoni M Marcolini
957 An Efficient and Highly Selective Synthesis of (Z)-Fluoroenol Phosphates from Hydroxy Difluorophosphonates P Beier R Pohl A V Alexandrova
963 Iodine-Catalyzed Three-Component Reaction A Rapid Synthesis of α-Alkoxy Azides and Homoallyl Ethers J S Yadav B V S Reddy G M Reddy R Narender
969 Rhodium(I)-Catalyzed Cycloisomerization of 13-Dienes with Alkenes in a Tether Y Oonishi A Saito M Mori Y Sato
980 Synthesis of New Optically Active D-GlucosaminendashPyrrole Derivatives B A Frontana-Uribe M V Escaacutercega-Bobadilla J Juaacuterez-Lagunas R A Toscano G A Garciacutea de la Mora M Salmoacuten
985 Partially Saturated Indeno[12-b]indole Derivatives via Deoxygenation of Heterocyclic α-Hydroxy-NO-hemiaminals H-J Hemmerling G Reiss
1000 Light-Induced Synthesis of Π-Extended Tetrathiafulvalenes Incorporating Ferrocenes An Efficient Route for the Synthesis of Electron-Donor Materials A A O Sarhan C Bolm
1007 Preparation of Nβ-Fmoc-Protected Aza-β3-Amino Acids with Nonproteinogenic Hydrophobic Side Chains for Solid-Phase Syntheses of Pseudopeptides M Laurencin P Bauchat M Baudy-Flocrsquoh
1014 Diastereomeric (η4-diene)Fe(CO)3 Complexes Containing Chiral Amide Groups A Convenient Method for the Resolution of Amino Acids M Schumacher G Coste L Miesch
1021 Palladium-Catalysed Heck Reactions of Alk-1-en-3-ones with Aryl Bromides A Very Simple Access to (E)-1-Arylalk-1-en-3-ones M Lemhadri Y Fall H Doucet M Santelli
1036 An Improved Process for the Synthesis of 4H-Imidazo[15-α][14]benzodiazepines J Yang Y Teng S Ara S Rallapalli J M Cook
1041 Meta- and Para-Difunctionalization of Arenes via an Ortho-Magnesiation and a Subsequent SulfoxidendashMagnesium Exchange L Melzig C B Rauhut P Knochel
XIII Forthcoming Articles
No 7 1049 Catalytic Transformations of Benzylic Carboxylates and Carbonates
R Kuwano 1062 A Simple and Practical Method for the Oxidation of Thebaine to 14-
Hydroxycodeinone by V2O5ndashH2O2 S Das Sharma D Konwar 1065 Umpolung with Sulfur Dioxide CarbonndashCarbon Cross-Coupling of Electron-
Rich 13-Dienes and Alkenes Application to the Enantioselective Synthesis of Long-Chain Polyketide Fragments M Turks C J Exner C Hamel P Vogel
1075 One-Pot Synthesis of 14-Diarylnaphthalenes via a WittigndashHorner Reaction[4+2] CycloadditionDehydrogenation Sequence Z Chen W Shou Y Wang
1081 A Novel and General Method for the Formation of S-Aryl Se-Aryl and Te-Aryl Phosphorochalcogenoates Y-X Gao G Tang Y Cao Y-F Zhao
1087 A Remarkable Access to γ-Fluoroalkylated Propargylamine Derivatives or Fluoroalkylated Dihydroisoxazoles via the Reaction of Fluoroalkylated Acetylides with Various Nitrones T Konno K Moriyasu T Ishihara
1095 Short and Practical Syntheses of (S)-(+)-3-(p-Tolylsulfinyl)furan-2(5H)-one and (S)-(+)-3-(p-Tolylsulfinyl)-56-dihydropyran-2-one D Cruz Cruz A Hernaacutendez Linares F Yuste M R Martiacuten J L Garciacutea Ruano
1099 Decarboxylative Aldol-Type Reaction of 2-(Trifluoroacetyl)-13-diazoles with Activated Acetic Acids P V Khodakovskiy D M Volochnyuk A A Tolmachev
1105 Synthesis of 2-[(Arylmethylene)amino]cyclopropanecarbonitriles via a Two-Step Ring Transformation of 2-(Cyanomethyl)aziridines S Mangelinckx M Drsquohooghe S Peeters N De Kimpe
1113 Synthesis of Dendrimeric Tumor-Associated Mucin-Type Glycopeptide Antigens T Becker A Kaiser H Kunz
1123 A Simple and Efficient Oxidation Procedure for the Synthesis of Acid-Sensitive Epoxides O Bortolini G Fantin M Fogagnolo
1127 Rapid Chemoselective Deprotection of Benzyl Esters by Nickel Boride J M Khurana R Arora
1131 Three-Component Coupling of Isoquinoline Activated Alkyne and Nitromethane A Facile Synthesis of Nitromethyl Derivatives of 12-Dihydroisoquinolines J S Yadav B V S Reddy N N Yadav M K Gupta
1137 Palladium Supported on a Polyionic Resin as an Efficient Ligand-Free and Recyclable Catalyst for Heck SuzukindashMiyaura and Sonogashira Reactions B Basu S Das P Das B Mandal D Banerjee F Almqvist
1147 Oxidation of 25-Dialkylpyrrole Derivatives with Cerium(IV) Ammonium Nitrate R Voloshchuk M Gałęzowski D T Gryko
1153 Practical Syntheses of Enantiomerically Pure Key Intermediates of Opioid Receptor-like 1 (ORL1) Antagonists T Yoshizumi A Ohno T Tsujita H Takahashi O Okamoto I Hayakawa H Kigoshi
1163 An Environmentally Benign TEMPO-Catalyzed Efficient Alcohol Oxidation System with a Recyclable Hypervalent Iodine(III) Reagent and Its Facile Preparation X-Q Li C Zhang
1170 Efficient and Stereoselective Rearrangement of BaylisndashHillman Acetates Catalyzed by Gold(I) ChlorideSilver(I) Trifluoromethanesulfonate Y Liu D Mao J Qian S Lou Z Xu Y Zhang
1175 The First Total Synthesis of Kynapcin-24 by Palladium Catalysis L-Y Yang C-F Chang Y-C Huang Y-J Lee C-C Hu T-H Tseng
1180 Enantioselective Synthesis of N-Protected α-Amino Acid Hydrazides M Bibian S El-Habnouni J Martinez J-A Fehrentz
1185 Synthesis of 11H-Indolo[32-c]quinoline-6-carboxylic Acids by Cascade AutoxidationndashRing Contractions A Becker S Kohfeld T Pies K Wieking L Preu C Kunick
1190 Reaction of N-Nonaflylbenzotriazole with Silyl Enol Ethers M Uhde T Ziegler
1195 2-(Benzoylimino)thiazolidin-4-ones Formation by an Alternative Ring Closure and Analysis of Rotational Barriers H-G Haumlcker P W Elsinghorst S Michels J Daniels G Schnakenburg M Guumltschow
1204 Microwave-Assisted Synthesis and Functionalization of Selenolopyrimidines S Hesse C Chenet D Thomae G Kirsch
1209 12-Disubstituted 4-Quinolones via Copper-Catalyzed Cyclization of 1-(2-Halophenyl)-2-en-3-amin-1-ones R Bernini S Cacchi G Fabrizi A Sferrazza
1220 A New Atom-Economical and Selective Synthesis of Secondary and Tertiary Alkylamines by Means of CpIridium Complex Catalyzed Multiple N-Alkylation of Ammonium Salts with Alcohols without Solvent R Yamaguchi Z Mingwen S Kawagoe C Asai K-i Fujita
1224 Synthesis of Regioisomerically Pure 5-Functionalized 27-Dichlorofluoresceins J C Castro A Malakhov K Burgess
XIII Forthcoming Articles
No 8 1227 Michael Additions to Activated Vinylphosphonates T Janecki J Kędzia
T Wąsek 1255 A Facile and General Synthesis of 2β-Aminosteroids X Ke H Hu
D Zhou W Xu Q Zhu N P Reddy X Hu 1261 Efficacious Preparation of Oppolzerrsquos Glycylsultam via the Deleacutepine
Reaction A Isleyen C Gonsky R C Ronald P Garner 1265 Synthesis of Masked Vicinal Amino Aldehydes of Pyrrolizine and Pyrrolo
[12-c]thiazole Series A V Tverdokhlebov A V Denisenko A A Tolmachev Y M Volovenko S V Shishkina O V Shishkin
1271 Preparation of 9-Substituted Pyridine-Stretched Adenines and Hypoxanthines J A Crawford W Fraser C A Ramsden
1279 A Versatile Synthesis of Heterocyclic Analogues of Neoflavonoids from Enamino Ketones V S Moskvina V P Khilya O V Turov U M Groth
1287 New Stereoselective Synthesis of Paeonilactone B F G Gatti S Serra 1291 The Use of NN-Dialkyltrimethylsilylamines in the Synthesis of
Pentamethinium Salts M Kořiacutenek M Rybaacutečkovaacute Boumlhm 1297 Synthesis of Triazoles via Regioselective Reactions of Aryl Azides with
Cyanoacetyl Pyrroles and Indoles N T Pokhodylo V S Matiychuk M D Obushak
1301 Gallium(III) Chloride Catalyzed Hydroarylation of Arylacetylenes with Naphthols and Phenols A Facile Synthesis of Vinylarenes J S Yadav B V S Reddy S Sengupta S K Biswas
1305 Electrophilic Bromination of meta-Substituted Anilines with N-Bromosuccinimide Regioselectivity and Solvent Effect S Bartoli A Cipollone A Squarcia A Madami D Fattori
1309 Cross-Coupling Reactions of Halopurines with Aryl- and Alkyltrifluoroborates The Scope and Limitations in the Synthesis of Modified Purines Z Hasniacutek R Pohl M Hocek
1318 A Convenient Method for Converting Hydroxyacetophenones into Their Ethylene or Trimethylene Acetals F Ono H Takenaka T Fujikawa M Mori T Sato
1323 γ-Chloromagnesio γ-Lactones and δ-Chloromagnesio δ-Lactones Generation Properties and Synthetic Uses H Shimizu S Fukuda S Sugiyama T Satoh
1336 Click Reactions with Nitroxides T Kaacutelai W L Hubbell K Hideg 1341 Synthesis of Novel 14-Benzoquinone-Containing 123-Triazoles An Entry
Into a New Library F Algi M Balci 1348 Efficient Synthesis of Two Sialylated Tetrasaccharides Found in Goat Milk
P K Mandal A K Misra 1355 Dendrimers of Vaccines Consisting of Tumor-Associated Glycopeptide
Antigens and T Cell Epitope Peptides S Keil A Kaiser F Syed H Kunz
1370 IBXTBAB-Mediated Oxidation of Primary Amines to Nitriles F Drouet P Fontaine G Masson J Zhu
1375 Chemoselectivity of Multicomponent Condensations of Barbituric Acids 5-Aminopyrazoles and Aldehydes E A Muravyova S V Shishkina V I Musatov I V Knyazeva O V Shishkin S M Desenko V A Chebanov
1386 Stereoselective Total Syntheses of Leiocarpin A and (ndash)-Galantinic Acid Starting from D-Mannitol K Nagaiah D Sreenu K V Purnima R S Rao J S Yadav
1393 A Facile Mild Deprotection Protocol for 13-Dithianes and 13-Dithiolanes with 30 Hydrogen Peroxide and Iodine Catalyst in Aqueous Micellar System N C Ganguly S K Barik
1400 Rhodium-Catalyzed Gram-Scale Synthesis of Highly Substituted Pyridine Derivatives K Parthasarathy C-H Cheng
1403 Enantioselective Synthesis of (R)-Propylene Carbonate from Ethyl (S)-Lactate J M Whitaker R C Ronald
XIII Forthcoming Articles
no 9 1405 Transition-Metal-Catalyzed Site-Selective Cross-Coupling of Di- and
Polyhalogenated Compounds J-R Wang K Manabe 1428 An Improved Synthesis of (4-4-Hydroxy-3-isopropyl-5-[(4-nitrophenyl)
ethynyl]benzyl-35-dimethylphenoxy)acetic Acid (NH-3) M B Gopinathan K S Rehder
1431 Copper-Catalyzed Tandem CndashN Bond Formation Reaction Selective Synthesis of 2-(Trifluoromethyl)benzimidazoles M-W Chen X-G Zhang P Zhong M-L Hu
1437 Synthesis and Thermochemical Properties of Stereoisomeric Dihydroxy- and Tetrahydroxyalkylammonium Salts M Thomas L Rothman J Hatcher P Agarkar R Ramkirath S Lall-Ramnarine R Engel
1445 Preparation of 5-Substituted 2-(2-Alkylaryl-1H-imidazol-4-yl)oxazoles and 5-Substituted 2-(2-Alkylarylthiazol-4-yl)oxazoles by Utilizing 5-Substituted 2-(2-Bromo-11-diethoxyethyl)oxazole as a Synthon D R St Laurent J L Romine
1459 Novel and Efficient Methods for the Synthesis of Symmetrical Trisulfides A Kertmen S Lach J Rachon D Witt
1463 An Environmentally Benign Electrochemical Process for the Reduction of Carboxylic Acid Hydrazides to Amides M Mentel M J Beier R Breinbauer
1469 Synthesis of 1-Chloroalkynes from Alkynylsilanes Using Trichloroisocyanuric Acid as Chlorinating Agent M H Vilhelmsen A S Andersson M B Nielsen
1473 A Convenient Approach to Enantioenriched Cyclopropanes Bearing Electron-Withdrawing Functionalities H Krawczyń K Wąsek J Kędzia
1477 Synthesis of Cyclopropenes via 12-Elimination of Bromocyclopropanes Catalyzed by Crown Ether W M Sherrill R Kim M Rubin
1485 A Base-Catalysed One-Pot Three-Component Coupling Reaction Leading to Nitrosubstituted Pyrroles I R Baxendale C D Buckle S V Ley L Tamborini
1494 Synthesis of 4-Alkylidene-4H-31-benzoxazine Derivatives by Acid-Catalyzed Cyclization of 2-Isocyanophenyl Ketones in the Presence of a Vinyl Ether K Kobayashi Y Okamura H Konishi
1499 Synthesis of Higher Helicenes via Olefin Metathesis and CndashH Activation J Cocircteacute S K Collins
1506 Azido- and Ethynyl-Substituted 2262-Terpyridines as Suitable Substrates for Click Reactions A Winter A Wild R Hoogenboom M W M Fijten M D Hager R-A Fallahpour U S Schubert
1513 Synthesis of 2-(Arylamino)ethanethiols via Lewis Acid Catalyzed Aminolysis of 22-Dimethylthiirane as Precursors of the 14-Benzothiazine Nucleus R Spogli S Sabatini G Manfroni O Tabarrini V Cecchetti
1520 Iron(III) Chloride A Versatile Catalyst for the Practical Synthesis of 3-Sulfenylindoles J S Yadav B V S Reddy Y J Reddy K Praneeth
1525 Organocatalytic Enantioselective Conjugate Addition of 2-Fluoromalonate to Nitroolefins Direct Synthesis of Chiral Fluorinated γ-Nitro Carboxylic Acid Derivatives H Li L Zu H Xie W Wang
1531 Asymmetric Transfer Hydrogenation of Ketimines with Trichlorosilane Structural Studies Z Zhang P Rooshenas H Hausmann P R Schreiner
1545 Prolinol Sulfinyl Ester Derivatives Organocatalytic Michael Addition of Ketones to Nitroolefins under Neat Conditions X Zeng G Zhong
1551 Asymmetric Oxidations of Electron-Poor Alkenes Promoted by the β-Amino AlcoholTBHP System A Russo A Lattanzi
1557 Enantioselectivity Switch in Direct Asymmetric Aminoxylation Catalyzed by Binaphthyl-Based Chiral Secondary Amines T Kano A Yamamoto F Shirozu K Maruoka
1564 Enantioselective Conjugate Addition of N-Heterocycles to αβ-Unsaturated Ketones Catalyzed by Chiral Primary Amines G Luo S Zhang W Duan W Wang
1573 Sulfonyl Hydrazine as New Functionality in Organocatalysis Camphorsulfonyl Hydrazine Catalyzed Enantioselective Aza-Michael Addition L-Y Chen H He B-J Pei W-H Chan A W M Lee
1578 Conversion of Primary Alcohols and Aldehydes into Methyl Esters by Ruthenium-Catalysed Hydrogen Transfer Reactions N A Owston T D Nixon A J Parker M K Whittlesey J M J Williams
1582 Addendum and Erratum XVII Forthcoming Articles
no 10 1583 Organocatalytic Formation of Quaternary Stereocenters M Bella
T Gasperi 1615 Regioselective Synthesis of 5H-Thiazolo[32-a]pyrimidin-5-ones from
MoritandashBaylisndashHillman Adduct Acetates under Solvent-Free and Base-Free Conditions W Zhong B Guo F Lin Y Liu W Su
1623 First Synthesis of 5-Cyanosalicylates by Formal [3+3] Cyclocondensations of 13-Bis(silyloxy)-13-butadienes A Riahi O Fatunsin M Shkoor R Dede H Reinke C Fischer P Langer
1635 Reaction of Isocyanides Dialkyl Acetylenedicarboxylates and a-Keto Lactones Unexpected Participation of an Ester Carbonyl Group in the Isocyanide-Based Three-Component Reaction A A Esmaeili H Vesalipoor
1639 An Efficient and Chemoselective Synthesis of 16-Naphthyridines and Pyrano[32-c]pyridines under Microwave Irradiation Z-G Han S-J Tu B Jiang S Yan X-H Zhang S-S Wu W-J Hao X-D Cao F Shi G Zhang N Ma
1647 N-Activation of N-Arylimidazoles Facile Syntheses of N-Alkyl-N-arylimidazolium Iodides from Less Expensive Chloro Substrates A M Oertel V Ritleng M J Chetcuti
1651 Synthesis of Polyhalogenated 2-(Phenylamino)pyridines by Thermal Amination Reactions S R Waldvogel A Faust W Barkmann R Froumlhlich O Wolff
1655 Cyanide Ion Promoted Addition of Acylphosphonates to Diethyl Cyanophosphonate Synthesis of Phosphonocyanohydrin O-Phosphates A S Demir A Aybey M Emrullahoglu
1659 Straightforward and Scalable Synthesis of Orthogonally Protected 37-Diazabicyclo[410]heptane H Schramm M Pavlova C Hoenke J Christoffers
1663 Hypervalent Iodine Mediated Oxidation of 12-Diaminobenzimidazole and Its Schiff Bases Efficient Synthesis of 3-Amino-124-benzotriazine and 2-Aryl-124-triazolo[15-a]benzimidazoles A Kumar M Parshad R K Gupta D Kumar
1667 Synthesis of the Reported Protoberberine Gusanlung D P B Wakchaure S Easwar N P Argade
1673 2-(Azidomethyl)arylboronic Acids in the Synthesis of Coumarin-Type Compounds M I Naumov A V Nuchev N S Sitnikov Y B Malysheva A S Shavyrin I P Beletskaya A E Gavryushin S Combes A Y Fedorov
1683 Asymmetric Synthesis of 12-anti-Disubstituted Taurine Derivatives D Enders D Iffland G Raabe
1689 A Novel One-Pot Three-Component Synthesis of 5-Imino-2358-tetrahydropyrazolo[12-a]pyridazin-1-one Derivatives B Qian M-J Fan Y-X Xie L-Y Wu Y Shi Y-M Liang
1694 One-Portion Synthesis of 2-Acetoxy Carbonyl Compounds from Aldehydes by Using an Acetylated Masked Acyl Cyanide H Nemoto T Kawamura K Kitasaki K Yatsuzuka M Kamiya Y Yoshioka
1703 Synthesis of 9-Anthryl Ethers from trans-910-Dihydro-910-dimethoxyanthracene by Acid-Catalyzed Transetherification K S Jang H Y Shin D Y Chi
1708 Efficient Synthesis of Azo Dye Labeled Terpenes Sugars and Steroids Using N-(4-Arylazobenzoyl)-1H-benzotriazoles A R Katritzky S R Tala N E Abo-Dya Z K Abdel-Samii
1715 Tandem CH-ActivationndashImine-Formation Reaction A New Route to Imidazo[21-a]phthalazines A Heim-Riether K R Gipson
1720 A Convenient and Efficient α-Sulfenylation of Carbonyl Compounds E Okragla S Demkowicz J Rachon D Witt
1725 Stereoselective Synthesis of β-Branched Phenylalanine Derivatives via Chelate-Claisen Rearrangement C Quirin U Kazmaier
1732 Catalyst-Free and Base-Free Water-Promoted SNAr Reaction of Heteroaryl Halides with Thiols B Sreedhar P S Reddy M A Reddy
1739 Convenient Methods for Synthesis of C2-Symmetric Diphenyltetrahydrothiophenes M Periasamy G Ramani G P Muthukumaragopal
1744 Highly Diastereoselective Conjugate AdditionndashElimination of Chiral Nickel(II) Glycinate with Activated Allylic Acetates for Asymmetric Synthesis of Glutamic Acid Derivatives J Wang J Shi X Zhang D Lin H Jiang H Liu
1753 Synthesis of 36-Dimethoxybenzene-12-diamine and of 47-Dimethoxy-2-methyl-1H-benzimidazole T Besset C Morin
1757 An Inexpensive Procedure for Reductive Aminations Using Dimethylamineborane on Millimolar and Molar Scale R Ortmann M Schlitzer
1760 Classics in Stereoselective Synthesis Edited by E M Carreira L Kvaerno Reviewed by Rolf Breinbauer
XV Forthcoming Articles
no 11 1761 Transition-Metal-Catalyzed Enantioselective Synthesis of Compounds with
Non-Centrochirality M Ogasawara S Watanabe 1786 One-Pot Synthesis of 3-Acyl-2-(alkylsulfanyl)indoles and 2-(Alkylsulfanyl)-
indole-3-carboxylates from (2-Isocyanophenyl)methyl Ketones or (2-Isocyanophenyl)acetates S Fukamachi H Konishi K Kobayashi
1791 Efficient and Recyclable Phthalocyanine-Based Sensitizers for Photooxygenation Reactions H Xu W-K Chan D K P Ng
1797 A Facile and Practical One-Pot Synthesis of β-Oxo Thioamides from β-Oxo Amides and Isothiocyanates P Huang D Xiang Y Zhou Y Liang T Na D Dong
1801 Microwave-Promoted Solid-Acid-Catalyzed One-Pot Synthesis of Phthalazinones V M Outerbridge S M Landge H Tamaki B Toumlroumlk
1807 Benzylic Brominations with N-Bromosuccinimide in (Trifluoromethyl)-benzene D Suarez G Laval S-M Tu D Jiang C L Robinson R Scott B T Golding
1811 Synthesis of Thioflavanone and Flavanone Derivatives by Cyclization of Chalcones W Konieczny M Konieczny
1815 A New and Expedient Total Synthesis of Ochratoxin A and d5-Ochratoxin A B Gabriele M Attya A Fazio L Di Donna P Plastina G Sindona
1821 Synthesis of Benzopyrrolizidinones by NorrishndashYang Cyclization of 3-(Acylmethyl)-2-alkylisoindol-1-ones J Wu W Zhang C Wang
1829 Reactions of MoritandashBaylisndashHillman Acetates with Huisgen Zwitterions A Novel Strategy for the Synthesis of β-Amino Acid Derivatives A Jose R R Paul R Mohan S C Mathew A T Biju E Suresh V Nair
1834 Peracetylated β-Allyl C-Glycosides of D-Ribofuranose and 2-Deoxy- D-ribofuranose in the Chemical Literature Until Now Mirages in the Literature H Otero Martinez H Reinke D Michalik C Vogel
1841 Core-Tetrasubstituted Naphthalene Diimides by Stille Cross-Coupling Reactions and Characterization of Their Optical and Redox Properties S-L Suraru F Wuumlrthner
1846 A Practical Synthesis of Indole-Based Heterocycles Using an Amidoaluminum-Mediated Strategy R Todd M M Hossain
1851 Synthesis of Fluorinated Pyrrolo[23-b]pyridine and Pyrrolo[23-d]pyrimidine Nucleosides V O Iaroshenko Y Wang D V Sevenard D M Volochnyuk
1858 Recyclization Reactions of 5-Formyl-13-dimethyluracil with Electron-Rich Amino Heterocycles A P Mityuk D M Volochnyuk S V Ryabukhin A S Plaskon A Shivanyuk A A Tolmachev
1865 Facile Synthesis of Fluorinated 1-Desazapurines V O Iaroshenko D V Sevenard D M Volochnyuk Y Wang A Martiloga A O Tolmachev
1876 A Practical Synthesis of 3-Diethoxyphosphoryl-12-pyridazine Derivatives J-C Monbaliu J Marchand-Brynaert
1881 Enantioselective Reduction of Prochiral Ketones Employing Sprouted Pisum sativa as Biocatalyst J S Yadav B V S Reddy C Sreelakshmi A B Rao
1886 Application of Phenolate Ion Mediated Intramolecular Epoxide Ring Opening in the Enantioselective Synthesis of Functionalized 23-Dihydrobenzofurans and 1-Benzopyrans S K Dinda S K Das G Panda
1897 Complementary Synthetic Approaches to Constitutionally Diverse N-Aminoalkylated Isoindolinones Application to the Synthesis of Falipamil and 5-HT1A Receptor Ligand Analogues M Lorion A Couture E Deniau P Grandclaudon
1904 Selective Deprotection of Silyl Ethers with Sodium Periodate J Li D Menche
1909 Micellar Solution of Sodium Dodecyl Sulfate (SDS) Catalyzes KabacknikndashFields Reaction in Aqueous Media S Sobhani A Vafaee
1916 Convenient Methods for the Synthesis of a Library of Hemilabile Phosphines M V Jimeacutenez J J Peacuterez-Torrente M I Bartolomeacute L A Oro
1923 Terminal Aziridines by Addition of Grignard Reagents or Organoceriums to an (α-Chloro)sulfinylimine D M Hodgson J Kloesges B Evans
1933 A Robust Synthesis of Nε-(Carboxymethyl)-L-lysine (CML) R Csuk S Stark A Barthel R Kluge D Stroumlhl
1935 One-Pot Curtius Rearrangement Processes from Carboxylic Acids O Leogane H Lebel
XV Forthcoming Articles
no 12 1941 The Chemistry of Deprotonated α-Aminonitriles T Opatz 1960 An Efficient Synthesis of Tetraalkyl 2345-Thiophenetetracarboxylate
Derivatives A Alizadeh R Hosseinpour 1963 Facile Deprotection of Bulky (Trialkylsilyl)acetylenes with Silver Fluoride
S Kim B Kim J In 1969 Highly Efficient and Reusable Ionic Liquids for the Catalyzed
Hydroamination of Alkenes with Sulfonamides Carbamates and Carboxamides L Yang L-W Xu C-G Xia
1975 Synthesis of 2391016172324-Octasubstituted Phthalocyaninatozinc(II) Complexes Mediated by Reductive Agents G A Gauna A C Monsalvo J Awruch
1979 A Short and Efficient Synthesis of 3-2-[2-(Bromomethyl)thiazol-4-yl]-ethynyl-5-fluorobenzonitrile A Precursor for PET Radioligand [18F]SP203 M B Gopinathan C Jin K S Rehder
1983 Synthesis of a Substituted Benzazepin-2-one Dihydrate S K Boini R K Vaid K P Moder D Mitchell
1987 Synthesis of Novel Trisubstituted Imidazolines F J Lakner M A Parker B Rogovoy A Khvat A Ivachtchenko
1991 A Novel Synthesis of N-But-3-enyl-α- and β-Amino Acids T T Van Nguyen R T C Brownlee A B Hughes
1999 Synthesis of Substituted 5-(3-Hydroxypropyl)pyrrolidin-2-ones and Pyrrolizidinones from Nitroethane via C3 Functionalized 56-Dihydro-4H-12-oxazines A Novel Approach to Some Analogues of the Antidepressant Rolipram A Yu Sukhorukov A V Lesiv Y A Khomutova S L Ioffe V A Tartakovsky
2009 Chiral Cyclobutanols and Cyclopentane Dimers via Samarium(II) Iodide Induced Keto-Olefin Cyclisations of Carbohydrate-Derived Unsaturated Ketones D B G Williams J Caddy K Blann J J C Groveacute C W Holzapfel
2015 Synthesis of Perfluoroalkylthio-Substituted Ferrocenes C Rhode J Lemke M Lieb N Metzler-Nolte
2019 Functionalization of Polyhedral Oligomeric Silsesquioxane (POSS) via Nucleophilic Substitution M Dutkiewicz H Maciejewski B Marciniec
2025 A Novel Synthesis of Aryl Mesylates via One-Pot DemethylationndashMesylation of Aryl Methyl Ethers Using a Mixture of Phosphorus Pentoxide in Methanesulfonic Acid B Kaboudin Y Abedi
2029 Anionic Cyclization of (NN-Dimethylamino)[2-(prop-2-yn-1-yloxy)aryl]-acetonitriles T Zdrojewski J Musielak A Jończyk
2035 Strecker-Type Reaction Catalyzed by Carboxylic Acids in Aqueous Media Z Xie G Li G Zhao J Wang
2040 Synthesis of Novel Structurally Simplified Estrogen Analogues with Electron-Donating Groups in Ring A L F Tietze C A Vock I K Krimmelbein L Nacke
2061 On the Resolution of Secondary Phosphine Oxides via Diastereomeric Complex Formation The Case of tert-Butylphenylphosphine Oxide J Holt A M Maj E P Schudde K M Pietrusiewicz L Sieroń W Wieczorek T Jerphagnon I W C E Arends U Hanefeld A J Minnaard
2066 Enantioselective Copper-Catalyzed Conjugate Addition of Dimethylzinc to 5-(1-Arylalkylidene) Meldrumrsquos Acids A Wilsily T Lou E Fillion
2073 SuzukindashMiyaura Coupling Reactions Using Phosphite Ligands M Jang Y Jo I-K Oh H M Jung S Lee
2076 Synthesis of 2-Methylindoline- and 2-Methyl-1234-tetrahydroquinoline-Derived Phosphoramidites and Their Applications in Iridium-Catalyzed Allylic Alkylation of Indoles W-B Liu H He L-X Dai S-L You
2083 Stereocontrolled Synthesis of 13-Amino Alcohols by Reduction of Substituted 2-1-[(tert-Butylsulfinyl)amino]alkylcyclohexanones J C Gonzaacutelez-Goacutemez F Foubelo M Yus
2089 Tunable Phosphoramidite Ligands for Asymmetric Hydrovinylation Ligands par excellence for Generation of All-Carbon Quaternary Centers C R Smith H J Lim A ZhangT V RajanBabu
2101 Copper-Catalyzed Asymmetric Ring-Opening Reaction of Oxabenzonorbornadienes with Grignard and Aluminum Reagents R Millet L Gremaud T Bernardez L Palais A Alexakis
2113 A Simplified Synthesis of Takemotorsquos Catalyst A Berkessel B Seelig 2116 Pharmaceutical Substances Syntheses Patents and Applications of the
Most Relevant AIPs Edited by Axel Kleeman Juumlrgen Engel Bernhard Kutscher Dietmar Reichert Reviewed by I Agranat
XV Forthcoming Articles
no 13 2117 Recent Advances in the Aza-Claisen Rearrangement K C Majumdar
T Bhattacharyya B Chattopadhyay B Sinha 2143 A Novel and Convenient Synthesis of lsquoReversedrsquo Diamidino 25-Aryl- and
25-Azaheterocycle-Substituted Furans L Hu D W Boykin 2146 Efficient and General Preparation of Pyranostilbenes First Total Synthesis
of Artocarbene and Pawhuskin B B H Park Y R Lee W S Lyoo 2155 Mild Oxidation of Diarylacetylenes to 12-Diketones Using Oxone in
Trifluoroacetic Acid J-H Chu Y-J Chen M-J Wu 2163 One-Pot Microwave-Assisted Selective Azido ReductionTandem Cyclization
in Condensed and Solid Phase with Nickel Boride N Shankaraiah N Markandeya M Espinoza-Moraga C Arancibia A Kamal L Silva Santos
2171 Pyrrolo[321-ij]quinolin-4-one and Pyrrolo[321-ij]quinolin-6-one H McNab D J Nelson E J Rozgowska
2175 Practical Synthesis of 5-Substituted Tetrazoles under Microwave Irradiation J Roh T V Artamonova K Vaacutevrovaacute G I Koldobskii A Hrabaacutelek
2179 A Simple Method for the Synthesis of 3-Arylthieno[23-b]pyridines via Iodine-Mediated Cyclization of 3-(1-Arylalkenyl)-2-[(1-phenylethyl)sulfanyl]pyridines K Kobayashi D Nakamura Y Shiroyama S Fukamachi H Konishi
2184 Synthesis of Four Lysine-Linked Cereulide Analogues Showing Ionophoric Activity Towards Potassium Cations as Lead Compounds for Emetic Toxin-Detection by Immunoassays A Makarasen T Nishikawa M Isobe
2205 Synthesis of α-Aliphatic and β-Aromatic Substituted Taurines via Regioselective Ring Opening of Thiiranes with Ammonia H Yu S Cao L Zhang G Liu J Xu
2210 Stability of 5(6)-Carboxyfluorescein in Microwave-Assisted Synthesis of Fluorescein-Labelled O-Dimannosylated Peptides R Kowalczyk P W R Harris R P Dunbar M A Brimble
2223 Diversity-Oriented Synthesis of Functionalized Diaryl Sulfones by Regioselective [3+3] Cyclizations of 13-Bis(siloxy)buta-13-dienes with 2-(Arylsulfonyl)-3-ethoxy-2-en-1-ones Scope and Limitations M Shkoor A Riahi O Fatunsin H Reinke C Fischer P Langer
2236 Synthesis of Functionalized Salicylates by Formal [3+3] Cyclocondensation of 13-Bis(silyloxy)buta-13-dienes with 3-Alkoxy-2-en-1-ones G Mroszlig S Ladzik H Reinke A Spannenberg C Fischer P Langer
2249 Synthetic Approach to Alkoxy-β-(trifluoromethyl)styrenes and Their Application in the Synthesis of New Trifluoromethylated Heterocycles V M Muzalevskiy V G Nenajdenko A V Shastin E S Balenkova G Haufe
2260 o-Benzenedisulfonimide as a Powerful and Recyclable Organocatalyst for the Nazarov Reaction M Barbero S Cadamuro A Deagostino S Dughera P Larini E G Occhiato C Prandi S Tabasso R Vulcano P Venturello
2267 The Catalytic Potential of 4-Guanidinylpyridines in Acylation Reactions I Held E Larionov C Bozler F Wagner H Zipse
2278 Iron(III) Chloride in EthanolndashWater Highly Efficient Catalytic System for the Synthesis of Garcia Gonzalez Polyhydroxyalkyl- and C-Glycosylfurans L Nagarapu M V Chary A Satyender B Supriya R Bantu
2283 Ruthenium-Catalyzed Addition of Primary Amides to Alkynes A Stereoselective Synthesis of Secondary Enamides L J Gooszligen M Blanchot K S M Salih K Gooszligen
2289 Binaphthyl-Modified Quaternary Phosphonium Salts as Chiral Phase Transfer Catalysts Application to Asymmetric Amination of β-Keto Esters R He K Maruoka
X Table of Contents XI Forthcoming Articles
no 14 2293 Direct Methods for Stereoselective Polypropionate Synthesis A Survey
J Li D Menche 2316 Synthesis of Symmetrical Ketones from Grignard Reagents and
11-Carbonyldiimidazole D Bottalico V Fiandanese G Marchese A Punzi
2319 Synthesis of 45-Substituted Imidazoles by a Fast Condensation of 12-Diketones and Urotropine in Heterogeneous Medium G Bratulescu
2321 (Arylsulfonyl)acetones and -acetonitriles New Activated Methylenic Building Blocks for Synthesis of 123-Triazoles N T Pokhodylo V S Matiychuk M D Obushak
2324 A Safe Convenient and Efficient One-Pot Synthesis of α-Chloroketone Acetals Directly from Ketones Using Iodobenzene Dichloride J Yu C Zhang
2329 An Efficient Oxidative Conversion of Aldehydes into 2-Substituted 2-Oxazolines Using 13-Diiodo-55-dimethylhydantoin S Takahashi H Togo
2333 A Novel Procedure for the Synthesis of Benzo[b][18]naphthyridine-3-carboxylate Derivatives from MoritandashBaylisndashHillman Adduct Acetates W Zhong F Lin R Chen W Su
2341 An Improved Synthesis of 147-Triazacyclononanes (tacns) and 14710-Tetraazacyclododecanes (cyclens) J Huang Z Zhou T H Chan
2345 The Ullmann Coupling between 2-Chlorobenzoic Acids and Amino Acids A Valuable Reaction for Preparing 2-Substituted 1-Acetyl-1H-indol-3-yl Acetates J C Rodriguez Dominguez X Gang G Kirsch
2349 gem-Dibromomethyl Aromatics Efficient Aldehyde Equivalents in the KnoevenagelndashDoebner Reaction J K Augustine Y A Naik S Poojari N Chowdappa B S Sherigara K Areppa
2357 Synthesis of Novel α-Aminophosphonates Containing Adamantyl Fragment M M Kabachnik L I Minaeva I P Beletskaya
2361 Efficient Fluoride-Mediated Synthesis of 5-Amino-Substituted Isothiazoles Y S Zubenko V I Potkin
2365 Phosphine-Catalyzed Reaction of Cyanohydrins with Activated Alkynes A Siby O Loreau F Taran
2371 Sulfanyl-Substituted [3]Cumulenes and Buta-13-dienes from a Tetrakis(pyridinium)-Substituted Butadiene A Schmidt A Rahimi M Gjikaj
2379 Efficient Synthesis of 2-Substituted Pyrido[32-d]pyrimidines Involving SNAr and Palladium-Catalyzed Cross-Coupling Reactions A Tikad S Routier M Akssira J-M Leacuteger C Jarry G Guillaumet
2385 Novel Synthesis of Medium-Sized Heterocycles by Palladium-Catalyzed Intramolecular Heck Reaction via 9-endo-trig Mode of Cyclization K C Majumdar B Chattopadhyay
2393 Facile Synthesis of Fluorinated Benzofuro- and Benzothieno[23-b]pyridines α-Carbolines and Nucleosides Containing the α-Carboline Framework V O Iaroshenko Y Wang B Zhang D Volochnyuk V Ya Sosnovskikh
2403 Synthesis of Functionalized N-Vinyl Nitrogen-Containing Heterocycles S M M Lopes A M Beja M Ramos Silva J A Paixatildeo F Palacios T M V D Pinho e Melo
2408 Kumada Cross-Coupling of Aryl Grignard Reagents with Aryl Halides Catalyzed by an Immobilized Nickel Catalyst X Chen L Wang J Liu
2413 Highly Enantioselective Synthesis of Heteroaromatic Alcohols Catalyzed by Chiral DiaminodiphosphinendashRuthenium(II) Complexes W-Y Shen Y-Y Li Z-R Dong J-X Gao
2418 Concise Total Synthesis of (+)-Disparlure and its trans-Isomer Using Asymmetric Organocatalysis S-G Kim
2423 Rhodium Carbenoid Induced [12]-Migration in an L-Lyxo-Configured α-Diazo β-Keto Ester Synthesis of a New Griseolic Acid Analogue N N Bhujbal K S A Kumar D D Dhavale
2430 Synthesis of 5-Arylthio-3-hydroxyphthalates by the First [4+2] Cycloadditions of 3-Arylthio-1-silyloxy-13-butadienes with Dimethyl Acetylenedicarboxylate I Iqbal M Imran P Langer
2435 Synthesis of Highly Functionalized Proline Derivatives via a One-Pot MichaelSN-AdditionCyclization Approach U Kazmaier C Schmidt
2440 RhodiumGraphite-Catalyzed Hydrogenation of Carbocyclic and Heterocyclic Aromatic Compounds G Falini A Gualandi D Savoia
2447 Potassium [1-(tert-Butoxycarbonyl)-1H-indol-2-yl]trifluoroborate as an Efficient Building Block in Palladium-Catalyzed SuzukindashMiyaura Cross Couplings P Kassis V Beacuteneacuteteau J-Y Meacuterour S Routier
2454 Syntheses of Substituted Furans and Pyrroles by Platinum-Catalyzed Cyclizations of Propargylic Oxiranes and Aziridines in Aqueous Media M Yoshida M Al-Amin K Shishido
2467 Transition-Metal-Free Oxidative Homocoupling of Aryl Alkenyl and Alkynyl Grignard Reagents with TEMPO M S Maji A Studer
XIII Forthcoming Articles
no 15 2471 Advances in Synthetic Approaches for the Preparation of Combretastatin-
Based Anti-Cancer Agents R Singh H Kaur 2492 Synthesis of Unsymmetrical Ureas by Sulfur-Assisted Carbonylation with
Carbon Monoxide and Oxidation with Molecular Oxygen under Mild Conditions T Mizuno T Nakai M Mihara
2497 Ring-OpeningRecyclization Reactions of (Dimethylamino)propenoyl-Substituted Cyclopropanes Facile Synthesis of Halogenated Pyridin-2(1H)-ones R Zhang Y Zhou Y Liang Z Jiang D Dong
2501 Facile and Efficient Total Synthesis of Taspine B Cheng S Zhang L Zhu J Zhang Q Li A Shan L He
2505 Oligomeric Iodosylbenzene Sulfate A Convenient Hypervalent Iodine Reagent for Oxidation of Organic Sulfides and Alkenes M S Yusubov R Y Yusubova T V Funk K-W Chi V V Zhdankin
2509 Pyrrolidine-Based Organocatalysts for Enantioselective Michael Addition of Cyclohexanone to trans-β-Nitrostyrene A P Carley S Dixon J D Kilburn
2517 CundashAl Hydrotalcite An Efficient and Reusable Ligand-Free Catalyst for the Coupling of Aryl Chlorides with Aliphatic Aromatic and N(H)-Heterocyclic Amines B Sreedhar R Arundhathi P L Reddy M A Reddy M L Kantam
2523 Highly Efficient Synthesis of trans-βγ-Unsaturated a-Keto Amides C Allais T Constantieux J Rodriguez
2531 Gas-Phase Synthesis of N-Unsubstituted 3-Hydroxypyrroles and 1H-Pyrrol-3(2H)-ones L Hill G A Hunter S H Imam H McNab W J OrsquoNeill
2535 3-Hydroxy-1H-pyrrole L Hill S H Imam H McNab W J OrsquoNeill 2539 123-Thiadiazoles with Unsaturated Side Chains Synthesis
Polymerization and Photocrosslinking M Al-Smadi N Hanold H Kalbitz H Meier
2547 Synthesis of 1112-Didehydrodibenzo[ae]cycloocten-5(6H)-one A Strained Eight-Membered Alkyne S C Kornmayer F Rominger R Gleiter
2553 Stannous Chloride Dihydrate A Novel and Efficient Catalyst for the Synthesis of gem-Dihydroperoxides from Ketones and Aldehydes D Azarifar K Khosravi F Soleimanei
2557 Synthesis of a Novel Class of Azacrown Macrocycles and Lariat Crown Ethers Containing Two 124-Triazole Rings as Subunits N Foroughifar A Mobinikhaledi S Ebrahimi
2561 Enantioselective Synthesis of the 3C-Protease Inhibitor (ndash)-Thysanone by a StauntonndashWeinreb Annulation Strategy J Sperry T Y Yuen M A Brimble
2570 Stereoselective Synthesis of Unnatural β-Amino Acids from Nitroethane via 56-Dihydro-4H-12-oxazin-3-ylacetates A Yu Sukhorukov A V Lesiv O L Eliseev Y A Khomutova S L Ioffe
2579 A Versatile Unexpected One-Pot Regioselective Synthesis of a New Class of 13-Diazepinoindolones by Reaction of Pyranoindolones with Monosubstituted Ureas D Livadiotou C A Tsoleridis J Stephanidou-Stephanatou
2584 Synthesis of a Trisaccharide and a Tetrasaccharide from the Cell-Wall Lipopolysaccharides of Azospirillum brasilense S17 S Pandey S Ghosh A K Misra
2591 Synthesis of Isoindoline Nitroxides by Electrocyclic Reactions T Kaacutelai J Jekı K Hideg
2596 Glycosylations of Tertiary Alcohols Synthesis of Fully Protected Disaccharides with Sterically Demanding Groups Attached to the Sugar Core A Holkenbrink J B Vicente D B Werz
2605 Copper-Catalyzed [13]-Dipolar Cycloaddition for the Synthesis of Macrocycles Containing Acyclic Aromatic and Steroidal Moieties G V Latyshev M S Baranom A V Kazantsev A D Averin N V Lukashev I P Beletskaya
2616 Aryl Ring Migration Reaction in the Synthesis of 24-Diaryl-4H-31-benzothiazines A V Butin F A Tsiunchik V T Abaev A V Gutnov D A Cheshkov
2627 Hydrogenation of β-N-Substituted and β-NN-Disubstituted Enamino Esters in the Presence of Iridium(I) Catalyst H Hebbache Z Hank C Bruneau J-L Renaud
2634 Stereoselective Olefination Reactions Promoted by Rieke Manganese J M Concelloacuten H Rodriacuteguez-Solla V del Amo P Diacuteaz
2646 Synthesis of Piperidinones through a Radical Cascade E Godineau Y Landais
2650 Asymmetric Organic Synthesis with Enzymes Edited by V Gotor I Alfonso E Garciacutea-Urdiales Reviewed by Steve Collier
XVII Forthcoming Articles
no 16 2651 Synthesis of Spirocyclic Ethers S Rosenberg R Leino 2674 Bimetallic PalladiumndashPlatinum-on-Carbon-Catalyzed HndashD Exchange
Reaction Synergistic Effect on Multiple Deuterium Incorporation T Maegawa N Ito K Oono Y Monguchi H Sajiki
2679 Efficient Copper-Catalyzed Synthesis of 2-Amino-4(3H)-quinazolinone and 2-Aminoquinazoline Derivatives X Huang H Yang H Fu R Qiao Y Zhao
2689 Synthesis and Chemoselective N- and O-Alkylation of Thiadiazolopyrimidine Nucleosides and Uridines A M L Hossion R Islam R K Kandahary T Nagamatsu
2697 Facile and Efficient Synthesis of a New Class of Indole-Substituted Pyridine Derivatives via One-Pot Multicomponent Reactions K Zhao X-P Xu S-L Zhu D-Q Shi Y Zhang S-J Ji
2709 Studies toward a Total Synthesis of Rhizoxin D Stereoselective Preparation of the C11ndashC19 Fragment S Padakanti C K Kumar E Ashok P Das
2715 A Short Synthesis of Enantiomeric Phytoprostanes B1 Type I W Perlikowska M Mikołajczyk
2719 Chemistry of Polyhalogenated Nitrobutadienes Part 7 A Novel Synthetic Access to Chlorinated Nitrile Oxides E Nutz V A Zapolrsquoskii D E Kaufmann
2725 Microwave-Assisted Silver(I)-Mediated Selective O-Alkylation of Aromatic Imidate Systems B K Singh C Cavalluzzo M De Maeyer Z Debyser V S Parmar E Van der Eycken
2729 Iodogen A Novel Reagent for the Oxidation of Urazoles under Heterogeneous Conditions A Khoramabadi A Shiri M A Zolfigol S Mallakpour
2733 An Unprecedented Synthesis of Eight-Membered-Ring Cyclic Thioimidic Esters by a Three-Component Reaction A Alizadeh R Hosseinpour
2737 A Novel Diastereoselective Synthesis of β-Phosphonato Unsaturated Thioimidates A Alizadeh N Zohreh
2741 Synthesis of 21-Benzisoxazoles by Nucleophilic Substitution of Hydrogen in Nitroarenes Activated by the Azole Ring N T Pokhodylo Y O Teslenko V S Matiychuk M D Obushak
2749 A Facile Synthesis of Two Series of Multifunctional Carbon Compounds from αα-Dihalo Ketones Using Allylsamarium Bromide X Liu S Zhang J Di
2756 Stereocontrolled Formation of Protected Aminodeoxyalditols from Simple Carbohydrate Precursors by Debenzylating Cycloetherification Y Jiang Z Fang Q Zheng H Jia J Cheng B Zheng
2761 trans-Stilbene as a Starting Material for the Synthesis of Tamoxifen Based on Palladium-Catalyzed Cross-Coupling Reactions C M Nunes J Limberger S Poersch M Seferin A L Monteiro
2766 Synthesis and Biological Evaluation of 6-Substituted Purinylcarbanucleosides with a Cyclopenta[b]thiophene Pseudosugar P Abeijoacuten J M Blanco O Caamantildeo F Fernaacutendez M D Garciacutea X Garciacutea-Mera J E Rodriacuteguez-Borges J Balzarini E De Clercq
2773 Synthesis and Electrochemical Signature of Novel Norbornyl-ferrocene Hybrids F A Khan S K Upadhyay
2778 A Regioselective TsujindashTrost Pentadienylation of 3-Allyltetronic Acid R Schobert B Barnickel
2785 Copper(I)-Catalyzed CarylndashCalkynyl Bond Formation of Aryl Iodides with Terminal Alkynes K G Thakur G Sekar
2790 Aminolysis of Epoxides Using Iridium Trichloride as an Efficient Catalyst J Agarwal A Duley R Rani R K Peddinti
2797 Preparation of Several Active N-Chloro Compounds from Trichloroisocyanuric Acid A Shiri A Khoramabadi-zad
2802 The First Mineral-Catalyzed One-Pot [3+1+2] Coupling Protocol for Multifunctionalized Fused-Ring Pyrimidines L D S Yadav A Rai
2809 Efficient Synthesis of Tetrahydro-β-carbolin-1-one and Dihydroisoquinolin-1-one Derivatives as Versatile Intermediates K E Judd M F Mahon L Caggiano
2818 A Concise Synthesis of ortho-Iodobenzyl Alcohols via Addition of ortho-Iodophenyl Grignard Reagent to Aldehydes and Ketones J Cvengroš D Stolz A Togni
XIII Forthcoming Articles
no 17 2825 Reactivity of Oxazol-5-(4H)-ones and Their Application toward Natural
Product Synthesis N M Hewlett C D Hupp J J Tepe 2840 Towards the Total Synthesis of 3-Hydroxyvibsanin E B D Schwartz
J R Denton P V Bernhardt H M L Davies C M Williams 2847 Structure Investigations of (ent)-Cladospolide D by De Novo Synthesis and
Kinetic and Thermodynamic Isomerization Y Xing J H Penn G A OrsquoDoherty
2855 New Applications of PhI(OAc)2 in Synthesis Total Synthesis and SAR Development of Potent Antitumor Natural Product PsymberinIrciniastatin A N Shao X Huang A Palani R Aslanian A Buevich J Piwinski R Huryk C Seidel-Dugan
2873 Total Synthesis of Largazole ndash Devolution of a Novel Synthetic Strategy B Wang C J Forsyth
2881 Formal Total Synthesis of Palmerolide A J Jaumlgel M E Maier 2893 Total Synthesis of Bongkrekic Acid via Sequential SuzukindashMiyaura Coupling
Reactions M Kanematsu M Shindo M Yoshida K Shishido 2905 Stereodivergent Approach to Both C28a-syn and C28a-anti Relative
Stereochemical Manifolds in the Lepadin Family via a TiCl4-Promoted G Li L J Carlson I K Sagamanova B W Slafer R P Hsung C Gilardi H M Sklenicka N Sydorenko
2915 Enantioselective Aldol Reaction of Tetrasubstituted Ketene Silyl Acetals with Achiral Aldehydes for the Construction of Asymmetric Tertiary Alcohols An Application for the Divergent Total Syntheses of Buergerinins F and G I Shiina T Iizumi Y-s Yamai Y-i Kawakita K Yokoyama Y-k Yamada
2927 Second-Generation Biomimetic Total Synthesis of Chaetominine A Coste G Karthikeyan F Couty G Evano
2935 Total Synthesis of (+)-Fostriecin and (+)-Phoslactomycin B S Shibahara M Fujino Y Tashiro N Okamoto T Esumi K Takahashi J Ishihara S Hatakeyama
2954 Stereochemical Assignments of the Chlorinated Residues in Victorin C A C Durow C Butts C L Willis
2963 Studies of the Asymmetric Total Synthesis of Clavilactone D by the lsquoLariatrsquo Cyclization Strategy T Yoshimitsu S Nojima M Hashimoto K Tsukamoto T Tanaka
2970 Total Synthesis of the Leucetta-Derived Alkaloid Calcaridine A P B Koswatta R Sivappa H V R Dias C J Lovely
2983 Formal Synthesis of Salinosporamide A Starting from D-Glucose T Momose Y Kaiya J-i Hasegawa T Sato N Chida
2992 Synthesis of Bioactive Natural Products by Asymmetric syn- and anti-Aldol Reactions A K Ghosh Z L Dawson
no 18 3003 Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural
Products B M Trost M K Brennan 3026 One-Pot Synthesis of Furo[34-b]pyridin-5(7H)-ones from 2-
Bromopyridine-3-carboxylic Acid and Carbonyl Compounds K Kobayashi T Kozuki H Konishi
3029 Iodocyclization of N-[2-(Methylthio)phenyl]propiolamides Selective Synthesis of 3-Iodo-15-benzothiazepin-4-ones T-S Jiang X-G Zhang J-H Li
3039 A Facile Synthetic Method for Fluorine-Containing 17-Phenanthrolines Pyridine-Ring Formation Reaction of N-Propargyl-68-bis(trifluoroacetyl)-quinolin-5-amine with Various Nucleophiles D Shibata E Okada M Hinoshita M Meacutedebielle
3047 Enantiotopic Discrimination in Palladium-Mediated Nucleophilic Substitutions on Achiral Substrates Chiral Ligand versus Chiral Nucleophile O Jacquet F Charnay J-C Fiaud J Ollivier
3051 Studies on the Chemistry of 2-[3-(2-Nitrophenyl)-2-oxopropyl]benzaldehydes Novel Syntheses of 5H-Benzo[b]carbazole-611-diones and Indolo[12-b]isoquinoline-611-diones M Fernaacutendez
3061 Studies on the C22ndashC23 Aldol Coupling of Spirangien M Lorenz N Bluhm M Kalesse
3067 One-Pot Synthesis of N-Alkyl Purine Pyrimidine and Azole Derivatives from Alcohols using Ph3PCCl4 A Rapid Route to Carboacyclic Nucleoside Synthesis M N Soltani Rad A Khalafi-Nezhad S Behrouz Z Asrari M Behrouz Z Amini
3077 Synthesis of 2-Amino-34-dihydroquinazolines and Imidazo[21-b]quinazoline-2-ones A Mishra S Batra
3089 Studies on the Reaction of Diimines with Thiourea Synthesis and Solvent-Induced cistrans-Isomerization of 135-Triazinane-2-thiones B Kaboudin T Ghasemi T Yokomatsu
3094 Suzuki Coupling of Heteroaromatic Chlorides Using Highly Electron-Donating ClickPhos Ligands S M Spinella Z-H Guan J Chen X Zhang
3099 Reaction of NN-Dioxyenamines with Anhydrides of Carboxylic and Sulfonic Acids A New Method for the Synthesis of a-Hydroxyoxime Derivatives A A Tabolin A V Lesiv S L Ioffe
3106 Directed ortho Metallation Chemistry and Phosphine Synthesis New Ligands for the SuzukindashMiyaura Reaction D B G Williams S J Evans H de Bod M S Mokhadinyana T Hughes
3113 New Functional Derivatives of 9-Phenylquinine P J Boratyński J SkarŜewski
3120 On the Synthesis of Asymmetric and Dissymmetric Amino Analogues of Troumlgerrsquos Base J Artacho K Waumlrnmark
3127 Synthesis of Polycyclic Sultams by Palladium-Catalyzed Intramolecular Cyclization K C Majumdar S Mondal N De
3136 Synthesis of Functionalized L-Cysteine and L-Methionine by Reaction with Electron-Deficient Acetylenes B A Trofimov A G Malrsquokina O A Shemyakina V V Nosyreva A P Borisova S S Khutsishvili L B Krivdin
3143 A lsquoClickrsquo Approach to the Synthesis of 3-[2-(1-Alkyltriazol-4-yl)ethyl]indoles M Petrini R R Shaikh
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
No 5 691 Transannulation Reactions in the Synthesis of Natural Products
P A Clarke A T Reeder J Winn 710 Synthesis of DL-erythro-Sphingosine Using a Tethered
Aminohydroxylation Reaction as the Key Step J A Morales-Serna Y Diacuteaz M I Matheu S Castilloacuten
713 Convenient Multigram Synthesis of 4-Chloropyridine-26-dicarbonyl Dichloride K Mitsui J R Parquette
715 A Novel and Efficient Synthesis of Dihydrexidine J P Cueva D E Nichols
721 Synthesis of 57-Dichloro-6-azaindoles and Functionalization via a Highly Selective LithiumndashChlorine Exchange N Lachance L-P Bonhomme-Beaulieu P Joly
731 A Convenient Synthesis of Fluorinated Pyrazolo[34-b]pyridine and Pyrazolo[34-d]pyrimidine Nucleosides V O Iaroshenko D V Sevenard A Kotljarov D M Volochnyuk A O Tolmachev V Y Sosnovskikh
741 Diastereoselective Synthesis of γ-Amino Acids and Their Derivatives from Nitroethane via Intermediacy of 56-Dihydro-4H-12-oxazines Bearing the CH2CH(CO2Me)2 Substituent at C3 A Y Sukhorukov A V Lesiv Y A Khomutova S L Ioffe
755 Synthesis of a New Pyrrolopyridoindole and Its Pyrrolopyridobenzimidazole Regioisomer F Bouchikhi M Sassatelli F Anizon M Prudhomme P Moreau
759 Practical Syntheses of Sphingosine-1-Phosphate and Analogues V Blot U Jacquemard H-U Reissig B Kleuser
767 A Facile Synthetic Route towards Substituted Thieno[32-e]indoles W Van Snick W Nulens S Jambon W Dehaen
775 Microwave-Assisted One-Pot Synthesis of (Aminoalkyl)naphthols and (Aminoalkyl)quinolinols by Using Ammonium Carbamate or Ammonium Hydrogen Carbonate as Solid Ammonia Source I Szatmaacuteri F Fuumlloumlp
779 Enantioselective Synthesis of Flavan-3-ols Using a Mitsunobu Cyclization K Krohn I Ahmed M John 787 Synthesis of a Novel γ-Folic AcidndashNτ-Histidine Conjugate Suitable for
Labeling with 99mTc and 188Re C Sparr U Michel R E Marti C Muumlller R Schibli R Moser V Groehn
793 Palladium-Catalyzed Intramolecular Biaryl Coupling A Highly Efficient Avenue for Benzannulated Pyranoquinolines and Julolidine Derivatives K C Majumdar A Taher P Debnath
801 Preparation of NN-Dimethyl-N-Arylureas Using SS-Dimethyl Dithiocarbonate as a Carbonylating Reagent I Degani R Fochi C Magistris M Migliaccio
809 Versatile Selective α-Carboxylic Acid Esterification of N-Protected Amino Acids and Peptides by Alcalase T Nuijens C Cusan J A W Kruijtzer D T S Rijkers R M J Liskamp P J L M Quaedflieg
815 Efficient Palladium-Catalyzed Amination of Aryl Chlorides Using Dicyclohexylamino[(26-dimethyl)morpholino]phenylphosphine as a PN2 Ligand S-E Park S B Kang K-J Jung J-E Won S-G Lee Y-J Yoon
824 A Clean Facile and Stereospecific Synthesis of α-Oxoketene OS-Acetals in Water Y Li Q Zhang X Cheng Q Liu X Xu
829 Sonogashira Cross-Coupling Reactions and Construction of the Indole Ring System Using a Robust Silica-Supported Palladium Catalyst E Tyrrell L Whiteman N Williams
836 Synthesis of Angular 78-Pyridazinocoumarins via the Transformation of a Hydroxy Group into a Carbonyl Group A Kotali I S Lafazanis P A Harris
841 Synthesis of New Cyclic and Acyclic 5-Halouridine Derivatives as Potential Antiviral Agents M F Elshehry J Balzarini C Meier
848 Dendritic Triphenylmethylium and Tetraphenylmethane Compounds H Meier S Kim A Oehlhof
853 Synthesis of Homoallylic Alcohols via Lewis Acid Assisted Enantioselective Desymmetrization B Yu F Menad N Isono M Lautens
860 Diastereoselective Synthesis of 123-Trisubstituted Indanes via Rhodium(I)-Catalyzed Tandem Conjugate Additions C Navarro A G Csaacutekyuml
864 Bakerrsquos Yeast for Sweet Dough Enables Large-Scale Synthesis of Enantiomerically Pure Bicyclo[331]nonane-26-dione C J Wallentin E Orentas E Butkus K Waumlrnmark
868 Addendum and Erratum XV Forthcoming Articles
No 6 869 Stereoselective Transformations of meso Bicyclic Hydrazines Versatile
Access to Functionalized Aminocyclopentanes C Bournaud F Chung A P Luna M Pasco G Errasti T Lecourt L Micouin
888 Synthesis of Glycoaminoxy Acids as Novel Sugar Building Blocks A Malapelle R Ramozzi J Xie
891 Electrophilic ipso-Halocyclization of N-Arylpropynamides with Polyfluoroalkyl Alcohols Selective Synthesis of 8-(Polyfluoroalkoxy) azaspiro[45]trienes Z-Q Wang B-X Tang H-P Zhang F Wang J-H Li
903 Electrooxidation of Alcohols in N-Oxyl-Immobilized Silica GelWater Disperse System Approach to Totally Closed System M Kuroboshi K Goto H Tanaka
909 Synthetic Routes to Aminotriamantanes Topological Analogues of the Neuroprotector Memantinereg A A Fokin A Merz N A Fokina H Schwertfeger S L Liu J E P Dahl R K M Carlson P R Schreiner
913 Parallel Synthesis of Drug-like 5-Amino-Substituted 124-Thiadiazole Libraries Using Cyclization Reactions of a Carboxamidine Dithiocarbamate Linker J Y Park I A Ryu J H Park D C Ha Y-D Gong
921 Copper-Catalyzed Selective S-Arylation of 12-Bis(o-amino-1H-pyrazolyl) Disulfides with Arylboronic Acids P-S Luo F Wang J-H Li R-Y Tang P Zhong
929 2-Iodoxybenzoic AcidTetraethylammonium BromideWater An Efficient Combination for Oxidative Cleavage of Acetals C Kuhakarn W Panchan S Chiampanichayakul N Samakkanad M Pohmakotr V Reutrakul T Jaipetch
935 Synthesis of Quinonoid Analogues of Diospyrin S Sagar I R Green 941 A One-Pot Method for the Iodination of Aryl Amines via Stable Aryl
Diazonium Silica Sulfates Under Solvent-Free Conditions A Zaroi A R Hajipour L Khazdooz
945 Poly(NN-dichloro-N-ethylbenzene-13-disulfonamide) and NNNN-Tetrachlorobenzene-13-disulfonamide as Novel Reagents for the Synthesis of N-Chloroamines Nitriles and Aldehydes R Ghorbani-Vaghei H Veisi
951 Synthesis of an (R)-Garner-type Aldehyde from L-Serine Useful Building Block for a (+)-Furanomycin Derivative G Bartoli G Di Antonio R Fiocchi S Giuli E Marcantoni M Marcolini
957 An Efficient and Highly Selective Synthesis of (Z)-Fluoroenol Phosphates from Hydroxy Difluorophosphonates P Beier R Pohl A V Alexandrova
963 Iodine-Catalyzed Three-Component Reaction A Rapid Synthesis of α-Alkoxy Azides and Homoallyl Ethers J S Yadav B V S Reddy G M Reddy R Narender
969 Rhodium(I)-Catalyzed Cycloisomerization of 13-Dienes with Alkenes in a Tether Y Oonishi A Saito M Mori Y Sato
980 Synthesis of New Optically Active D-GlucosaminendashPyrrole Derivatives B A Frontana-Uribe M V Escaacutercega-Bobadilla J Juaacuterez-Lagunas R A Toscano G A Garciacutea de la Mora M Salmoacuten
985 Partially Saturated Indeno[12-b]indole Derivatives via Deoxygenation of Heterocyclic α-Hydroxy-NO-hemiaminals H-J Hemmerling G Reiss
1000 Light-Induced Synthesis of Π-Extended Tetrathiafulvalenes Incorporating Ferrocenes An Efficient Route for the Synthesis of Electron-Donor Materials A A O Sarhan C Bolm
1007 Preparation of Nβ-Fmoc-Protected Aza-β3-Amino Acids with Nonproteinogenic Hydrophobic Side Chains for Solid-Phase Syntheses of Pseudopeptides M Laurencin P Bauchat M Baudy-Flocrsquoh
1014 Diastereomeric (η4-diene)Fe(CO)3 Complexes Containing Chiral Amide Groups A Convenient Method for the Resolution of Amino Acids M Schumacher G Coste L Miesch
1021 Palladium-Catalysed Heck Reactions of Alk-1-en-3-ones with Aryl Bromides A Very Simple Access to (E)-1-Arylalk-1-en-3-ones M Lemhadri Y Fall H Doucet M Santelli
1036 An Improved Process for the Synthesis of 4H-Imidazo[15-α][14]benzodiazepines J Yang Y Teng S Ara S Rallapalli J M Cook
1041 Meta- and Para-Difunctionalization of Arenes via an Ortho-Magnesiation and a Subsequent SulfoxidendashMagnesium Exchange L Melzig C B Rauhut P Knochel
XIII Forthcoming Articles
No 7 1049 Catalytic Transformations of Benzylic Carboxylates and Carbonates
R Kuwano 1062 A Simple and Practical Method for the Oxidation of Thebaine to 14-
Hydroxycodeinone by V2O5ndashH2O2 S Das Sharma D Konwar 1065 Umpolung with Sulfur Dioxide CarbonndashCarbon Cross-Coupling of Electron-
Rich 13-Dienes and Alkenes Application to the Enantioselective Synthesis of Long-Chain Polyketide Fragments M Turks C J Exner C Hamel P Vogel
1075 One-Pot Synthesis of 14-Diarylnaphthalenes via a WittigndashHorner Reaction[4+2] CycloadditionDehydrogenation Sequence Z Chen W Shou Y Wang
1081 A Novel and General Method for the Formation of S-Aryl Se-Aryl and Te-Aryl Phosphorochalcogenoates Y-X Gao G Tang Y Cao Y-F Zhao
1087 A Remarkable Access to γ-Fluoroalkylated Propargylamine Derivatives or Fluoroalkylated Dihydroisoxazoles via the Reaction of Fluoroalkylated Acetylides with Various Nitrones T Konno K Moriyasu T Ishihara
1095 Short and Practical Syntheses of (S)-(+)-3-(p-Tolylsulfinyl)furan-2(5H)-one and (S)-(+)-3-(p-Tolylsulfinyl)-56-dihydropyran-2-one D Cruz Cruz A Hernaacutendez Linares F Yuste M R Martiacuten J L Garciacutea Ruano
1099 Decarboxylative Aldol-Type Reaction of 2-(Trifluoroacetyl)-13-diazoles with Activated Acetic Acids P V Khodakovskiy D M Volochnyuk A A Tolmachev
1105 Synthesis of 2-[(Arylmethylene)amino]cyclopropanecarbonitriles via a Two-Step Ring Transformation of 2-(Cyanomethyl)aziridines S Mangelinckx M Drsquohooghe S Peeters N De Kimpe
1113 Synthesis of Dendrimeric Tumor-Associated Mucin-Type Glycopeptide Antigens T Becker A Kaiser H Kunz
1123 A Simple and Efficient Oxidation Procedure for the Synthesis of Acid-Sensitive Epoxides O Bortolini G Fantin M Fogagnolo
1127 Rapid Chemoselective Deprotection of Benzyl Esters by Nickel Boride J M Khurana R Arora
1131 Three-Component Coupling of Isoquinoline Activated Alkyne and Nitromethane A Facile Synthesis of Nitromethyl Derivatives of 12-Dihydroisoquinolines J S Yadav B V S Reddy N N Yadav M K Gupta
1137 Palladium Supported on a Polyionic Resin as an Efficient Ligand-Free and Recyclable Catalyst for Heck SuzukindashMiyaura and Sonogashira Reactions B Basu S Das P Das B Mandal D Banerjee F Almqvist
1147 Oxidation of 25-Dialkylpyrrole Derivatives with Cerium(IV) Ammonium Nitrate R Voloshchuk M Gałęzowski D T Gryko
1153 Practical Syntheses of Enantiomerically Pure Key Intermediates of Opioid Receptor-like 1 (ORL1) Antagonists T Yoshizumi A Ohno T Tsujita H Takahashi O Okamoto I Hayakawa H Kigoshi
1163 An Environmentally Benign TEMPO-Catalyzed Efficient Alcohol Oxidation System with a Recyclable Hypervalent Iodine(III) Reagent and Its Facile Preparation X-Q Li C Zhang
1170 Efficient and Stereoselective Rearrangement of BaylisndashHillman Acetates Catalyzed by Gold(I) ChlorideSilver(I) Trifluoromethanesulfonate Y Liu D Mao J Qian S Lou Z Xu Y Zhang
1175 The First Total Synthesis of Kynapcin-24 by Palladium Catalysis L-Y Yang C-F Chang Y-C Huang Y-J Lee C-C Hu T-H Tseng
1180 Enantioselective Synthesis of N-Protected α-Amino Acid Hydrazides M Bibian S El-Habnouni J Martinez J-A Fehrentz
1185 Synthesis of 11H-Indolo[32-c]quinoline-6-carboxylic Acids by Cascade AutoxidationndashRing Contractions A Becker S Kohfeld T Pies K Wieking L Preu C Kunick
1190 Reaction of N-Nonaflylbenzotriazole with Silyl Enol Ethers M Uhde T Ziegler
1195 2-(Benzoylimino)thiazolidin-4-ones Formation by an Alternative Ring Closure and Analysis of Rotational Barriers H-G Haumlcker P W Elsinghorst S Michels J Daniels G Schnakenburg M Guumltschow
1204 Microwave-Assisted Synthesis and Functionalization of Selenolopyrimidines S Hesse C Chenet D Thomae G Kirsch
1209 12-Disubstituted 4-Quinolones via Copper-Catalyzed Cyclization of 1-(2-Halophenyl)-2-en-3-amin-1-ones R Bernini S Cacchi G Fabrizi A Sferrazza
1220 A New Atom-Economical and Selective Synthesis of Secondary and Tertiary Alkylamines by Means of CpIridium Complex Catalyzed Multiple N-Alkylation of Ammonium Salts with Alcohols without Solvent R Yamaguchi Z Mingwen S Kawagoe C Asai K-i Fujita
1224 Synthesis of Regioisomerically Pure 5-Functionalized 27-Dichlorofluoresceins J C Castro A Malakhov K Burgess
XIII Forthcoming Articles
No 8 1227 Michael Additions to Activated Vinylphosphonates T Janecki J Kędzia
T Wąsek 1255 A Facile and General Synthesis of 2β-Aminosteroids X Ke H Hu
D Zhou W Xu Q Zhu N P Reddy X Hu 1261 Efficacious Preparation of Oppolzerrsquos Glycylsultam via the Deleacutepine
Reaction A Isleyen C Gonsky R C Ronald P Garner 1265 Synthesis of Masked Vicinal Amino Aldehydes of Pyrrolizine and Pyrrolo
[12-c]thiazole Series A V Tverdokhlebov A V Denisenko A A Tolmachev Y M Volovenko S V Shishkina O V Shishkin
1271 Preparation of 9-Substituted Pyridine-Stretched Adenines and Hypoxanthines J A Crawford W Fraser C A Ramsden
1279 A Versatile Synthesis of Heterocyclic Analogues of Neoflavonoids from Enamino Ketones V S Moskvina V P Khilya O V Turov U M Groth
1287 New Stereoselective Synthesis of Paeonilactone B F G Gatti S Serra 1291 The Use of NN-Dialkyltrimethylsilylamines in the Synthesis of
Pentamethinium Salts M Kořiacutenek M Rybaacutečkovaacute Boumlhm 1297 Synthesis of Triazoles via Regioselective Reactions of Aryl Azides with
Cyanoacetyl Pyrroles and Indoles N T Pokhodylo V S Matiychuk M D Obushak
1301 Gallium(III) Chloride Catalyzed Hydroarylation of Arylacetylenes with Naphthols and Phenols A Facile Synthesis of Vinylarenes J S Yadav B V S Reddy S Sengupta S K Biswas
1305 Electrophilic Bromination of meta-Substituted Anilines with N-Bromosuccinimide Regioselectivity and Solvent Effect S Bartoli A Cipollone A Squarcia A Madami D Fattori
1309 Cross-Coupling Reactions of Halopurines with Aryl- and Alkyltrifluoroborates The Scope and Limitations in the Synthesis of Modified Purines Z Hasniacutek R Pohl M Hocek
1318 A Convenient Method for Converting Hydroxyacetophenones into Their Ethylene or Trimethylene Acetals F Ono H Takenaka T Fujikawa M Mori T Sato
1323 γ-Chloromagnesio γ-Lactones and δ-Chloromagnesio δ-Lactones Generation Properties and Synthetic Uses H Shimizu S Fukuda S Sugiyama T Satoh
1336 Click Reactions with Nitroxides T Kaacutelai W L Hubbell K Hideg 1341 Synthesis of Novel 14-Benzoquinone-Containing 123-Triazoles An Entry
Into a New Library F Algi M Balci 1348 Efficient Synthesis of Two Sialylated Tetrasaccharides Found in Goat Milk
P K Mandal A K Misra 1355 Dendrimers of Vaccines Consisting of Tumor-Associated Glycopeptide
Antigens and T Cell Epitope Peptides S Keil A Kaiser F Syed H Kunz
1370 IBXTBAB-Mediated Oxidation of Primary Amines to Nitriles F Drouet P Fontaine G Masson J Zhu
1375 Chemoselectivity of Multicomponent Condensations of Barbituric Acids 5-Aminopyrazoles and Aldehydes E A Muravyova S V Shishkina V I Musatov I V Knyazeva O V Shishkin S M Desenko V A Chebanov
1386 Stereoselective Total Syntheses of Leiocarpin A and (ndash)-Galantinic Acid Starting from D-Mannitol K Nagaiah D Sreenu K V Purnima R S Rao J S Yadav
1393 A Facile Mild Deprotection Protocol for 13-Dithianes and 13-Dithiolanes with 30 Hydrogen Peroxide and Iodine Catalyst in Aqueous Micellar System N C Ganguly S K Barik
1400 Rhodium-Catalyzed Gram-Scale Synthesis of Highly Substituted Pyridine Derivatives K Parthasarathy C-H Cheng
1403 Enantioselective Synthesis of (R)-Propylene Carbonate from Ethyl (S)-Lactate J M Whitaker R C Ronald
XIII Forthcoming Articles
no 9 1405 Transition-Metal-Catalyzed Site-Selective Cross-Coupling of Di- and
Polyhalogenated Compounds J-R Wang K Manabe 1428 An Improved Synthesis of (4-4-Hydroxy-3-isopropyl-5-[(4-nitrophenyl)
ethynyl]benzyl-35-dimethylphenoxy)acetic Acid (NH-3) M B Gopinathan K S Rehder
1431 Copper-Catalyzed Tandem CndashN Bond Formation Reaction Selective Synthesis of 2-(Trifluoromethyl)benzimidazoles M-W Chen X-G Zhang P Zhong M-L Hu
1437 Synthesis and Thermochemical Properties of Stereoisomeric Dihydroxy- and Tetrahydroxyalkylammonium Salts M Thomas L Rothman J Hatcher P Agarkar R Ramkirath S Lall-Ramnarine R Engel
1445 Preparation of 5-Substituted 2-(2-Alkylaryl-1H-imidazol-4-yl)oxazoles and 5-Substituted 2-(2-Alkylarylthiazol-4-yl)oxazoles by Utilizing 5-Substituted 2-(2-Bromo-11-diethoxyethyl)oxazole as a Synthon D R St Laurent J L Romine
1459 Novel and Efficient Methods for the Synthesis of Symmetrical Trisulfides A Kertmen S Lach J Rachon D Witt
1463 An Environmentally Benign Electrochemical Process for the Reduction of Carboxylic Acid Hydrazides to Amides M Mentel M J Beier R Breinbauer
1469 Synthesis of 1-Chloroalkynes from Alkynylsilanes Using Trichloroisocyanuric Acid as Chlorinating Agent M H Vilhelmsen A S Andersson M B Nielsen
1473 A Convenient Approach to Enantioenriched Cyclopropanes Bearing Electron-Withdrawing Functionalities H Krawczyń K Wąsek J Kędzia
1477 Synthesis of Cyclopropenes via 12-Elimination of Bromocyclopropanes Catalyzed by Crown Ether W M Sherrill R Kim M Rubin
1485 A Base-Catalysed One-Pot Three-Component Coupling Reaction Leading to Nitrosubstituted Pyrroles I R Baxendale C D Buckle S V Ley L Tamborini
1494 Synthesis of 4-Alkylidene-4H-31-benzoxazine Derivatives by Acid-Catalyzed Cyclization of 2-Isocyanophenyl Ketones in the Presence of a Vinyl Ether K Kobayashi Y Okamura H Konishi
1499 Synthesis of Higher Helicenes via Olefin Metathesis and CndashH Activation J Cocircteacute S K Collins
1506 Azido- and Ethynyl-Substituted 2262-Terpyridines as Suitable Substrates for Click Reactions A Winter A Wild R Hoogenboom M W M Fijten M D Hager R-A Fallahpour U S Schubert
1513 Synthesis of 2-(Arylamino)ethanethiols via Lewis Acid Catalyzed Aminolysis of 22-Dimethylthiirane as Precursors of the 14-Benzothiazine Nucleus R Spogli S Sabatini G Manfroni O Tabarrini V Cecchetti
1520 Iron(III) Chloride A Versatile Catalyst for the Practical Synthesis of 3-Sulfenylindoles J S Yadav B V S Reddy Y J Reddy K Praneeth
1525 Organocatalytic Enantioselective Conjugate Addition of 2-Fluoromalonate to Nitroolefins Direct Synthesis of Chiral Fluorinated γ-Nitro Carboxylic Acid Derivatives H Li L Zu H Xie W Wang
1531 Asymmetric Transfer Hydrogenation of Ketimines with Trichlorosilane Structural Studies Z Zhang P Rooshenas H Hausmann P R Schreiner
1545 Prolinol Sulfinyl Ester Derivatives Organocatalytic Michael Addition of Ketones to Nitroolefins under Neat Conditions X Zeng G Zhong
1551 Asymmetric Oxidations of Electron-Poor Alkenes Promoted by the β-Amino AlcoholTBHP System A Russo A Lattanzi
1557 Enantioselectivity Switch in Direct Asymmetric Aminoxylation Catalyzed by Binaphthyl-Based Chiral Secondary Amines T Kano A Yamamoto F Shirozu K Maruoka
1564 Enantioselective Conjugate Addition of N-Heterocycles to αβ-Unsaturated Ketones Catalyzed by Chiral Primary Amines G Luo S Zhang W Duan W Wang
1573 Sulfonyl Hydrazine as New Functionality in Organocatalysis Camphorsulfonyl Hydrazine Catalyzed Enantioselective Aza-Michael Addition L-Y Chen H He B-J Pei W-H Chan A W M Lee
1578 Conversion of Primary Alcohols and Aldehydes into Methyl Esters by Ruthenium-Catalysed Hydrogen Transfer Reactions N A Owston T D Nixon A J Parker M K Whittlesey J M J Williams
1582 Addendum and Erratum XVII Forthcoming Articles
no 10 1583 Organocatalytic Formation of Quaternary Stereocenters M Bella
T Gasperi 1615 Regioselective Synthesis of 5H-Thiazolo[32-a]pyrimidin-5-ones from
MoritandashBaylisndashHillman Adduct Acetates under Solvent-Free and Base-Free Conditions W Zhong B Guo F Lin Y Liu W Su
1623 First Synthesis of 5-Cyanosalicylates by Formal [3+3] Cyclocondensations of 13-Bis(silyloxy)-13-butadienes A Riahi O Fatunsin M Shkoor R Dede H Reinke C Fischer P Langer
1635 Reaction of Isocyanides Dialkyl Acetylenedicarboxylates and a-Keto Lactones Unexpected Participation of an Ester Carbonyl Group in the Isocyanide-Based Three-Component Reaction A A Esmaeili H Vesalipoor
1639 An Efficient and Chemoselective Synthesis of 16-Naphthyridines and Pyrano[32-c]pyridines under Microwave Irradiation Z-G Han S-J Tu B Jiang S Yan X-H Zhang S-S Wu W-J Hao X-D Cao F Shi G Zhang N Ma
1647 N-Activation of N-Arylimidazoles Facile Syntheses of N-Alkyl-N-arylimidazolium Iodides from Less Expensive Chloro Substrates A M Oertel V Ritleng M J Chetcuti
1651 Synthesis of Polyhalogenated 2-(Phenylamino)pyridines by Thermal Amination Reactions S R Waldvogel A Faust W Barkmann R Froumlhlich O Wolff
1655 Cyanide Ion Promoted Addition of Acylphosphonates to Diethyl Cyanophosphonate Synthesis of Phosphonocyanohydrin O-Phosphates A S Demir A Aybey M Emrullahoglu
1659 Straightforward and Scalable Synthesis of Orthogonally Protected 37-Diazabicyclo[410]heptane H Schramm M Pavlova C Hoenke J Christoffers
1663 Hypervalent Iodine Mediated Oxidation of 12-Diaminobenzimidazole and Its Schiff Bases Efficient Synthesis of 3-Amino-124-benzotriazine and 2-Aryl-124-triazolo[15-a]benzimidazoles A Kumar M Parshad R K Gupta D Kumar
1667 Synthesis of the Reported Protoberberine Gusanlung D P B Wakchaure S Easwar N P Argade
1673 2-(Azidomethyl)arylboronic Acids in the Synthesis of Coumarin-Type Compounds M I Naumov A V Nuchev N S Sitnikov Y B Malysheva A S Shavyrin I P Beletskaya A E Gavryushin S Combes A Y Fedorov
1683 Asymmetric Synthesis of 12-anti-Disubstituted Taurine Derivatives D Enders D Iffland G Raabe
1689 A Novel One-Pot Three-Component Synthesis of 5-Imino-2358-tetrahydropyrazolo[12-a]pyridazin-1-one Derivatives B Qian M-J Fan Y-X Xie L-Y Wu Y Shi Y-M Liang
1694 One-Portion Synthesis of 2-Acetoxy Carbonyl Compounds from Aldehydes by Using an Acetylated Masked Acyl Cyanide H Nemoto T Kawamura K Kitasaki K Yatsuzuka M Kamiya Y Yoshioka
1703 Synthesis of 9-Anthryl Ethers from trans-910-Dihydro-910-dimethoxyanthracene by Acid-Catalyzed Transetherification K S Jang H Y Shin D Y Chi
1708 Efficient Synthesis of Azo Dye Labeled Terpenes Sugars and Steroids Using N-(4-Arylazobenzoyl)-1H-benzotriazoles A R Katritzky S R Tala N E Abo-Dya Z K Abdel-Samii
1715 Tandem CH-ActivationndashImine-Formation Reaction A New Route to Imidazo[21-a]phthalazines A Heim-Riether K R Gipson
1720 A Convenient and Efficient α-Sulfenylation of Carbonyl Compounds E Okragla S Demkowicz J Rachon D Witt
1725 Stereoselective Synthesis of β-Branched Phenylalanine Derivatives via Chelate-Claisen Rearrangement C Quirin U Kazmaier
1732 Catalyst-Free and Base-Free Water-Promoted SNAr Reaction of Heteroaryl Halides with Thiols B Sreedhar P S Reddy M A Reddy
1739 Convenient Methods for Synthesis of C2-Symmetric Diphenyltetrahydrothiophenes M Periasamy G Ramani G P Muthukumaragopal
1744 Highly Diastereoselective Conjugate AdditionndashElimination of Chiral Nickel(II) Glycinate with Activated Allylic Acetates for Asymmetric Synthesis of Glutamic Acid Derivatives J Wang J Shi X Zhang D Lin H Jiang H Liu
1753 Synthesis of 36-Dimethoxybenzene-12-diamine and of 47-Dimethoxy-2-methyl-1H-benzimidazole T Besset C Morin
1757 An Inexpensive Procedure for Reductive Aminations Using Dimethylamineborane on Millimolar and Molar Scale R Ortmann M Schlitzer
1760 Classics in Stereoselective Synthesis Edited by E M Carreira L Kvaerno Reviewed by Rolf Breinbauer
XV Forthcoming Articles
no 11 1761 Transition-Metal-Catalyzed Enantioselective Synthesis of Compounds with
Non-Centrochirality M Ogasawara S Watanabe 1786 One-Pot Synthesis of 3-Acyl-2-(alkylsulfanyl)indoles and 2-(Alkylsulfanyl)-
indole-3-carboxylates from (2-Isocyanophenyl)methyl Ketones or (2-Isocyanophenyl)acetates S Fukamachi H Konishi K Kobayashi
1791 Efficient and Recyclable Phthalocyanine-Based Sensitizers for Photooxygenation Reactions H Xu W-K Chan D K P Ng
1797 A Facile and Practical One-Pot Synthesis of β-Oxo Thioamides from β-Oxo Amides and Isothiocyanates P Huang D Xiang Y Zhou Y Liang T Na D Dong
1801 Microwave-Promoted Solid-Acid-Catalyzed One-Pot Synthesis of Phthalazinones V M Outerbridge S M Landge H Tamaki B Toumlroumlk
1807 Benzylic Brominations with N-Bromosuccinimide in (Trifluoromethyl)-benzene D Suarez G Laval S-M Tu D Jiang C L Robinson R Scott B T Golding
1811 Synthesis of Thioflavanone and Flavanone Derivatives by Cyclization of Chalcones W Konieczny M Konieczny
1815 A New and Expedient Total Synthesis of Ochratoxin A and d5-Ochratoxin A B Gabriele M Attya A Fazio L Di Donna P Plastina G Sindona
1821 Synthesis of Benzopyrrolizidinones by NorrishndashYang Cyclization of 3-(Acylmethyl)-2-alkylisoindol-1-ones J Wu W Zhang C Wang
1829 Reactions of MoritandashBaylisndashHillman Acetates with Huisgen Zwitterions A Novel Strategy for the Synthesis of β-Amino Acid Derivatives A Jose R R Paul R Mohan S C Mathew A T Biju E Suresh V Nair
1834 Peracetylated β-Allyl C-Glycosides of D-Ribofuranose and 2-Deoxy- D-ribofuranose in the Chemical Literature Until Now Mirages in the Literature H Otero Martinez H Reinke D Michalik C Vogel
1841 Core-Tetrasubstituted Naphthalene Diimides by Stille Cross-Coupling Reactions and Characterization of Their Optical and Redox Properties S-L Suraru F Wuumlrthner
1846 A Practical Synthesis of Indole-Based Heterocycles Using an Amidoaluminum-Mediated Strategy R Todd M M Hossain
1851 Synthesis of Fluorinated Pyrrolo[23-b]pyridine and Pyrrolo[23-d]pyrimidine Nucleosides V O Iaroshenko Y Wang D V Sevenard D M Volochnyuk
1858 Recyclization Reactions of 5-Formyl-13-dimethyluracil with Electron-Rich Amino Heterocycles A P Mityuk D M Volochnyuk S V Ryabukhin A S Plaskon A Shivanyuk A A Tolmachev
1865 Facile Synthesis of Fluorinated 1-Desazapurines V O Iaroshenko D V Sevenard D M Volochnyuk Y Wang A Martiloga A O Tolmachev
1876 A Practical Synthesis of 3-Diethoxyphosphoryl-12-pyridazine Derivatives J-C Monbaliu J Marchand-Brynaert
1881 Enantioselective Reduction of Prochiral Ketones Employing Sprouted Pisum sativa as Biocatalyst J S Yadav B V S Reddy C Sreelakshmi A B Rao
1886 Application of Phenolate Ion Mediated Intramolecular Epoxide Ring Opening in the Enantioselective Synthesis of Functionalized 23-Dihydrobenzofurans and 1-Benzopyrans S K Dinda S K Das G Panda
1897 Complementary Synthetic Approaches to Constitutionally Diverse N-Aminoalkylated Isoindolinones Application to the Synthesis of Falipamil and 5-HT1A Receptor Ligand Analogues M Lorion A Couture E Deniau P Grandclaudon
1904 Selective Deprotection of Silyl Ethers with Sodium Periodate J Li D Menche
1909 Micellar Solution of Sodium Dodecyl Sulfate (SDS) Catalyzes KabacknikndashFields Reaction in Aqueous Media S Sobhani A Vafaee
1916 Convenient Methods for the Synthesis of a Library of Hemilabile Phosphines M V Jimeacutenez J J Peacuterez-Torrente M I Bartolomeacute L A Oro
1923 Terminal Aziridines by Addition of Grignard Reagents or Organoceriums to an (α-Chloro)sulfinylimine D M Hodgson J Kloesges B Evans
1933 A Robust Synthesis of Nε-(Carboxymethyl)-L-lysine (CML) R Csuk S Stark A Barthel R Kluge D Stroumlhl
1935 One-Pot Curtius Rearrangement Processes from Carboxylic Acids O Leogane H Lebel
XV Forthcoming Articles
no 12 1941 The Chemistry of Deprotonated α-Aminonitriles T Opatz 1960 An Efficient Synthesis of Tetraalkyl 2345-Thiophenetetracarboxylate
Derivatives A Alizadeh R Hosseinpour 1963 Facile Deprotection of Bulky (Trialkylsilyl)acetylenes with Silver Fluoride
S Kim B Kim J In 1969 Highly Efficient and Reusable Ionic Liquids for the Catalyzed
Hydroamination of Alkenes with Sulfonamides Carbamates and Carboxamides L Yang L-W Xu C-G Xia
1975 Synthesis of 2391016172324-Octasubstituted Phthalocyaninatozinc(II) Complexes Mediated by Reductive Agents G A Gauna A C Monsalvo J Awruch
1979 A Short and Efficient Synthesis of 3-2-[2-(Bromomethyl)thiazol-4-yl]-ethynyl-5-fluorobenzonitrile A Precursor for PET Radioligand [18F]SP203 M B Gopinathan C Jin K S Rehder
1983 Synthesis of a Substituted Benzazepin-2-one Dihydrate S K Boini R K Vaid K P Moder D Mitchell
1987 Synthesis of Novel Trisubstituted Imidazolines F J Lakner M A Parker B Rogovoy A Khvat A Ivachtchenko
1991 A Novel Synthesis of N-But-3-enyl-α- and β-Amino Acids T T Van Nguyen R T C Brownlee A B Hughes
1999 Synthesis of Substituted 5-(3-Hydroxypropyl)pyrrolidin-2-ones and Pyrrolizidinones from Nitroethane via C3 Functionalized 56-Dihydro-4H-12-oxazines A Novel Approach to Some Analogues of the Antidepressant Rolipram A Yu Sukhorukov A V Lesiv Y A Khomutova S L Ioffe V A Tartakovsky
2009 Chiral Cyclobutanols and Cyclopentane Dimers via Samarium(II) Iodide Induced Keto-Olefin Cyclisations of Carbohydrate-Derived Unsaturated Ketones D B G Williams J Caddy K Blann J J C Groveacute C W Holzapfel
2015 Synthesis of Perfluoroalkylthio-Substituted Ferrocenes C Rhode J Lemke M Lieb N Metzler-Nolte
2019 Functionalization of Polyhedral Oligomeric Silsesquioxane (POSS) via Nucleophilic Substitution M Dutkiewicz H Maciejewski B Marciniec
2025 A Novel Synthesis of Aryl Mesylates via One-Pot DemethylationndashMesylation of Aryl Methyl Ethers Using a Mixture of Phosphorus Pentoxide in Methanesulfonic Acid B Kaboudin Y Abedi
2029 Anionic Cyclization of (NN-Dimethylamino)[2-(prop-2-yn-1-yloxy)aryl]-acetonitriles T Zdrojewski J Musielak A Jończyk
2035 Strecker-Type Reaction Catalyzed by Carboxylic Acids in Aqueous Media Z Xie G Li G Zhao J Wang
2040 Synthesis of Novel Structurally Simplified Estrogen Analogues with Electron-Donating Groups in Ring A L F Tietze C A Vock I K Krimmelbein L Nacke
2061 On the Resolution of Secondary Phosphine Oxides via Diastereomeric Complex Formation The Case of tert-Butylphenylphosphine Oxide J Holt A M Maj E P Schudde K M Pietrusiewicz L Sieroń W Wieczorek T Jerphagnon I W C E Arends U Hanefeld A J Minnaard
2066 Enantioselective Copper-Catalyzed Conjugate Addition of Dimethylzinc to 5-(1-Arylalkylidene) Meldrumrsquos Acids A Wilsily T Lou E Fillion
2073 SuzukindashMiyaura Coupling Reactions Using Phosphite Ligands M Jang Y Jo I-K Oh H M Jung S Lee
2076 Synthesis of 2-Methylindoline- and 2-Methyl-1234-tetrahydroquinoline-Derived Phosphoramidites and Their Applications in Iridium-Catalyzed Allylic Alkylation of Indoles W-B Liu H He L-X Dai S-L You
2083 Stereocontrolled Synthesis of 13-Amino Alcohols by Reduction of Substituted 2-1-[(tert-Butylsulfinyl)amino]alkylcyclohexanones J C Gonzaacutelez-Goacutemez F Foubelo M Yus
2089 Tunable Phosphoramidite Ligands for Asymmetric Hydrovinylation Ligands par excellence for Generation of All-Carbon Quaternary Centers C R Smith H J Lim A ZhangT V RajanBabu
2101 Copper-Catalyzed Asymmetric Ring-Opening Reaction of Oxabenzonorbornadienes with Grignard and Aluminum Reagents R Millet L Gremaud T Bernardez L Palais A Alexakis
2113 A Simplified Synthesis of Takemotorsquos Catalyst A Berkessel B Seelig 2116 Pharmaceutical Substances Syntheses Patents and Applications of the
Most Relevant AIPs Edited by Axel Kleeman Juumlrgen Engel Bernhard Kutscher Dietmar Reichert Reviewed by I Agranat
XV Forthcoming Articles
no 13 2117 Recent Advances in the Aza-Claisen Rearrangement K C Majumdar
T Bhattacharyya B Chattopadhyay B Sinha 2143 A Novel and Convenient Synthesis of lsquoReversedrsquo Diamidino 25-Aryl- and
25-Azaheterocycle-Substituted Furans L Hu D W Boykin 2146 Efficient and General Preparation of Pyranostilbenes First Total Synthesis
of Artocarbene and Pawhuskin B B H Park Y R Lee W S Lyoo 2155 Mild Oxidation of Diarylacetylenes to 12-Diketones Using Oxone in
Trifluoroacetic Acid J-H Chu Y-J Chen M-J Wu 2163 One-Pot Microwave-Assisted Selective Azido ReductionTandem Cyclization
in Condensed and Solid Phase with Nickel Boride N Shankaraiah N Markandeya M Espinoza-Moraga C Arancibia A Kamal L Silva Santos
2171 Pyrrolo[321-ij]quinolin-4-one and Pyrrolo[321-ij]quinolin-6-one H McNab D J Nelson E J Rozgowska
2175 Practical Synthesis of 5-Substituted Tetrazoles under Microwave Irradiation J Roh T V Artamonova K Vaacutevrovaacute G I Koldobskii A Hrabaacutelek
2179 A Simple Method for the Synthesis of 3-Arylthieno[23-b]pyridines via Iodine-Mediated Cyclization of 3-(1-Arylalkenyl)-2-[(1-phenylethyl)sulfanyl]pyridines K Kobayashi D Nakamura Y Shiroyama S Fukamachi H Konishi
2184 Synthesis of Four Lysine-Linked Cereulide Analogues Showing Ionophoric Activity Towards Potassium Cations as Lead Compounds for Emetic Toxin-Detection by Immunoassays A Makarasen T Nishikawa M Isobe
2205 Synthesis of α-Aliphatic and β-Aromatic Substituted Taurines via Regioselective Ring Opening of Thiiranes with Ammonia H Yu S Cao L Zhang G Liu J Xu
2210 Stability of 5(6)-Carboxyfluorescein in Microwave-Assisted Synthesis of Fluorescein-Labelled O-Dimannosylated Peptides R Kowalczyk P W R Harris R P Dunbar M A Brimble
2223 Diversity-Oriented Synthesis of Functionalized Diaryl Sulfones by Regioselective [3+3] Cyclizations of 13-Bis(siloxy)buta-13-dienes with 2-(Arylsulfonyl)-3-ethoxy-2-en-1-ones Scope and Limitations M Shkoor A Riahi O Fatunsin H Reinke C Fischer P Langer
2236 Synthesis of Functionalized Salicylates by Formal [3+3] Cyclocondensation of 13-Bis(silyloxy)buta-13-dienes with 3-Alkoxy-2-en-1-ones G Mroszlig S Ladzik H Reinke A Spannenberg C Fischer P Langer
2249 Synthetic Approach to Alkoxy-β-(trifluoromethyl)styrenes and Their Application in the Synthesis of New Trifluoromethylated Heterocycles V M Muzalevskiy V G Nenajdenko A V Shastin E S Balenkova G Haufe
2260 o-Benzenedisulfonimide as a Powerful and Recyclable Organocatalyst for the Nazarov Reaction M Barbero S Cadamuro A Deagostino S Dughera P Larini E G Occhiato C Prandi S Tabasso R Vulcano P Venturello
2267 The Catalytic Potential of 4-Guanidinylpyridines in Acylation Reactions I Held E Larionov C Bozler F Wagner H Zipse
2278 Iron(III) Chloride in EthanolndashWater Highly Efficient Catalytic System for the Synthesis of Garcia Gonzalez Polyhydroxyalkyl- and C-Glycosylfurans L Nagarapu M V Chary A Satyender B Supriya R Bantu
2283 Ruthenium-Catalyzed Addition of Primary Amides to Alkynes A Stereoselective Synthesis of Secondary Enamides L J Gooszligen M Blanchot K S M Salih K Gooszligen
2289 Binaphthyl-Modified Quaternary Phosphonium Salts as Chiral Phase Transfer Catalysts Application to Asymmetric Amination of β-Keto Esters R He K Maruoka
X Table of Contents XI Forthcoming Articles
no 14 2293 Direct Methods for Stereoselective Polypropionate Synthesis A Survey
J Li D Menche 2316 Synthesis of Symmetrical Ketones from Grignard Reagents and
11-Carbonyldiimidazole D Bottalico V Fiandanese G Marchese A Punzi
2319 Synthesis of 45-Substituted Imidazoles by a Fast Condensation of 12-Diketones and Urotropine in Heterogeneous Medium G Bratulescu
2321 (Arylsulfonyl)acetones and -acetonitriles New Activated Methylenic Building Blocks for Synthesis of 123-Triazoles N T Pokhodylo V S Matiychuk M D Obushak
2324 A Safe Convenient and Efficient One-Pot Synthesis of α-Chloroketone Acetals Directly from Ketones Using Iodobenzene Dichloride J Yu C Zhang
2329 An Efficient Oxidative Conversion of Aldehydes into 2-Substituted 2-Oxazolines Using 13-Diiodo-55-dimethylhydantoin S Takahashi H Togo
2333 A Novel Procedure for the Synthesis of Benzo[b][18]naphthyridine-3-carboxylate Derivatives from MoritandashBaylisndashHillman Adduct Acetates W Zhong F Lin R Chen W Su
2341 An Improved Synthesis of 147-Triazacyclononanes (tacns) and 14710-Tetraazacyclododecanes (cyclens) J Huang Z Zhou T H Chan
2345 The Ullmann Coupling between 2-Chlorobenzoic Acids and Amino Acids A Valuable Reaction for Preparing 2-Substituted 1-Acetyl-1H-indol-3-yl Acetates J C Rodriguez Dominguez X Gang G Kirsch
2349 gem-Dibromomethyl Aromatics Efficient Aldehyde Equivalents in the KnoevenagelndashDoebner Reaction J K Augustine Y A Naik S Poojari N Chowdappa B S Sherigara K Areppa
2357 Synthesis of Novel α-Aminophosphonates Containing Adamantyl Fragment M M Kabachnik L I Minaeva I P Beletskaya
2361 Efficient Fluoride-Mediated Synthesis of 5-Amino-Substituted Isothiazoles Y S Zubenko V I Potkin
2365 Phosphine-Catalyzed Reaction of Cyanohydrins with Activated Alkynes A Siby O Loreau F Taran
2371 Sulfanyl-Substituted [3]Cumulenes and Buta-13-dienes from a Tetrakis(pyridinium)-Substituted Butadiene A Schmidt A Rahimi M Gjikaj
2379 Efficient Synthesis of 2-Substituted Pyrido[32-d]pyrimidines Involving SNAr and Palladium-Catalyzed Cross-Coupling Reactions A Tikad S Routier M Akssira J-M Leacuteger C Jarry G Guillaumet
2385 Novel Synthesis of Medium-Sized Heterocycles by Palladium-Catalyzed Intramolecular Heck Reaction via 9-endo-trig Mode of Cyclization K C Majumdar B Chattopadhyay
2393 Facile Synthesis of Fluorinated Benzofuro- and Benzothieno[23-b]pyridines α-Carbolines and Nucleosides Containing the α-Carboline Framework V O Iaroshenko Y Wang B Zhang D Volochnyuk V Ya Sosnovskikh
2403 Synthesis of Functionalized N-Vinyl Nitrogen-Containing Heterocycles S M M Lopes A M Beja M Ramos Silva J A Paixatildeo F Palacios T M V D Pinho e Melo
2408 Kumada Cross-Coupling of Aryl Grignard Reagents with Aryl Halides Catalyzed by an Immobilized Nickel Catalyst X Chen L Wang J Liu
2413 Highly Enantioselective Synthesis of Heteroaromatic Alcohols Catalyzed by Chiral DiaminodiphosphinendashRuthenium(II) Complexes W-Y Shen Y-Y Li Z-R Dong J-X Gao
2418 Concise Total Synthesis of (+)-Disparlure and its trans-Isomer Using Asymmetric Organocatalysis S-G Kim
2423 Rhodium Carbenoid Induced [12]-Migration in an L-Lyxo-Configured α-Diazo β-Keto Ester Synthesis of a New Griseolic Acid Analogue N N Bhujbal K S A Kumar D D Dhavale
2430 Synthesis of 5-Arylthio-3-hydroxyphthalates by the First [4+2] Cycloadditions of 3-Arylthio-1-silyloxy-13-butadienes with Dimethyl Acetylenedicarboxylate I Iqbal M Imran P Langer
2435 Synthesis of Highly Functionalized Proline Derivatives via a One-Pot MichaelSN-AdditionCyclization Approach U Kazmaier C Schmidt
2440 RhodiumGraphite-Catalyzed Hydrogenation of Carbocyclic and Heterocyclic Aromatic Compounds G Falini A Gualandi D Savoia
2447 Potassium [1-(tert-Butoxycarbonyl)-1H-indol-2-yl]trifluoroborate as an Efficient Building Block in Palladium-Catalyzed SuzukindashMiyaura Cross Couplings P Kassis V Beacuteneacuteteau J-Y Meacuterour S Routier
2454 Syntheses of Substituted Furans and Pyrroles by Platinum-Catalyzed Cyclizations of Propargylic Oxiranes and Aziridines in Aqueous Media M Yoshida M Al-Amin K Shishido
2467 Transition-Metal-Free Oxidative Homocoupling of Aryl Alkenyl and Alkynyl Grignard Reagents with TEMPO M S Maji A Studer
XIII Forthcoming Articles
no 15 2471 Advances in Synthetic Approaches for the Preparation of Combretastatin-
Based Anti-Cancer Agents R Singh H Kaur 2492 Synthesis of Unsymmetrical Ureas by Sulfur-Assisted Carbonylation with
Carbon Monoxide and Oxidation with Molecular Oxygen under Mild Conditions T Mizuno T Nakai M Mihara
2497 Ring-OpeningRecyclization Reactions of (Dimethylamino)propenoyl-Substituted Cyclopropanes Facile Synthesis of Halogenated Pyridin-2(1H)-ones R Zhang Y Zhou Y Liang Z Jiang D Dong
2501 Facile and Efficient Total Synthesis of Taspine B Cheng S Zhang L Zhu J Zhang Q Li A Shan L He
2505 Oligomeric Iodosylbenzene Sulfate A Convenient Hypervalent Iodine Reagent for Oxidation of Organic Sulfides and Alkenes M S Yusubov R Y Yusubova T V Funk K-W Chi V V Zhdankin
2509 Pyrrolidine-Based Organocatalysts for Enantioselective Michael Addition of Cyclohexanone to trans-β-Nitrostyrene A P Carley S Dixon J D Kilburn
2517 CundashAl Hydrotalcite An Efficient and Reusable Ligand-Free Catalyst for the Coupling of Aryl Chlorides with Aliphatic Aromatic and N(H)-Heterocyclic Amines B Sreedhar R Arundhathi P L Reddy M A Reddy M L Kantam
2523 Highly Efficient Synthesis of trans-βγ-Unsaturated a-Keto Amides C Allais T Constantieux J Rodriguez
2531 Gas-Phase Synthesis of N-Unsubstituted 3-Hydroxypyrroles and 1H-Pyrrol-3(2H)-ones L Hill G A Hunter S H Imam H McNab W J OrsquoNeill
2535 3-Hydroxy-1H-pyrrole L Hill S H Imam H McNab W J OrsquoNeill 2539 123-Thiadiazoles with Unsaturated Side Chains Synthesis
Polymerization and Photocrosslinking M Al-Smadi N Hanold H Kalbitz H Meier
2547 Synthesis of 1112-Didehydrodibenzo[ae]cycloocten-5(6H)-one A Strained Eight-Membered Alkyne S C Kornmayer F Rominger R Gleiter
2553 Stannous Chloride Dihydrate A Novel and Efficient Catalyst for the Synthesis of gem-Dihydroperoxides from Ketones and Aldehydes D Azarifar K Khosravi F Soleimanei
2557 Synthesis of a Novel Class of Azacrown Macrocycles and Lariat Crown Ethers Containing Two 124-Triazole Rings as Subunits N Foroughifar A Mobinikhaledi S Ebrahimi
2561 Enantioselective Synthesis of the 3C-Protease Inhibitor (ndash)-Thysanone by a StauntonndashWeinreb Annulation Strategy J Sperry T Y Yuen M A Brimble
2570 Stereoselective Synthesis of Unnatural β-Amino Acids from Nitroethane via 56-Dihydro-4H-12-oxazin-3-ylacetates A Yu Sukhorukov A V Lesiv O L Eliseev Y A Khomutova S L Ioffe
2579 A Versatile Unexpected One-Pot Regioselective Synthesis of a New Class of 13-Diazepinoindolones by Reaction of Pyranoindolones with Monosubstituted Ureas D Livadiotou C A Tsoleridis J Stephanidou-Stephanatou
2584 Synthesis of a Trisaccharide and a Tetrasaccharide from the Cell-Wall Lipopolysaccharides of Azospirillum brasilense S17 S Pandey S Ghosh A K Misra
2591 Synthesis of Isoindoline Nitroxides by Electrocyclic Reactions T Kaacutelai J Jekı K Hideg
2596 Glycosylations of Tertiary Alcohols Synthesis of Fully Protected Disaccharides with Sterically Demanding Groups Attached to the Sugar Core A Holkenbrink J B Vicente D B Werz
2605 Copper-Catalyzed [13]-Dipolar Cycloaddition for the Synthesis of Macrocycles Containing Acyclic Aromatic and Steroidal Moieties G V Latyshev M S Baranom A V Kazantsev A D Averin N V Lukashev I P Beletskaya
2616 Aryl Ring Migration Reaction in the Synthesis of 24-Diaryl-4H-31-benzothiazines A V Butin F A Tsiunchik V T Abaev A V Gutnov D A Cheshkov
2627 Hydrogenation of β-N-Substituted and β-NN-Disubstituted Enamino Esters in the Presence of Iridium(I) Catalyst H Hebbache Z Hank C Bruneau J-L Renaud
2634 Stereoselective Olefination Reactions Promoted by Rieke Manganese J M Concelloacuten H Rodriacuteguez-Solla V del Amo P Diacuteaz
2646 Synthesis of Piperidinones through a Radical Cascade E Godineau Y Landais
2650 Asymmetric Organic Synthesis with Enzymes Edited by V Gotor I Alfonso E Garciacutea-Urdiales Reviewed by Steve Collier
XVII Forthcoming Articles
no 16 2651 Synthesis of Spirocyclic Ethers S Rosenberg R Leino 2674 Bimetallic PalladiumndashPlatinum-on-Carbon-Catalyzed HndashD Exchange
Reaction Synergistic Effect on Multiple Deuterium Incorporation T Maegawa N Ito K Oono Y Monguchi H Sajiki
2679 Efficient Copper-Catalyzed Synthesis of 2-Amino-4(3H)-quinazolinone and 2-Aminoquinazoline Derivatives X Huang H Yang H Fu R Qiao Y Zhao
2689 Synthesis and Chemoselective N- and O-Alkylation of Thiadiazolopyrimidine Nucleosides and Uridines A M L Hossion R Islam R K Kandahary T Nagamatsu
2697 Facile and Efficient Synthesis of a New Class of Indole-Substituted Pyridine Derivatives via One-Pot Multicomponent Reactions K Zhao X-P Xu S-L Zhu D-Q Shi Y Zhang S-J Ji
2709 Studies toward a Total Synthesis of Rhizoxin D Stereoselective Preparation of the C11ndashC19 Fragment S Padakanti C K Kumar E Ashok P Das
2715 A Short Synthesis of Enantiomeric Phytoprostanes B1 Type I W Perlikowska M Mikołajczyk
2719 Chemistry of Polyhalogenated Nitrobutadienes Part 7 A Novel Synthetic Access to Chlorinated Nitrile Oxides E Nutz V A Zapolrsquoskii D E Kaufmann
2725 Microwave-Assisted Silver(I)-Mediated Selective O-Alkylation of Aromatic Imidate Systems B K Singh C Cavalluzzo M De Maeyer Z Debyser V S Parmar E Van der Eycken
2729 Iodogen A Novel Reagent for the Oxidation of Urazoles under Heterogeneous Conditions A Khoramabadi A Shiri M A Zolfigol S Mallakpour
2733 An Unprecedented Synthesis of Eight-Membered-Ring Cyclic Thioimidic Esters by a Three-Component Reaction A Alizadeh R Hosseinpour
2737 A Novel Diastereoselective Synthesis of β-Phosphonato Unsaturated Thioimidates A Alizadeh N Zohreh
2741 Synthesis of 21-Benzisoxazoles by Nucleophilic Substitution of Hydrogen in Nitroarenes Activated by the Azole Ring N T Pokhodylo Y O Teslenko V S Matiychuk M D Obushak
2749 A Facile Synthesis of Two Series of Multifunctional Carbon Compounds from αα-Dihalo Ketones Using Allylsamarium Bromide X Liu S Zhang J Di
2756 Stereocontrolled Formation of Protected Aminodeoxyalditols from Simple Carbohydrate Precursors by Debenzylating Cycloetherification Y Jiang Z Fang Q Zheng H Jia J Cheng B Zheng
2761 trans-Stilbene as a Starting Material for the Synthesis of Tamoxifen Based on Palladium-Catalyzed Cross-Coupling Reactions C M Nunes J Limberger S Poersch M Seferin A L Monteiro
2766 Synthesis and Biological Evaluation of 6-Substituted Purinylcarbanucleosides with a Cyclopenta[b]thiophene Pseudosugar P Abeijoacuten J M Blanco O Caamantildeo F Fernaacutendez M D Garciacutea X Garciacutea-Mera J E Rodriacuteguez-Borges J Balzarini E De Clercq
2773 Synthesis and Electrochemical Signature of Novel Norbornyl-ferrocene Hybrids F A Khan S K Upadhyay
2778 A Regioselective TsujindashTrost Pentadienylation of 3-Allyltetronic Acid R Schobert B Barnickel
2785 Copper(I)-Catalyzed CarylndashCalkynyl Bond Formation of Aryl Iodides with Terminal Alkynes K G Thakur G Sekar
2790 Aminolysis of Epoxides Using Iridium Trichloride as an Efficient Catalyst J Agarwal A Duley R Rani R K Peddinti
2797 Preparation of Several Active N-Chloro Compounds from Trichloroisocyanuric Acid A Shiri A Khoramabadi-zad
2802 The First Mineral-Catalyzed One-Pot [3+1+2] Coupling Protocol for Multifunctionalized Fused-Ring Pyrimidines L D S Yadav A Rai
2809 Efficient Synthesis of Tetrahydro-β-carbolin-1-one and Dihydroisoquinolin-1-one Derivatives as Versatile Intermediates K E Judd M F Mahon L Caggiano
2818 A Concise Synthesis of ortho-Iodobenzyl Alcohols via Addition of ortho-Iodophenyl Grignard Reagent to Aldehydes and Ketones J Cvengroš D Stolz A Togni
XIII Forthcoming Articles
no 17 2825 Reactivity of Oxazol-5-(4H)-ones and Their Application toward Natural
Product Synthesis N M Hewlett C D Hupp J J Tepe 2840 Towards the Total Synthesis of 3-Hydroxyvibsanin E B D Schwartz
J R Denton P V Bernhardt H M L Davies C M Williams 2847 Structure Investigations of (ent)-Cladospolide D by De Novo Synthesis and
Kinetic and Thermodynamic Isomerization Y Xing J H Penn G A OrsquoDoherty
2855 New Applications of PhI(OAc)2 in Synthesis Total Synthesis and SAR Development of Potent Antitumor Natural Product PsymberinIrciniastatin A N Shao X Huang A Palani R Aslanian A Buevich J Piwinski R Huryk C Seidel-Dugan
2873 Total Synthesis of Largazole ndash Devolution of a Novel Synthetic Strategy B Wang C J Forsyth
2881 Formal Total Synthesis of Palmerolide A J Jaumlgel M E Maier 2893 Total Synthesis of Bongkrekic Acid via Sequential SuzukindashMiyaura Coupling
Reactions M Kanematsu M Shindo M Yoshida K Shishido 2905 Stereodivergent Approach to Both C28a-syn and C28a-anti Relative
Stereochemical Manifolds in the Lepadin Family via a TiCl4-Promoted G Li L J Carlson I K Sagamanova B W Slafer R P Hsung C Gilardi H M Sklenicka N Sydorenko
2915 Enantioselective Aldol Reaction of Tetrasubstituted Ketene Silyl Acetals with Achiral Aldehydes for the Construction of Asymmetric Tertiary Alcohols An Application for the Divergent Total Syntheses of Buergerinins F and G I Shiina T Iizumi Y-s Yamai Y-i Kawakita K Yokoyama Y-k Yamada
2927 Second-Generation Biomimetic Total Synthesis of Chaetominine A Coste G Karthikeyan F Couty G Evano
2935 Total Synthesis of (+)-Fostriecin and (+)-Phoslactomycin B S Shibahara M Fujino Y Tashiro N Okamoto T Esumi K Takahashi J Ishihara S Hatakeyama
2954 Stereochemical Assignments of the Chlorinated Residues in Victorin C A C Durow C Butts C L Willis
2963 Studies of the Asymmetric Total Synthesis of Clavilactone D by the lsquoLariatrsquo Cyclization Strategy T Yoshimitsu S Nojima M Hashimoto K Tsukamoto T Tanaka
2970 Total Synthesis of the Leucetta-Derived Alkaloid Calcaridine A P B Koswatta R Sivappa H V R Dias C J Lovely
2983 Formal Synthesis of Salinosporamide A Starting from D-Glucose T Momose Y Kaiya J-i Hasegawa T Sato N Chida
2992 Synthesis of Bioactive Natural Products by Asymmetric syn- and anti-Aldol Reactions A K Ghosh Z L Dawson
no 18 3003 Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural
Products B M Trost M K Brennan 3026 One-Pot Synthesis of Furo[34-b]pyridin-5(7H)-ones from 2-
Bromopyridine-3-carboxylic Acid and Carbonyl Compounds K Kobayashi T Kozuki H Konishi
3029 Iodocyclization of N-[2-(Methylthio)phenyl]propiolamides Selective Synthesis of 3-Iodo-15-benzothiazepin-4-ones T-S Jiang X-G Zhang J-H Li
3039 A Facile Synthetic Method for Fluorine-Containing 17-Phenanthrolines Pyridine-Ring Formation Reaction of N-Propargyl-68-bis(trifluoroacetyl)-quinolin-5-amine with Various Nucleophiles D Shibata E Okada M Hinoshita M Meacutedebielle
3047 Enantiotopic Discrimination in Palladium-Mediated Nucleophilic Substitutions on Achiral Substrates Chiral Ligand versus Chiral Nucleophile O Jacquet F Charnay J-C Fiaud J Ollivier
3051 Studies on the Chemistry of 2-[3-(2-Nitrophenyl)-2-oxopropyl]benzaldehydes Novel Syntheses of 5H-Benzo[b]carbazole-611-diones and Indolo[12-b]isoquinoline-611-diones M Fernaacutendez
3061 Studies on the C22ndashC23 Aldol Coupling of Spirangien M Lorenz N Bluhm M Kalesse
3067 One-Pot Synthesis of N-Alkyl Purine Pyrimidine and Azole Derivatives from Alcohols using Ph3PCCl4 A Rapid Route to Carboacyclic Nucleoside Synthesis M N Soltani Rad A Khalafi-Nezhad S Behrouz Z Asrari M Behrouz Z Amini
3077 Synthesis of 2-Amino-34-dihydroquinazolines and Imidazo[21-b]quinazoline-2-ones A Mishra S Batra
3089 Studies on the Reaction of Diimines with Thiourea Synthesis and Solvent-Induced cistrans-Isomerization of 135-Triazinane-2-thiones B Kaboudin T Ghasemi T Yokomatsu
3094 Suzuki Coupling of Heteroaromatic Chlorides Using Highly Electron-Donating ClickPhos Ligands S M Spinella Z-H Guan J Chen X Zhang
3099 Reaction of NN-Dioxyenamines with Anhydrides of Carboxylic and Sulfonic Acids A New Method for the Synthesis of a-Hydroxyoxime Derivatives A A Tabolin A V Lesiv S L Ioffe
3106 Directed ortho Metallation Chemistry and Phosphine Synthesis New Ligands for the SuzukindashMiyaura Reaction D B G Williams S J Evans H de Bod M S Mokhadinyana T Hughes
3113 New Functional Derivatives of 9-Phenylquinine P J Boratyński J SkarŜewski
3120 On the Synthesis of Asymmetric and Dissymmetric Amino Analogues of Troumlgerrsquos Base J Artacho K Waumlrnmark
3127 Synthesis of Polycyclic Sultams by Palladium-Catalyzed Intramolecular Cyclization K C Majumdar S Mondal N De
3136 Synthesis of Functionalized L-Cysteine and L-Methionine by Reaction with Electron-Deficient Acetylenes B A Trofimov A G Malrsquokina O A Shemyakina V V Nosyreva A P Borisova S S Khutsishvili L B Krivdin
3143 A lsquoClickrsquo Approach to the Synthesis of 3-[2-(1-Alkyltriazol-4-yl)ethyl]indoles M Petrini R R Shaikh
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
824 A Clean Facile and Stereospecific Synthesis of α-Oxoketene OS-Acetals in Water Y Li Q Zhang X Cheng Q Liu X Xu
829 Sonogashira Cross-Coupling Reactions and Construction of the Indole Ring System Using a Robust Silica-Supported Palladium Catalyst E Tyrrell L Whiteman N Williams
836 Synthesis of Angular 78-Pyridazinocoumarins via the Transformation of a Hydroxy Group into a Carbonyl Group A Kotali I S Lafazanis P A Harris
841 Synthesis of New Cyclic and Acyclic 5-Halouridine Derivatives as Potential Antiviral Agents M F Elshehry J Balzarini C Meier
848 Dendritic Triphenylmethylium and Tetraphenylmethane Compounds H Meier S Kim A Oehlhof
853 Synthesis of Homoallylic Alcohols via Lewis Acid Assisted Enantioselective Desymmetrization B Yu F Menad N Isono M Lautens
860 Diastereoselective Synthesis of 123-Trisubstituted Indanes via Rhodium(I)-Catalyzed Tandem Conjugate Additions C Navarro A G Csaacutekyuml
864 Bakerrsquos Yeast for Sweet Dough Enables Large-Scale Synthesis of Enantiomerically Pure Bicyclo[331]nonane-26-dione C J Wallentin E Orentas E Butkus K Waumlrnmark
868 Addendum and Erratum XV Forthcoming Articles
No 6 869 Stereoselective Transformations of meso Bicyclic Hydrazines Versatile
Access to Functionalized Aminocyclopentanes C Bournaud F Chung A P Luna M Pasco G Errasti T Lecourt L Micouin
888 Synthesis of Glycoaminoxy Acids as Novel Sugar Building Blocks A Malapelle R Ramozzi J Xie
891 Electrophilic ipso-Halocyclization of N-Arylpropynamides with Polyfluoroalkyl Alcohols Selective Synthesis of 8-(Polyfluoroalkoxy) azaspiro[45]trienes Z-Q Wang B-X Tang H-P Zhang F Wang J-H Li
903 Electrooxidation of Alcohols in N-Oxyl-Immobilized Silica GelWater Disperse System Approach to Totally Closed System M Kuroboshi K Goto H Tanaka
909 Synthetic Routes to Aminotriamantanes Topological Analogues of the Neuroprotector Memantinereg A A Fokin A Merz N A Fokina H Schwertfeger S L Liu J E P Dahl R K M Carlson P R Schreiner
913 Parallel Synthesis of Drug-like 5-Amino-Substituted 124-Thiadiazole Libraries Using Cyclization Reactions of a Carboxamidine Dithiocarbamate Linker J Y Park I A Ryu J H Park D C Ha Y-D Gong
921 Copper-Catalyzed Selective S-Arylation of 12-Bis(o-amino-1H-pyrazolyl) Disulfides with Arylboronic Acids P-S Luo F Wang J-H Li R-Y Tang P Zhong
929 2-Iodoxybenzoic AcidTetraethylammonium BromideWater An Efficient Combination for Oxidative Cleavage of Acetals C Kuhakarn W Panchan S Chiampanichayakul N Samakkanad M Pohmakotr V Reutrakul T Jaipetch
935 Synthesis of Quinonoid Analogues of Diospyrin S Sagar I R Green 941 A One-Pot Method for the Iodination of Aryl Amines via Stable Aryl
Diazonium Silica Sulfates Under Solvent-Free Conditions A Zaroi A R Hajipour L Khazdooz
945 Poly(NN-dichloro-N-ethylbenzene-13-disulfonamide) and NNNN-Tetrachlorobenzene-13-disulfonamide as Novel Reagents for the Synthesis of N-Chloroamines Nitriles and Aldehydes R Ghorbani-Vaghei H Veisi
951 Synthesis of an (R)-Garner-type Aldehyde from L-Serine Useful Building Block for a (+)-Furanomycin Derivative G Bartoli G Di Antonio R Fiocchi S Giuli E Marcantoni M Marcolini
957 An Efficient and Highly Selective Synthesis of (Z)-Fluoroenol Phosphates from Hydroxy Difluorophosphonates P Beier R Pohl A V Alexandrova
963 Iodine-Catalyzed Three-Component Reaction A Rapid Synthesis of α-Alkoxy Azides and Homoallyl Ethers J S Yadav B V S Reddy G M Reddy R Narender
969 Rhodium(I)-Catalyzed Cycloisomerization of 13-Dienes with Alkenes in a Tether Y Oonishi A Saito M Mori Y Sato
980 Synthesis of New Optically Active D-GlucosaminendashPyrrole Derivatives B A Frontana-Uribe M V Escaacutercega-Bobadilla J Juaacuterez-Lagunas R A Toscano G A Garciacutea de la Mora M Salmoacuten
985 Partially Saturated Indeno[12-b]indole Derivatives via Deoxygenation of Heterocyclic α-Hydroxy-NO-hemiaminals H-J Hemmerling G Reiss
1000 Light-Induced Synthesis of Π-Extended Tetrathiafulvalenes Incorporating Ferrocenes An Efficient Route for the Synthesis of Electron-Donor Materials A A O Sarhan C Bolm
1007 Preparation of Nβ-Fmoc-Protected Aza-β3-Amino Acids with Nonproteinogenic Hydrophobic Side Chains for Solid-Phase Syntheses of Pseudopeptides M Laurencin P Bauchat M Baudy-Flocrsquoh
1014 Diastereomeric (η4-diene)Fe(CO)3 Complexes Containing Chiral Amide Groups A Convenient Method for the Resolution of Amino Acids M Schumacher G Coste L Miesch
1021 Palladium-Catalysed Heck Reactions of Alk-1-en-3-ones with Aryl Bromides A Very Simple Access to (E)-1-Arylalk-1-en-3-ones M Lemhadri Y Fall H Doucet M Santelli
1036 An Improved Process for the Synthesis of 4H-Imidazo[15-α][14]benzodiazepines J Yang Y Teng S Ara S Rallapalli J M Cook
1041 Meta- and Para-Difunctionalization of Arenes via an Ortho-Magnesiation and a Subsequent SulfoxidendashMagnesium Exchange L Melzig C B Rauhut P Knochel
XIII Forthcoming Articles
No 7 1049 Catalytic Transformations of Benzylic Carboxylates and Carbonates
R Kuwano 1062 A Simple and Practical Method for the Oxidation of Thebaine to 14-
Hydroxycodeinone by V2O5ndashH2O2 S Das Sharma D Konwar 1065 Umpolung with Sulfur Dioxide CarbonndashCarbon Cross-Coupling of Electron-
Rich 13-Dienes and Alkenes Application to the Enantioselective Synthesis of Long-Chain Polyketide Fragments M Turks C J Exner C Hamel P Vogel
1075 One-Pot Synthesis of 14-Diarylnaphthalenes via a WittigndashHorner Reaction[4+2] CycloadditionDehydrogenation Sequence Z Chen W Shou Y Wang
1081 A Novel and General Method for the Formation of S-Aryl Se-Aryl and Te-Aryl Phosphorochalcogenoates Y-X Gao G Tang Y Cao Y-F Zhao
1087 A Remarkable Access to γ-Fluoroalkylated Propargylamine Derivatives or Fluoroalkylated Dihydroisoxazoles via the Reaction of Fluoroalkylated Acetylides with Various Nitrones T Konno K Moriyasu T Ishihara
1095 Short and Practical Syntheses of (S)-(+)-3-(p-Tolylsulfinyl)furan-2(5H)-one and (S)-(+)-3-(p-Tolylsulfinyl)-56-dihydropyran-2-one D Cruz Cruz A Hernaacutendez Linares F Yuste M R Martiacuten J L Garciacutea Ruano
1099 Decarboxylative Aldol-Type Reaction of 2-(Trifluoroacetyl)-13-diazoles with Activated Acetic Acids P V Khodakovskiy D M Volochnyuk A A Tolmachev
1105 Synthesis of 2-[(Arylmethylene)amino]cyclopropanecarbonitriles via a Two-Step Ring Transformation of 2-(Cyanomethyl)aziridines S Mangelinckx M Drsquohooghe S Peeters N De Kimpe
1113 Synthesis of Dendrimeric Tumor-Associated Mucin-Type Glycopeptide Antigens T Becker A Kaiser H Kunz
1123 A Simple and Efficient Oxidation Procedure for the Synthesis of Acid-Sensitive Epoxides O Bortolini G Fantin M Fogagnolo
1127 Rapid Chemoselective Deprotection of Benzyl Esters by Nickel Boride J M Khurana R Arora
1131 Three-Component Coupling of Isoquinoline Activated Alkyne and Nitromethane A Facile Synthesis of Nitromethyl Derivatives of 12-Dihydroisoquinolines J S Yadav B V S Reddy N N Yadav M K Gupta
1137 Palladium Supported on a Polyionic Resin as an Efficient Ligand-Free and Recyclable Catalyst for Heck SuzukindashMiyaura and Sonogashira Reactions B Basu S Das P Das B Mandal D Banerjee F Almqvist
1147 Oxidation of 25-Dialkylpyrrole Derivatives with Cerium(IV) Ammonium Nitrate R Voloshchuk M Gałęzowski D T Gryko
1153 Practical Syntheses of Enantiomerically Pure Key Intermediates of Opioid Receptor-like 1 (ORL1) Antagonists T Yoshizumi A Ohno T Tsujita H Takahashi O Okamoto I Hayakawa H Kigoshi
1163 An Environmentally Benign TEMPO-Catalyzed Efficient Alcohol Oxidation System with a Recyclable Hypervalent Iodine(III) Reagent and Its Facile Preparation X-Q Li C Zhang
1170 Efficient and Stereoselective Rearrangement of BaylisndashHillman Acetates Catalyzed by Gold(I) ChlorideSilver(I) Trifluoromethanesulfonate Y Liu D Mao J Qian S Lou Z Xu Y Zhang
1175 The First Total Synthesis of Kynapcin-24 by Palladium Catalysis L-Y Yang C-F Chang Y-C Huang Y-J Lee C-C Hu T-H Tseng
1180 Enantioselective Synthesis of N-Protected α-Amino Acid Hydrazides M Bibian S El-Habnouni J Martinez J-A Fehrentz
1185 Synthesis of 11H-Indolo[32-c]quinoline-6-carboxylic Acids by Cascade AutoxidationndashRing Contractions A Becker S Kohfeld T Pies K Wieking L Preu C Kunick
1190 Reaction of N-Nonaflylbenzotriazole with Silyl Enol Ethers M Uhde T Ziegler
1195 2-(Benzoylimino)thiazolidin-4-ones Formation by an Alternative Ring Closure and Analysis of Rotational Barriers H-G Haumlcker P W Elsinghorst S Michels J Daniels G Schnakenburg M Guumltschow
1204 Microwave-Assisted Synthesis and Functionalization of Selenolopyrimidines S Hesse C Chenet D Thomae G Kirsch
1209 12-Disubstituted 4-Quinolones via Copper-Catalyzed Cyclization of 1-(2-Halophenyl)-2-en-3-amin-1-ones R Bernini S Cacchi G Fabrizi A Sferrazza
1220 A New Atom-Economical and Selective Synthesis of Secondary and Tertiary Alkylamines by Means of CpIridium Complex Catalyzed Multiple N-Alkylation of Ammonium Salts with Alcohols without Solvent R Yamaguchi Z Mingwen S Kawagoe C Asai K-i Fujita
1224 Synthesis of Regioisomerically Pure 5-Functionalized 27-Dichlorofluoresceins J C Castro A Malakhov K Burgess
XIII Forthcoming Articles
No 8 1227 Michael Additions to Activated Vinylphosphonates T Janecki J Kędzia
T Wąsek 1255 A Facile and General Synthesis of 2β-Aminosteroids X Ke H Hu
D Zhou W Xu Q Zhu N P Reddy X Hu 1261 Efficacious Preparation of Oppolzerrsquos Glycylsultam via the Deleacutepine
Reaction A Isleyen C Gonsky R C Ronald P Garner 1265 Synthesis of Masked Vicinal Amino Aldehydes of Pyrrolizine and Pyrrolo
[12-c]thiazole Series A V Tverdokhlebov A V Denisenko A A Tolmachev Y M Volovenko S V Shishkina O V Shishkin
1271 Preparation of 9-Substituted Pyridine-Stretched Adenines and Hypoxanthines J A Crawford W Fraser C A Ramsden
1279 A Versatile Synthesis of Heterocyclic Analogues of Neoflavonoids from Enamino Ketones V S Moskvina V P Khilya O V Turov U M Groth
1287 New Stereoselective Synthesis of Paeonilactone B F G Gatti S Serra 1291 The Use of NN-Dialkyltrimethylsilylamines in the Synthesis of
Pentamethinium Salts M Kořiacutenek M Rybaacutečkovaacute Boumlhm 1297 Synthesis of Triazoles via Regioselective Reactions of Aryl Azides with
Cyanoacetyl Pyrroles and Indoles N T Pokhodylo V S Matiychuk M D Obushak
1301 Gallium(III) Chloride Catalyzed Hydroarylation of Arylacetylenes with Naphthols and Phenols A Facile Synthesis of Vinylarenes J S Yadav B V S Reddy S Sengupta S K Biswas
1305 Electrophilic Bromination of meta-Substituted Anilines with N-Bromosuccinimide Regioselectivity and Solvent Effect S Bartoli A Cipollone A Squarcia A Madami D Fattori
1309 Cross-Coupling Reactions of Halopurines with Aryl- and Alkyltrifluoroborates The Scope and Limitations in the Synthesis of Modified Purines Z Hasniacutek R Pohl M Hocek
1318 A Convenient Method for Converting Hydroxyacetophenones into Their Ethylene or Trimethylene Acetals F Ono H Takenaka T Fujikawa M Mori T Sato
1323 γ-Chloromagnesio γ-Lactones and δ-Chloromagnesio δ-Lactones Generation Properties and Synthetic Uses H Shimizu S Fukuda S Sugiyama T Satoh
1336 Click Reactions with Nitroxides T Kaacutelai W L Hubbell K Hideg 1341 Synthesis of Novel 14-Benzoquinone-Containing 123-Triazoles An Entry
Into a New Library F Algi M Balci 1348 Efficient Synthesis of Two Sialylated Tetrasaccharides Found in Goat Milk
P K Mandal A K Misra 1355 Dendrimers of Vaccines Consisting of Tumor-Associated Glycopeptide
Antigens and T Cell Epitope Peptides S Keil A Kaiser F Syed H Kunz
1370 IBXTBAB-Mediated Oxidation of Primary Amines to Nitriles F Drouet P Fontaine G Masson J Zhu
1375 Chemoselectivity of Multicomponent Condensations of Barbituric Acids 5-Aminopyrazoles and Aldehydes E A Muravyova S V Shishkina V I Musatov I V Knyazeva O V Shishkin S M Desenko V A Chebanov
1386 Stereoselective Total Syntheses of Leiocarpin A and (ndash)-Galantinic Acid Starting from D-Mannitol K Nagaiah D Sreenu K V Purnima R S Rao J S Yadav
1393 A Facile Mild Deprotection Protocol for 13-Dithianes and 13-Dithiolanes with 30 Hydrogen Peroxide and Iodine Catalyst in Aqueous Micellar System N C Ganguly S K Barik
1400 Rhodium-Catalyzed Gram-Scale Synthesis of Highly Substituted Pyridine Derivatives K Parthasarathy C-H Cheng
1403 Enantioselective Synthesis of (R)-Propylene Carbonate from Ethyl (S)-Lactate J M Whitaker R C Ronald
XIII Forthcoming Articles
no 9 1405 Transition-Metal-Catalyzed Site-Selective Cross-Coupling of Di- and
Polyhalogenated Compounds J-R Wang K Manabe 1428 An Improved Synthesis of (4-4-Hydroxy-3-isopropyl-5-[(4-nitrophenyl)
ethynyl]benzyl-35-dimethylphenoxy)acetic Acid (NH-3) M B Gopinathan K S Rehder
1431 Copper-Catalyzed Tandem CndashN Bond Formation Reaction Selective Synthesis of 2-(Trifluoromethyl)benzimidazoles M-W Chen X-G Zhang P Zhong M-L Hu
1437 Synthesis and Thermochemical Properties of Stereoisomeric Dihydroxy- and Tetrahydroxyalkylammonium Salts M Thomas L Rothman J Hatcher P Agarkar R Ramkirath S Lall-Ramnarine R Engel
1445 Preparation of 5-Substituted 2-(2-Alkylaryl-1H-imidazol-4-yl)oxazoles and 5-Substituted 2-(2-Alkylarylthiazol-4-yl)oxazoles by Utilizing 5-Substituted 2-(2-Bromo-11-diethoxyethyl)oxazole as a Synthon D R St Laurent J L Romine
1459 Novel and Efficient Methods for the Synthesis of Symmetrical Trisulfides A Kertmen S Lach J Rachon D Witt
1463 An Environmentally Benign Electrochemical Process for the Reduction of Carboxylic Acid Hydrazides to Amides M Mentel M J Beier R Breinbauer
1469 Synthesis of 1-Chloroalkynes from Alkynylsilanes Using Trichloroisocyanuric Acid as Chlorinating Agent M H Vilhelmsen A S Andersson M B Nielsen
1473 A Convenient Approach to Enantioenriched Cyclopropanes Bearing Electron-Withdrawing Functionalities H Krawczyń K Wąsek J Kędzia
1477 Synthesis of Cyclopropenes via 12-Elimination of Bromocyclopropanes Catalyzed by Crown Ether W M Sherrill R Kim M Rubin
1485 A Base-Catalysed One-Pot Three-Component Coupling Reaction Leading to Nitrosubstituted Pyrroles I R Baxendale C D Buckle S V Ley L Tamborini
1494 Synthesis of 4-Alkylidene-4H-31-benzoxazine Derivatives by Acid-Catalyzed Cyclization of 2-Isocyanophenyl Ketones in the Presence of a Vinyl Ether K Kobayashi Y Okamura H Konishi
1499 Synthesis of Higher Helicenes via Olefin Metathesis and CndashH Activation J Cocircteacute S K Collins
1506 Azido- and Ethynyl-Substituted 2262-Terpyridines as Suitable Substrates for Click Reactions A Winter A Wild R Hoogenboom M W M Fijten M D Hager R-A Fallahpour U S Schubert
1513 Synthesis of 2-(Arylamino)ethanethiols via Lewis Acid Catalyzed Aminolysis of 22-Dimethylthiirane as Precursors of the 14-Benzothiazine Nucleus R Spogli S Sabatini G Manfroni O Tabarrini V Cecchetti
1520 Iron(III) Chloride A Versatile Catalyst for the Practical Synthesis of 3-Sulfenylindoles J S Yadav B V S Reddy Y J Reddy K Praneeth
1525 Organocatalytic Enantioselective Conjugate Addition of 2-Fluoromalonate to Nitroolefins Direct Synthesis of Chiral Fluorinated γ-Nitro Carboxylic Acid Derivatives H Li L Zu H Xie W Wang
1531 Asymmetric Transfer Hydrogenation of Ketimines with Trichlorosilane Structural Studies Z Zhang P Rooshenas H Hausmann P R Schreiner
1545 Prolinol Sulfinyl Ester Derivatives Organocatalytic Michael Addition of Ketones to Nitroolefins under Neat Conditions X Zeng G Zhong
1551 Asymmetric Oxidations of Electron-Poor Alkenes Promoted by the β-Amino AlcoholTBHP System A Russo A Lattanzi
1557 Enantioselectivity Switch in Direct Asymmetric Aminoxylation Catalyzed by Binaphthyl-Based Chiral Secondary Amines T Kano A Yamamoto F Shirozu K Maruoka
1564 Enantioselective Conjugate Addition of N-Heterocycles to αβ-Unsaturated Ketones Catalyzed by Chiral Primary Amines G Luo S Zhang W Duan W Wang
1573 Sulfonyl Hydrazine as New Functionality in Organocatalysis Camphorsulfonyl Hydrazine Catalyzed Enantioselective Aza-Michael Addition L-Y Chen H He B-J Pei W-H Chan A W M Lee
1578 Conversion of Primary Alcohols and Aldehydes into Methyl Esters by Ruthenium-Catalysed Hydrogen Transfer Reactions N A Owston T D Nixon A J Parker M K Whittlesey J M J Williams
1582 Addendum and Erratum XVII Forthcoming Articles
no 10 1583 Organocatalytic Formation of Quaternary Stereocenters M Bella
T Gasperi 1615 Regioselective Synthesis of 5H-Thiazolo[32-a]pyrimidin-5-ones from
MoritandashBaylisndashHillman Adduct Acetates under Solvent-Free and Base-Free Conditions W Zhong B Guo F Lin Y Liu W Su
1623 First Synthesis of 5-Cyanosalicylates by Formal [3+3] Cyclocondensations of 13-Bis(silyloxy)-13-butadienes A Riahi O Fatunsin M Shkoor R Dede H Reinke C Fischer P Langer
1635 Reaction of Isocyanides Dialkyl Acetylenedicarboxylates and a-Keto Lactones Unexpected Participation of an Ester Carbonyl Group in the Isocyanide-Based Three-Component Reaction A A Esmaeili H Vesalipoor
1639 An Efficient and Chemoselective Synthesis of 16-Naphthyridines and Pyrano[32-c]pyridines under Microwave Irradiation Z-G Han S-J Tu B Jiang S Yan X-H Zhang S-S Wu W-J Hao X-D Cao F Shi G Zhang N Ma
1647 N-Activation of N-Arylimidazoles Facile Syntheses of N-Alkyl-N-arylimidazolium Iodides from Less Expensive Chloro Substrates A M Oertel V Ritleng M J Chetcuti
1651 Synthesis of Polyhalogenated 2-(Phenylamino)pyridines by Thermal Amination Reactions S R Waldvogel A Faust W Barkmann R Froumlhlich O Wolff
1655 Cyanide Ion Promoted Addition of Acylphosphonates to Diethyl Cyanophosphonate Synthesis of Phosphonocyanohydrin O-Phosphates A S Demir A Aybey M Emrullahoglu
1659 Straightforward and Scalable Synthesis of Orthogonally Protected 37-Diazabicyclo[410]heptane H Schramm M Pavlova C Hoenke J Christoffers
1663 Hypervalent Iodine Mediated Oxidation of 12-Diaminobenzimidazole and Its Schiff Bases Efficient Synthesis of 3-Amino-124-benzotriazine and 2-Aryl-124-triazolo[15-a]benzimidazoles A Kumar M Parshad R K Gupta D Kumar
1667 Synthesis of the Reported Protoberberine Gusanlung D P B Wakchaure S Easwar N P Argade
1673 2-(Azidomethyl)arylboronic Acids in the Synthesis of Coumarin-Type Compounds M I Naumov A V Nuchev N S Sitnikov Y B Malysheva A S Shavyrin I P Beletskaya A E Gavryushin S Combes A Y Fedorov
1683 Asymmetric Synthesis of 12-anti-Disubstituted Taurine Derivatives D Enders D Iffland G Raabe
1689 A Novel One-Pot Three-Component Synthesis of 5-Imino-2358-tetrahydropyrazolo[12-a]pyridazin-1-one Derivatives B Qian M-J Fan Y-X Xie L-Y Wu Y Shi Y-M Liang
1694 One-Portion Synthesis of 2-Acetoxy Carbonyl Compounds from Aldehydes by Using an Acetylated Masked Acyl Cyanide H Nemoto T Kawamura K Kitasaki K Yatsuzuka M Kamiya Y Yoshioka
1703 Synthesis of 9-Anthryl Ethers from trans-910-Dihydro-910-dimethoxyanthracene by Acid-Catalyzed Transetherification K S Jang H Y Shin D Y Chi
1708 Efficient Synthesis of Azo Dye Labeled Terpenes Sugars and Steroids Using N-(4-Arylazobenzoyl)-1H-benzotriazoles A R Katritzky S R Tala N E Abo-Dya Z K Abdel-Samii
1715 Tandem CH-ActivationndashImine-Formation Reaction A New Route to Imidazo[21-a]phthalazines A Heim-Riether K R Gipson
1720 A Convenient and Efficient α-Sulfenylation of Carbonyl Compounds E Okragla S Demkowicz J Rachon D Witt
1725 Stereoselective Synthesis of β-Branched Phenylalanine Derivatives via Chelate-Claisen Rearrangement C Quirin U Kazmaier
1732 Catalyst-Free and Base-Free Water-Promoted SNAr Reaction of Heteroaryl Halides with Thiols B Sreedhar P S Reddy M A Reddy
1739 Convenient Methods for Synthesis of C2-Symmetric Diphenyltetrahydrothiophenes M Periasamy G Ramani G P Muthukumaragopal
1744 Highly Diastereoselective Conjugate AdditionndashElimination of Chiral Nickel(II) Glycinate with Activated Allylic Acetates for Asymmetric Synthesis of Glutamic Acid Derivatives J Wang J Shi X Zhang D Lin H Jiang H Liu
1753 Synthesis of 36-Dimethoxybenzene-12-diamine and of 47-Dimethoxy-2-methyl-1H-benzimidazole T Besset C Morin
1757 An Inexpensive Procedure for Reductive Aminations Using Dimethylamineborane on Millimolar and Molar Scale R Ortmann M Schlitzer
1760 Classics in Stereoselective Synthesis Edited by E M Carreira L Kvaerno Reviewed by Rolf Breinbauer
XV Forthcoming Articles
no 11 1761 Transition-Metal-Catalyzed Enantioselective Synthesis of Compounds with
Non-Centrochirality M Ogasawara S Watanabe 1786 One-Pot Synthesis of 3-Acyl-2-(alkylsulfanyl)indoles and 2-(Alkylsulfanyl)-
indole-3-carboxylates from (2-Isocyanophenyl)methyl Ketones or (2-Isocyanophenyl)acetates S Fukamachi H Konishi K Kobayashi
1791 Efficient and Recyclable Phthalocyanine-Based Sensitizers for Photooxygenation Reactions H Xu W-K Chan D K P Ng
1797 A Facile and Practical One-Pot Synthesis of β-Oxo Thioamides from β-Oxo Amides and Isothiocyanates P Huang D Xiang Y Zhou Y Liang T Na D Dong
1801 Microwave-Promoted Solid-Acid-Catalyzed One-Pot Synthesis of Phthalazinones V M Outerbridge S M Landge H Tamaki B Toumlroumlk
1807 Benzylic Brominations with N-Bromosuccinimide in (Trifluoromethyl)-benzene D Suarez G Laval S-M Tu D Jiang C L Robinson R Scott B T Golding
1811 Synthesis of Thioflavanone and Flavanone Derivatives by Cyclization of Chalcones W Konieczny M Konieczny
1815 A New and Expedient Total Synthesis of Ochratoxin A and d5-Ochratoxin A B Gabriele M Attya A Fazio L Di Donna P Plastina G Sindona
1821 Synthesis of Benzopyrrolizidinones by NorrishndashYang Cyclization of 3-(Acylmethyl)-2-alkylisoindol-1-ones J Wu W Zhang C Wang
1829 Reactions of MoritandashBaylisndashHillman Acetates with Huisgen Zwitterions A Novel Strategy for the Synthesis of β-Amino Acid Derivatives A Jose R R Paul R Mohan S C Mathew A T Biju E Suresh V Nair
1834 Peracetylated β-Allyl C-Glycosides of D-Ribofuranose and 2-Deoxy- D-ribofuranose in the Chemical Literature Until Now Mirages in the Literature H Otero Martinez H Reinke D Michalik C Vogel
1841 Core-Tetrasubstituted Naphthalene Diimides by Stille Cross-Coupling Reactions and Characterization of Their Optical and Redox Properties S-L Suraru F Wuumlrthner
1846 A Practical Synthesis of Indole-Based Heterocycles Using an Amidoaluminum-Mediated Strategy R Todd M M Hossain
1851 Synthesis of Fluorinated Pyrrolo[23-b]pyridine and Pyrrolo[23-d]pyrimidine Nucleosides V O Iaroshenko Y Wang D V Sevenard D M Volochnyuk
1858 Recyclization Reactions of 5-Formyl-13-dimethyluracil with Electron-Rich Amino Heterocycles A P Mityuk D M Volochnyuk S V Ryabukhin A S Plaskon A Shivanyuk A A Tolmachev
1865 Facile Synthesis of Fluorinated 1-Desazapurines V O Iaroshenko D V Sevenard D M Volochnyuk Y Wang A Martiloga A O Tolmachev
1876 A Practical Synthesis of 3-Diethoxyphosphoryl-12-pyridazine Derivatives J-C Monbaliu J Marchand-Brynaert
1881 Enantioselective Reduction of Prochiral Ketones Employing Sprouted Pisum sativa as Biocatalyst J S Yadav B V S Reddy C Sreelakshmi A B Rao
1886 Application of Phenolate Ion Mediated Intramolecular Epoxide Ring Opening in the Enantioselective Synthesis of Functionalized 23-Dihydrobenzofurans and 1-Benzopyrans S K Dinda S K Das G Panda
1897 Complementary Synthetic Approaches to Constitutionally Diverse N-Aminoalkylated Isoindolinones Application to the Synthesis of Falipamil and 5-HT1A Receptor Ligand Analogues M Lorion A Couture E Deniau P Grandclaudon
1904 Selective Deprotection of Silyl Ethers with Sodium Periodate J Li D Menche
1909 Micellar Solution of Sodium Dodecyl Sulfate (SDS) Catalyzes KabacknikndashFields Reaction in Aqueous Media S Sobhani A Vafaee
1916 Convenient Methods for the Synthesis of a Library of Hemilabile Phosphines M V Jimeacutenez J J Peacuterez-Torrente M I Bartolomeacute L A Oro
1923 Terminal Aziridines by Addition of Grignard Reagents or Organoceriums to an (α-Chloro)sulfinylimine D M Hodgson J Kloesges B Evans
1933 A Robust Synthesis of Nε-(Carboxymethyl)-L-lysine (CML) R Csuk S Stark A Barthel R Kluge D Stroumlhl
1935 One-Pot Curtius Rearrangement Processes from Carboxylic Acids O Leogane H Lebel
XV Forthcoming Articles
no 12 1941 The Chemistry of Deprotonated α-Aminonitriles T Opatz 1960 An Efficient Synthesis of Tetraalkyl 2345-Thiophenetetracarboxylate
Derivatives A Alizadeh R Hosseinpour 1963 Facile Deprotection of Bulky (Trialkylsilyl)acetylenes with Silver Fluoride
S Kim B Kim J In 1969 Highly Efficient and Reusable Ionic Liquids for the Catalyzed
Hydroamination of Alkenes with Sulfonamides Carbamates and Carboxamides L Yang L-W Xu C-G Xia
1975 Synthesis of 2391016172324-Octasubstituted Phthalocyaninatozinc(II) Complexes Mediated by Reductive Agents G A Gauna A C Monsalvo J Awruch
1979 A Short and Efficient Synthesis of 3-2-[2-(Bromomethyl)thiazol-4-yl]-ethynyl-5-fluorobenzonitrile A Precursor for PET Radioligand [18F]SP203 M B Gopinathan C Jin K S Rehder
1983 Synthesis of a Substituted Benzazepin-2-one Dihydrate S K Boini R K Vaid K P Moder D Mitchell
1987 Synthesis of Novel Trisubstituted Imidazolines F J Lakner M A Parker B Rogovoy A Khvat A Ivachtchenko
1991 A Novel Synthesis of N-But-3-enyl-α- and β-Amino Acids T T Van Nguyen R T C Brownlee A B Hughes
1999 Synthesis of Substituted 5-(3-Hydroxypropyl)pyrrolidin-2-ones and Pyrrolizidinones from Nitroethane via C3 Functionalized 56-Dihydro-4H-12-oxazines A Novel Approach to Some Analogues of the Antidepressant Rolipram A Yu Sukhorukov A V Lesiv Y A Khomutova S L Ioffe V A Tartakovsky
2009 Chiral Cyclobutanols and Cyclopentane Dimers via Samarium(II) Iodide Induced Keto-Olefin Cyclisations of Carbohydrate-Derived Unsaturated Ketones D B G Williams J Caddy K Blann J J C Groveacute C W Holzapfel
2015 Synthesis of Perfluoroalkylthio-Substituted Ferrocenes C Rhode J Lemke M Lieb N Metzler-Nolte
2019 Functionalization of Polyhedral Oligomeric Silsesquioxane (POSS) via Nucleophilic Substitution M Dutkiewicz H Maciejewski B Marciniec
2025 A Novel Synthesis of Aryl Mesylates via One-Pot DemethylationndashMesylation of Aryl Methyl Ethers Using a Mixture of Phosphorus Pentoxide in Methanesulfonic Acid B Kaboudin Y Abedi
2029 Anionic Cyclization of (NN-Dimethylamino)[2-(prop-2-yn-1-yloxy)aryl]-acetonitriles T Zdrojewski J Musielak A Jończyk
2035 Strecker-Type Reaction Catalyzed by Carboxylic Acids in Aqueous Media Z Xie G Li G Zhao J Wang
2040 Synthesis of Novel Structurally Simplified Estrogen Analogues with Electron-Donating Groups in Ring A L F Tietze C A Vock I K Krimmelbein L Nacke
2061 On the Resolution of Secondary Phosphine Oxides via Diastereomeric Complex Formation The Case of tert-Butylphenylphosphine Oxide J Holt A M Maj E P Schudde K M Pietrusiewicz L Sieroń W Wieczorek T Jerphagnon I W C E Arends U Hanefeld A J Minnaard
2066 Enantioselective Copper-Catalyzed Conjugate Addition of Dimethylzinc to 5-(1-Arylalkylidene) Meldrumrsquos Acids A Wilsily T Lou E Fillion
2073 SuzukindashMiyaura Coupling Reactions Using Phosphite Ligands M Jang Y Jo I-K Oh H M Jung S Lee
2076 Synthesis of 2-Methylindoline- and 2-Methyl-1234-tetrahydroquinoline-Derived Phosphoramidites and Their Applications in Iridium-Catalyzed Allylic Alkylation of Indoles W-B Liu H He L-X Dai S-L You
2083 Stereocontrolled Synthesis of 13-Amino Alcohols by Reduction of Substituted 2-1-[(tert-Butylsulfinyl)amino]alkylcyclohexanones J C Gonzaacutelez-Goacutemez F Foubelo M Yus
2089 Tunable Phosphoramidite Ligands for Asymmetric Hydrovinylation Ligands par excellence for Generation of All-Carbon Quaternary Centers C R Smith H J Lim A ZhangT V RajanBabu
2101 Copper-Catalyzed Asymmetric Ring-Opening Reaction of Oxabenzonorbornadienes with Grignard and Aluminum Reagents R Millet L Gremaud T Bernardez L Palais A Alexakis
2113 A Simplified Synthesis of Takemotorsquos Catalyst A Berkessel B Seelig 2116 Pharmaceutical Substances Syntheses Patents and Applications of the
Most Relevant AIPs Edited by Axel Kleeman Juumlrgen Engel Bernhard Kutscher Dietmar Reichert Reviewed by I Agranat
XV Forthcoming Articles
no 13 2117 Recent Advances in the Aza-Claisen Rearrangement K C Majumdar
T Bhattacharyya B Chattopadhyay B Sinha 2143 A Novel and Convenient Synthesis of lsquoReversedrsquo Diamidino 25-Aryl- and
25-Azaheterocycle-Substituted Furans L Hu D W Boykin 2146 Efficient and General Preparation of Pyranostilbenes First Total Synthesis
of Artocarbene and Pawhuskin B B H Park Y R Lee W S Lyoo 2155 Mild Oxidation of Diarylacetylenes to 12-Diketones Using Oxone in
Trifluoroacetic Acid J-H Chu Y-J Chen M-J Wu 2163 One-Pot Microwave-Assisted Selective Azido ReductionTandem Cyclization
in Condensed and Solid Phase with Nickel Boride N Shankaraiah N Markandeya M Espinoza-Moraga C Arancibia A Kamal L Silva Santos
2171 Pyrrolo[321-ij]quinolin-4-one and Pyrrolo[321-ij]quinolin-6-one H McNab D J Nelson E J Rozgowska
2175 Practical Synthesis of 5-Substituted Tetrazoles under Microwave Irradiation J Roh T V Artamonova K Vaacutevrovaacute G I Koldobskii A Hrabaacutelek
2179 A Simple Method for the Synthesis of 3-Arylthieno[23-b]pyridines via Iodine-Mediated Cyclization of 3-(1-Arylalkenyl)-2-[(1-phenylethyl)sulfanyl]pyridines K Kobayashi D Nakamura Y Shiroyama S Fukamachi H Konishi
2184 Synthesis of Four Lysine-Linked Cereulide Analogues Showing Ionophoric Activity Towards Potassium Cations as Lead Compounds for Emetic Toxin-Detection by Immunoassays A Makarasen T Nishikawa M Isobe
2205 Synthesis of α-Aliphatic and β-Aromatic Substituted Taurines via Regioselective Ring Opening of Thiiranes with Ammonia H Yu S Cao L Zhang G Liu J Xu
2210 Stability of 5(6)-Carboxyfluorescein in Microwave-Assisted Synthesis of Fluorescein-Labelled O-Dimannosylated Peptides R Kowalczyk P W R Harris R P Dunbar M A Brimble
2223 Diversity-Oriented Synthesis of Functionalized Diaryl Sulfones by Regioselective [3+3] Cyclizations of 13-Bis(siloxy)buta-13-dienes with 2-(Arylsulfonyl)-3-ethoxy-2-en-1-ones Scope and Limitations M Shkoor A Riahi O Fatunsin H Reinke C Fischer P Langer
2236 Synthesis of Functionalized Salicylates by Formal [3+3] Cyclocondensation of 13-Bis(silyloxy)buta-13-dienes with 3-Alkoxy-2-en-1-ones G Mroszlig S Ladzik H Reinke A Spannenberg C Fischer P Langer
2249 Synthetic Approach to Alkoxy-β-(trifluoromethyl)styrenes and Their Application in the Synthesis of New Trifluoromethylated Heterocycles V M Muzalevskiy V G Nenajdenko A V Shastin E S Balenkova G Haufe
2260 o-Benzenedisulfonimide as a Powerful and Recyclable Organocatalyst for the Nazarov Reaction M Barbero S Cadamuro A Deagostino S Dughera P Larini E G Occhiato C Prandi S Tabasso R Vulcano P Venturello
2267 The Catalytic Potential of 4-Guanidinylpyridines in Acylation Reactions I Held E Larionov C Bozler F Wagner H Zipse
2278 Iron(III) Chloride in EthanolndashWater Highly Efficient Catalytic System for the Synthesis of Garcia Gonzalez Polyhydroxyalkyl- and C-Glycosylfurans L Nagarapu M V Chary A Satyender B Supriya R Bantu
2283 Ruthenium-Catalyzed Addition of Primary Amides to Alkynes A Stereoselective Synthesis of Secondary Enamides L J Gooszligen M Blanchot K S M Salih K Gooszligen
2289 Binaphthyl-Modified Quaternary Phosphonium Salts as Chiral Phase Transfer Catalysts Application to Asymmetric Amination of β-Keto Esters R He K Maruoka
X Table of Contents XI Forthcoming Articles
no 14 2293 Direct Methods for Stereoselective Polypropionate Synthesis A Survey
J Li D Menche 2316 Synthesis of Symmetrical Ketones from Grignard Reagents and
11-Carbonyldiimidazole D Bottalico V Fiandanese G Marchese A Punzi
2319 Synthesis of 45-Substituted Imidazoles by a Fast Condensation of 12-Diketones and Urotropine in Heterogeneous Medium G Bratulescu
2321 (Arylsulfonyl)acetones and -acetonitriles New Activated Methylenic Building Blocks for Synthesis of 123-Triazoles N T Pokhodylo V S Matiychuk M D Obushak
2324 A Safe Convenient and Efficient One-Pot Synthesis of α-Chloroketone Acetals Directly from Ketones Using Iodobenzene Dichloride J Yu C Zhang
2329 An Efficient Oxidative Conversion of Aldehydes into 2-Substituted 2-Oxazolines Using 13-Diiodo-55-dimethylhydantoin S Takahashi H Togo
2333 A Novel Procedure for the Synthesis of Benzo[b][18]naphthyridine-3-carboxylate Derivatives from MoritandashBaylisndashHillman Adduct Acetates W Zhong F Lin R Chen W Su
2341 An Improved Synthesis of 147-Triazacyclononanes (tacns) and 14710-Tetraazacyclododecanes (cyclens) J Huang Z Zhou T H Chan
2345 The Ullmann Coupling between 2-Chlorobenzoic Acids and Amino Acids A Valuable Reaction for Preparing 2-Substituted 1-Acetyl-1H-indol-3-yl Acetates J C Rodriguez Dominguez X Gang G Kirsch
2349 gem-Dibromomethyl Aromatics Efficient Aldehyde Equivalents in the KnoevenagelndashDoebner Reaction J K Augustine Y A Naik S Poojari N Chowdappa B S Sherigara K Areppa
2357 Synthesis of Novel α-Aminophosphonates Containing Adamantyl Fragment M M Kabachnik L I Minaeva I P Beletskaya
2361 Efficient Fluoride-Mediated Synthesis of 5-Amino-Substituted Isothiazoles Y S Zubenko V I Potkin
2365 Phosphine-Catalyzed Reaction of Cyanohydrins with Activated Alkynes A Siby O Loreau F Taran
2371 Sulfanyl-Substituted [3]Cumulenes and Buta-13-dienes from a Tetrakis(pyridinium)-Substituted Butadiene A Schmidt A Rahimi M Gjikaj
2379 Efficient Synthesis of 2-Substituted Pyrido[32-d]pyrimidines Involving SNAr and Palladium-Catalyzed Cross-Coupling Reactions A Tikad S Routier M Akssira J-M Leacuteger C Jarry G Guillaumet
2385 Novel Synthesis of Medium-Sized Heterocycles by Palladium-Catalyzed Intramolecular Heck Reaction via 9-endo-trig Mode of Cyclization K C Majumdar B Chattopadhyay
2393 Facile Synthesis of Fluorinated Benzofuro- and Benzothieno[23-b]pyridines α-Carbolines and Nucleosides Containing the α-Carboline Framework V O Iaroshenko Y Wang B Zhang D Volochnyuk V Ya Sosnovskikh
2403 Synthesis of Functionalized N-Vinyl Nitrogen-Containing Heterocycles S M M Lopes A M Beja M Ramos Silva J A Paixatildeo F Palacios T M V D Pinho e Melo
2408 Kumada Cross-Coupling of Aryl Grignard Reagents with Aryl Halides Catalyzed by an Immobilized Nickel Catalyst X Chen L Wang J Liu
2413 Highly Enantioselective Synthesis of Heteroaromatic Alcohols Catalyzed by Chiral DiaminodiphosphinendashRuthenium(II) Complexes W-Y Shen Y-Y Li Z-R Dong J-X Gao
2418 Concise Total Synthesis of (+)-Disparlure and its trans-Isomer Using Asymmetric Organocatalysis S-G Kim
2423 Rhodium Carbenoid Induced [12]-Migration in an L-Lyxo-Configured α-Diazo β-Keto Ester Synthesis of a New Griseolic Acid Analogue N N Bhujbal K S A Kumar D D Dhavale
2430 Synthesis of 5-Arylthio-3-hydroxyphthalates by the First [4+2] Cycloadditions of 3-Arylthio-1-silyloxy-13-butadienes with Dimethyl Acetylenedicarboxylate I Iqbal M Imran P Langer
2435 Synthesis of Highly Functionalized Proline Derivatives via a One-Pot MichaelSN-AdditionCyclization Approach U Kazmaier C Schmidt
2440 RhodiumGraphite-Catalyzed Hydrogenation of Carbocyclic and Heterocyclic Aromatic Compounds G Falini A Gualandi D Savoia
2447 Potassium [1-(tert-Butoxycarbonyl)-1H-indol-2-yl]trifluoroborate as an Efficient Building Block in Palladium-Catalyzed SuzukindashMiyaura Cross Couplings P Kassis V Beacuteneacuteteau J-Y Meacuterour S Routier
2454 Syntheses of Substituted Furans and Pyrroles by Platinum-Catalyzed Cyclizations of Propargylic Oxiranes and Aziridines in Aqueous Media M Yoshida M Al-Amin K Shishido
2467 Transition-Metal-Free Oxidative Homocoupling of Aryl Alkenyl and Alkynyl Grignard Reagents with TEMPO M S Maji A Studer
XIII Forthcoming Articles
no 15 2471 Advances in Synthetic Approaches for the Preparation of Combretastatin-
Based Anti-Cancer Agents R Singh H Kaur 2492 Synthesis of Unsymmetrical Ureas by Sulfur-Assisted Carbonylation with
Carbon Monoxide and Oxidation with Molecular Oxygen under Mild Conditions T Mizuno T Nakai M Mihara
2497 Ring-OpeningRecyclization Reactions of (Dimethylamino)propenoyl-Substituted Cyclopropanes Facile Synthesis of Halogenated Pyridin-2(1H)-ones R Zhang Y Zhou Y Liang Z Jiang D Dong
2501 Facile and Efficient Total Synthesis of Taspine B Cheng S Zhang L Zhu J Zhang Q Li A Shan L He
2505 Oligomeric Iodosylbenzene Sulfate A Convenient Hypervalent Iodine Reagent for Oxidation of Organic Sulfides and Alkenes M S Yusubov R Y Yusubova T V Funk K-W Chi V V Zhdankin
2509 Pyrrolidine-Based Organocatalysts for Enantioselective Michael Addition of Cyclohexanone to trans-β-Nitrostyrene A P Carley S Dixon J D Kilburn
2517 CundashAl Hydrotalcite An Efficient and Reusable Ligand-Free Catalyst for the Coupling of Aryl Chlorides with Aliphatic Aromatic and N(H)-Heterocyclic Amines B Sreedhar R Arundhathi P L Reddy M A Reddy M L Kantam
2523 Highly Efficient Synthesis of trans-βγ-Unsaturated a-Keto Amides C Allais T Constantieux J Rodriguez
2531 Gas-Phase Synthesis of N-Unsubstituted 3-Hydroxypyrroles and 1H-Pyrrol-3(2H)-ones L Hill G A Hunter S H Imam H McNab W J OrsquoNeill
2535 3-Hydroxy-1H-pyrrole L Hill S H Imam H McNab W J OrsquoNeill 2539 123-Thiadiazoles with Unsaturated Side Chains Synthesis
Polymerization and Photocrosslinking M Al-Smadi N Hanold H Kalbitz H Meier
2547 Synthesis of 1112-Didehydrodibenzo[ae]cycloocten-5(6H)-one A Strained Eight-Membered Alkyne S C Kornmayer F Rominger R Gleiter
2553 Stannous Chloride Dihydrate A Novel and Efficient Catalyst for the Synthesis of gem-Dihydroperoxides from Ketones and Aldehydes D Azarifar K Khosravi F Soleimanei
2557 Synthesis of a Novel Class of Azacrown Macrocycles and Lariat Crown Ethers Containing Two 124-Triazole Rings as Subunits N Foroughifar A Mobinikhaledi S Ebrahimi
2561 Enantioselective Synthesis of the 3C-Protease Inhibitor (ndash)-Thysanone by a StauntonndashWeinreb Annulation Strategy J Sperry T Y Yuen M A Brimble
2570 Stereoselective Synthesis of Unnatural β-Amino Acids from Nitroethane via 56-Dihydro-4H-12-oxazin-3-ylacetates A Yu Sukhorukov A V Lesiv O L Eliseev Y A Khomutova S L Ioffe
2579 A Versatile Unexpected One-Pot Regioselective Synthesis of a New Class of 13-Diazepinoindolones by Reaction of Pyranoindolones with Monosubstituted Ureas D Livadiotou C A Tsoleridis J Stephanidou-Stephanatou
2584 Synthesis of a Trisaccharide and a Tetrasaccharide from the Cell-Wall Lipopolysaccharides of Azospirillum brasilense S17 S Pandey S Ghosh A K Misra
2591 Synthesis of Isoindoline Nitroxides by Electrocyclic Reactions T Kaacutelai J Jekı K Hideg
2596 Glycosylations of Tertiary Alcohols Synthesis of Fully Protected Disaccharides with Sterically Demanding Groups Attached to the Sugar Core A Holkenbrink J B Vicente D B Werz
2605 Copper-Catalyzed [13]-Dipolar Cycloaddition for the Synthesis of Macrocycles Containing Acyclic Aromatic and Steroidal Moieties G V Latyshev M S Baranom A V Kazantsev A D Averin N V Lukashev I P Beletskaya
2616 Aryl Ring Migration Reaction in the Synthesis of 24-Diaryl-4H-31-benzothiazines A V Butin F A Tsiunchik V T Abaev A V Gutnov D A Cheshkov
2627 Hydrogenation of β-N-Substituted and β-NN-Disubstituted Enamino Esters in the Presence of Iridium(I) Catalyst H Hebbache Z Hank C Bruneau J-L Renaud
2634 Stereoselective Olefination Reactions Promoted by Rieke Manganese J M Concelloacuten H Rodriacuteguez-Solla V del Amo P Diacuteaz
2646 Synthesis of Piperidinones through a Radical Cascade E Godineau Y Landais
2650 Asymmetric Organic Synthesis with Enzymes Edited by V Gotor I Alfonso E Garciacutea-Urdiales Reviewed by Steve Collier
XVII Forthcoming Articles
no 16 2651 Synthesis of Spirocyclic Ethers S Rosenberg R Leino 2674 Bimetallic PalladiumndashPlatinum-on-Carbon-Catalyzed HndashD Exchange
Reaction Synergistic Effect on Multiple Deuterium Incorporation T Maegawa N Ito K Oono Y Monguchi H Sajiki
2679 Efficient Copper-Catalyzed Synthesis of 2-Amino-4(3H)-quinazolinone and 2-Aminoquinazoline Derivatives X Huang H Yang H Fu R Qiao Y Zhao
2689 Synthesis and Chemoselective N- and O-Alkylation of Thiadiazolopyrimidine Nucleosides and Uridines A M L Hossion R Islam R K Kandahary T Nagamatsu
2697 Facile and Efficient Synthesis of a New Class of Indole-Substituted Pyridine Derivatives via One-Pot Multicomponent Reactions K Zhao X-P Xu S-L Zhu D-Q Shi Y Zhang S-J Ji
2709 Studies toward a Total Synthesis of Rhizoxin D Stereoselective Preparation of the C11ndashC19 Fragment S Padakanti C K Kumar E Ashok P Das
2715 A Short Synthesis of Enantiomeric Phytoprostanes B1 Type I W Perlikowska M Mikołajczyk
2719 Chemistry of Polyhalogenated Nitrobutadienes Part 7 A Novel Synthetic Access to Chlorinated Nitrile Oxides E Nutz V A Zapolrsquoskii D E Kaufmann
2725 Microwave-Assisted Silver(I)-Mediated Selective O-Alkylation of Aromatic Imidate Systems B K Singh C Cavalluzzo M De Maeyer Z Debyser V S Parmar E Van der Eycken
2729 Iodogen A Novel Reagent for the Oxidation of Urazoles under Heterogeneous Conditions A Khoramabadi A Shiri M A Zolfigol S Mallakpour
2733 An Unprecedented Synthesis of Eight-Membered-Ring Cyclic Thioimidic Esters by a Three-Component Reaction A Alizadeh R Hosseinpour
2737 A Novel Diastereoselective Synthesis of β-Phosphonato Unsaturated Thioimidates A Alizadeh N Zohreh
2741 Synthesis of 21-Benzisoxazoles by Nucleophilic Substitution of Hydrogen in Nitroarenes Activated by the Azole Ring N T Pokhodylo Y O Teslenko V S Matiychuk M D Obushak
2749 A Facile Synthesis of Two Series of Multifunctional Carbon Compounds from αα-Dihalo Ketones Using Allylsamarium Bromide X Liu S Zhang J Di
2756 Stereocontrolled Formation of Protected Aminodeoxyalditols from Simple Carbohydrate Precursors by Debenzylating Cycloetherification Y Jiang Z Fang Q Zheng H Jia J Cheng B Zheng
2761 trans-Stilbene as a Starting Material for the Synthesis of Tamoxifen Based on Palladium-Catalyzed Cross-Coupling Reactions C M Nunes J Limberger S Poersch M Seferin A L Monteiro
2766 Synthesis and Biological Evaluation of 6-Substituted Purinylcarbanucleosides with a Cyclopenta[b]thiophene Pseudosugar P Abeijoacuten J M Blanco O Caamantildeo F Fernaacutendez M D Garciacutea X Garciacutea-Mera J E Rodriacuteguez-Borges J Balzarini E De Clercq
2773 Synthesis and Electrochemical Signature of Novel Norbornyl-ferrocene Hybrids F A Khan S K Upadhyay
2778 A Regioselective TsujindashTrost Pentadienylation of 3-Allyltetronic Acid R Schobert B Barnickel
2785 Copper(I)-Catalyzed CarylndashCalkynyl Bond Formation of Aryl Iodides with Terminal Alkynes K G Thakur G Sekar
2790 Aminolysis of Epoxides Using Iridium Trichloride as an Efficient Catalyst J Agarwal A Duley R Rani R K Peddinti
2797 Preparation of Several Active N-Chloro Compounds from Trichloroisocyanuric Acid A Shiri A Khoramabadi-zad
2802 The First Mineral-Catalyzed One-Pot [3+1+2] Coupling Protocol for Multifunctionalized Fused-Ring Pyrimidines L D S Yadav A Rai
2809 Efficient Synthesis of Tetrahydro-β-carbolin-1-one and Dihydroisoquinolin-1-one Derivatives as Versatile Intermediates K E Judd M F Mahon L Caggiano
2818 A Concise Synthesis of ortho-Iodobenzyl Alcohols via Addition of ortho-Iodophenyl Grignard Reagent to Aldehydes and Ketones J Cvengroš D Stolz A Togni
XIII Forthcoming Articles
no 17 2825 Reactivity of Oxazol-5-(4H)-ones and Their Application toward Natural
Product Synthesis N M Hewlett C D Hupp J J Tepe 2840 Towards the Total Synthesis of 3-Hydroxyvibsanin E B D Schwartz
J R Denton P V Bernhardt H M L Davies C M Williams 2847 Structure Investigations of (ent)-Cladospolide D by De Novo Synthesis and
Kinetic and Thermodynamic Isomerization Y Xing J H Penn G A OrsquoDoherty
2855 New Applications of PhI(OAc)2 in Synthesis Total Synthesis and SAR Development of Potent Antitumor Natural Product PsymberinIrciniastatin A N Shao X Huang A Palani R Aslanian A Buevich J Piwinski R Huryk C Seidel-Dugan
2873 Total Synthesis of Largazole ndash Devolution of a Novel Synthetic Strategy B Wang C J Forsyth
2881 Formal Total Synthesis of Palmerolide A J Jaumlgel M E Maier 2893 Total Synthesis of Bongkrekic Acid via Sequential SuzukindashMiyaura Coupling
Reactions M Kanematsu M Shindo M Yoshida K Shishido 2905 Stereodivergent Approach to Both C28a-syn and C28a-anti Relative
Stereochemical Manifolds in the Lepadin Family via a TiCl4-Promoted G Li L J Carlson I K Sagamanova B W Slafer R P Hsung C Gilardi H M Sklenicka N Sydorenko
2915 Enantioselective Aldol Reaction of Tetrasubstituted Ketene Silyl Acetals with Achiral Aldehydes for the Construction of Asymmetric Tertiary Alcohols An Application for the Divergent Total Syntheses of Buergerinins F and G I Shiina T Iizumi Y-s Yamai Y-i Kawakita K Yokoyama Y-k Yamada
2927 Second-Generation Biomimetic Total Synthesis of Chaetominine A Coste G Karthikeyan F Couty G Evano
2935 Total Synthesis of (+)-Fostriecin and (+)-Phoslactomycin B S Shibahara M Fujino Y Tashiro N Okamoto T Esumi K Takahashi J Ishihara S Hatakeyama
2954 Stereochemical Assignments of the Chlorinated Residues in Victorin C A C Durow C Butts C L Willis
2963 Studies of the Asymmetric Total Synthesis of Clavilactone D by the lsquoLariatrsquo Cyclization Strategy T Yoshimitsu S Nojima M Hashimoto K Tsukamoto T Tanaka
2970 Total Synthesis of the Leucetta-Derived Alkaloid Calcaridine A P B Koswatta R Sivappa H V R Dias C J Lovely
2983 Formal Synthesis of Salinosporamide A Starting from D-Glucose T Momose Y Kaiya J-i Hasegawa T Sato N Chida
2992 Synthesis of Bioactive Natural Products by Asymmetric syn- and anti-Aldol Reactions A K Ghosh Z L Dawson
no 18 3003 Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural
Products B M Trost M K Brennan 3026 One-Pot Synthesis of Furo[34-b]pyridin-5(7H)-ones from 2-
Bromopyridine-3-carboxylic Acid and Carbonyl Compounds K Kobayashi T Kozuki H Konishi
3029 Iodocyclization of N-[2-(Methylthio)phenyl]propiolamides Selective Synthesis of 3-Iodo-15-benzothiazepin-4-ones T-S Jiang X-G Zhang J-H Li
3039 A Facile Synthetic Method for Fluorine-Containing 17-Phenanthrolines Pyridine-Ring Formation Reaction of N-Propargyl-68-bis(trifluoroacetyl)-quinolin-5-amine with Various Nucleophiles D Shibata E Okada M Hinoshita M Meacutedebielle
3047 Enantiotopic Discrimination in Palladium-Mediated Nucleophilic Substitutions on Achiral Substrates Chiral Ligand versus Chiral Nucleophile O Jacquet F Charnay J-C Fiaud J Ollivier
3051 Studies on the Chemistry of 2-[3-(2-Nitrophenyl)-2-oxopropyl]benzaldehydes Novel Syntheses of 5H-Benzo[b]carbazole-611-diones and Indolo[12-b]isoquinoline-611-diones M Fernaacutendez
3061 Studies on the C22ndashC23 Aldol Coupling of Spirangien M Lorenz N Bluhm M Kalesse
3067 One-Pot Synthesis of N-Alkyl Purine Pyrimidine and Azole Derivatives from Alcohols using Ph3PCCl4 A Rapid Route to Carboacyclic Nucleoside Synthesis M N Soltani Rad A Khalafi-Nezhad S Behrouz Z Asrari M Behrouz Z Amini
3077 Synthesis of 2-Amino-34-dihydroquinazolines and Imidazo[21-b]quinazoline-2-ones A Mishra S Batra
3089 Studies on the Reaction of Diimines with Thiourea Synthesis and Solvent-Induced cistrans-Isomerization of 135-Triazinane-2-thiones B Kaboudin T Ghasemi T Yokomatsu
3094 Suzuki Coupling of Heteroaromatic Chlorides Using Highly Electron-Donating ClickPhos Ligands S M Spinella Z-H Guan J Chen X Zhang
3099 Reaction of NN-Dioxyenamines with Anhydrides of Carboxylic and Sulfonic Acids A New Method for the Synthesis of a-Hydroxyoxime Derivatives A A Tabolin A V Lesiv S L Ioffe
3106 Directed ortho Metallation Chemistry and Phosphine Synthesis New Ligands for the SuzukindashMiyaura Reaction D B G Williams S J Evans H de Bod M S Mokhadinyana T Hughes
3113 New Functional Derivatives of 9-Phenylquinine P J Boratyński J SkarŜewski
3120 On the Synthesis of Asymmetric and Dissymmetric Amino Analogues of Troumlgerrsquos Base J Artacho K Waumlrnmark
3127 Synthesis of Polycyclic Sultams by Palladium-Catalyzed Intramolecular Cyclization K C Majumdar S Mondal N De
3136 Synthesis of Functionalized L-Cysteine and L-Methionine by Reaction with Electron-Deficient Acetylenes B A Trofimov A G Malrsquokina O A Shemyakina V V Nosyreva A P Borisova S S Khutsishvili L B Krivdin
3143 A lsquoClickrsquo Approach to the Synthesis of 3-[2-(1-Alkyltriazol-4-yl)ethyl]indoles M Petrini R R Shaikh
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
No 6 869 Stereoselective Transformations of meso Bicyclic Hydrazines Versatile
Access to Functionalized Aminocyclopentanes C Bournaud F Chung A P Luna M Pasco G Errasti T Lecourt L Micouin
888 Synthesis of Glycoaminoxy Acids as Novel Sugar Building Blocks A Malapelle R Ramozzi J Xie
891 Electrophilic ipso-Halocyclization of N-Arylpropynamides with Polyfluoroalkyl Alcohols Selective Synthesis of 8-(Polyfluoroalkoxy) azaspiro[45]trienes Z-Q Wang B-X Tang H-P Zhang F Wang J-H Li
903 Electrooxidation of Alcohols in N-Oxyl-Immobilized Silica GelWater Disperse System Approach to Totally Closed System M Kuroboshi K Goto H Tanaka
909 Synthetic Routes to Aminotriamantanes Topological Analogues of the Neuroprotector Memantinereg A A Fokin A Merz N A Fokina H Schwertfeger S L Liu J E P Dahl R K M Carlson P R Schreiner
913 Parallel Synthesis of Drug-like 5-Amino-Substituted 124-Thiadiazole Libraries Using Cyclization Reactions of a Carboxamidine Dithiocarbamate Linker J Y Park I A Ryu J H Park D C Ha Y-D Gong
921 Copper-Catalyzed Selective S-Arylation of 12-Bis(o-amino-1H-pyrazolyl) Disulfides with Arylboronic Acids P-S Luo F Wang J-H Li R-Y Tang P Zhong
929 2-Iodoxybenzoic AcidTetraethylammonium BromideWater An Efficient Combination for Oxidative Cleavage of Acetals C Kuhakarn W Panchan S Chiampanichayakul N Samakkanad M Pohmakotr V Reutrakul T Jaipetch
935 Synthesis of Quinonoid Analogues of Diospyrin S Sagar I R Green 941 A One-Pot Method for the Iodination of Aryl Amines via Stable Aryl
Diazonium Silica Sulfates Under Solvent-Free Conditions A Zaroi A R Hajipour L Khazdooz
945 Poly(NN-dichloro-N-ethylbenzene-13-disulfonamide) and NNNN-Tetrachlorobenzene-13-disulfonamide as Novel Reagents for the Synthesis of N-Chloroamines Nitriles and Aldehydes R Ghorbani-Vaghei H Veisi
951 Synthesis of an (R)-Garner-type Aldehyde from L-Serine Useful Building Block for a (+)-Furanomycin Derivative G Bartoli G Di Antonio R Fiocchi S Giuli E Marcantoni M Marcolini
957 An Efficient and Highly Selective Synthesis of (Z)-Fluoroenol Phosphates from Hydroxy Difluorophosphonates P Beier R Pohl A V Alexandrova
963 Iodine-Catalyzed Three-Component Reaction A Rapid Synthesis of α-Alkoxy Azides and Homoallyl Ethers J S Yadav B V S Reddy G M Reddy R Narender
969 Rhodium(I)-Catalyzed Cycloisomerization of 13-Dienes with Alkenes in a Tether Y Oonishi A Saito M Mori Y Sato
980 Synthesis of New Optically Active D-GlucosaminendashPyrrole Derivatives B A Frontana-Uribe M V Escaacutercega-Bobadilla J Juaacuterez-Lagunas R A Toscano G A Garciacutea de la Mora M Salmoacuten
985 Partially Saturated Indeno[12-b]indole Derivatives via Deoxygenation of Heterocyclic α-Hydroxy-NO-hemiaminals H-J Hemmerling G Reiss
1000 Light-Induced Synthesis of Π-Extended Tetrathiafulvalenes Incorporating Ferrocenes An Efficient Route for the Synthesis of Electron-Donor Materials A A O Sarhan C Bolm
1007 Preparation of Nβ-Fmoc-Protected Aza-β3-Amino Acids with Nonproteinogenic Hydrophobic Side Chains for Solid-Phase Syntheses of Pseudopeptides M Laurencin P Bauchat M Baudy-Flocrsquoh
1014 Diastereomeric (η4-diene)Fe(CO)3 Complexes Containing Chiral Amide Groups A Convenient Method for the Resolution of Amino Acids M Schumacher G Coste L Miesch
1021 Palladium-Catalysed Heck Reactions of Alk-1-en-3-ones with Aryl Bromides A Very Simple Access to (E)-1-Arylalk-1-en-3-ones M Lemhadri Y Fall H Doucet M Santelli
1036 An Improved Process for the Synthesis of 4H-Imidazo[15-α][14]benzodiazepines J Yang Y Teng S Ara S Rallapalli J M Cook
1041 Meta- and Para-Difunctionalization of Arenes via an Ortho-Magnesiation and a Subsequent SulfoxidendashMagnesium Exchange L Melzig C B Rauhut P Knochel
XIII Forthcoming Articles
No 7 1049 Catalytic Transformations of Benzylic Carboxylates and Carbonates
R Kuwano 1062 A Simple and Practical Method for the Oxidation of Thebaine to 14-
Hydroxycodeinone by V2O5ndashH2O2 S Das Sharma D Konwar 1065 Umpolung with Sulfur Dioxide CarbonndashCarbon Cross-Coupling of Electron-
Rich 13-Dienes and Alkenes Application to the Enantioselective Synthesis of Long-Chain Polyketide Fragments M Turks C J Exner C Hamel P Vogel
1075 One-Pot Synthesis of 14-Diarylnaphthalenes via a WittigndashHorner Reaction[4+2] CycloadditionDehydrogenation Sequence Z Chen W Shou Y Wang
1081 A Novel and General Method for the Formation of S-Aryl Se-Aryl and Te-Aryl Phosphorochalcogenoates Y-X Gao G Tang Y Cao Y-F Zhao
1087 A Remarkable Access to γ-Fluoroalkylated Propargylamine Derivatives or Fluoroalkylated Dihydroisoxazoles via the Reaction of Fluoroalkylated Acetylides with Various Nitrones T Konno K Moriyasu T Ishihara
1095 Short and Practical Syntheses of (S)-(+)-3-(p-Tolylsulfinyl)furan-2(5H)-one and (S)-(+)-3-(p-Tolylsulfinyl)-56-dihydropyran-2-one D Cruz Cruz A Hernaacutendez Linares F Yuste M R Martiacuten J L Garciacutea Ruano
1099 Decarboxylative Aldol-Type Reaction of 2-(Trifluoroacetyl)-13-diazoles with Activated Acetic Acids P V Khodakovskiy D M Volochnyuk A A Tolmachev
1105 Synthesis of 2-[(Arylmethylene)amino]cyclopropanecarbonitriles via a Two-Step Ring Transformation of 2-(Cyanomethyl)aziridines S Mangelinckx M Drsquohooghe S Peeters N De Kimpe
1113 Synthesis of Dendrimeric Tumor-Associated Mucin-Type Glycopeptide Antigens T Becker A Kaiser H Kunz
1123 A Simple and Efficient Oxidation Procedure for the Synthesis of Acid-Sensitive Epoxides O Bortolini G Fantin M Fogagnolo
1127 Rapid Chemoselective Deprotection of Benzyl Esters by Nickel Boride J M Khurana R Arora
1131 Three-Component Coupling of Isoquinoline Activated Alkyne and Nitromethane A Facile Synthesis of Nitromethyl Derivatives of 12-Dihydroisoquinolines J S Yadav B V S Reddy N N Yadav M K Gupta
1137 Palladium Supported on a Polyionic Resin as an Efficient Ligand-Free and Recyclable Catalyst for Heck SuzukindashMiyaura and Sonogashira Reactions B Basu S Das P Das B Mandal D Banerjee F Almqvist
1147 Oxidation of 25-Dialkylpyrrole Derivatives with Cerium(IV) Ammonium Nitrate R Voloshchuk M Gałęzowski D T Gryko
1153 Practical Syntheses of Enantiomerically Pure Key Intermediates of Opioid Receptor-like 1 (ORL1) Antagonists T Yoshizumi A Ohno T Tsujita H Takahashi O Okamoto I Hayakawa H Kigoshi
1163 An Environmentally Benign TEMPO-Catalyzed Efficient Alcohol Oxidation System with a Recyclable Hypervalent Iodine(III) Reagent and Its Facile Preparation X-Q Li C Zhang
1170 Efficient and Stereoselective Rearrangement of BaylisndashHillman Acetates Catalyzed by Gold(I) ChlorideSilver(I) Trifluoromethanesulfonate Y Liu D Mao J Qian S Lou Z Xu Y Zhang
1175 The First Total Synthesis of Kynapcin-24 by Palladium Catalysis L-Y Yang C-F Chang Y-C Huang Y-J Lee C-C Hu T-H Tseng
1180 Enantioselective Synthesis of N-Protected α-Amino Acid Hydrazides M Bibian S El-Habnouni J Martinez J-A Fehrentz
1185 Synthesis of 11H-Indolo[32-c]quinoline-6-carboxylic Acids by Cascade AutoxidationndashRing Contractions A Becker S Kohfeld T Pies K Wieking L Preu C Kunick
1190 Reaction of N-Nonaflylbenzotriazole with Silyl Enol Ethers M Uhde T Ziegler
1195 2-(Benzoylimino)thiazolidin-4-ones Formation by an Alternative Ring Closure and Analysis of Rotational Barriers H-G Haumlcker P W Elsinghorst S Michels J Daniels G Schnakenburg M Guumltschow
1204 Microwave-Assisted Synthesis and Functionalization of Selenolopyrimidines S Hesse C Chenet D Thomae G Kirsch
1209 12-Disubstituted 4-Quinolones via Copper-Catalyzed Cyclization of 1-(2-Halophenyl)-2-en-3-amin-1-ones R Bernini S Cacchi G Fabrizi A Sferrazza
1220 A New Atom-Economical and Selective Synthesis of Secondary and Tertiary Alkylamines by Means of CpIridium Complex Catalyzed Multiple N-Alkylation of Ammonium Salts with Alcohols without Solvent R Yamaguchi Z Mingwen S Kawagoe C Asai K-i Fujita
1224 Synthesis of Regioisomerically Pure 5-Functionalized 27-Dichlorofluoresceins J C Castro A Malakhov K Burgess
XIII Forthcoming Articles
No 8 1227 Michael Additions to Activated Vinylphosphonates T Janecki J Kędzia
T Wąsek 1255 A Facile and General Synthesis of 2β-Aminosteroids X Ke H Hu
D Zhou W Xu Q Zhu N P Reddy X Hu 1261 Efficacious Preparation of Oppolzerrsquos Glycylsultam via the Deleacutepine
Reaction A Isleyen C Gonsky R C Ronald P Garner 1265 Synthesis of Masked Vicinal Amino Aldehydes of Pyrrolizine and Pyrrolo
[12-c]thiazole Series A V Tverdokhlebov A V Denisenko A A Tolmachev Y M Volovenko S V Shishkina O V Shishkin
1271 Preparation of 9-Substituted Pyridine-Stretched Adenines and Hypoxanthines J A Crawford W Fraser C A Ramsden
1279 A Versatile Synthesis of Heterocyclic Analogues of Neoflavonoids from Enamino Ketones V S Moskvina V P Khilya O V Turov U M Groth
1287 New Stereoselective Synthesis of Paeonilactone B F G Gatti S Serra 1291 The Use of NN-Dialkyltrimethylsilylamines in the Synthesis of
Pentamethinium Salts M Kořiacutenek M Rybaacutečkovaacute Boumlhm 1297 Synthesis of Triazoles via Regioselective Reactions of Aryl Azides with
Cyanoacetyl Pyrroles and Indoles N T Pokhodylo V S Matiychuk M D Obushak
1301 Gallium(III) Chloride Catalyzed Hydroarylation of Arylacetylenes with Naphthols and Phenols A Facile Synthesis of Vinylarenes J S Yadav B V S Reddy S Sengupta S K Biswas
1305 Electrophilic Bromination of meta-Substituted Anilines with N-Bromosuccinimide Regioselectivity and Solvent Effect S Bartoli A Cipollone A Squarcia A Madami D Fattori
1309 Cross-Coupling Reactions of Halopurines with Aryl- and Alkyltrifluoroborates The Scope and Limitations in the Synthesis of Modified Purines Z Hasniacutek R Pohl M Hocek
1318 A Convenient Method for Converting Hydroxyacetophenones into Their Ethylene or Trimethylene Acetals F Ono H Takenaka T Fujikawa M Mori T Sato
1323 γ-Chloromagnesio γ-Lactones and δ-Chloromagnesio δ-Lactones Generation Properties and Synthetic Uses H Shimizu S Fukuda S Sugiyama T Satoh
1336 Click Reactions with Nitroxides T Kaacutelai W L Hubbell K Hideg 1341 Synthesis of Novel 14-Benzoquinone-Containing 123-Triazoles An Entry
Into a New Library F Algi M Balci 1348 Efficient Synthesis of Two Sialylated Tetrasaccharides Found in Goat Milk
P K Mandal A K Misra 1355 Dendrimers of Vaccines Consisting of Tumor-Associated Glycopeptide
Antigens and T Cell Epitope Peptides S Keil A Kaiser F Syed H Kunz
1370 IBXTBAB-Mediated Oxidation of Primary Amines to Nitriles F Drouet P Fontaine G Masson J Zhu
1375 Chemoselectivity of Multicomponent Condensations of Barbituric Acids 5-Aminopyrazoles and Aldehydes E A Muravyova S V Shishkina V I Musatov I V Knyazeva O V Shishkin S M Desenko V A Chebanov
1386 Stereoselective Total Syntheses of Leiocarpin A and (ndash)-Galantinic Acid Starting from D-Mannitol K Nagaiah D Sreenu K V Purnima R S Rao J S Yadav
1393 A Facile Mild Deprotection Protocol for 13-Dithianes and 13-Dithiolanes with 30 Hydrogen Peroxide and Iodine Catalyst in Aqueous Micellar System N C Ganguly S K Barik
1400 Rhodium-Catalyzed Gram-Scale Synthesis of Highly Substituted Pyridine Derivatives K Parthasarathy C-H Cheng
1403 Enantioselective Synthesis of (R)-Propylene Carbonate from Ethyl (S)-Lactate J M Whitaker R C Ronald
XIII Forthcoming Articles
no 9 1405 Transition-Metal-Catalyzed Site-Selective Cross-Coupling of Di- and
Polyhalogenated Compounds J-R Wang K Manabe 1428 An Improved Synthesis of (4-4-Hydroxy-3-isopropyl-5-[(4-nitrophenyl)
ethynyl]benzyl-35-dimethylphenoxy)acetic Acid (NH-3) M B Gopinathan K S Rehder
1431 Copper-Catalyzed Tandem CndashN Bond Formation Reaction Selective Synthesis of 2-(Trifluoromethyl)benzimidazoles M-W Chen X-G Zhang P Zhong M-L Hu
1437 Synthesis and Thermochemical Properties of Stereoisomeric Dihydroxy- and Tetrahydroxyalkylammonium Salts M Thomas L Rothman J Hatcher P Agarkar R Ramkirath S Lall-Ramnarine R Engel
1445 Preparation of 5-Substituted 2-(2-Alkylaryl-1H-imidazol-4-yl)oxazoles and 5-Substituted 2-(2-Alkylarylthiazol-4-yl)oxazoles by Utilizing 5-Substituted 2-(2-Bromo-11-diethoxyethyl)oxazole as a Synthon D R St Laurent J L Romine
1459 Novel and Efficient Methods for the Synthesis of Symmetrical Trisulfides A Kertmen S Lach J Rachon D Witt
1463 An Environmentally Benign Electrochemical Process for the Reduction of Carboxylic Acid Hydrazides to Amides M Mentel M J Beier R Breinbauer
1469 Synthesis of 1-Chloroalkynes from Alkynylsilanes Using Trichloroisocyanuric Acid as Chlorinating Agent M H Vilhelmsen A S Andersson M B Nielsen
1473 A Convenient Approach to Enantioenriched Cyclopropanes Bearing Electron-Withdrawing Functionalities H Krawczyń K Wąsek J Kędzia
1477 Synthesis of Cyclopropenes via 12-Elimination of Bromocyclopropanes Catalyzed by Crown Ether W M Sherrill R Kim M Rubin
1485 A Base-Catalysed One-Pot Three-Component Coupling Reaction Leading to Nitrosubstituted Pyrroles I R Baxendale C D Buckle S V Ley L Tamborini
1494 Synthesis of 4-Alkylidene-4H-31-benzoxazine Derivatives by Acid-Catalyzed Cyclization of 2-Isocyanophenyl Ketones in the Presence of a Vinyl Ether K Kobayashi Y Okamura H Konishi
1499 Synthesis of Higher Helicenes via Olefin Metathesis and CndashH Activation J Cocircteacute S K Collins
1506 Azido- and Ethynyl-Substituted 2262-Terpyridines as Suitable Substrates for Click Reactions A Winter A Wild R Hoogenboom M W M Fijten M D Hager R-A Fallahpour U S Schubert
1513 Synthesis of 2-(Arylamino)ethanethiols via Lewis Acid Catalyzed Aminolysis of 22-Dimethylthiirane as Precursors of the 14-Benzothiazine Nucleus R Spogli S Sabatini G Manfroni O Tabarrini V Cecchetti
1520 Iron(III) Chloride A Versatile Catalyst for the Practical Synthesis of 3-Sulfenylindoles J S Yadav B V S Reddy Y J Reddy K Praneeth
1525 Organocatalytic Enantioselective Conjugate Addition of 2-Fluoromalonate to Nitroolefins Direct Synthesis of Chiral Fluorinated γ-Nitro Carboxylic Acid Derivatives H Li L Zu H Xie W Wang
1531 Asymmetric Transfer Hydrogenation of Ketimines with Trichlorosilane Structural Studies Z Zhang P Rooshenas H Hausmann P R Schreiner
1545 Prolinol Sulfinyl Ester Derivatives Organocatalytic Michael Addition of Ketones to Nitroolefins under Neat Conditions X Zeng G Zhong
1551 Asymmetric Oxidations of Electron-Poor Alkenes Promoted by the β-Amino AlcoholTBHP System A Russo A Lattanzi
1557 Enantioselectivity Switch in Direct Asymmetric Aminoxylation Catalyzed by Binaphthyl-Based Chiral Secondary Amines T Kano A Yamamoto F Shirozu K Maruoka
1564 Enantioselective Conjugate Addition of N-Heterocycles to αβ-Unsaturated Ketones Catalyzed by Chiral Primary Amines G Luo S Zhang W Duan W Wang
1573 Sulfonyl Hydrazine as New Functionality in Organocatalysis Camphorsulfonyl Hydrazine Catalyzed Enantioselective Aza-Michael Addition L-Y Chen H He B-J Pei W-H Chan A W M Lee
1578 Conversion of Primary Alcohols and Aldehydes into Methyl Esters by Ruthenium-Catalysed Hydrogen Transfer Reactions N A Owston T D Nixon A J Parker M K Whittlesey J M J Williams
1582 Addendum and Erratum XVII Forthcoming Articles
no 10 1583 Organocatalytic Formation of Quaternary Stereocenters M Bella
T Gasperi 1615 Regioselective Synthesis of 5H-Thiazolo[32-a]pyrimidin-5-ones from
MoritandashBaylisndashHillman Adduct Acetates under Solvent-Free and Base-Free Conditions W Zhong B Guo F Lin Y Liu W Su
1623 First Synthesis of 5-Cyanosalicylates by Formal [3+3] Cyclocondensations of 13-Bis(silyloxy)-13-butadienes A Riahi O Fatunsin M Shkoor R Dede H Reinke C Fischer P Langer
1635 Reaction of Isocyanides Dialkyl Acetylenedicarboxylates and a-Keto Lactones Unexpected Participation of an Ester Carbonyl Group in the Isocyanide-Based Three-Component Reaction A A Esmaeili H Vesalipoor
1639 An Efficient and Chemoselective Synthesis of 16-Naphthyridines and Pyrano[32-c]pyridines under Microwave Irradiation Z-G Han S-J Tu B Jiang S Yan X-H Zhang S-S Wu W-J Hao X-D Cao F Shi G Zhang N Ma
1647 N-Activation of N-Arylimidazoles Facile Syntheses of N-Alkyl-N-arylimidazolium Iodides from Less Expensive Chloro Substrates A M Oertel V Ritleng M J Chetcuti
1651 Synthesis of Polyhalogenated 2-(Phenylamino)pyridines by Thermal Amination Reactions S R Waldvogel A Faust W Barkmann R Froumlhlich O Wolff
1655 Cyanide Ion Promoted Addition of Acylphosphonates to Diethyl Cyanophosphonate Synthesis of Phosphonocyanohydrin O-Phosphates A S Demir A Aybey M Emrullahoglu
1659 Straightforward and Scalable Synthesis of Orthogonally Protected 37-Diazabicyclo[410]heptane H Schramm M Pavlova C Hoenke J Christoffers
1663 Hypervalent Iodine Mediated Oxidation of 12-Diaminobenzimidazole and Its Schiff Bases Efficient Synthesis of 3-Amino-124-benzotriazine and 2-Aryl-124-triazolo[15-a]benzimidazoles A Kumar M Parshad R K Gupta D Kumar
1667 Synthesis of the Reported Protoberberine Gusanlung D P B Wakchaure S Easwar N P Argade
1673 2-(Azidomethyl)arylboronic Acids in the Synthesis of Coumarin-Type Compounds M I Naumov A V Nuchev N S Sitnikov Y B Malysheva A S Shavyrin I P Beletskaya A E Gavryushin S Combes A Y Fedorov
1683 Asymmetric Synthesis of 12-anti-Disubstituted Taurine Derivatives D Enders D Iffland G Raabe
1689 A Novel One-Pot Three-Component Synthesis of 5-Imino-2358-tetrahydropyrazolo[12-a]pyridazin-1-one Derivatives B Qian M-J Fan Y-X Xie L-Y Wu Y Shi Y-M Liang
1694 One-Portion Synthesis of 2-Acetoxy Carbonyl Compounds from Aldehydes by Using an Acetylated Masked Acyl Cyanide H Nemoto T Kawamura K Kitasaki K Yatsuzuka M Kamiya Y Yoshioka
1703 Synthesis of 9-Anthryl Ethers from trans-910-Dihydro-910-dimethoxyanthracene by Acid-Catalyzed Transetherification K S Jang H Y Shin D Y Chi
1708 Efficient Synthesis of Azo Dye Labeled Terpenes Sugars and Steroids Using N-(4-Arylazobenzoyl)-1H-benzotriazoles A R Katritzky S R Tala N E Abo-Dya Z K Abdel-Samii
1715 Tandem CH-ActivationndashImine-Formation Reaction A New Route to Imidazo[21-a]phthalazines A Heim-Riether K R Gipson
1720 A Convenient and Efficient α-Sulfenylation of Carbonyl Compounds E Okragla S Demkowicz J Rachon D Witt
1725 Stereoselective Synthesis of β-Branched Phenylalanine Derivatives via Chelate-Claisen Rearrangement C Quirin U Kazmaier
1732 Catalyst-Free and Base-Free Water-Promoted SNAr Reaction of Heteroaryl Halides with Thiols B Sreedhar P S Reddy M A Reddy
1739 Convenient Methods for Synthesis of C2-Symmetric Diphenyltetrahydrothiophenes M Periasamy G Ramani G P Muthukumaragopal
1744 Highly Diastereoselective Conjugate AdditionndashElimination of Chiral Nickel(II) Glycinate with Activated Allylic Acetates for Asymmetric Synthesis of Glutamic Acid Derivatives J Wang J Shi X Zhang D Lin H Jiang H Liu
1753 Synthesis of 36-Dimethoxybenzene-12-diamine and of 47-Dimethoxy-2-methyl-1H-benzimidazole T Besset C Morin
1757 An Inexpensive Procedure for Reductive Aminations Using Dimethylamineborane on Millimolar and Molar Scale R Ortmann M Schlitzer
1760 Classics in Stereoselective Synthesis Edited by E M Carreira L Kvaerno Reviewed by Rolf Breinbauer
XV Forthcoming Articles
no 11 1761 Transition-Metal-Catalyzed Enantioselective Synthesis of Compounds with
Non-Centrochirality M Ogasawara S Watanabe 1786 One-Pot Synthesis of 3-Acyl-2-(alkylsulfanyl)indoles and 2-(Alkylsulfanyl)-
indole-3-carboxylates from (2-Isocyanophenyl)methyl Ketones or (2-Isocyanophenyl)acetates S Fukamachi H Konishi K Kobayashi
1791 Efficient and Recyclable Phthalocyanine-Based Sensitizers for Photooxygenation Reactions H Xu W-K Chan D K P Ng
1797 A Facile and Practical One-Pot Synthesis of β-Oxo Thioamides from β-Oxo Amides and Isothiocyanates P Huang D Xiang Y Zhou Y Liang T Na D Dong
1801 Microwave-Promoted Solid-Acid-Catalyzed One-Pot Synthesis of Phthalazinones V M Outerbridge S M Landge H Tamaki B Toumlroumlk
1807 Benzylic Brominations with N-Bromosuccinimide in (Trifluoromethyl)-benzene D Suarez G Laval S-M Tu D Jiang C L Robinson R Scott B T Golding
1811 Synthesis of Thioflavanone and Flavanone Derivatives by Cyclization of Chalcones W Konieczny M Konieczny
1815 A New and Expedient Total Synthesis of Ochratoxin A and d5-Ochratoxin A B Gabriele M Attya A Fazio L Di Donna P Plastina G Sindona
1821 Synthesis of Benzopyrrolizidinones by NorrishndashYang Cyclization of 3-(Acylmethyl)-2-alkylisoindol-1-ones J Wu W Zhang C Wang
1829 Reactions of MoritandashBaylisndashHillman Acetates with Huisgen Zwitterions A Novel Strategy for the Synthesis of β-Amino Acid Derivatives A Jose R R Paul R Mohan S C Mathew A T Biju E Suresh V Nair
1834 Peracetylated β-Allyl C-Glycosides of D-Ribofuranose and 2-Deoxy- D-ribofuranose in the Chemical Literature Until Now Mirages in the Literature H Otero Martinez H Reinke D Michalik C Vogel
1841 Core-Tetrasubstituted Naphthalene Diimides by Stille Cross-Coupling Reactions and Characterization of Their Optical and Redox Properties S-L Suraru F Wuumlrthner
1846 A Practical Synthesis of Indole-Based Heterocycles Using an Amidoaluminum-Mediated Strategy R Todd M M Hossain
1851 Synthesis of Fluorinated Pyrrolo[23-b]pyridine and Pyrrolo[23-d]pyrimidine Nucleosides V O Iaroshenko Y Wang D V Sevenard D M Volochnyuk
1858 Recyclization Reactions of 5-Formyl-13-dimethyluracil with Electron-Rich Amino Heterocycles A P Mityuk D M Volochnyuk S V Ryabukhin A S Plaskon A Shivanyuk A A Tolmachev
1865 Facile Synthesis of Fluorinated 1-Desazapurines V O Iaroshenko D V Sevenard D M Volochnyuk Y Wang A Martiloga A O Tolmachev
1876 A Practical Synthesis of 3-Diethoxyphosphoryl-12-pyridazine Derivatives J-C Monbaliu J Marchand-Brynaert
1881 Enantioselective Reduction of Prochiral Ketones Employing Sprouted Pisum sativa as Biocatalyst J S Yadav B V S Reddy C Sreelakshmi A B Rao
1886 Application of Phenolate Ion Mediated Intramolecular Epoxide Ring Opening in the Enantioselective Synthesis of Functionalized 23-Dihydrobenzofurans and 1-Benzopyrans S K Dinda S K Das G Panda
1897 Complementary Synthetic Approaches to Constitutionally Diverse N-Aminoalkylated Isoindolinones Application to the Synthesis of Falipamil and 5-HT1A Receptor Ligand Analogues M Lorion A Couture E Deniau P Grandclaudon
1904 Selective Deprotection of Silyl Ethers with Sodium Periodate J Li D Menche
1909 Micellar Solution of Sodium Dodecyl Sulfate (SDS) Catalyzes KabacknikndashFields Reaction in Aqueous Media S Sobhani A Vafaee
1916 Convenient Methods for the Synthesis of a Library of Hemilabile Phosphines M V Jimeacutenez J J Peacuterez-Torrente M I Bartolomeacute L A Oro
1923 Terminal Aziridines by Addition of Grignard Reagents or Organoceriums to an (α-Chloro)sulfinylimine D M Hodgson J Kloesges B Evans
1933 A Robust Synthesis of Nε-(Carboxymethyl)-L-lysine (CML) R Csuk S Stark A Barthel R Kluge D Stroumlhl
1935 One-Pot Curtius Rearrangement Processes from Carboxylic Acids O Leogane H Lebel
XV Forthcoming Articles
no 12 1941 The Chemistry of Deprotonated α-Aminonitriles T Opatz 1960 An Efficient Synthesis of Tetraalkyl 2345-Thiophenetetracarboxylate
Derivatives A Alizadeh R Hosseinpour 1963 Facile Deprotection of Bulky (Trialkylsilyl)acetylenes with Silver Fluoride
S Kim B Kim J In 1969 Highly Efficient and Reusable Ionic Liquids for the Catalyzed
Hydroamination of Alkenes with Sulfonamides Carbamates and Carboxamides L Yang L-W Xu C-G Xia
1975 Synthesis of 2391016172324-Octasubstituted Phthalocyaninatozinc(II) Complexes Mediated by Reductive Agents G A Gauna A C Monsalvo J Awruch
1979 A Short and Efficient Synthesis of 3-2-[2-(Bromomethyl)thiazol-4-yl]-ethynyl-5-fluorobenzonitrile A Precursor for PET Radioligand [18F]SP203 M B Gopinathan C Jin K S Rehder
1983 Synthesis of a Substituted Benzazepin-2-one Dihydrate S K Boini R K Vaid K P Moder D Mitchell
1987 Synthesis of Novel Trisubstituted Imidazolines F J Lakner M A Parker B Rogovoy A Khvat A Ivachtchenko
1991 A Novel Synthesis of N-But-3-enyl-α- and β-Amino Acids T T Van Nguyen R T C Brownlee A B Hughes
1999 Synthesis of Substituted 5-(3-Hydroxypropyl)pyrrolidin-2-ones and Pyrrolizidinones from Nitroethane via C3 Functionalized 56-Dihydro-4H-12-oxazines A Novel Approach to Some Analogues of the Antidepressant Rolipram A Yu Sukhorukov A V Lesiv Y A Khomutova S L Ioffe V A Tartakovsky
2009 Chiral Cyclobutanols and Cyclopentane Dimers via Samarium(II) Iodide Induced Keto-Olefin Cyclisations of Carbohydrate-Derived Unsaturated Ketones D B G Williams J Caddy K Blann J J C Groveacute C W Holzapfel
2015 Synthesis of Perfluoroalkylthio-Substituted Ferrocenes C Rhode J Lemke M Lieb N Metzler-Nolte
2019 Functionalization of Polyhedral Oligomeric Silsesquioxane (POSS) via Nucleophilic Substitution M Dutkiewicz H Maciejewski B Marciniec
2025 A Novel Synthesis of Aryl Mesylates via One-Pot DemethylationndashMesylation of Aryl Methyl Ethers Using a Mixture of Phosphorus Pentoxide in Methanesulfonic Acid B Kaboudin Y Abedi
2029 Anionic Cyclization of (NN-Dimethylamino)[2-(prop-2-yn-1-yloxy)aryl]-acetonitriles T Zdrojewski J Musielak A Jończyk
2035 Strecker-Type Reaction Catalyzed by Carboxylic Acids in Aqueous Media Z Xie G Li G Zhao J Wang
2040 Synthesis of Novel Structurally Simplified Estrogen Analogues with Electron-Donating Groups in Ring A L F Tietze C A Vock I K Krimmelbein L Nacke
2061 On the Resolution of Secondary Phosphine Oxides via Diastereomeric Complex Formation The Case of tert-Butylphenylphosphine Oxide J Holt A M Maj E P Schudde K M Pietrusiewicz L Sieroń W Wieczorek T Jerphagnon I W C E Arends U Hanefeld A J Minnaard
2066 Enantioselective Copper-Catalyzed Conjugate Addition of Dimethylzinc to 5-(1-Arylalkylidene) Meldrumrsquos Acids A Wilsily T Lou E Fillion
2073 SuzukindashMiyaura Coupling Reactions Using Phosphite Ligands M Jang Y Jo I-K Oh H M Jung S Lee
2076 Synthesis of 2-Methylindoline- and 2-Methyl-1234-tetrahydroquinoline-Derived Phosphoramidites and Their Applications in Iridium-Catalyzed Allylic Alkylation of Indoles W-B Liu H He L-X Dai S-L You
2083 Stereocontrolled Synthesis of 13-Amino Alcohols by Reduction of Substituted 2-1-[(tert-Butylsulfinyl)amino]alkylcyclohexanones J C Gonzaacutelez-Goacutemez F Foubelo M Yus
2089 Tunable Phosphoramidite Ligands for Asymmetric Hydrovinylation Ligands par excellence for Generation of All-Carbon Quaternary Centers C R Smith H J Lim A ZhangT V RajanBabu
2101 Copper-Catalyzed Asymmetric Ring-Opening Reaction of Oxabenzonorbornadienes with Grignard and Aluminum Reagents R Millet L Gremaud T Bernardez L Palais A Alexakis
2113 A Simplified Synthesis of Takemotorsquos Catalyst A Berkessel B Seelig 2116 Pharmaceutical Substances Syntheses Patents and Applications of the
Most Relevant AIPs Edited by Axel Kleeman Juumlrgen Engel Bernhard Kutscher Dietmar Reichert Reviewed by I Agranat
XV Forthcoming Articles
no 13 2117 Recent Advances in the Aza-Claisen Rearrangement K C Majumdar
T Bhattacharyya B Chattopadhyay B Sinha 2143 A Novel and Convenient Synthesis of lsquoReversedrsquo Diamidino 25-Aryl- and
25-Azaheterocycle-Substituted Furans L Hu D W Boykin 2146 Efficient and General Preparation of Pyranostilbenes First Total Synthesis
of Artocarbene and Pawhuskin B B H Park Y R Lee W S Lyoo 2155 Mild Oxidation of Diarylacetylenes to 12-Diketones Using Oxone in
Trifluoroacetic Acid J-H Chu Y-J Chen M-J Wu 2163 One-Pot Microwave-Assisted Selective Azido ReductionTandem Cyclization
in Condensed and Solid Phase with Nickel Boride N Shankaraiah N Markandeya M Espinoza-Moraga C Arancibia A Kamal L Silva Santos
2171 Pyrrolo[321-ij]quinolin-4-one and Pyrrolo[321-ij]quinolin-6-one H McNab D J Nelson E J Rozgowska
2175 Practical Synthesis of 5-Substituted Tetrazoles under Microwave Irradiation J Roh T V Artamonova K Vaacutevrovaacute G I Koldobskii A Hrabaacutelek
2179 A Simple Method for the Synthesis of 3-Arylthieno[23-b]pyridines via Iodine-Mediated Cyclization of 3-(1-Arylalkenyl)-2-[(1-phenylethyl)sulfanyl]pyridines K Kobayashi D Nakamura Y Shiroyama S Fukamachi H Konishi
2184 Synthesis of Four Lysine-Linked Cereulide Analogues Showing Ionophoric Activity Towards Potassium Cations as Lead Compounds for Emetic Toxin-Detection by Immunoassays A Makarasen T Nishikawa M Isobe
2205 Synthesis of α-Aliphatic and β-Aromatic Substituted Taurines via Regioselective Ring Opening of Thiiranes with Ammonia H Yu S Cao L Zhang G Liu J Xu
2210 Stability of 5(6)-Carboxyfluorescein in Microwave-Assisted Synthesis of Fluorescein-Labelled O-Dimannosylated Peptides R Kowalczyk P W R Harris R P Dunbar M A Brimble
2223 Diversity-Oriented Synthesis of Functionalized Diaryl Sulfones by Regioselective [3+3] Cyclizations of 13-Bis(siloxy)buta-13-dienes with 2-(Arylsulfonyl)-3-ethoxy-2-en-1-ones Scope and Limitations M Shkoor A Riahi O Fatunsin H Reinke C Fischer P Langer
2236 Synthesis of Functionalized Salicylates by Formal [3+3] Cyclocondensation of 13-Bis(silyloxy)buta-13-dienes with 3-Alkoxy-2-en-1-ones G Mroszlig S Ladzik H Reinke A Spannenberg C Fischer P Langer
2249 Synthetic Approach to Alkoxy-β-(trifluoromethyl)styrenes and Their Application in the Synthesis of New Trifluoromethylated Heterocycles V M Muzalevskiy V G Nenajdenko A V Shastin E S Balenkova G Haufe
2260 o-Benzenedisulfonimide as a Powerful and Recyclable Organocatalyst for the Nazarov Reaction M Barbero S Cadamuro A Deagostino S Dughera P Larini E G Occhiato C Prandi S Tabasso R Vulcano P Venturello
2267 The Catalytic Potential of 4-Guanidinylpyridines in Acylation Reactions I Held E Larionov C Bozler F Wagner H Zipse
2278 Iron(III) Chloride in EthanolndashWater Highly Efficient Catalytic System for the Synthesis of Garcia Gonzalez Polyhydroxyalkyl- and C-Glycosylfurans L Nagarapu M V Chary A Satyender B Supriya R Bantu
2283 Ruthenium-Catalyzed Addition of Primary Amides to Alkynes A Stereoselective Synthesis of Secondary Enamides L J Gooszligen M Blanchot K S M Salih K Gooszligen
2289 Binaphthyl-Modified Quaternary Phosphonium Salts as Chiral Phase Transfer Catalysts Application to Asymmetric Amination of β-Keto Esters R He K Maruoka
X Table of Contents XI Forthcoming Articles
no 14 2293 Direct Methods for Stereoselective Polypropionate Synthesis A Survey
J Li D Menche 2316 Synthesis of Symmetrical Ketones from Grignard Reagents and
11-Carbonyldiimidazole D Bottalico V Fiandanese G Marchese A Punzi
2319 Synthesis of 45-Substituted Imidazoles by a Fast Condensation of 12-Diketones and Urotropine in Heterogeneous Medium G Bratulescu
2321 (Arylsulfonyl)acetones and -acetonitriles New Activated Methylenic Building Blocks for Synthesis of 123-Triazoles N T Pokhodylo V S Matiychuk M D Obushak
2324 A Safe Convenient and Efficient One-Pot Synthesis of α-Chloroketone Acetals Directly from Ketones Using Iodobenzene Dichloride J Yu C Zhang
2329 An Efficient Oxidative Conversion of Aldehydes into 2-Substituted 2-Oxazolines Using 13-Diiodo-55-dimethylhydantoin S Takahashi H Togo
2333 A Novel Procedure for the Synthesis of Benzo[b][18]naphthyridine-3-carboxylate Derivatives from MoritandashBaylisndashHillman Adduct Acetates W Zhong F Lin R Chen W Su
2341 An Improved Synthesis of 147-Triazacyclononanes (tacns) and 14710-Tetraazacyclododecanes (cyclens) J Huang Z Zhou T H Chan
2345 The Ullmann Coupling between 2-Chlorobenzoic Acids and Amino Acids A Valuable Reaction for Preparing 2-Substituted 1-Acetyl-1H-indol-3-yl Acetates J C Rodriguez Dominguez X Gang G Kirsch
2349 gem-Dibromomethyl Aromatics Efficient Aldehyde Equivalents in the KnoevenagelndashDoebner Reaction J K Augustine Y A Naik S Poojari N Chowdappa B S Sherigara K Areppa
2357 Synthesis of Novel α-Aminophosphonates Containing Adamantyl Fragment M M Kabachnik L I Minaeva I P Beletskaya
2361 Efficient Fluoride-Mediated Synthesis of 5-Amino-Substituted Isothiazoles Y S Zubenko V I Potkin
2365 Phosphine-Catalyzed Reaction of Cyanohydrins with Activated Alkynes A Siby O Loreau F Taran
2371 Sulfanyl-Substituted [3]Cumulenes and Buta-13-dienes from a Tetrakis(pyridinium)-Substituted Butadiene A Schmidt A Rahimi M Gjikaj
2379 Efficient Synthesis of 2-Substituted Pyrido[32-d]pyrimidines Involving SNAr and Palladium-Catalyzed Cross-Coupling Reactions A Tikad S Routier M Akssira J-M Leacuteger C Jarry G Guillaumet
2385 Novel Synthesis of Medium-Sized Heterocycles by Palladium-Catalyzed Intramolecular Heck Reaction via 9-endo-trig Mode of Cyclization K C Majumdar B Chattopadhyay
2393 Facile Synthesis of Fluorinated Benzofuro- and Benzothieno[23-b]pyridines α-Carbolines and Nucleosides Containing the α-Carboline Framework V O Iaroshenko Y Wang B Zhang D Volochnyuk V Ya Sosnovskikh
2403 Synthesis of Functionalized N-Vinyl Nitrogen-Containing Heterocycles S M M Lopes A M Beja M Ramos Silva J A Paixatildeo F Palacios T M V D Pinho e Melo
2408 Kumada Cross-Coupling of Aryl Grignard Reagents with Aryl Halides Catalyzed by an Immobilized Nickel Catalyst X Chen L Wang J Liu
2413 Highly Enantioselective Synthesis of Heteroaromatic Alcohols Catalyzed by Chiral DiaminodiphosphinendashRuthenium(II) Complexes W-Y Shen Y-Y Li Z-R Dong J-X Gao
2418 Concise Total Synthesis of (+)-Disparlure and its trans-Isomer Using Asymmetric Organocatalysis S-G Kim
2423 Rhodium Carbenoid Induced [12]-Migration in an L-Lyxo-Configured α-Diazo β-Keto Ester Synthesis of a New Griseolic Acid Analogue N N Bhujbal K S A Kumar D D Dhavale
2430 Synthesis of 5-Arylthio-3-hydroxyphthalates by the First [4+2] Cycloadditions of 3-Arylthio-1-silyloxy-13-butadienes with Dimethyl Acetylenedicarboxylate I Iqbal M Imran P Langer
2435 Synthesis of Highly Functionalized Proline Derivatives via a One-Pot MichaelSN-AdditionCyclization Approach U Kazmaier C Schmidt
2440 RhodiumGraphite-Catalyzed Hydrogenation of Carbocyclic and Heterocyclic Aromatic Compounds G Falini A Gualandi D Savoia
2447 Potassium [1-(tert-Butoxycarbonyl)-1H-indol-2-yl]trifluoroborate as an Efficient Building Block in Palladium-Catalyzed SuzukindashMiyaura Cross Couplings P Kassis V Beacuteneacuteteau J-Y Meacuterour S Routier
2454 Syntheses of Substituted Furans and Pyrroles by Platinum-Catalyzed Cyclizations of Propargylic Oxiranes and Aziridines in Aqueous Media M Yoshida M Al-Amin K Shishido
2467 Transition-Metal-Free Oxidative Homocoupling of Aryl Alkenyl and Alkynyl Grignard Reagents with TEMPO M S Maji A Studer
XIII Forthcoming Articles
no 15 2471 Advances in Synthetic Approaches for the Preparation of Combretastatin-
Based Anti-Cancer Agents R Singh H Kaur 2492 Synthesis of Unsymmetrical Ureas by Sulfur-Assisted Carbonylation with
Carbon Monoxide and Oxidation with Molecular Oxygen under Mild Conditions T Mizuno T Nakai M Mihara
2497 Ring-OpeningRecyclization Reactions of (Dimethylamino)propenoyl-Substituted Cyclopropanes Facile Synthesis of Halogenated Pyridin-2(1H)-ones R Zhang Y Zhou Y Liang Z Jiang D Dong
2501 Facile and Efficient Total Synthesis of Taspine B Cheng S Zhang L Zhu J Zhang Q Li A Shan L He
2505 Oligomeric Iodosylbenzene Sulfate A Convenient Hypervalent Iodine Reagent for Oxidation of Organic Sulfides and Alkenes M S Yusubov R Y Yusubova T V Funk K-W Chi V V Zhdankin
2509 Pyrrolidine-Based Organocatalysts for Enantioselective Michael Addition of Cyclohexanone to trans-β-Nitrostyrene A P Carley S Dixon J D Kilburn
2517 CundashAl Hydrotalcite An Efficient and Reusable Ligand-Free Catalyst for the Coupling of Aryl Chlorides with Aliphatic Aromatic and N(H)-Heterocyclic Amines B Sreedhar R Arundhathi P L Reddy M A Reddy M L Kantam
2523 Highly Efficient Synthesis of trans-βγ-Unsaturated a-Keto Amides C Allais T Constantieux J Rodriguez
2531 Gas-Phase Synthesis of N-Unsubstituted 3-Hydroxypyrroles and 1H-Pyrrol-3(2H)-ones L Hill G A Hunter S H Imam H McNab W J OrsquoNeill
2535 3-Hydroxy-1H-pyrrole L Hill S H Imam H McNab W J OrsquoNeill 2539 123-Thiadiazoles with Unsaturated Side Chains Synthesis
Polymerization and Photocrosslinking M Al-Smadi N Hanold H Kalbitz H Meier
2547 Synthesis of 1112-Didehydrodibenzo[ae]cycloocten-5(6H)-one A Strained Eight-Membered Alkyne S C Kornmayer F Rominger R Gleiter
2553 Stannous Chloride Dihydrate A Novel and Efficient Catalyst for the Synthesis of gem-Dihydroperoxides from Ketones and Aldehydes D Azarifar K Khosravi F Soleimanei
2557 Synthesis of a Novel Class of Azacrown Macrocycles and Lariat Crown Ethers Containing Two 124-Triazole Rings as Subunits N Foroughifar A Mobinikhaledi S Ebrahimi
2561 Enantioselective Synthesis of the 3C-Protease Inhibitor (ndash)-Thysanone by a StauntonndashWeinreb Annulation Strategy J Sperry T Y Yuen M A Brimble
2570 Stereoselective Synthesis of Unnatural β-Amino Acids from Nitroethane via 56-Dihydro-4H-12-oxazin-3-ylacetates A Yu Sukhorukov A V Lesiv O L Eliseev Y A Khomutova S L Ioffe
2579 A Versatile Unexpected One-Pot Regioselective Synthesis of a New Class of 13-Diazepinoindolones by Reaction of Pyranoindolones with Monosubstituted Ureas D Livadiotou C A Tsoleridis J Stephanidou-Stephanatou
2584 Synthesis of a Trisaccharide and a Tetrasaccharide from the Cell-Wall Lipopolysaccharides of Azospirillum brasilense S17 S Pandey S Ghosh A K Misra
2591 Synthesis of Isoindoline Nitroxides by Electrocyclic Reactions T Kaacutelai J Jekı K Hideg
2596 Glycosylations of Tertiary Alcohols Synthesis of Fully Protected Disaccharides with Sterically Demanding Groups Attached to the Sugar Core A Holkenbrink J B Vicente D B Werz
2605 Copper-Catalyzed [13]-Dipolar Cycloaddition for the Synthesis of Macrocycles Containing Acyclic Aromatic and Steroidal Moieties G V Latyshev M S Baranom A V Kazantsev A D Averin N V Lukashev I P Beletskaya
2616 Aryl Ring Migration Reaction in the Synthesis of 24-Diaryl-4H-31-benzothiazines A V Butin F A Tsiunchik V T Abaev A V Gutnov D A Cheshkov
2627 Hydrogenation of β-N-Substituted and β-NN-Disubstituted Enamino Esters in the Presence of Iridium(I) Catalyst H Hebbache Z Hank C Bruneau J-L Renaud
2634 Stereoselective Olefination Reactions Promoted by Rieke Manganese J M Concelloacuten H Rodriacuteguez-Solla V del Amo P Diacuteaz
2646 Synthesis of Piperidinones through a Radical Cascade E Godineau Y Landais
2650 Asymmetric Organic Synthesis with Enzymes Edited by V Gotor I Alfonso E Garciacutea-Urdiales Reviewed by Steve Collier
XVII Forthcoming Articles
no 16 2651 Synthesis of Spirocyclic Ethers S Rosenberg R Leino 2674 Bimetallic PalladiumndashPlatinum-on-Carbon-Catalyzed HndashD Exchange
Reaction Synergistic Effect on Multiple Deuterium Incorporation T Maegawa N Ito K Oono Y Monguchi H Sajiki
2679 Efficient Copper-Catalyzed Synthesis of 2-Amino-4(3H)-quinazolinone and 2-Aminoquinazoline Derivatives X Huang H Yang H Fu R Qiao Y Zhao
2689 Synthesis and Chemoselective N- and O-Alkylation of Thiadiazolopyrimidine Nucleosides and Uridines A M L Hossion R Islam R K Kandahary T Nagamatsu
2697 Facile and Efficient Synthesis of a New Class of Indole-Substituted Pyridine Derivatives via One-Pot Multicomponent Reactions K Zhao X-P Xu S-L Zhu D-Q Shi Y Zhang S-J Ji
2709 Studies toward a Total Synthesis of Rhizoxin D Stereoselective Preparation of the C11ndashC19 Fragment S Padakanti C K Kumar E Ashok P Das
2715 A Short Synthesis of Enantiomeric Phytoprostanes B1 Type I W Perlikowska M Mikołajczyk
2719 Chemistry of Polyhalogenated Nitrobutadienes Part 7 A Novel Synthetic Access to Chlorinated Nitrile Oxides E Nutz V A Zapolrsquoskii D E Kaufmann
2725 Microwave-Assisted Silver(I)-Mediated Selective O-Alkylation of Aromatic Imidate Systems B K Singh C Cavalluzzo M De Maeyer Z Debyser V S Parmar E Van der Eycken
2729 Iodogen A Novel Reagent for the Oxidation of Urazoles under Heterogeneous Conditions A Khoramabadi A Shiri M A Zolfigol S Mallakpour
2733 An Unprecedented Synthesis of Eight-Membered-Ring Cyclic Thioimidic Esters by a Three-Component Reaction A Alizadeh R Hosseinpour
2737 A Novel Diastereoselective Synthesis of β-Phosphonato Unsaturated Thioimidates A Alizadeh N Zohreh
2741 Synthesis of 21-Benzisoxazoles by Nucleophilic Substitution of Hydrogen in Nitroarenes Activated by the Azole Ring N T Pokhodylo Y O Teslenko V S Matiychuk M D Obushak
2749 A Facile Synthesis of Two Series of Multifunctional Carbon Compounds from αα-Dihalo Ketones Using Allylsamarium Bromide X Liu S Zhang J Di
2756 Stereocontrolled Formation of Protected Aminodeoxyalditols from Simple Carbohydrate Precursors by Debenzylating Cycloetherification Y Jiang Z Fang Q Zheng H Jia J Cheng B Zheng
2761 trans-Stilbene as a Starting Material for the Synthesis of Tamoxifen Based on Palladium-Catalyzed Cross-Coupling Reactions C M Nunes J Limberger S Poersch M Seferin A L Monteiro
2766 Synthesis and Biological Evaluation of 6-Substituted Purinylcarbanucleosides with a Cyclopenta[b]thiophene Pseudosugar P Abeijoacuten J M Blanco O Caamantildeo F Fernaacutendez M D Garciacutea X Garciacutea-Mera J E Rodriacuteguez-Borges J Balzarini E De Clercq
2773 Synthesis and Electrochemical Signature of Novel Norbornyl-ferrocene Hybrids F A Khan S K Upadhyay
2778 A Regioselective TsujindashTrost Pentadienylation of 3-Allyltetronic Acid R Schobert B Barnickel
2785 Copper(I)-Catalyzed CarylndashCalkynyl Bond Formation of Aryl Iodides with Terminal Alkynes K G Thakur G Sekar
2790 Aminolysis of Epoxides Using Iridium Trichloride as an Efficient Catalyst J Agarwal A Duley R Rani R K Peddinti
2797 Preparation of Several Active N-Chloro Compounds from Trichloroisocyanuric Acid A Shiri A Khoramabadi-zad
2802 The First Mineral-Catalyzed One-Pot [3+1+2] Coupling Protocol for Multifunctionalized Fused-Ring Pyrimidines L D S Yadav A Rai
2809 Efficient Synthesis of Tetrahydro-β-carbolin-1-one and Dihydroisoquinolin-1-one Derivatives as Versatile Intermediates K E Judd M F Mahon L Caggiano
2818 A Concise Synthesis of ortho-Iodobenzyl Alcohols via Addition of ortho-Iodophenyl Grignard Reagent to Aldehydes and Ketones J Cvengroš D Stolz A Togni
XIII Forthcoming Articles
no 17 2825 Reactivity of Oxazol-5-(4H)-ones and Their Application toward Natural
Product Synthesis N M Hewlett C D Hupp J J Tepe 2840 Towards the Total Synthesis of 3-Hydroxyvibsanin E B D Schwartz
J R Denton P V Bernhardt H M L Davies C M Williams 2847 Structure Investigations of (ent)-Cladospolide D by De Novo Synthesis and
Kinetic and Thermodynamic Isomerization Y Xing J H Penn G A OrsquoDoherty
2855 New Applications of PhI(OAc)2 in Synthesis Total Synthesis and SAR Development of Potent Antitumor Natural Product PsymberinIrciniastatin A N Shao X Huang A Palani R Aslanian A Buevich J Piwinski R Huryk C Seidel-Dugan
2873 Total Synthesis of Largazole ndash Devolution of a Novel Synthetic Strategy B Wang C J Forsyth
2881 Formal Total Synthesis of Palmerolide A J Jaumlgel M E Maier 2893 Total Synthesis of Bongkrekic Acid via Sequential SuzukindashMiyaura Coupling
Reactions M Kanematsu M Shindo M Yoshida K Shishido 2905 Stereodivergent Approach to Both C28a-syn and C28a-anti Relative
Stereochemical Manifolds in the Lepadin Family via a TiCl4-Promoted G Li L J Carlson I K Sagamanova B W Slafer R P Hsung C Gilardi H M Sklenicka N Sydorenko
2915 Enantioselective Aldol Reaction of Tetrasubstituted Ketene Silyl Acetals with Achiral Aldehydes for the Construction of Asymmetric Tertiary Alcohols An Application for the Divergent Total Syntheses of Buergerinins F and G I Shiina T Iizumi Y-s Yamai Y-i Kawakita K Yokoyama Y-k Yamada
2927 Second-Generation Biomimetic Total Synthesis of Chaetominine A Coste G Karthikeyan F Couty G Evano
2935 Total Synthesis of (+)-Fostriecin and (+)-Phoslactomycin B S Shibahara M Fujino Y Tashiro N Okamoto T Esumi K Takahashi J Ishihara S Hatakeyama
2954 Stereochemical Assignments of the Chlorinated Residues in Victorin C A C Durow C Butts C L Willis
2963 Studies of the Asymmetric Total Synthesis of Clavilactone D by the lsquoLariatrsquo Cyclization Strategy T Yoshimitsu S Nojima M Hashimoto K Tsukamoto T Tanaka
2970 Total Synthesis of the Leucetta-Derived Alkaloid Calcaridine A P B Koswatta R Sivappa H V R Dias C J Lovely
2983 Formal Synthesis of Salinosporamide A Starting from D-Glucose T Momose Y Kaiya J-i Hasegawa T Sato N Chida
2992 Synthesis of Bioactive Natural Products by Asymmetric syn- and anti-Aldol Reactions A K Ghosh Z L Dawson
no 18 3003 Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural
Products B M Trost M K Brennan 3026 One-Pot Synthesis of Furo[34-b]pyridin-5(7H)-ones from 2-
Bromopyridine-3-carboxylic Acid and Carbonyl Compounds K Kobayashi T Kozuki H Konishi
3029 Iodocyclization of N-[2-(Methylthio)phenyl]propiolamides Selective Synthesis of 3-Iodo-15-benzothiazepin-4-ones T-S Jiang X-G Zhang J-H Li
3039 A Facile Synthetic Method for Fluorine-Containing 17-Phenanthrolines Pyridine-Ring Formation Reaction of N-Propargyl-68-bis(trifluoroacetyl)-quinolin-5-amine with Various Nucleophiles D Shibata E Okada M Hinoshita M Meacutedebielle
3047 Enantiotopic Discrimination in Palladium-Mediated Nucleophilic Substitutions on Achiral Substrates Chiral Ligand versus Chiral Nucleophile O Jacquet F Charnay J-C Fiaud J Ollivier
3051 Studies on the Chemistry of 2-[3-(2-Nitrophenyl)-2-oxopropyl]benzaldehydes Novel Syntheses of 5H-Benzo[b]carbazole-611-diones and Indolo[12-b]isoquinoline-611-diones M Fernaacutendez
3061 Studies on the C22ndashC23 Aldol Coupling of Spirangien M Lorenz N Bluhm M Kalesse
3067 One-Pot Synthesis of N-Alkyl Purine Pyrimidine and Azole Derivatives from Alcohols using Ph3PCCl4 A Rapid Route to Carboacyclic Nucleoside Synthesis M N Soltani Rad A Khalafi-Nezhad S Behrouz Z Asrari M Behrouz Z Amini
3077 Synthesis of 2-Amino-34-dihydroquinazolines and Imidazo[21-b]quinazoline-2-ones A Mishra S Batra
3089 Studies on the Reaction of Diimines with Thiourea Synthesis and Solvent-Induced cistrans-Isomerization of 135-Triazinane-2-thiones B Kaboudin T Ghasemi T Yokomatsu
3094 Suzuki Coupling of Heteroaromatic Chlorides Using Highly Electron-Donating ClickPhos Ligands S M Spinella Z-H Guan J Chen X Zhang
3099 Reaction of NN-Dioxyenamines with Anhydrides of Carboxylic and Sulfonic Acids A New Method for the Synthesis of a-Hydroxyoxime Derivatives A A Tabolin A V Lesiv S L Ioffe
3106 Directed ortho Metallation Chemistry and Phosphine Synthesis New Ligands for the SuzukindashMiyaura Reaction D B G Williams S J Evans H de Bod M S Mokhadinyana T Hughes
3113 New Functional Derivatives of 9-Phenylquinine P J Boratyński J SkarŜewski
3120 On the Synthesis of Asymmetric and Dissymmetric Amino Analogues of Troumlgerrsquos Base J Artacho K Waumlrnmark
3127 Synthesis of Polycyclic Sultams by Palladium-Catalyzed Intramolecular Cyclization K C Majumdar S Mondal N De
3136 Synthesis of Functionalized L-Cysteine and L-Methionine by Reaction with Electron-Deficient Acetylenes B A Trofimov A G Malrsquokina O A Shemyakina V V Nosyreva A P Borisova S S Khutsishvili L B Krivdin
3143 A lsquoClickrsquo Approach to the Synthesis of 3-[2-(1-Alkyltriazol-4-yl)ethyl]indoles M Petrini R R Shaikh
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
1000 Light-Induced Synthesis of Π-Extended Tetrathiafulvalenes Incorporating Ferrocenes An Efficient Route for the Synthesis of Electron-Donor Materials A A O Sarhan C Bolm
1007 Preparation of Nβ-Fmoc-Protected Aza-β3-Amino Acids with Nonproteinogenic Hydrophobic Side Chains for Solid-Phase Syntheses of Pseudopeptides M Laurencin P Bauchat M Baudy-Flocrsquoh
1014 Diastereomeric (η4-diene)Fe(CO)3 Complexes Containing Chiral Amide Groups A Convenient Method for the Resolution of Amino Acids M Schumacher G Coste L Miesch
1021 Palladium-Catalysed Heck Reactions of Alk-1-en-3-ones with Aryl Bromides A Very Simple Access to (E)-1-Arylalk-1-en-3-ones M Lemhadri Y Fall H Doucet M Santelli
1036 An Improved Process for the Synthesis of 4H-Imidazo[15-α][14]benzodiazepines J Yang Y Teng S Ara S Rallapalli J M Cook
1041 Meta- and Para-Difunctionalization of Arenes via an Ortho-Magnesiation and a Subsequent SulfoxidendashMagnesium Exchange L Melzig C B Rauhut P Knochel
XIII Forthcoming Articles
No 7 1049 Catalytic Transformations of Benzylic Carboxylates and Carbonates
R Kuwano 1062 A Simple and Practical Method for the Oxidation of Thebaine to 14-
Hydroxycodeinone by V2O5ndashH2O2 S Das Sharma D Konwar 1065 Umpolung with Sulfur Dioxide CarbonndashCarbon Cross-Coupling of Electron-
Rich 13-Dienes and Alkenes Application to the Enantioselective Synthesis of Long-Chain Polyketide Fragments M Turks C J Exner C Hamel P Vogel
1075 One-Pot Synthesis of 14-Diarylnaphthalenes via a WittigndashHorner Reaction[4+2] CycloadditionDehydrogenation Sequence Z Chen W Shou Y Wang
1081 A Novel and General Method for the Formation of S-Aryl Se-Aryl and Te-Aryl Phosphorochalcogenoates Y-X Gao G Tang Y Cao Y-F Zhao
1087 A Remarkable Access to γ-Fluoroalkylated Propargylamine Derivatives or Fluoroalkylated Dihydroisoxazoles via the Reaction of Fluoroalkylated Acetylides with Various Nitrones T Konno K Moriyasu T Ishihara
1095 Short and Practical Syntheses of (S)-(+)-3-(p-Tolylsulfinyl)furan-2(5H)-one and (S)-(+)-3-(p-Tolylsulfinyl)-56-dihydropyran-2-one D Cruz Cruz A Hernaacutendez Linares F Yuste M R Martiacuten J L Garciacutea Ruano
1099 Decarboxylative Aldol-Type Reaction of 2-(Trifluoroacetyl)-13-diazoles with Activated Acetic Acids P V Khodakovskiy D M Volochnyuk A A Tolmachev
1105 Synthesis of 2-[(Arylmethylene)amino]cyclopropanecarbonitriles via a Two-Step Ring Transformation of 2-(Cyanomethyl)aziridines S Mangelinckx M Drsquohooghe S Peeters N De Kimpe
1113 Synthesis of Dendrimeric Tumor-Associated Mucin-Type Glycopeptide Antigens T Becker A Kaiser H Kunz
1123 A Simple and Efficient Oxidation Procedure for the Synthesis of Acid-Sensitive Epoxides O Bortolini G Fantin M Fogagnolo
1127 Rapid Chemoselective Deprotection of Benzyl Esters by Nickel Boride J M Khurana R Arora
1131 Three-Component Coupling of Isoquinoline Activated Alkyne and Nitromethane A Facile Synthesis of Nitromethyl Derivatives of 12-Dihydroisoquinolines J S Yadav B V S Reddy N N Yadav M K Gupta
1137 Palladium Supported on a Polyionic Resin as an Efficient Ligand-Free and Recyclable Catalyst for Heck SuzukindashMiyaura and Sonogashira Reactions B Basu S Das P Das B Mandal D Banerjee F Almqvist
1147 Oxidation of 25-Dialkylpyrrole Derivatives with Cerium(IV) Ammonium Nitrate R Voloshchuk M Gałęzowski D T Gryko
1153 Practical Syntheses of Enantiomerically Pure Key Intermediates of Opioid Receptor-like 1 (ORL1) Antagonists T Yoshizumi A Ohno T Tsujita H Takahashi O Okamoto I Hayakawa H Kigoshi
1163 An Environmentally Benign TEMPO-Catalyzed Efficient Alcohol Oxidation System with a Recyclable Hypervalent Iodine(III) Reagent and Its Facile Preparation X-Q Li C Zhang
1170 Efficient and Stereoselective Rearrangement of BaylisndashHillman Acetates Catalyzed by Gold(I) ChlorideSilver(I) Trifluoromethanesulfonate Y Liu D Mao J Qian S Lou Z Xu Y Zhang
1175 The First Total Synthesis of Kynapcin-24 by Palladium Catalysis L-Y Yang C-F Chang Y-C Huang Y-J Lee C-C Hu T-H Tseng
1180 Enantioselective Synthesis of N-Protected α-Amino Acid Hydrazides M Bibian S El-Habnouni J Martinez J-A Fehrentz
1185 Synthesis of 11H-Indolo[32-c]quinoline-6-carboxylic Acids by Cascade AutoxidationndashRing Contractions A Becker S Kohfeld T Pies K Wieking L Preu C Kunick
1190 Reaction of N-Nonaflylbenzotriazole with Silyl Enol Ethers M Uhde T Ziegler
1195 2-(Benzoylimino)thiazolidin-4-ones Formation by an Alternative Ring Closure and Analysis of Rotational Barriers H-G Haumlcker P W Elsinghorst S Michels J Daniels G Schnakenburg M Guumltschow
1204 Microwave-Assisted Synthesis and Functionalization of Selenolopyrimidines S Hesse C Chenet D Thomae G Kirsch
1209 12-Disubstituted 4-Quinolones via Copper-Catalyzed Cyclization of 1-(2-Halophenyl)-2-en-3-amin-1-ones R Bernini S Cacchi G Fabrizi A Sferrazza
1220 A New Atom-Economical and Selective Synthesis of Secondary and Tertiary Alkylamines by Means of CpIridium Complex Catalyzed Multiple N-Alkylation of Ammonium Salts with Alcohols without Solvent R Yamaguchi Z Mingwen S Kawagoe C Asai K-i Fujita
1224 Synthesis of Regioisomerically Pure 5-Functionalized 27-Dichlorofluoresceins J C Castro A Malakhov K Burgess
XIII Forthcoming Articles
No 8 1227 Michael Additions to Activated Vinylphosphonates T Janecki J Kędzia
T Wąsek 1255 A Facile and General Synthesis of 2β-Aminosteroids X Ke H Hu
D Zhou W Xu Q Zhu N P Reddy X Hu 1261 Efficacious Preparation of Oppolzerrsquos Glycylsultam via the Deleacutepine
Reaction A Isleyen C Gonsky R C Ronald P Garner 1265 Synthesis of Masked Vicinal Amino Aldehydes of Pyrrolizine and Pyrrolo
[12-c]thiazole Series A V Tverdokhlebov A V Denisenko A A Tolmachev Y M Volovenko S V Shishkina O V Shishkin
1271 Preparation of 9-Substituted Pyridine-Stretched Adenines and Hypoxanthines J A Crawford W Fraser C A Ramsden
1279 A Versatile Synthesis of Heterocyclic Analogues of Neoflavonoids from Enamino Ketones V S Moskvina V P Khilya O V Turov U M Groth
1287 New Stereoselective Synthesis of Paeonilactone B F G Gatti S Serra 1291 The Use of NN-Dialkyltrimethylsilylamines in the Synthesis of
Pentamethinium Salts M Kořiacutenek M Rybaacutečkovaacute Boumlhm 1297 Synthesis of Triazoles via Regioselective Reactions of Aryl Azides with
Cyanoacetyl Pyrroles and Indoles N T Pokhodylo V S Matiychuk M D Obushak
1301 Gallium(III) Chloride Catalyzed Hydroarylation of Arylacetylenes with Naphthols and Phenols A Facile Synthesis of Vinylarenes J S Yadav B V S Reddy S Sengupta S K Biswas
1305 Electrophilic Bromination of meta-Substituted Anilines with N-Bromosuccinimide Regioselectivity and Solvent Effect S Bartoli A Cipollone A Squarcia A Madami D Fattori
1309 Cross-Coupling Reactions of Halopurines with Aryl- and Alkyltrifluoroborates The Scope and Limitations in the Synthesis of Modified Purines Z Hasniacutek R Pohl M Hocek
1318 A Convenient Method for Converting Hydroxyacetophenones into Their Ethylene or Trimethylene Acetals F Ono H Takenaka T Fujikawa M Mori T Sato
1323 γ-Chloromagnesio γ-Lactones and δ-Chloromagnesio δ-Lactones Generation Properties and Synthetic Uses H Shimizu S Fukuda S Sugiyama T Satoh
1336 Click Reactions with Nitroxides T Kaacutelai W L Hubbell K Hideg 1341 Synthesis of Novel 14-Benzoquinone-Containing 123-Triazoles An Entry
Into a New Library F Algi M Balci 1348 Efficient Synthesis of Two Sialylated Tetrasaccharides Found in Goat Milk
P K Mandal A K Misra 1355 Dendrimers of Vaccines Consisting of Tumor-Associated Glycopeptide
Antigens and T Cell Epitope Peptides S Keil A Kaiser F Syed H Kunz
1370 IBXTBAB-Mediated Oxidation of Primary Amines to Nitriles F Drouet P Fontaine G Masson J Zhu
1375 Chemoselectivity of Multicomponent Condensations of Barbituric Acids 5-Aminopyrazoles and Aldehydes E A Muravyova S V Shishkina V I Musatov I V Knyazeva O V Shishkin S M Desenko V A Chebanov
1386 Stereoselective Total Syntheses of Leiocarpin A and (ndash)-Galantinic Acid Starting from D-Mannitol K Nagaiah D Sreenu K V Purnima R S Rao J S Yadav
1393 A Facile Mild Deprotection Protocol for 13-Dithianes and 13-Dithiolanes with 30 Hydrogen Peroxide and Iodine Catalyst in Aqueous Micellar System N C Ganguly S K Barik
1400 Rhodium-Catalyzed Gram-Scale Synthesis of Highly Substituted Pyridine Derivatives K Parthasarathy C-H Cheng
1403 Enantioselective Synthesis of (R)-Propylene Carbonate from Ethyl (S)-Lactate J M Whitaker R C Ronald
XIII Forthcoming Articles
no 9 1405 Transition-Metal-Catalyzed Site-Selective Cross-Coupling of Di- and
Polyhalogenated Compounds J-R Wang K Manabe 1428 An Improved Synthesis of (4-4-Hydroxy-3-isopropyl-5-[(4-nitrophenyl)
ethynyl]benzyl-35-dimethylphenoxy)acetic Acid (NH-3) M B Gopinathan K S Rehder
1431 Copper-Catalyzed Tandem CndashN Bond Formation Reaction Selective Synthesis of 2-(Trifluoromethyl)benzimidazoles M-W Chen X-G Zhang P Zhong M-L Hu
1437 Synthesis and Thermochemical Properties of Stereoisomeric Dihydroxy- and Tetrahydroxyalkylammonium Salts M Thomas L Rothman J Hatcher P Agarkar R Ramkirath S Lall-Ramnarine R Engel
1445 Preparation of 5-Substituted 2-(2-Alkylaryl-1H-imidazol-4-yl)oxazoles and 5-Substituted 2-(2-Alkylarylthiazol-4-yl)oxazoles by Utilizing 5-Substituted 2-(2-Bromo-11-diethoxyethyl)oxazole as a Synthon D R St Laurent J L Romine
1459 Novel and Efficient Methods for the Synthesis of Symmetrical Trisulfides A Kertmen S Lach J Rachon D Witt
1463 An Environmentally Benign Electrochemical Process for the Reduction of Carboxylic Acid Hydrazides to Amides M Mentel M J Beier R Breinbauer
1469 Synthesis of 1-Chloroalkynes from Alkynylsilanes Using Trichloroisocyanuric Acid as Chlorinating Agent M H Vilhelmsen A S Andersson M B Nielsen
1473 A Convenient Approach to Enantioenriched Cyclopropanes Bearing Electron-Withdrawing Functionalities H Krawczyń K Wąsek J Kędzia
1477 Synthesis of Cyclopropenes via 12-Elimination of Bromocyclopropanes Catalyzed by Crown Ether W M Sherrill R Kim M Rubin
1485 A Base-Catalysed One-Pot Three-Component Coupling Reaction Leading to Nitrosubstituted Pyrroles I R Baxendale C D Buckle S V Ley L Tamborini
1494 Synthesis of 4-Alkylidene-4H-31-benzoxazine Derivatives by Acid-Catalyzed Cyclization of 2-Isocyanophenyl Ketones in the Presence of a Vinyl Ether K Kobayashi Y Okamura H Konishi
1499 Synthesis of Higher Helicenes via Olefin Metathesis and CndashH Activation J Cocircteacute S K Collins
1506 Azido- and Ethynyl-Substituted 2262-Terpyridines as Suitable Substrates for Click Reactions A Winter A Wild R Hoogenboom M W M Fijten M D Hager R-A Fallahpour U S Schubert
1513 Synthesis of 2-(Arylamino)ethanethiols via Lewis Acid Catalyzed Aminolysis of 22-Dimethylthiirane as Precursors of the 14-Benzothiazine Nucleus R Spogli S Sabatini G Manfroni O Tabarrini V Cecchetti
1520 Iron(III) Chloride A Versatile Catalyst for the Practical Synthesis of 3-Sulfenylindoles J S Yadav B V S Reddy Y J Reddy K Praneeth
1525 Organocatalytic Enantioselective Conjugate Addition of 2-Fluoromalonate to Nitroolefins Direct Synthesis of Chiral Fluorinated γ-Nitro Carboxylic Acid Derivatives H Li L Zu H Xie W Wang
1531 Asymmetric Transfer Hydrogenation of Ketimines with Trichlorosilane Structural Studies Z Zhang P Rooshenas H Hausmann P R Schreiner
1545 Prolinol Sulfinyl Ester Derivatives Organocatalytic Michael Addition of Ketones to Nitroolefins under Neat Conditions X Zeng G Zhong
1551 Asymmetric Oxidations of Electron-Poor Alkenes Promoted by the β-Amino AlcoholTBHP System A Russo A Lattanzi
1557 Enantioselectivity Switch in Direct Asymmetric Aminoxylation Catalyzed by Binaphthyl-Based Chiral Secondary Amines T Kano A Yamamoto F Shirozu K Maruoka
1564 Enantioselective Conjugate Addition of N-Heterocycles to αβ-Unsaturated Ketones Catalyzed by Chiral Primary Amines G Luo S Zhang W Duan W Wang
1573 Sulfonyl Hydrazine as New Functionality in Organocatalysis Camphorsulfonyl Hydrazine Catalyzed Enantioselective Aza-Michael Addition L-Y Chen H He B-J Pei W-H Chan A W M Lee
1578 Conversion of Primary Alcohols and Aldehydes into Methyl Esters by Ruthenium-Catalysed Hydrogen Transfer Reactions N A Owston T D Nixon A J Parker M K Whittlesey J M J Williams
1582 Addendum and Erratum XVII Forthcoming Articles
no 10 1583 Organocatalytic Formation of Quaternary Stereocenters M Bella
T Gasperi 1615 Regioselective Synthesis of 5H-Thiazolo[32-a]pyrimidin-5-ones from
MoritandashBaylisndashHillman Adduct Acetates under Solvent-Free and Base-Free Conditions W Zhong B Guo F Lin Y Liu W Su
1623 First Synthesis of 5-Cyanosalicylates by Formal [3+3] Cyclocondensations of 13-Bis(silyloxy)-13-butadienes A Riahi O Fatunsin M Shkoor R Dede H Reinke C Fischer P Langer
1635 Reaction of Isocyanides Dialkyl Acetylenedicarboxylates and a-Keto Lactones Unexpected Participation of an Ester Carbonyl Group in the Isocyanide-Based Three-Component Reaction A A Esmaeili H Vesalipoor
1639 An Efficient and Chemoselective Synthesis of 16-Naphthyridines and Pyrano[32-c]pyridines under Microwave Irradiation Z-G Han S-J Tu B Jiang S Yan X-H Zhang S-S Wu W-J Hao X-D Cao F Shi G Zhang N Ma
1647 N-Activation of N-Arylimidazoles Facile Syntheses of N-Alkyl-N-arylimidazolium Iodides from Less Expensive Chloro Substrates A M Oertel V Ritleng M J Chetcuti
1651 Synthesis of Polyhalogenated 2-(Phenylamino)pyridines by Thermal Amination Reactions S R Waldvogel A Faust W Barkmann R Froumlhlich O Wolff
1655 Cyanide Ion Promoted Addition of Acylphosphonates to Diethyl Cyanophosphonate Synthesis of Phosphonocyanohydrin O-Phosphates A S Demir A Aybey M Emrullahoglu
1659 Straightforward and Scalable Synthesis of Orthogonally Protected 37-Diazabicyclo[410]heptane H Schramm M Pavlova C Hoenke J Christoffers
1663 Hypervalent Iodine Mediated Oxidation of 12-Diaminobenzimidazole and Its Schiff Bases Efficient Synthesis of 3-Amino-124-benzotriazine and 2-Aryl-124-triazolo[15-a]benzimidazoles A Kumar M Parshad R K Gupta D Kumar
1667 Synthesis of the Reported Protoberberine Gusanlung D P B Wakchaure S Easwar N P Argade
1673 2-(Azidomethyl)arylboronic Acids in the Synthesis of Coumarin-Type Compounds M I Naumov A V Nuchev N S Sitnikov Y B Malysheva A S Shavyrin I P Beletskaya A E Gavryushin S Combes A Y Fedorov
1683 Asymmetric Synthesis of 12-anti-Disubstituted Taurine Derivatives D Enders D Iffland G Raabe
1689 A Novel One-Pot Three-Component Synthesis of 5-Imino-2358-tetrahydropyrazolo[12-a]pyridazin-1-one Derivatives B Qian M-J Fan Y-X Xie L-Y Wu Y Shi Y-M Liang
1694 One-Portion Synthesis of 2-Acetoxy Carbonyl Compounds from Aldehydes by Using an Acetylated Masked Acyl Cyanide H Nemoto T Kawamura K Kitasaki K Yatsuzuka M Kamiya Y Yoshioka
1703 Synthesis of 9-Anthryl Ethers from trans-910-Dihydro-910-dimethoxyanthracene by Acid-Catalyzed Transetherification K S Jang H Y Shin D Y Chi
1708 Efficient Synthesis of Azo Dye Labeled Terpenes Sugars and Steroids Using N-(4-Arylazobenzoyl)-1H-benzotriazoles A R Katritzky S R Tala N E Abo-Dya Z K Abdel-Samii
1715 Tandem CH-ActivationndashImine-Formation Reaction A New Route to Imidazo[21-a]phthalazines A Heim-Riether K R Gipson
1720 A Convenient and Efficient α-Sulfenylation of Carbonyl Compounds E Okragla S Demkowicz J Rachon D Witt
1725 Stereoselective Synthesis of β-Branched Phenylalanine Derivatives via Chelate-Claisen Rearrangement C Quirin U Kazmaier
1732 Catalyst-Free and Base-Free Water-Promoted SNAr Reaction of Heteroaryl Halides with Thiols B Sreedhar P S Reddy M A Reddy
1739 Convenient Methods for Synthesis of C2-Symmetric Diphenyltetrahydrothiophenes M Periasamy G Ramani G P Muthukumaragopal
1744 Highly Diastereoselective Conjugate AdditionndashElimination of Chiral Nickel(II) Glycinate with Activated Allylic Acetates for Asymmetric Synthesis of Glutamic Acid Derivatives J Wang J Shi X Zhang D Lin H Jiang H Liu
1753 Synthesis of 36-Dimethoxybenzene-12-diamine and of 47-Dimethoxy-2-methyl-1H-benzimidazole T Besset C Morin
1757 An Inexpensive Procedure for Reductive Aminations Using Dimethylamineborane on Millimolar and Molar Scale R Ortmann M Schlitzer
1760 Classics in Stereoselective Synthesis Edited by E M Carreira L Kvaerno Reviewed by Rolf Breinbauer
XV Forthcoming Articles
no 11 1761 Transition-Metal-Catalyzed Enantioselective Synthesis of Compounds with
Non-Centrochirality M Ogasawara S Watanabe 1786 One-Pot Synthesis of 3-Acyl-2-(alkylsulfanyl)indoles and 2-(Alkylsulfanyl)-
indole-3-carboxylates from (2-Isocyanophenyl)methyl Ketones or (2-Isocyanophenyl)acetates S Fukamachi H Konishi K Kobayashi
1791 Efficient and Recyclable Phthalocyanine-Based Sensitizers for Photooxygenation Reactions H Xu W-K Chan D K P Ng
1797 A Facile and Practical One-Pot Synthesis of β-Oxo Thioamides from β-Oxo Amides and Isothiocyanates P Huang D Xiang Y Zhou Y Liang T Na D Dong
1801 Microwave-Promoted Solid-Acid-Catalyzed One-Pot Synthesis of Phthalazinones V M Outerbridge S M Landge H Tamaki B Toumlroumlk
1807 Benzylic Brominations with N-Bromosuccinimide in (Trifluoromethyl)-benzene D Suarez G Laval S-M Tu D Jiang C L Robinson R Scott B T Golding
1811 Synthesis of Thioflavanone and Flavanone Derivatives by Cyclization of Chalcones W Konieczny M Konieczny
1815 A New and Expedient Total Synthesis of Ochratoxin A and d5-Ochratoxin A B Gabriele M Attya A Fazio L Di Donna P Plastina G Sindona
1821 Synthesis of Benzopyrrolizidinones by NorrishndashYang Cyclization of 3-(Acylmethyl)-2-alkylisoindol-1-ones J Wu W Zhang C Wang
1829 Reactions of MoritandashBaylisndashHillman Acetates with Huisgen Zwitterions A Novel Strategy for the Synthesis of β-Amino Acid Derivatives A Jose R R Paul R Mohan S C Mathew A T Biju E Suresh V Nair
1834 Peracetylated β-Allyl C-Glycosides of D-Ribofuranose and 2-Deoxy- D-ribofuranose in the Chemical Literature Until Now Mirages in the Literature H Otero Martinez H Reinke D Michalik C Vogel
1841 Core-Tetrasubstituted Naphthalene Diimides by Stille Cross-Coupling Reactions and Characterization of Their Optical and Redox Properties S-L Suraru F Wuumlrthner
1846 A Practical Synthesis of Indole-Based Heterocycles Using an Amidoaluminum-Mediated Strategy R Todd M M Hossain
1851 Synthesis of Fluorinated Pyrrolo[23-b]pyridine and Pyrrolo[23-d]pyrimidine Nucleosides V O Iaroshenko Y Wang D V Sevenard D M Volochnyuk
1858 Recyclization Reactions of 5-Formyl-13-dimethyluracil with Electron-Rich Amino Heterocycles A P Mityuk D M Volochnyuk S V Ryabukhin A S Plaskon A Shivanyuk A A Tolmachev
1865 Facile Synthesis of Fluorinated 1-Desazapurines V O Iaroshenko D V Sevenard D M Volochnyuk Y Wang A Martiloga A O Tolmachev
1876 A Practical Synthesis of 3-Diethoxyphosphoryl-12-pyridazine Derivatives J-C Monbaliu J Marchand-Brynaert
1881 Enantioselective Reduction of Prochiral Ketones Employing Sprouted Pisum sativa as Biocatalyst J S Yadav B V S Reddy C Sreelakshmi A B Rao
1886 Application of Phenolate Ion Mediated Intramolecular Epoxide Ring Opening in the Enantioselective Synthesis of Functionalized 23-Dihydrobenzofurans and 1-Benzopyrans S K Dinda S K Das G Panda
1897 Complementary Synthetic Approaches to Constitutionally Diverse N-Aminoalkylated Isoindolinones Application to the Synthesis of Falipamil and 5-HT1A Receptor Ligand Analogues M Lorion A Couture E Deniau P Grandclaudon
1904 Selective Deprotection of Silyl Ethers with Sodium Periodate J Li D Menche
1909 Micellar Solution of Sodium Dodecyl Sulfate (SDS) Catalyzes KabacknikndashFields Reaction in Aqueous Media S Sobhani A Vafaee
1916 Convenient Methods for the Synthesis of a Library of Hemilabile Phosphines M V Jimeacutenez J J Peacuterez-Torrente M I Bartolomeacute L A Oro
1923 Terminal Aziridines by Addition of Grignard Reagents or Organoceriums to an (α-Chloro)sulfinylimine D M Hodgson J Kloesges B Evans
1933 A Robust Synthesis of Nε-(Carboxymethyl)-L-lysine (CML) R Csuk S Stark A Barthel R Kluge D Stroumlhl
1935 One-Pot Curtius Rearrangement Processes from Carboxylic Acids O Leogane H Lebel
XV Forthcoming Articles
no 12 1941 The Chemistry of Deprotonated α-Aminonitriles T Opatz 1960 An Efficient Synthesis of Tetraalkyl 2345-Thiophenetetracarboxylate
Derivatives A Alizadeh R Hosseinpour 1963 Facile Deprotection of Bulky (Trialkylsilyl)acetylenes with Silver Fluoride
S Kim B Kim J In 1969 Highly Efficient and Reusable Ionic Liquids for the Catalyzed
Hydroamination of Alkenes with Sulfonamides Carbamates and Carboxamides L Yang L-W Xu C-G Xia
1975 Synthesis of 2391016172324-Octasubstituted Phthalocyaninatozinc(II) Complexes Mediated by Reductive Agents G A Gauna A C Monsalvo J Awruch
1979 A Short and Efficient Synthesis of 3-2-[2-(Bromomethyl)thiazol-4-yl]-ethynyl-5-fluorobenzonitrile A Precursor for PET Radioligand [18F]SP203 M B Gopinathan C Jin K S Rehder
1983 Synthesis of a Substituted Benzazepin-2-one Dihydrate S K Boini R K Vaid K P Moder D Mitchell
1987 Synthesis of Novel Trisubstituted Imidazolines F J Lakner M A Parker B Rogovoy A Khvat A Ivachtchenko
1991 A Novel Synthesis of N-But-3-enyl-α- and β-Amino Acids T T Van Nguyen R T C Brownlee A B Hughes
1999 Synthesis of Substituted 5-(3-Hydroxypropyl)pyrrolidin-2-ones and Pyrrolizidinones from Nitroethane via C3 Functionalized 56-Dihydro-4H-12-oxazines A Novel Approach to Some Analogues of the Antidepressant Rolipram A Yu Sukhorukov A V Lesiv Y A Khomutova S L Ioffe V A Tartakovsky
2009 Chiral Cyclobutanols and Cyclopentane Dimers via Samarium(II) Iodide Induced Keto-Olefin Cyclisations of Carbohydrate-Derived Unsaturated Ketones D B G Williams J Caddy K Blann J J C Groveacute C W Holzapfel
2015 Synthesis of Perfluoroalkylthio-Substituted Ferrocenes C Rhode J Lemke M Lieb N Metzler-Nolte
2019 Functionalization of Polyhedral Oligomeric Silsesquioxane (POSS) via Nucleophilic Substitution M Dutkiewicz H Maciejewski B Marciniec
2025 A Novel Synthesis of Aryl Mesylates via One-Pot DemethylationndashMesylation of Aryl Methyl Ethers Using a Mixture of Phosphorus Pentoxide in Methanesulfonic Acid B Kaboudin Y Abedi
2029 Anionic Cyclization of (NN-Dimethylamino)[2-(prop-2-yn-1-yloxy)aryl]-acetonitriles T Zdrojewski J Musielak A Jończyk
2035 Strecker-Type Reaction Catalyzed by Carboxylic Acids in Aqueous Media Z Xie G Li G Zhao J Wang
2040 Synthesis of Novel Structurally Simplified Estrogen Analogues with Electron-Donating Groups in Ring A L F Tietze C A Vock I K Krimmelbein L Nacke
2061 On the Resolution of Secondary Phosphine Oxides via Diastereomeric Complex Formation The Case of tert-Butylphenylphosphine Oxide J Holt A M Maj E P Schudde K M Pietrusiewicz L Sieroń W Wieczorek T Jerphagnon I W C E Arends U Hanefeld A J Minnaard
2066 Enantioselective Copper-Catalyzed Conjugate Addition of Dimethylzinc to 5-(1-Arylalkylidene) Meldrumrsquos Acids A Wilsily T Lou E Fillion
2073 SuzukindashMiyaura Coupling Reactions Using Phosphite Ligands M Jang Y Jo I-K Oh H M Jung S Lee
2076 Synthesis of 2-Methylindoline- and 2-Methyl-1234-tetrahydroquinoline-Derived Phosphoramidites and Their Applications in Iridium-Catalyzed Allylic Alkylation of Indoles W-B Liu H He L-X Dai S-L You
2083 Stereocontrolled Synthesis of 13-Amino Alcohols by Reduction of Substituted 2-1-[(tert-Butylsulfinyl)amino]alkylcyclohexanones J C Gonzaacutelez-Goacutemez F Foubelo M Yus
2089 Tunable Phosphoramidite Ligands for Asymmetric Hydrovinylation Ligands par excellence for Generation of All-Carbon Quaternary Centers C R Smith H J Lim A ZhangT V RajanBabu
2101 Copper-Catalyzed Asymmetric Ring-Opening Reaction of Oxabenzonorbornadienes with Grignard and Aluminum Reagents R Millet L Gremaud T Bernardez L Palais A Alexakis
2113 A Simplified Synthesis of Takemotorsquos Catalyst A Berkessel B Seelig 2116 Pharmaceutical Substances Syntheses Patents and Applications of the
Most Relevant AIPs Edited by Axel Kleeman Juumlrgen Engel Bernhard Kutscher Dietmar Reichert Reviewed by I Agranat
XV Forthcoming Articles
no 13 2117 Recent Advances in the Aza-Claisen Rearrangement K C Majumdar
T Bhattacharyya B Chattopadhyay B Sinha 2143 A Novel and Convenient Synthesis of lsquoReversedrsquo Diamidino 25-Aryl- and
25-Azaheterocycle-Substituted Furans L Hu D W Boykin 2146 Efficient and General Preparation of Pyranostilbenes First Total Synthesis
of Artocarbene and Pawhuskin B B H Park Y R Lee W S Lyoo 2155 Mild Oxidation of Diarylacetylenes to 12-Diketones Using Oxone in
Trifluoroacetic Acid J-H Chu Y-J Chen M-J Wu 2163 One-Pot Microwave-Assisted Selective Azido ReductionTandem Cyclization
in Condensed and Solid Phase with Nickel Boride N Shankaraiah N Markandeya M Espinoza-Moraga C Arancibia A Kamal L Silva Santos
2171 Pyrrolo[321-ij]quinolin-4-one and Pyrrolo[321-ij]quinolin-6-one H McNab D J Nelson E J Rozgowska
2175 Practical Synthesis of 5-Substituted Tetrazoles under Microwave Irradiation J Roh T V Artamonova K Vaacutevrovaacute G I Koldobskii A Hrabaacutelek
2179 A Simple Method for the Synthesis of 3-Arylthieno[23-b]pyridines via Iodine-Mediated Cyclization of 3-(1-Arylalkenyl)-2-[(1-phenylethyl)sulfanyl]pyridines K Kobayashi D Nakamura Y Shiroyama S Fukamachi H Konishi
2184 Synthesis of Four Lysine-Linked Cereulide Analogues Showing Ionophoric Activity Towards Potassium Cations as Lead Compounds for Emetic Toxin-Detection by Immunoassays A Makarasen T Nishikawa M Isobe
2205 Synthesis of α-Aliphatic and β-Aromatic Substituted Taurines via Regioselective Ring Opening of Thiiranes with Ammonia H Yu S Cao L Zhang G Liu J Xu
2210 Stability of 5(6)-Carboxyfluorescein in Microwave-Assisted Synthesis of Fluorescein-Labelled O-Dimannosylated Peptides R Kowalczyk P W R Harris R P Dunbar M A Brimble
2223 Diversity-Oriented Synthesis of Functionalized Diaryl Sulfones by Regioselective [3+3] Cyclizations of 13-Bis(siloxy)buta-13-dienes with 2-(Arylsulfonyl)-3-ethoxy-2-en-1-ones Scope and Limitations M Shkoor A Riahi O Fatunsin H Reinke C Fischer P Langer
2236 Synthesis of Functionalized Salicylates by Formal [3+3] Cyclocondensation of 13-Bis(silyloxy)buta-13-dienes with 3-Alkoxy-2-en-1-ones G Mroszlig S Ladzik H Reinke A Spannenberg C Fischer P Langer
2249 Synthetic Approach to Alkoxy-β-(trifluoromethyl)styrenes and Their Application in the Synthesis of New Trifluoromethylated Heterocycles V M Muzalevskiy V G Nenajdenko A V Shastin E S Balenkova G Haufe
2260 o-Benzenedisulfonimide as a Powerful and Recyclable Organocatalyst for the Nazarov Reaction M Barbero S Cadamuro A Deagostino S Dughera P Larini E G Occhiato C Prandi S Tabasso R Vulcano P Venturello
2267 The Catalytic Potential of 4-Guanidinylpyridines in Acylation Reactions I Held E Larionov C Bozler F Wagner H Zipse
2278 Iron(III) Chloride in EthanolndashWater Highly Efficient Catalytic System for the Synthesis of Garcia Gonzalez Polyhydroxyalkyl- and C-Glycosylfurans L Nagarapu M V Chary A Satyender B Supriya R Bantu
2283 Ruthenium-Catalyzed Addition of Primary Amides to Alkynes A Stereoselective Synthesis of Secondary Enamides L J Gooszligen M Blanchot K S M Salih K Gooszligen
2289 Binaphthyl-Modified Quaternary Phosphonium Salts as Chiral Phase Transfer Catalysts Application to Asymmetric Amination of β-Keto Esters R He K Maruoka
X Table of Contents XI Forthcoming Articles
no 14 2293 Direct Methods for Stereoselective Polypropionate Synthesis A Survey
J Li D Menche 2316 Synthesis of Symmetrical Ketones from Grignard Reagents and
11-Carbonyldiimidazole D Bottalico V Fiandanese G Marchese A Punzi
2319 Synthesis of 45-Substituted Imidazoles by a Fast Condensation of 12-Diketones and Urotropine in Heterogeneous Medium G Bratulescu
2321 (Arylsulfonyl)acetones and -acetonitriles New Activated Methylenic Building Blocks for Synthesis of 123-Triazoles N T Pokhodylo V S Matiychuk M D Obushak
2324 A Safe Convenient and Efficient One-Pot Synthesis of α-Chloroketone Acetals Directly from Ketones Using Iodobenzene Dichloride J Yu C Zhang
2329 An Efficient Oxidative Conversion of Aldehydes into 2-Substituted 2-Oxazolines Using 13-Diiodo-55-dimethylhydantoin S Takahashi H Togo
2333 A Novel Procedure for the Synthesis of Benzo[b][18]naphthyridine-3-carboxylate Derivatives from MoritandashBaylisndashHillman Adduct Acetates W Zhong F Lin R Chen W Su
2341 An Improved Synthesis of 147-Triazacyclononanes (tacns) and 14710-Tetraazacyclododecanes (cyclens) J Huang Z Zhou T H Chan
2345 The Ullmann Coupling between 2-Chlorobenzoic Acids and Amino Acids A Valuable Reaction for Preparing 2-Substituted 1-Acetyl-1H-indol-3-yl Acetates J C Rodriguez Dominguez X Gang G Kirsch
2349 gem-Dibromomethyl Aromatics Efficient Aldehyde Equivalents in the KnoevenagelndashDoebner Reaction J K Augustine Y A Naik S Poojari N Chowdappa B S Sherigara K Areppa
2357 Synthesis of Novel α-Aminophosphonates Containing Adamantyl Fragment M M Kabachnik L I Minaeva I P Beletskaya
2361 Efficient Fluoride-Mediated Synthesis of 5-Amino-Substituted Isothiazoles Y S Zubenko V I Potkin
2365 Phosphine-Catalyzed Reaction of Cyanohydrins with Activated Alkynes A Siby O Loreau F Taran
2371 Sulfanyl-Substituted [3]Cumulenes and Buta-13-dienes from a Tetrakis(pyridinium)-Substituted Butadiene A Schmidt A Rahimi M Gjikaj
2379 Efficient Synthesis of 2-Substituted Pyrido[32-d]pyrimidines Involving SNAr and Palladium-Catalyzed Cross-Coupling Reactions A Tikad S Routier M Akssira J-M Leacuteger C Jarry G Guillaumet
2385 Novel Synthesis of Medium-Sized Heterocycles by Palladium-Catalyzed Intramolecular Heck Reaction via 9-endo-trig Mode of Cyclization K C Majumdar B Chattopadhyay
2393 Facile Synthesis of Fluorinated Benzofuro- and Benzothieno[23-b]pyridines α-Carbolines and Nucleosides Containing the α-Carboline Framework V O Iaroshenko Y Wang B Zhang D Volochnyuk V Ya Sosnovskikh
2403 Synthesis of Functionalized N-Vinyl Nitrogen-Containing Heterocycles S M M Lopes A M Beja M Ramos Silva J A Paixatildeo F Palacios T M V D Pinho e Melo
2408 Kumada Cross-Coupling of Aryl Grignard Reagents with Aryl Halides Catalyzed by an Immobilized Nickel Catalyst X Chen L Wang J Liu
2413 Highly Enantioselective Synthesis of Heteroaromatic Alcohols Catalyzed by Chiral DiaminodiphosphinendashRuthenium(II) Complexes W-Y Shen Y-Y Li Z-R Dong J-X Gao
2418 Concise Total Synthesis of (+)-Disparlure and its trans-Isomer Using Asymmetric Organocatalysis S-G Kim
2423 Rhodium Carbenoid Induced [12]-Migration in an L-Lyxo-Configured α-Diazo β-Keto Ester Synthesis of a New Griseolic Acid Analogue N N Bhujbal K S A Kumar D D Dhavale
2430 Synthesis of 5-Arylthio-3-hydroxyphthalates by the First [4+2] Cycloadditions of 3-Arylthio-1-silyloxy-13-butadienes with Dimethyl Acetylenedicarboxylate I Iqbal M Imran P Langer
2435 Synthesis of Highly Functionalized Proline Derivatives via a One-Pot MichaelSN-AdditionCyclization Approach U Kazmaier C Schmidt
2440 RhodiumGraphite-Catalyzed Hydrogenation of Carbocyclic and Heterocyclic Aromatic Compounds G Falini A Gualandi D Savoia
2447 Potassium [1-(tert-Butoxycarbonyl)-1H-indol-2-yl]trifluoroborate as an Efficient Building Block in Palladium-Catalyzed SuzukindashMiyaura Cross Couplings P Kassis V Beacuteneacuteteau J-Y Meacuterour S Routier
2454 Syntheses of Substituted Furans and Pyrroles by Platinum-Catalyzed Cyclizations of Propargylic Oxiranes and Aziridines in Aqueous Media M Yoshida M Al-Amin K Shishido
2467 Transition-Metal-Free Oxidative Homocoupling of Aryl Alkenyl and Alkynyl Grignard Reagents with TEMPO M S Maji A Studer
XIII Forthcoming Articles
no 15 2471 Advances in Synthetic Approaches for the Preparation of Combretastatin-
Based Anti-Cancer Agents R Singh H Kaur 2492 Synthesis of Unsymmetrical Ureas by Sulfur-Assisted Carbonylation with
Carbon Monoxide and Oxidation with Molecular Oxygen under Mild Conditions T Mizuno T Nakai M Mihara
2497 Ring-OpeningRecyclization Reactions of (Dimethylamino)propenoyl-Substituted Cyclopropanes Facile Synthesis of Halogenated Pyridin-2(1H)-ones R Zhang Y Zhou Y Liang Z Jiang D Dong
2501 Facile and Efficient Total Synthesis of Taspine B Cheng S Zhang L Zhu J Zhang Q Li A Shan L He
2505 Oligomeric Iodosylbenzene Sulfate A Convenient Hypervalent Iodine Reagent for Oxidation of Organic Sulfides and Alkenes M S Yusubov R Y Yusubova T V Funk K-W Chi V V Zhdankin
2509 Pyrrolidine-Based Organocatalysts for Enantioselective Michael Addition of Cyclohexanone to trans-β-Nitrostyrene A P Carley S Dixon J D Kilburn
2517 CundashAl Hydrotalcite An Efficient and Reusable Ligand-Free Catalyst for the Coupling of Aryl Chlorides with Aliphatic Aromatic and N(H)-Heterocyclic Amines B Sreedhar R Arundhathi P L Reddy M A Reddy M L Kantam
2523 Highly Efficient Synthesis of trans-βγ-Unsaturated a-Keto Amides C Allais T Constantieux J Rodriguez
2531 Gas-Phase Synthesis of N-Unsubstituted 3-Hydroxypyrroles and 1H-Pyrrol-3(2H)-ones L Hill G A Hunter S H Imam H McNab W J OrsquoNeill
2535 3-Hydroxy-1H-pyrrole L Hill S H Imam H McNab W J OrsquoNeill 2539 123-Thiadiazoles with Unsaturated Side Chains Synthesis
Polymerization and Photocrosslinking M Al-Smadi N Hanold H Kalbitz H Meier
2547 Synthesis of 1112-Didehydrodibenzo[ae]cycloocten-5(6H)-one A Strained Eight-Membered Alkyne S C Kornmayer F Rominger R Gleiter
2553 Stannous Chloride Dihydrate A Novel and Efficient Catalyst for the Synthesis of gem-Dihydroperoxides from Ketones and Aldehydes D Azarifar K Khosravi F Soleimanei
2557 Synthesis of a Novel Class of Azacrown Macrocycles and Lariat Crown Ethers Containing Two 124-Triazole Rings as Subunits N Foroughifar A Mobinikhaledi S Ebrahimi
2561 Enantioselective Synthesis of the 3C-Protease Inhibitor (ndash)-Thysanone by a StauntonndashWeinreb Annulation Strategy J Sperry T Y Yuen M A Brimble
2570 Stereoselective Synthesis of Unnatural β-Amino Acids from Nitroethane via 56-Dihydro-4H-12-oxazin-3-ylacetates A Yu Sukhorukov A V Lesiv O L Eliseev Y A Khomutova S L Ioffe
2579 A Versatile Unexpected One-Pot Regioselective Synthesis of a New Class of 13-Diazepinoindolones by Reaction of Pyranoindolones with Monosubstituted Ureas D Livadiotou C A Tsoleridis J Stephanidou-Stephanatou
2584 Synthesis of a Trisaccharide and a Tetrasaccharide from the Cell-Wall Lipopolysaccharides of Azospirillum brasilense S17 S Pandey S Ghosh A K Misra
2591 Synthesis of Isoindoline Nitroxides by Electrocyclic Reactions T Kaacutelai J Jekı K Hideg
2596 Glycosylations of Tertiary Alcohols Synthesis of Fully Protected Disaccharides with Sterically Demanding Groups Attached to the Sugar Core A Holkenbrink J B Vicente D B Werz
2605 Copper-Catalyzed [13]-Dipolar Cycloaddition for the Synthesis of Macrocycles Containing Acyclic Aromatic and Steroidal Moieties G V Latyshev M S Baranom A V Kazantsev A D Averin N V Lukashev I P Beletskaya
2616 Aryl Ring Migration Reaction in the Synthesis of 24-Diaryl-4H-31-benzothiazines A V Butin F A Tsiunchik V T Abaev A V Gutnov D A Cheshkov
2627 Hydrogenation of β-N-Substituted and β-NN-Disubstituted Enamino Esters in the Presence of Iridium(I) Catalyst H Hebbache Z Hank C Bruneau J-L Renaud
2634 Stereoselective Olefination Reactions Promoted by Rieke Manganese J M Concelloacuten H Rodriacuteguez-Solla V del Amo P Diacuteaz
2646 Synthesis of Piperidinones through a Radical Cascade E Godineau Y Landais
2650 Asymmetric Organic Synthesis with Enzymes Edited by V Gotor I Alfonso E Garciacutea-Urdiales Reviewed by Steve Collier
XVII Forthcoming Articles
no 16 2651 Synthesis of Spirocyclic Ethers S Rosenberg R Leino 2674 Bimetallic PalladiumndashPlatinum-on-Carbon-Catalyzed HndashD Exchange
Reaction Synergistic Effect on Multiple Deuterium Incorporation T Maegawa N Ito K Oono Y Monguchi H Sajiki
2679 Efficient Copper-Catalyzed Synthesis of 2-Amino-4(3H)-quinazolinone and 2-Aminoquinazoline Derivatives X Huang H Yang H Fu R Qiao Y Zhao
2689 Synthesis and Chemoselective N- and O-Alkylation of Thiadiazolopyrimidine Nucleosides and Uridines A M L Hossion R Islam R K Kandahary T Nagamatsu
2697 Facile and Efficient Synthesis of a New Class of Indole-Substituted Pyridine Derivatives via One-Pot Multicomponent Reactions K Zhao X-P Xu S-L Zhu D-Q Shi Y Zhang S-J Ji
2709 Studies toward a Total Synthesis of Rhizoxin D Stereoselective Preparation of the C11ndashC19 Fragment S Padakanti C K Kumar E Ashok P Das
2715 A Short Synthesis of Enantiomeric Phytoprostanes B1 Type I W Perlikowska M Mikołajczyk
2719 Chemistry of Polyhalogenated Nitrobutadienes Part 7 A Novel Synthetic Access to Chlorinated Nitrile Oxides E Nutz V A Zapolrsquoskii D E Kaufmann
2725 Microwave-Assisted Silver(I)-Mediated Selective O-Alkylation of Aromatic Imidate Systems B K Singh C Cavalluzzo M De Maeyer Z Debyser V S Parmar E Van der Eycken
2729 Iodogen A Novel Reagent for the Oxidation of Urazoles under Heterogeneous Conditions A Khoramabadi A Shiri M A Zolfigol S Mallakpour
2733 An Unprecedented Synthesis of Eight-Membered-Ring Cyclic Thioimidic Esters by a Three-Component Reaction A Alizadeh R Hosseinpour
2737 A Novel Diastereoselective Synthesis of β-Phosphonato Unsaturated Thioimidates A Alizadeh N Zohreh
2741 Synthesis of 21-Benzisoxazoles by Nucleophilic Substitution of Hydrogen in Nitroarenes Activated by the Azole Ring N T Pokhodylo Y O Teslenko V S Matiychuk M D Obushak
2749 A Facile Synthesis of Two Series of Multifunctional Carbon Compounds from αα-Dihalo Ketones Using Allylsamarium Bromide X Liu S Zhang J Di
2756 Stereocontrolled Formation of Protected Aminodeoxyalditols from Simple Carbohydrate Precursors by Debenzylating Cycloetherification Y Jiang Z Fang Q Zheng H Jia J Cheng B Zheng
2761 trans-Stilbene as a Starting Material for the Synthesis of Tamoxifen Based on Palladium-Catalyzed Cross-Coupling Reactions C M Nunes J Limberger S Poersch M Seferin A L Monteiro
2766 Synthesis and Biological Evaluation of 6-Substituted Purinylcarbanucleosides with a Cyclopenta[b]thiophene Pseudosugar P Abeijoacuten J M Blanco O Caamantildeo F Fernaacutendez M D Garciacutea X Garciacutea-Mera J E Rodriacuteguez-Borges J Balzarini E De Clercq
2773 Synthesis and Electrochemical Signature of Novel Norbornyl-ferrocene Hybrids F A Khan S K Upadhyay
2778 A Regioselective TsujindashTrost Pentadienylation of 3-Allyltetronic Acid R Schobert B Barnickel
2785 Copper(I)-Catalyzed CarylndashCalkynyl Bond Formation of Aryl Iodides with Terminal Alkynes K G Thakur G Sekar
2790 Aminolysis of Epoxides Using Iridium Trichloride as an Efficient Catalyst J Agarwal A Duley R Rani R K Peddinti
2797 Preparation of Several Active N-Chloro Compounds from Trichloroisocyanuric Acid A Shiri A Khoramabadi-zad
2802 The First Mineral-Catalyzed One-Pot [3+1+2] Coupling Protocol for Multifunctionalized Fused-Ring Pyrimidines L D S Yadav A Rai
2809 Efficient Synthesis of Tetrahydro-β-carbolin-1-one and Dihydroisoquinolin-1-one Derivatives as Versatile Intermediates K E Judd M F Mahon L Caggiano
2818 A Concise Synthesis of ortho-Iodobenzyl Alcohols via Addition of ortho-Iodophenyl Grignard Reagent to Aldehydes and Ketones J Cvengroš D Stolz A Togni
XIII Forthcoming Articles
no 17 2825 Reactivity of Oxazol-5-(4H)-ones and Their Application toward Natural
Product Synthesis N M Hewlett C D Hupp J J Tepe 2840 Towards the Total Synthesis of 3-Hydroxyvibsanin E B D Schwartz
J R Denton P V Bernhardt H M L Davies C M Williams 2847 Structure Investigations of (ent)-Cladospolide D by De Novo Synthesis and
Kinetic and Thermodynamic Isomerization Y Xing J H Penn G A OrsquoDoherty
2855 New Applications of PhI(OAc)2 in Synthesis Total Synthesis and SAR Development of Potent Antitumor Natural Product PsymberinIrciniastatin A N Shao X Huang A Palani R Aslanian A Buevich J Piwinski R Huryk C Seidel-Dugan
2873 Total Synthesis of Largazole ndash Devolution of a Novel Synthetic Strategy B Wang C J Forsyth
2881 Formal Total Synthesis of Palmerolide A J Jaumlgel M E Maier 2893 Total Synthesis of Bongkrekic Acid via Sequential SuzukindashMiyaura Coupling
Reactions M Kanematsu M Shindo M Yoshida K Shishido 2905 Stereodivergent Approach to Both C28a-syn and C28a-anti Relative
Stereochemical Manifolds in the Lepadin Family via a TiCl4-Promoted G Li L J Carlson I K Sagamanova B W Slafer R P Hsung C Gilardi H M Sklenicka N Sydorenko
2915 Enantioselective Aldol Reaction of Tetrasubstituted Ketene Silyl Acetals with Achiral Aldehydes for the Construction of Asymmetric Tertiary Alcohols An Application for the Divergent Total Syntheses of Buergerinins F and G I Shiina T Iizumi Y-s Yamai Y-i Kawakita K Yokoyama Y-k Yamada
2927 Second-Generation Biomimetic Total Synthesis of Chaetominine A Coste G Karthikeyan F Couty G Evano
2935 Total Synthesis of (+)-Fostriecin and (+)-Phoslactomycin B S Shibahara M Fujino Y Tashiro N Okamoto T Esumi K Takahashi J Ishihara S Hatakeyama
2954 Stereochemical Assignments of the Chlorinated Residues in Victorin C A C Durow C Butts C L Willis
2963 Studies of the Asymmetric Total Synthesis of Clavilactone D by the lsquoLariatrsquo Cyclization Strategy T Yoshimitsu S Nojima M Hashimoto K Tsukamoto T Tanaka
2970 Total Synthesis of the Leucetta-Derived Alkaloid Calcaridine A P B Koswatta R Sivappa H V R Dias C J Lovely
2983 Formal Synthesis of Salinosporamide A Starting from D-Glucose T Momose Y Kaiya J-i Hasegawa T Sato N Chida
2992 Synthesis of Bioactive Natural Products by Asymmetric syn- and anti-Aldol Reactions A K Ghosh Z L Dawson
no 18 3003 Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural
Products B M Trost M K Brennan 3026 One-Pot Synthesis of Furo[34-b]pyridin-5(7H)-ones from 2-
Bromopyridine-3-carboxylic Acid and Carbonyl Compounds K Kobayashi T Kozuki H Konishi
3029 Iodocyclization of N-[2-(Methylthio)phenyl]propiolamides Selective Synthesis of 3-Iodo-15-benzothiazepin-4-ones T-S Jiang X-G Zhang J-H Li
3039 A Facile Synthetic Method for Fluorine-Containing 17-Phenanthrolines Pyridine-Ring Formation Reaction of N-Propargyl-68-bis(trifluoroacetyl)-quinolin-5-amine with Various Nucleophiles D Shibata E Okada M Hinoshita M Meacutedebielle
3047 Enantiotopic Discrimination in Palladium-Mediated Nucleophilic Substitutions on Achiral Substrates Chiral Ligand versus Chiral Nucleophile O Jacquet F Charnay J-C Fiaud J Ollivier
3051 Studies on the Chemistry of 2-[3-(2-Nitrophenyl)-2-oxopropyl]benzaldehydes Novel Syntheses of 5H-Benzo[b]carbazole-611-diones and Indolo[12-b]isoquinoline-611-diones M Fernaacutendez
3061 Studies on the C22ndashC23 Aldol Coupling of Spirangien M Lorenz N Bluhm M Kalesse
3067 One-Pot Synthesis of N-Alkyl Purine Pyrimidine and Azole Derivatives from Alcohols using Ph3PCCl4 A Rapid Route to Carboacyclic Nucleoside Synthesis M N Soltani Rad A Khalafi-Nezhad S Behrouz Z Asrari M Behrouz Z Amini
3077 Synthesis of 2-Amino-34-dihydroquinazolines and Imidazo[21-b]quinazoline-2-ones A Mishra S Batra
3089 Studies on the Reaction of Diimines with Thiourea Synthesis and Solvent-Induced cistrans-Isomerization of 135-Triazinane-2-thiones B Kaboudin T Ghasemi T Yokomatsu
3094 Suzuki Coupling of Heteroaromatic Chlorides Using Highly Electron-Donating ClickPhos Ligands S M Spinella Z-H Guan J Chen X Zhang
3099 Reaction of NN-Dioxyenamines with Anhydrides of Carboxylic and Sulfonic Acids A New Method for the Synthesis of a-Hydroxyoxime Derivatives A A Tabolin A V Lesiv S L Ioffe
3106 Directed ortho Metallation Chemistry and Phosphine Synthesis New Ligands for the SuzukindashMiyaura Reaction D B G Williams S J Evans H de Bod M S Mokhadinyana T Hughes
3113 New Functional Derivatives of 9-Phenylquinine P J Boratyński J SkarŜewski
3120 On the Synthesis of Asymmetric and Dissymmetric Amino Analogues of Troumlgerrsquos Base J Artacho K Waumlrnmark
3127 Synthesis of Polycyclic Sultams by Palladium-Catalyzed Intramolecular Cyclization K C Majumdar S Mondal N De
3136 Synthesis of Functionalized L-Cysteine and L-Methionine by Reaction with Electron-Deficient Acetylenes B A Trofimov A G Malrsquokina O A Shemyakina V V Nosyreva A P Borisova S S Khutsishvili L B Krivdin
3143 A lsquoClickrsquo Approach to the Synthesis of 3-[2-(1-Alkyltriazol-4-yl)ethyl]indoles M Petrini R R Shaikh
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
No 7 1049 Catalytic Transformations of Benzylic Carboxylates and Carbonates
R Kuwano 1062 A Simple and Practical Method for the Oxidation of Thebaine to 14-
Hydroxycodeinone by V2O5ndashH2O2 S Das Sharma D Konwar 1065 Umpolung with Sulfur Dioxide CarbonndashCarbon Cross-Coupling of Electron-
Rich 13-Dienes and Alkenes Application to the Enantioselective Synthesis of Long-Chain Polyketide Fragments M Turks C J Exner C Hamel P Vogel
1075 One-Pot Synthesis of 14-Diarylnaphthalenes via a WittigndashHorner Reaction[4+2] CycloadditionDehydrogenation Sequence Z Chen W Shou Y Wang
1081 A Novel and General Method for the Formation of S-Aryl Se-Aryl and Te-Aryl Phosphorochalcogenoates Y-X Gao G Tang Y Cao Y-F Zhao
1087 A Remarkable Access to γ-Fluoroalkylated Propargylamine Derivatives or Fluoroalkylated Dihydroisoxazoles via the Reaction of Fluoroalkylated Acetylides with Various Nitrones T Konno K Moriyasu T Ishihara
1095 Short and Practical Syntheses of (S)-(+)-3-(p-Tolylsulfinyl)furan-2(5H)-one and (S)-(+)-3-(p-Tolylsulfinyl)-56-dihydropyran-2-one D Cruz Cruz A Hernaacutendez Linares F Yuste M R Martiacuten J L Garciacutea Ruano
1099 Decarboxylative Aldol-Type Reaction of 2-(Trifluoroacetyl)-13-diazoles with Activated Acetic Acids P V Khodakovskiy D M Volochnyuk A A Tolmachev
1105 Synthesis of 2-[(Arylmethylene)amino]cyclopropanecarbonitriles via a Two-Step Ring Transformation of 2-(Cyanomethyl)aziridines S Mangelinckx M Drsquohooghe S Peeters N De Kimpe
1113 Synthesis of Dendrimeric Tumor-Associated Mucin-Type Glycopeptide Antigens T Becker A Kaiser H Kunz
1123 A Simple and Efficient Oxidation Procedure for the Synthesis of Acid-Sensitive Epoxides O Bortolini G Fantin M Fogagnolo
1127 Rapid Chemoselective Deprotection of Benzyl Esters by Nickel Boride J M Khurana R Arora
1131 Three-Component Coupling of Isoquinoline Activated Alkyne and Nitromethane A Facile Synthesis of Nitromethyl Derivatives of 12-Dihydroisoquinolines J S Yadav B V S Reddy N N Yadav M K Gupta
1137 Palladium Supported on a Polyionic Resin as an Efficient Ligand-Free and Recyclable Catalyst for Heck SuzukindashMiyaura and Sonogashira Reactions B Basu S Das P Das B Mandal D Banerjee F Almqvist
1147 Oxidation of 25-Dialkylpyrrole Derivatives with Cerium(IV) Ammonium Nitrate R Voloshchuk M Gałęzowski D T Gryko
1153 Practical Syntheses of Enantiomerically Pure Key Intermediates of Opioid Receptor-like 1 (ORL1) Antagonists T Yoshizumi A Ohno T Tsujita H Takahashi O Okamoto I Hayakawa H Kigoshi
1163 An Environmentally Benign TEMPO-Catalyzed Efficient Alcohol Oxidation System with a Recyclable Hypervalent Iodine(III) Reagent and Its Facile Preparation X-Q Li C Zhang
1170 Efficient and Stereoselective Rearrangement of BaylisndashHillman Acetates Catalyzed by Gold(I) ChlorideSilver(I) Trifluoromethanesulfonate Y Liu D Mao J Qian S Lou Z Xu Y Zhang
1175 The First Total Synthesis of Kynapcin-24 by Palladium Catalysis L-Y Yang C-F Chang Y-C Huang Y-J Lee C-C Hu T-H Tseng
1180 Enantioselective Synthesis of N-Protected α-Amino Acid Hydrazides M Bibian S El-Habnouni J Martinez J-A Fehrentz
1185 Synthesis of 11H-Indolo[32-c]quinoline-6-carboxylic Acids by Cascade AutoxidationndashRing Contractions A Becker S Kohfeld T Pies K Wieking L Preu C Kunick
1190 Reaction of N-Nonaflylbenzotriazole with Silyl Enol Ethers M Uhde T Ziegler
1195 2-(Benzoylimino)thiazolidin-4-ones Formation by an Alternative Ring Closure and Analysis of Rotational Barriers H-G Haumlcker P W Elsinghorst S Michels J Daniels G Schnakenburg M Guumltschow
1204 Microwave-Assisted Synthesis and Functionalization of Selenolopyrimidines S Hesse C Chenet D Thomae G Kirsch
1209 12-Disubstituted 4-Quinolones via Copper-Catalyzed Cyclization of 1-(2-Halophenyl)-2-en-3-amin-1-ones R Bernini S Cacchi G Fabrizi A Sferrazza
1220 A New Atom-Economical and Selective Synthesis of Secondary and Tertiary Alkylamines by Means of CpIridium Complex Catalyzed Multiple N-Alkylation of Ammonium Salts with Alcohols without Solvent R Yamaguchi Z Mingwen S Kawagoe C Asai K-i Fujita
1224 Synthesis of Regioisomerically Pure 5-Functionalized 27-Dichlorofluoresceins J C Castro A Malakhov K Burgess
XIII Forthcoming Articles
No 8 1227 Michael Additions to Activated Vinylphosphonates T Janecki J Kędzia
T Wąsek 1255 A Facile and General Synthesis of 2β-Aminosteroids X Ke H Hu
D Zhou W Xu Q Zhu N P Reddy X Hu 1261 Efficacious Preparation of Oppolzerrsquos Glycylsultam via the Deleacutepine
Reaction A Isleyen C Gonsky R C Ronald P Garner 1265 Synthesis of Masked Vicinal Amino Aldehydes of Pyrrolizine and Pyrrolo
[12-c]thiazole Series A V Tverdokhlebov A V Denisenko A A Tolmachev Y M Volovenko S V Shishkina O V Shishkin
1271 Preparation of 9-Substituted Pyridine-Stretched Adenines and Hypoxanthines J A Crawford W Fraser C A Ramsden
1279 A Versatile Synthesis of Heterocyclic Analogues of Neoflavonoids from Enamino Ketones V S Moskvina V P Khilya O V Turov U M Groth
1287 New Stereoselective Synthesis of Paeonilactone B F G Gatti S Serra 1291 The Use of NN-Dialkyltrimethylsilylamines in the Synthesis of
Pentamethinium Salts M Kořiacutenek M Rybaacutečkovaacute Boumlhm 1297 Synthesis of Triazoles via Regioselective Reactions of Aryl Azides with
Cyanoacetyl Pyrroles and Indoles N T Pokhodylo V S Matiychuk M D Obushak
1301 Gallium(III) Chloride Catalyzed Hydroarylation of Arylacetylenes with Naphthols and Phenols A Facile Synthesis of Vinylarenes J S Yadav B V S Reddy S Sengupta S K Biswas
1305 Electrophilic Bromination of meta-Substituted Anilines with N-Bromosuccinimide Regioselectivity and Solvent Effect S Bartoli A Cipollone A Squarcia A Madami D Fattori
1309 Cross-Coupling Reactions of Halopurines with Aryl- and Alkyltrifluoroborates The Scope and Limitations in the Synthesis of Modified Purines Z Hasniacutek R Pohl M Hocek
1318 A Convenient Method for Converting Hydroxyacetophenones into Their Ethylene or Trimethylene Acetals F Ono H Takenaka T Fujikawa M Mori T Sato
1323 γ-Chloromagnesio γ-Lactones and δ-Chloromagnesio δ-Lactones Generation Properties and Synthetic Uses H Shimizu S Fukuda S Sugiyama T Satoh
1336 Click Reactions with Nitroxides T Kaacutelai W L Hubbell K Hideg 1341 Synthesis of Novel 14-Benzoquinone-Containing 123-Triazoles An Entry
Into a New Library F Algi M Balci 1348 Efficient Synthesis of Two Sialylated Tetrasaccharides Found in Goat Milk
P K Mandal A K Misra 1355 Dendrimers of Vaccines Consisting of Tumor-Associated Glycopeptide
Antigens and T Cell Epitope Peptides S Keil A Kaiser F Syed H Kunz
1370 IBXTBAB-Mediated Oxidation of Primary Amines to Nitriles F Drouet P Fontaine G Masson J Zhu
1375 Chemoselectivity of Multicomponent Condensations of Barbituric Acids 5-Aminopyrazoles and Aldehydes E A Muravyova S V Shishkina V I Musatov I V Knyazeva O V Shishkin S M Desenko V A Chebanov
1386 Stereoselective Total Syntheses of Leiocarpin A and (ndash)-Galantinic Acid Starting from D-Mannitol K Nagaiah D Sreenu K V Purnima R S Rao J S Yadav
1393 A Facile Mild Deprotection Protocol for 13-Dithianes and 13-Dithiolanes with 30 Hydrogen Peroxide and Iodine Catalyst in Aqueous Micellar System N C Ganguly S K Barik
1400 Rhodium-Catalyzed Gram-Scale Synthesis of Highly Substituted Pyridine Derivatives K Parthasarathy C-H Cheng
1403 Enantioselective Synthesis of (R)-Propylene Carbonate from Ethyl (S)-Lactate J M Whitaker R C Ronald
XIII Forthcoming Articles
no 9 1405 Transition-Metal-Catalyzed Site-Selective Cross-Coupling of Di- and
Polyhalogenated Compounds J-R Wang K Manabe 1428 An Improved Synthesis of (4-4-Hydroxy-3-isopropyl-5-[(4-nitrophenyl)
ethynyl]benzyl-35-dimethylphenoxy)acetic Acid (NH-3) M B Gopinathan K S Rehder
1431 Copper-Catalyzed Tandem CndashN Bond Formation Reaction Selective Synthesis of 2-(Trifluoromethyl)benzimidazoles M-W Chen X-G Zhang P Zhong M-L Hu
1437 Synthesis and Thermochemical Properties of Stereoisomeric Dihydroxy- and Tetrahydroxyalkylammonium Salts M Thomas L Rothman J Hatcher P Agarkar R Ramkirath S Lall-Ramnarine R Engel
1445 Preparation of 5-Substituted 2-(2-Alkylaryl-1H-imidazol-4-yl)oxazoles and 5-Substituted 2-(2-Alkylarylthiazol-4-yl)oxazoles by Utilizing 5-Substituted 2-(2-Bromo-11-diethoxyethyl)oxazole as a Synthon D R St Laurent J L Romine
1459 Novel and Efficient Methods for the Synthesis of Symmetrical Trisulfides A Kertmen S Lach J Rachon D Witt
1463 An Environmentally Benign Electrochemical Process for the Reduction of Carboxylic Acid Hydrazides to Amides M Mentel M J Beier R Breinbauer
1469 Synthesis of 1-Chloroalkynes from Alkynylsilanes Using Trichloroisocyanuric Acid as Chlorinating Agent M H Vilhelmsen A S Andersson M B Nielsen
1473 A Convenient Approach to Enantioenriched Cyclopropanes Bearing Electron-Withdrawing Functionalities H Krawczyń K Wąsek J Kędzia
1477 Synthesis of Cyclopropenes via 12-Elimination of Bromocyclopropanes Catalyzed by Crown Ether W M Sherrill R Kim M Rubin
1485 A Base-Catalysed One-Pot Three-Component Coupling Reaction Leading to Nitrosubstituted Pyrroles I R Baxendale C D Buckle S V Ley L Tamborini
1494 Synthesis of 4-Alkylidene-4H-31-benzoxazine Derivatives by Acid-Catalyzed Cyclization of 2-Isocyanophenyl Ketones in the Presence of a Vinyl Ether K Kobayashi Y Okamura H Konishi
1499 Synthesis of Higher Helicenes via Olefin Metathesis and CndashH Activation J Cocircteacute S K Collins
1506 Azido- and Ethynyl-Substituted 2262-Terpyridines as Suitable Substrates for Click Reactions A Winter A Wild R Hoogenboom M W M Fijten M D Hager R-A Fallahpour U S Schubert
1513 Synthesis of 2-(Arylamino)ethanethiols via Lewis Acid Catalyzed Aminolysis of 22-Dimethylthiirane as Precursors of the 14-Benzothiazine Nucleus R Spogli S Sabatini G Manfroni O Tabarrini V Cecchetti
1520 Iron(III) Chloride A Versatile Catalyst for the Practical Synthesis of 3-Sulfenylindoles J S Yadav B V S Reddy Y J Reddy K Praneeth
1525 Organocatalytic Enantioselective Conjugate Addition of 2-Fluoromalonate to Nitroolefins Direct Synthesis of Chiral Fluorinated γ-Nitro Carboxylic Acid Derivatives H Li L Zu H Xie W Wang
1531 Asymmetric Transfer Hydrogenation of Ketimines with Trichlorosilane Structural Studies Z Zhang P Rooshenas H Hausmann P R Schreiner
1545 Prolinol Sulfinyl Ester Derivatives Organocatalytic Michael Addition of Ketones to Nitroolefins under Neat Conditions X Zeng G Zhong
1551 Asymmetric Oxidations of Electron-Poor Alkenes Promoted by the β-Amino AlcoholTBHP System A Russo A Lattanzi
1557 Enantioselectivity Switch in Direct Asymmetric Aminoxylation Catalyzed by Binaphthyl-Based Chiral Secondary Amines T Kano A Yamamoto F Shirozu K Maruoka
1564 Enantioselective Conjugate Addition of N-Heterocycles to αβ-Unsaturated Ketones Catalyzed by Chiral Primary Amines G Luo S Zhang W Duan W Wang
1573 Sulfonyl Hydrazine as New Functionality in Organocatalysis Camphorsulfonyl Hydrazine Catalyzed Enantioselective Aza-Michael Addition L-Y Chen H He B-J Pei W-H Chan A W M Lee
1578 Conversion of Primary Alcohols and Aldehydes into Methyl Esters by Ruthenium-Catalysed Hydrogen Transfer Reactions N A Owston T D Nixon A J Parker M K Whittlesey J M J Williams
1582 Addendum and Erratum XVII Forthcoming Articles
no 10 1583 Organocatalytic Formation of Quaternary Stereocenters M Bella
T Gasperi 1615 Regioselective Synthesis of 5H-Thiazolo[32-a]pyrimidin-5-ones from
MoritandashBaylisndashHillman Adduct Acetates under Solvent-Free and Base-Free Conditions W Zhong B Guo F Lin Y Liu W Su
1623 First Synthesis of 5-Cyanosalicylates by Formal [3+3] Cyclocondensations of 13-Bis(silyloxy)-13-butadienes A Riahi O Fatunsin M Shkoor R Dede H Reinke C Fischer P Langer
1635 Reaction of Isocyanides Dialkyl Acetylenedicarboxylates and a-Keto Lactones Unexpected Participation of an Ester Carbonyl Group in the Isocyanide-Based Three-Component Reaction A A Esmaeili H Vesalipoor
1639 An Efficient and Chemoselective Synthesis of 16-Naphthyridines and Pyrano[32-c]pyridines under Microwave Irradiation Z-G Han S-J Tu B Jiang S Yan X-H Zhang S-S Wu W-J Hao X-D Cao F Shi G Zhang N Ma
1647 N-Activation of N-Arylimidazoles Facile Syntheses of N-Alkyl-N-arylimidazolium Iodides from Less Expensive Chloro Substrates A M Oertel V Ritleng M J Chetcuti
1651 Synthesis of Polyhalogenated 2-(Phenylamino)pyridines by Thermal Amination Reactions S R Waldvogel A Faust W Barkmann R Froumlhlich O Wolff
1655 Cyanide Ion Promoted Addition of Acylphosphonates to Diethyl Cyanophosphonate Synthesis of Phosphonocyanohydrin O-Phosphates A S Demir A Aybey M Emrullahoglu
1659 Straightforward and Scalable Synthesis of Orthogonally Protected 37-Diazabicyclo[410]heptane H Schramm M Pavlova C Hoenke J Christoffers
1663 Hypervalent Iodine Mediated Oxidation of 12-Diaminobenzimidazole and Its Schiff Bases Efficient Synthesis of 3-Amino-124-benzotriazine and 2-Aryl-124-triazolo[15-a]benzimidazoles A Kumar M Parshad R K Gupta D Kumar
1667 Synthesis of the Reported Protoberberine Gusanlung D P B Wakchaure S Easwar N P Argade
1673 2-(Azidomethyl)arylboronic Acids in the Synthesis of Coumarin-Type Compounds M I Naumov A V Nuchev N S Sitnikov Y B Malysheva A S Shavyrin I P Beletskaya A E Gavryushin S Combes A Y Fedorov
1683 Asymmetric Synthesis of 12-anti-Disubstituted Taurine Derivatives D Enders D Iffland G Raabe
1689 A Novel One-Pot Three-Component Synthesis of 5-Imino-2358-tetrahydropyrazolo[12-a]pyridazin-1-one Derivatives B Qian M-J Fan Y-X Xie L-Y Wu Y Shi Y-M Liang
1694 One-Portion Synthesis of 2-Acetoxy Carbonyl Compounds from Aldehydes by Using an Acetylated Masked Acyl Cyanide H Nemoto T Kawamura K Kitasaki K Yatsuzuka M Kamiya Y Yoshioka
1703 Synthesis of 9-Anthryl Ethers from trans-910-Dihydro-910-dimethoxyanthracene by Acid-Catalyzed Transetherification K S Jang H Y Shin D Y Chi
1708 Efficient Synthesis of Azo Dye Labeled Terpenes Sugars and Steroids Using N-(4-Arylazobenzoyl)-1H-benzotriazoles A R Katritzky S R Tala N E Abo-Dya Z K Abdel-Samii
1715 Tandem CH-ActivationndashImine-Formation Reaction A New Route to Imidazo[21-a]phthalazines A Heim-Riether K R Gipson
1720 A Convenient and Efficient α-Sulfenylation of Carbonyl Compounds E Okragla S Demkowicz J Rachon D Witt
1725 Stereoselective Synthesis of β-Branched Phenylalanine Derivatives via Chelate-Claisen Rearrangement C Quirin U Kazmaier
1732 Catalyst-Free and Base-Free Water-Promoted SNAr Reaction of Heteroaryl Halides with Thiols B Sreedhar P S Reddy M A Reddy
1739 Convenient Methods for Synthesis of C2-Symmetric Diphenyltetrahydrothiophenes M Periasamy G Ramani G P Muthukumaragopal
1744 Highly Diastereoselective Conjugate AdditionndashElimination of Chiral Nickel(II) Glycinate with Activated Allylic Acetates for Asymmetric Synthesis of Glutamic Acid Derivatives J Wang J Shi X Zhang D Lin H Jiang H Liu
1753 Synthesis of 36-Dimethoxybenzene-12-diamine and of 47-Dimethoxy-2-methyl-1H-benzimidazole T Besset C Morin
1757 An Inexpensive Procedure for Reductive Aminations Using Dimethylamineborane on Millimolar and Molar Scale R Ortmann M Schlitzer
1760 Classics in Stereoselective Synthesis Edited by E M Carreira L Kvaerno Reviewed by Rolf Breinbauer
XV Forthcoming Articles
no 11 1761 Transition-Metal-Catalyzed Enantioselective Synthesis of Compounds with
Non-Centrochirality M Ogasawara S Watanabe 1786 One-Pot Synthesis of 3-Acyl-2-(alkylsulfanyl)indoles and 2-(Alkylsulfanyl)-
indole-3-carboxylates from (2-Isocyanophenyl)methyl Ketones or (2-Isocyanophenyl)acetates S Fukamachi H Konishi K Kobayashi
1791 Efficient and Recyclable Phthalocyanine-Based Sensitizers for Photooxygenation Reactions H Xu W-K Chan D K P Ng
1797 A Facile and Practical One-Pot Synthesis of β-Oxo Thioamides from β-Oxo Amides and Isothiocyanates P Huang D Xiang Y Zhou Y Liang T Na D Dong
1801 Microwave-Promoted Solid-Acid-Catalyzed One-Pot Synthesis of Phthalazinones V M Outerbridge S M Landge H Tamaki B Toumlroumlk
1807 Benzylic Brominations with N-Bromosuccinimide in (Trifluoromethyl)-benzene D Suarez G Laval S-M Tu D Jiang C L Robinson R Scott B T Golding
1811 Synthesis of Thioflavanone and Flavanone Derivatives by Cyclization of Chalcones W Konieczny M Konieczny
1815 A New and Expedient Total Synthesis of Ochratoxin A and d5-Ochratoxin A B Gabriele M Attya A Fazio L Di Donna P Plastina G Sindona
1821 Synthesis of Benzopyrrolizidinones by NorrishndashYang Cyclization of 3-(Acylmethyl)-2-alkylisoindol-1-ones J Wu W Zhang C Wang
1829 Reactions of MoritandashBaylisndashHillman Acetates with Huisgen Zwitterions A Novel Strategy for the Synthesis of β-Amino Acid Derivatives A Jose R R Paul R Mohan S C Mathew A T Biju E Suresh V Nair
1834 Peracetylated β-Allyl C-Glycosides of D-Ribofuranose and 2-Deoxy- D-ribofuranose in the Chemical Literature Until Now Mirages in the Literature H Otero Martinez H Reinke D Michalik C Vogel
1841 Core-Tetrasubstituted Naphthalene Diimides by Stille Cross-Coupling Reactions and Characterization of Their Optical and Redox Properties S-L Suraru F Wuumlrthner
1846 A Practical Synthesis of Indole-Based Heterocycles Using an Amidoaluminum-Mediated Strategy R Todd M M Hossain
1851 Synthesis of Fluorinated Pyrrolo[23-b]pyridine and Pyrrolo[23-d]pyrimidine Nucleosides V O Iaroshenko Y Wang D V Sevenard D M Volochnyuk
1858 Recyclization Reactions of 5-Formyl-13-dimethyluracil with Electron-Rich Amino Heterocycles A P Mityuk D M Volochnyuk S V Ryabukhin A S Plaskon A Shivanyuk A A Tolmachev
1865 Facile Synthesis of Fluorinated 1-Desazapurines V O Iaroshenko D V Sevenard D M Volochnyuk Y Wang A Martiloga A O Tolmachev
1876 A Practical Synthesis of 3-Diethoxyphosphoryl-12-pyridazine Derivatives J-C Monbaliu J Marchand-Brynaert
1881 Enantioselective Reduction of Prochiral Ketones Employing Sprouted Pisum sativa as Biocatalyst J S Yadav B V S Reddy C Sreelakshmi A B Rao
1886 Application of Phenolate Ion Mediated Intramolecular Epoxide Ring Opening in the Enantioselective Synthesis of Functionalized 23-Dihydrobenzofurans and 1-Benzopyrans S K Dinda S K Das G Panda
1897 Complementary Synthetic Approaches to Constitutionally Diverse N-Aminoalkylated Isoindolinones Application to the Synthesis of Falipamil and 5-HT1A Receptor Ligand Analogues M Lorion A Couture E Deniau P Grandclaudon
1904 Selective Deprotection of Silyl Ethers with Sodium Periodate J Li D Menche
1909 Micellar Solution of Sodium Dodecyl Sulfate (SDS) Catalyzes KabacknikndashFields Reaction in Aqueous Media S Sobhani A Vafaee
1916 Convenient Methods for the Synthesis of a Library of Hemilabile Phosphines M V Jimeacutenez J J Peacuterez-Torrente M I Bartolomeacute L A Oro
1923 Terminal Aziridines by Addition of Grignard Reagents or Organoceriums to an (α-Chloro)sulfinylimine D M Hodgson J Kloesges B Evans
1933 A Robust Synthesis of Nε-(Carboxymethyl)-L-lysine (CML) R Csuk S Stark A Barthel R Kluge D Stroumlhl
1935 One-Pot Curtius Rearrangement Processes from Carboxylic Acids O Leogane H Lebel
XV Forthcoming Articles
no 12 1941 The Chemistry of Deprotonated α-Aminonitriles T Opatz 1960 An Efficient Synthesis of Tetraalkyl 2345-Thiophenetetracarboxylate
Derivatives A Alizadeh R Hosseinpour 1963 Facile Deprotection of Bulky (Trialkylsilyl)acetylenes with Silver Fluoride
S Kim B Kim J In 1969 Highly Efficient and Reusable Ionic Liquids for the Catalyzed
Hydroamination of Alkenes with Sulfonamides Carbamates and Carboxamides L Yang L-W Xu C-G Xia
1975 Synthesis of 2391016172324-Octasubstituted Phthalocyaninatozinc(II) Complexes Mediated by Reductive Agents G A Gauna A C Monsalvo J Awruch
1979 A Short and Efficient Synthesis of 3-2-[2-(Bromomethyl)thiazol-4-yl]-ethynyl-5-fluorobenzonitrile A Precursor for PET Radioligand [18F]SP203 M B Gopinathan C Jin K S Rehder
1983 Synthesis of a Substituted Benzazepin-2-one Dihydrate S K Boini R K Vaid K P Moder D Mitchell
1987 Synthesis of Novel Trisubstituted Imidazolines F J Lakner M A Parker B Rogovoy A Khvat A Ivachtchenko
1991 A Novel Synthesis of N-But-3-enyl-α- and β-Amino Acids T T Van Nguyen R T C Brownlee A B Hughes
1999 Synthesis of Substituted 5-(3-Hydroxypropyl)pyrrolidin-2-ones and Pyrrolizidinones from Nitroethane via C3 Functionalized 56-Dihydro-4H-12-oxazines A Novel Approach to Some Analogues of the Antidepressant Rolipram A Yu Sukhorukov A V Lesiv Y A Khomutova S L Ioffe V A Tartakovsky
2009 Chiral Cyclobutanols and Cyclopentane Dimers via Samarium(II) Iodide Induced Keto-Olefin Cyclisations of Carbohydrate-Derived Unsaturated Ketones D B G Williams J Caddy K Blann J J C Groveacute C W Holzapfel
2015 Synthesis of Perfluoroalkylthio-Substituted Ferrocenes C Rhode J Lemke M Lieb N Metzler-Nolte
2019 Functionalization of Polyhedral Oligomeric Silsesquioxane (POSS) via Nucleophilic Substitution M Dutkiewicz H Maciejewski B Marciniec
2025 A Novel Synthesis of Aryl Mesylates via One-Pot DemethylationndashMesylation of Aryl Methyl Ethers Using a Mixture of Phosphorus Pentoxide in Methanesulfonic Acid B Kaboudin Y Abedi
2029 Anionic Cyclization of (NN-Dimethylamino)[2-(prop-2-yn-1-yloxy)aryl]-acetonitriles T Zdrojewski J Musielak A Jończyk
2035 Strecker-Type Reaction Catalyzed by Carboxylic Acids in Aqueous Media Z Xie G Li G Zhao J Wang
2040 Synthesis of Novel Structurally Simplified Estrogen Analogues with Electron-Donating Groups in Ring A L F Tietze C A Vock I K Krimmelbein L Nacke
2061 On the Resolution of Secondary Phosphine Oxides via Diastereomeric Complex Formation The Case of tert-Butylphenylphosphine Oxide J Holt A M Maj E P Schudde K M Pietrusiewicz L Sieroń W Wieczorek T Jerphagnon I W C E Arends U Hanefeld A J Minnaard
2066 Enantioselective Copper-Catalyzed Conjugate Addition of Dimethylzinc to 5-(1-Arylalkylidene) Meldrumrsquos Acids A Wilsily T Lou E Fillion
2073 SuzukindashMiyaura Coupling Reactions Using Phosphite Ligands M Jang Y Jo I-K Oh H M Jung S Lee
2076 Synthesis of 2-Methylindoline- and 2-Methyl-1234-tetrahydroquinoline-Derived Phosphoramidites and Their Applications in Iridium-Catalyzed Allylic Alkylation of Indoles W-B Liu H He L-X Dai S-L You
2083 Stereocontrolled Synthesis of 13-Amino Alcohols by Reduction of Substituted 2-1-[(tert-Butylsulfinyl)amino]alkylcyclohexanones J C Gonzaacutelez-Goacutemez F Foubelo M Yus
2089 Tunable Phosphoramidite Ligands for Asymmetric Hydrovinylation Ligands par excellence for Generation of All-Carbon Quaternary Centers C R Smith H J Lim A ZhangT V RajanBabu
2101 Copper-Catalyzed Asymmetric Ring-Opening Reaction of Oxabenzonorbornadienes with Grignard and Aluminum Reagents R Millet L Gremaud T Bernardez L Palais A Alexakis
2113 A Simplified Synthesis of Takemotorsquos Catalyst A Berkessel B Seelig 2116 Pharmaceutical Substances Syntheses Patents and Applications of the
Most Relevant AIPs Edited by Axel Kleeman Juumlrgen Engel Bernhard Kutscher Dietmar Reichert Reviewed by I Agranat
XV Forthcoming Articles
no 13 2117 Recent Advances in the Aza-Claisen Rearrangement K C Majumdar
T Bhattacharyya B Chattopadhyay B Sinha 2143 A Novel and Convenient Synthesis of lsquoReversedrsquo Diamidino 25-Aryl- and
25-Azaheterocycle-Substituted Furans L Hu D W Boykin 2146 Efficient and General Preparation of Pyranostilbenes First Total Synthesis
of Artocarbene and Pawhuskin B B H Park Y R Lee W S Lyoo 2155 Mild Oxidation of Diarylacetylenes to 12-Diketones Using Oxone in
Trifluoroacetic Acid J-H Chu Y-J Chen M-J Wu 2163 One-Pot Microwave-Assisted Selective Azido ReductionTandem Cyclization
in Condensed and Solid Phase with Nickel Boride N Shankaraiah N Markandeya M Espinoza-Moraga C Arancibia A Kamal L Silva Santos
2171 Pyrrolo[321-ij]quinolin-4-one and Pyrrolo[321-ij]quinolin-6-one H McNab D J Nelson E J Rozgowska
2175 Practical Synthesis of 5-Substituted Tetrazoles under Microwave Irradiation J Roh T V Artamonova K Vaacutevrovaacute G I Koldobskii A Hrabaacutelek
2179 A Simple Method for the Synthesis of 3-Arylthieno[23-b]pyridines via Iodine-Mediated Cyclization of 3-(1-Arylalkenyl)-2-[(1-phenylethyl)sulfanyl]pyridines K Kobayashi D Nakamura Y Shiroyama S Fukamachi H Konishi
2184 Synthesis of Four Lysine-Linked Cereulide Analogues Showing Ionophoric Activity Towards Potassium Cations as Lead Compounds for Emetic Toxin-Detection by Immunoassays A Makarasen T Nishikawa M Isobe
2205 Synthesis of α-Aliphatic and β-Aromatic Substituted Taurines via Regioselective Ring Opening of Thiiranes with Ammonia H Yu S Cao L Zhang G Liu J Xu
2210 Stability of 5(6)-Carboxyfluorescein in Microwave-Assisted Synthesis of Fluorescein-Labelled O-Dimannosylated Peptides R Kowalczyk P W R Harris R P Dunbar M A Brimble
2223 Diversity-Oriented Synthesis of Functionalized Diaryl Sulfones by Regioselective [3+3] Cyclizations of 13-Bis(siloxy)buta-13-dienes with 2-(Arylsulfonyl)-3-ethoxy-2-en-1-ones Scope and Limitations M Shkoor A Riahi O Fatunsin H Reinke C Fischer P Langer
2236 Synthesis of Functionalized Salicylates by Formal [3+3] Cyclocondensation of 13-Bis(silyloxy)buta-13-dienes with 3-Alkoxy-2-en-1-ones G Mroszlig S Ladzik H Reinke A Spannenberg C Fischer P Langer
2249 Synthetic Approach to Alkoxy-β-(trifluoromethyl)styrenes and Their Application in the Synthesis of New Trifluoromethylated Heterocycles V M Muzalevskiy V G Nenajdenko A V Shastin E S Balenkova G Haufe
2260 o-Benzenedisulfonimide as a Powerful and Recyclable Organocatalyst for the Nazarov Reaction M Barbero S Cadamuro A Deagostino S Dughera P Larini E G Occhiato C Prandi S Tabasso R Vulcano P Venturello
2267 The Catalytic Potential of 4-Guanidinylpyridines in Acylation Reactions I Held E Larionov C Bozler F Wagner H Zipse
2278 Iron(III) Chloride in EthanolndashWater Highly Efficient Catalytic System for the Synthesis of Garcia Gonzalez Polyhydroxyalkyl- and C-Glycosylfurans L Nagarapu M V Chary A Satyender B Supriya R Bantu
2283 Ruthenium-Catalyzed Addition of Primary Amides to Alkynes A Stereoselective Synthesis of Secondary Enamides L J Gooszligen M Blanchot K S M Salih K Gooszligen
2289 Binaphthyl-Modified Quaternary Phosphonium Salts as Chiral Phase Transfer Catalysts Application to Asymmetric Amination of β-Keto Esters R He K Maruoka
X Table of Contents XI Forthcoming Articles
no 14 2293 Direct Methods for Stereoselective Polypropionate Synthesis A Survey
J Li D Menche 2316 Synthesis of Symmetrical Ketones from Grignard Reagents and
11-Carbonyldiimidazole D Bottalico V Fiandanese G Marchese A Punzi
2319 Synthesis of 45-Substituted Imidazoles by a Fast Condensation of 12-Diketones and Urotropine in Heterogeneous Medium G Bratulescu
2321 (Arylsulfonyl)acetones and -acetonitriles New Activated Methylenic Building Blocks for Synthesis of 123-Triazoles N T Pokhodylo V S Matiychuk M D Obushak
2324 A Safe Convenient and Efficient One-Pot Synthesis of α-Chloroketone Acetals Directly from Ketones Using Iodobenzene Dichloride J Yu C Zhang
2329 An Efficient Oxidative Conversion of Aldehydes into 2-Substituted 2-Oxazolines Using 13-Diiodo-55-dimethylhydantoin S Takahashi H Togo
2333 A Novel Procedure for the Synthesis of Benzo[b][18]naphthyridine-3-carboxylate Derivatives from MoritandashBaylisndashHillman Adduct Acetates W Zhong F Lin R Chen W Su
2341 An Improved Synthesis of 147-Triazacyclononanes (tacns) and 14710-Tetraazacyclododecanes (cyclens) J Huang Z Zhou T H Chan
2345 The Ullmann Coupling between 2-Chlorobenzoic Acids and Amino Acids A Valuable Reaction for Preparing 2-Substituted 1-Acetyl-1H-indol-3-yl Acetates J C Rodriguez Dominguez X Gang G Kirsch
2349 gem-Dibromomethyl Aromatics Efficient Aldehyde Equivalents in the KnoevenagelndashDoebner Reaction J K Augustine Y A Naik S Poojari N Chowdappa B S Sherigara K Areppa
2357 Synthesis of Novel α-Aminophosphonates Containing Adamantyl Fragment M M Kabachnik L I Minaeva I P Beletskaya
2361 Efficient Fluoride-Mediated Synthesis of 5-Amino-Substituted Isothiazoles Y S Zubenko V I Potkin
2365 Phosphine-Catalyzed Reaction of Cyanohydrins with Activated Alkynes A Siby O Loreau F Taran
2371 Sulfanyl-Substituted [3]Cumulenes and Buta-13-dienes from a Tetrakis(pyridinium)-Substituted Butadiene A Schmidt A Rahimi M Gjikaj
2379 Efficient Synthesis of 2-Substituted Pyrido[32-d]pyrimidines Involving SNAr and Palladium-Catalyzed Cross-Coupling Reactions A Tikad S Routier M Akssira J-M Leacuteger C Jarry G Guillaumet
2385 Novel Synthesis of Medium-Sized Heterocycles by Palladium-Catalyzed Intramolecular Heck Reaction via 9-endo-trig Mode of Cyclization K C Majumdar B Chattopadhyay
2393 Facile Synthesis of Fluorinated Benzofuro- and Benzothieno[23-b]pyridines α-Carbolines and Nucleosides Containing the α-Carboline Framework V O Iaroshenko Y Wang B Zhang D Volochnyuk V Ya Sosnovskikh
2403 Synthesis of Functionalized N-Vinyl Nitrogen-Containing Heterocycles S M M Lopes A M Beja M Ramos Silva J A Paixatildeo F Palacios T M V D Pinho e Melo
2408 Kumada Cross-Coupling of Aryl Grignard Reagents with Aryl Halides Catalyzed by an Immobilized Nickel Catalyst X Chen L Wang J Liu
2413 Highly Enantioselective Synthesis of Heteroaromatic Alcohols Catalyzed by Chiral DiaminodiphosphinendashRuthenium(II) Complexes W-Y Shen Y-Y Li Z-R Dong J-X Gao
2418 Concise Total Synthesis of (+)-Disparlure and its trans-Isomer Using Asymmetric Organocatalysis S-G Kim
2423 Rhodium Carbenoid Induced [12]-Migration in an L-Lyxo-Configured α-Diazo β-Keto Ester Synthesis of a New Griseolic Acid Analogue N N Bhujbal K S A Kumar D D Dhavale
2430 Synthesis of 5-Arylthio-3-hydroxyphthalates by the First [4+2] Cycloadditions of 3-Arylthio-1-silyloxy-13-butadienes with Dimethyl Acetylenedicarboxylate I Iqbal M Imran P Langer
2435 Synthesis of Highly Functionalized Proline Derivatives via a One-Pot MichaelSN-AdditionCyclization Approach U Kazmaier C Schmidt
2440 RhodiumGraphite-Catalyzed Hydrogenation of Carbocyclic and Heterocyclic Aromatic Compounds G Falini A Gualandi D Savoia
2447 Potassium [1-(tert-Butoxycarbonyl)-1H-indol-2-yl]trifluoroborate as an Efficient Building Block in Palladium-Catalyzed SuzukindashMiyaura Cross Couplings P Kassis V Beacuteneacuteteau J-Y Meacuterour S Routier
2454 Syntheses of Substituted Furans and Pyrroles by Platinum-Catalyzed Cyclizations of Propargylic Oxiranes and Aziridines in Aqueous Media M Yoshida M Al-Amin K Shishido
2467 Transition-Metal-Free Oxidative Homocoupling of Aryl Alkenyl and Alkynyl Grignard Reagents with TEMPO M S Maji A Studer
XIII Forthcoming Articles
no 15 2471 Advances in Synthetic Approaches for the Preparation of Combretastatin-
Based Anti-Cancer Agents R Singh H Kaur 2492 Synthesis of Unsymmetrical Ureas by Sulfur-Assisted Carbonylation with
Carbon Monoxide and Oxidation with Molecular Oxygen under Mild Conditions T Mizuno T Nakai M Mihara
2497 Ring-OpeningRecyclization Reactions of (Dimethylamino)propenoyl-Substituted Cyclopropanes Facile Synthesis of Halogenated Pyridin-2(1H)-ones R Zhang Y Zhou Y Liang Z Jiang D Dong
2501 Facile and Efficient Total Synthesis of Taspine B Cheng S Zhang L Zhu J Zhang Q Li A Shan L He
2505 Oligomeric Iodosylbenzene Sulfate A Convenient Hypervalent Iodine Reagent for Oxidation of Organic Sulfides and Alkenes M S Yusubov R Y Yusubova T V Funk K-W Chi V V Zhdankin
2509 Pyrrolidine-Based Organocatalysts for Enantioselective Michael Addition of Cyclohexanone to trans-β-Nitrostyrene A P Carley S Dixon J D Kilburn
2517 CundashAl Hydrotalcite An Efficient and Reusable Ligand-Free Catalyst for the Coupling of Aryl Chlorides with Aliphatic Aromatic and N(H)-Heterocyclic Amines B Sreedhar R Arundhathi P L Reddy M A Reddy M L Kantam
2523 Highly Efficient Synthesis of trans-βγ-Unsaturated a-Keto Amides C Allais T Constantieux J Rodriguez
2531 Gas-Phase Synthesis of N-Unsubstituted 3-Hydroxypyrroles and 1H-Pyrrol-3(2H)-ones L Hill G A Hunter S H Imam H McNab W J OrsquoNeill
2535 3-Hydroxy-1H-pyrrole L Hill S H Imam H McNab W J OrsquoNeill 2539 123-Thiadiazoles with Unsaturated Side Chains Synthesis
Polymerization and Photocrosslinking M Al-Smadi N Hanold H Kalbitz H Meier
2547 Synthesis of 1112-Didehydrodibenzo[ae]cycloocten-5(6H)-one A Strained Eight-Membered Alkyne S C Kornmayer F Rominger R Gleiter
2553 Stannous Chloride Dihydrate A Novel and Efficient Catalyst for the Synthesis of gem-Dihydroperoxides from Ketones and Aldehydes D Azarifar K Khosravi F Soleimanei
2557 Synthesis of a Novel Class of Azacrown Macrocycles and Lariat Crown Ethers Containing Two 124-Triazole Rings as Subunits N Foroughifar A Mobinikhaledi S Ebrahimi
2561 Enantioselective Synthesis of the 3C-Protease Inhibitor (ndash)-Thysanone by a StauntonndashWeinreb Annulation Strategy J Sperry T Y Yuen M A Brimble
2570 Stereoselective Synthesis of Unnatural β-Amino Acids from Nitroethane via 56-Dihydro-4H-12-oxazin-3-ylacetates A Yu Sukhorukov A V Lesiv O L Eliseev Y A Khomutova S L Ioffe
2579 A Versatile Unexpected One-Pot Regioselective Synthesis of a New Class of 13-Diazepinoindolones by Reaction of Pyranoindolones with Monosubstituted Ureas D Livadiotou C A Tsoleridis J Stephanidou-Stephanatou
2584 Synthesis of a Trisaccharide and a Tetrasaccharide from the Cell-Wall Lipopolysaccharides of Azospirillum brasilense S17 S Pandey S Ghosh A K Misra
2591 Synthesis of Isoindoline Nitroxides by Electrocyclic Reactions T Kaacutelai J Jekı K Hideg
2596 Glycosylations of Tertiary Alcohols Synthesis of Fully Protected Disaccharides with Sterically Demanding Groups Attached to the Sugar Core A Holkenbrink J B Vicente D B Werz
2605 Copper-Catalyzed [13]-Dipolar Cycloaddition for the Synthesis of Macrocycles Containing Acyclic Aromatic and Steroidal Moieties G V Latyshev M S Baranom A V Kazantsev A D Averin N V Lukashev I P Beletskaya
2616 Aryl Ring Migration Reaction in the Synthesis of 24-Diaryl-4H-31-benzothiazines A V Butin F A Tsiunchik V T Abaev A V Gutnov D A Cheshkov
2627 Hydrogenation of β-N-Substituted and β-NN-Disubstituted Enamino Esters in the Presence of Iridium(I) Catalyst H Hebbache Z Hank C Bruneau J-L Renaud
2634 Stereoselective Olefination Reactions Promoted by Rieke Manganese J M Concelloacuten H Rodriacuteguez-Solla V del Amo P Diacuteaz
2646 Synthesis of Piperidinones through a Radical Cascade E Godineau Y Landais
2650 Asymmetric Organic Synthesis with Enzymes Edited by V Gotor I Alfonso E Garciacutea-Urdiales Reviewed by Steve Collier
XVII Forthcoming Articles
no 16 2651 Synthesis of Spirocyclic Ethers S Rosenberg R Leino 2674 Bimetallic PalladiumndashPlatinum-on-Carbon-Catalyzed HndashD Exchange
Reaction Synergistic Effect on Multiple Deuterium Incorporation T Maegawa N Ito K Oono Y Monguchi H Sajiki
2679 Efficient Copper-Catalyzed Synthesis of 2-Amino-4(3H)-quinazolinone and 2-Aminoquinazoline Derivatives X Huang H Yang H Fu R Qiao Y Zhao
2689 Synthesis and Chemoselective N- and O-Alkylation of Thiadiazolopyrimidine Nucleosides and Uridines A M L Hossion R Islam R K Kandahary T Nagamatsu
2697 Facile and Efficient Synthesis of a New Class of Indole-Substituted Pyridine Derivatives via One-Pot Multicomponent Reactions K Zhao X-P Xu S-L Zhu D-Q Shi Y Zhang S-J Ji
2709 Studies toward a Total Synthesis of Rhizoxin D Stereoselective Preparation of the C11ndashC19 Fragment S Padakanti C K Kumar E Ashok P Das
2715 A Short Synthesis of Enantiomeric Phytoprostanes B1 Type I W Perlikowska M Mikołajczyk
2719 Chemistry of Polyhalogenated Nitrobutadienes Part 7 A Novel Synthetic Access to Chlorinated Nitrile Oxides E Nutz V A Zapolrsquoskii D E Kaufmann
2725 Microwave-Assisted Silver(I)-Mediated Selective O-Alkylation of Aromatic Imidate Systems B K Singh C Cavalluzzo M De Maeyer Z Debyser V S Parmar E Van der Eycken
2729 Iodogen A Novel Reagent for the Oxidation of Urazoles under Heterogeneous Conditions A Khoramabadi A Shiri M A Zolfigol S Mallakpour
2733 An Unprecedented Synthesis of Eight-Membered-Ring Cyclic Thioimidic Esters by a Three-Component Reaction A Alizadeh R Hosseinpour
2737 A Novel Diastereoselective Synthesis of β-Phosphonato Unsaturated Thioimidates A Alizadeh N Zohreh
2741 Synthesis of 21-Benzisoxazoles by Nucleophilic Substitution of Hydrogen in Nitroarenes Activated by the Azole Ring N T Pokhodylo Y O Teslenko V S Matiychuk M D Obushak
2749 A Facile Synthesis of Two Series of Multifunctional Carbon Compounds from αα-Dihalo Ketones Using Allylsamarium Bromide X Liu S Zhang J Di
2756 Stereocontrolled Formation of Protected Aminodeoxyalditols from Simple Carbohydrate Precursors by Debenzylating Cycloetherification Y Jiang Z Fang Q Zheng H Jia J Cheng B Zheng
2761 trans-Stilbene as a Starting Material for the Synthesis of Tamoxifen Based on Palladium-Catalyzed Cross-Coupling Reactions C M Nunes J Limberger S Poersch M Seferin A L Monteiro
2766 Synthesis and Biological Evaluation of 6-Substituted Purinylcarbanucleosides with a Cyclopenta[b]thiophene Pseudosugar P Abeijoacuten J M Blanco O Caamantildeo F Fernaacutendez M D Garciacutea X Garciacutea-Mera J E Rodriacuteguez-Borges J Balzarini E De Clercq
2773 Synthesis and Electrochemical Signature of Novel Norbornyl-ferrocene Hybrids F A Khan S K Upadhyay
2778 A Regioselective TsujindashTrost Pentadienylation of 3-Allyltetronic Acid R Schobert B Barnickel
2785 Copper(I)-Catalyzed CarylndashCalkynyl Bond Formation of Aryl Iodides with Terminal Alkynes K G Thakur G Sekar
2790 Aminolysis of Epoxides Using Iridium Trichloride as an Efficient Catalyst J Agarwal A Duley R Rani R K Peddinti
2797 Preparation of Several Active N-Chloro Compounds from Trichloroisocyanuric Acid A Shiri A Khoramabadi-zad
2802 The First Mineral-Catalyzed One-Pot [3+1+2] Coupling Protocol for Multifunctionalized Fused-Ring Pyrimidines L D S Yadav A Rai
2809 Efficient Synthesis of Tetrahydro-β-carbolin-1-one and Dihydroisoquinolin-1-one Derivatives as Versatile Intermediates K E Judd M F Mahon L Caggiano
2818 A Concise Synthesis of ortho-Iodobenzyl Alcohols via Addition of ortho-Iodophenyl Grignard Reagent to Aldehydes and Ketones J Cvengroš D Stolz A Togni
XIII Forthcoming Articles
no 17 2825 Reactivity of Oxazol-5-(4H)-ones and Their Application toward Natural
Product Synthesis N M Hewlett C D Hupp J J Tepe 2840 Towards the Total Synthesis of 3-Hydroxyvibsanin E B D Schwartz
J R Denton P V Bernhardt H M L Davies C M Williams 2847 Structure Investigations of (ent)-Cladospolide D by De Novo Synthesis and
Kinetic and Thermodynamic Isomerization Y Xing J H Penn G A OrsquoDoherty
2855 New Applications of PhI(OAc)2 in Synthesis Total Synthesis and SAR Development of Potent Antitumor Natural Product PsymberinIrciniastatin A N Shao X Huang A Palani R Aslanian A Buevich J Piwinski R Huryk C Seidel-Dugan
2873 Total Synthesis of Largazole ndash Devolution of a Novel Synthetic Strategy B Wang C J Forsyth
2881 Formal Total Synthesis of Palmerolide A J Jaumlgel M E Maier 2893 Total Synthesis of Bongkrekic Acid via Sequential SuzukindashMiyaura Coupling
Reactions M Kanematsu M Shindo M Yoshida K Shishido 2905 Stereodivergent Approach to Both C28a-syn and C28a-anti Relative
Stereochemical Manifolds in the Lepadin Family via a TiCl4-Promoted G Li L J Carlson I K Sagamanova B W Slafer R P Hsung C Gilardi H M Sklenicka N Sydorenko
2915 Enantioselective Aldol Reaction of Tetrasubstituted Ketene Silyl Acetals with Achiral Aldehydes for the Construction of Asymmetric Tertiary Alcohols An Application for the Divergent Total Syntheses of Buergerinins F and G I Shiina T Iizumi Y-s Yamai Y-i Kawakita K Yokoyama Y-k Yamada
2927 Second-Generation Biomimetic Total Synthesis of Chaetominine A Coste G Karthikeyan F Couty G Evano
2935 Total Synthesis of (+)-Fostriecin and (+)-Phoslactomycin B S Shibahara M Fujino Y Tashiro N Okamoto T Esumi K Takahashi J Ishihara S Hatakeyama
2954 Stereochemical Assignments of the Chlorinated Residues in Victorin C A C Durow C Butts C L Willis
2963 Studies of the Asymmetric Total Synthesis of Clavilactone D by the lsquoLariatrsquo Cyclization Strategy T Yoshimitsu S Nojima M Hashimoto K Tsukamoto T Tanaka
2970 Total Synthesis of the Leucetta-Derived Alkaloid Calcaridine A P B Koswatta R Sivappa H V R Dias C J Lovely
2983 Formal Synthesis of Salinosporamide A Starting from D-Glucose T Momose Y Kaiya J-i Hasegawa T Sato N Chida
2992 Synthesis of Bioactive Natural Products by Asymmetric syn- and anti-Aldol Reactions A K Ghosh Z L Dawson
no 18 3003 Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural
Products B M Trost M K Brennan 3026 One-Pot Synthesis of Furo[34-b]pyridin-5(7H)-ones from 2-
Bromopyridine-3-carboxylic Acid and Carbonyl Compounds K Kobayashi T Kozuki H Konishi
3029 Iodocyclization of N-[2-(Methylthio)phenyl]propiolamides Selective Synthesis of 3-Iodo-15-benzothiazepin-4-ones T-S Jiang X-G Zhang J-H Li
3039 A Facile Synthetic Method for Fluorine-Containing 17-Phenanthrolines Pyridine-Ring Formation Reaction of N-Propargyl-68-bis(trifluoroacetyl)-quinolin-5-amine with Various Nucleophiles D Shibata E Okada M Hinoshita M Meacutedebielle
3047 Enantiotopic Discrimination in Palladium-Mediated Nucleophilic Substitutions on Achiral Substrates Chiral Ligand versus Chiral Nucleophile O Jacquet F Charnay J-C Fiaud J Ollivier
3051 Studies on the Chemistry of 2-[3-(2-Nitrophenyl)-2-oxopropyl]benzaldehydes Novel Syntheses of 5H-Benzo[b]carbazole-611-diones and Indolo[12-b]isoquinoline-611-diones M Fernaacutendez
3061 Studies on the C22ndashC23 Aldol Coupling of Spirangien M Lorenz N Bluhm M Kalesse
3067 One-Pot Synthesis of N-Alkyl Purine Pyrimidine and Azole Derivatives from Alcohols using Ph3PCCl4 A Rapid Route to Carboacyclic Nucleoside Synthesis M N Soltani Rad A Khalafi-Nezhad S Behrouz Z Asrari M Behrouz Z Amini
3077 Synthesis of 2-Amino-34-dihydroquinazolines and Imidazo[21-b]quinazoline-2-ones A Mishra S Batra
3089 Studies on the Reaction of Diimines with Thiourea Synthesis and Solvent-Induced cistrans-Isomerization of 135-Triazinane-2-thiones B Kaboudin T Ghasemi T Yokomatsu
3094 Suzuki Coupling of Heteroaromatic Chlorides Using Highly Electron-Donating ClickPhos Ligands S M Spinella Z-H Guan J Chen X Zhang
3099 Reaction of NN-Dioxyenamines with Anhydrides of Carboxylic and Sulfonic Acids A New Method for the Synthesis of a-Hydroxyoxime Derivatives A A Tabolin A V Lesiv S L Ioffe
3106 Directed ortho Metallation Chemistry and Phosphine Synthesis New Ligands for the SuzukindashMiyaura Reaction D B G Williams S J Evans H de Bod M S Mokhadinyana T Hughes
3113 New Functional Derivatives of 9-Phenylquinine P J Boratyński J SkarŜewski
3120 On the Synthesis of Asymmetric and Dissymmetric Amino Analogues of Troumlgerrsquos Base J Artacho K Waumlrnmark
3127 Synthesis of Polycyclic Sultams by Palladium-Catalyzed Intramolecular Cyclization K C Majumdar S Mondal N De
3136 Synthesis of Functionalized L-Cysteine and L-Methionine by Reaction with Electron-Deficient Acetylenes B A Trofimov A G Malrsquokina O A Shemyakina V V Nosyreva A P Borisova S S Khutsishvili L B Krivdin
3143 A lsquoClickrsquo Approach to the Synthesis of 3-[2-(1-Alkyltriazol-4-yl)ethyl]indoles M Petrini R R Shaikh
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
1175 The First Total Synthesis of Kynapcin-24 by Palladium Catalysis L-Y Yang C-F Chang Y-C Huang Y-J Lee C-C Hu T-H Tseng
1180 Enantioselective Synthesis of N-Protected α-Amino Acid Hydrazides M Bibian S El-Habnouni J Martinez J-A Fehrentz
1185 Synthesis of 11H-Indolo[32-c]quinoline-6-carboxylic Acids by Cascade AutoxidationndashRing Contractions A Becker S Kohfeld T Pies K Wieking L Preu C Kunick
1190 Reaction of N-Nonaflylbenzotriazole with Silyl Enol Ethers M Uhde T Ziegler
1195 2-(Benzoylimino)thiazolidin-4-ones Formation by an Alternative Ring Closure and Analysis of Rotational Barriers H-G Haumlcker P W Elsinghorst S Michels J Daniels G Schnakenburg M Guumltschow
1204 Microwave-Assisted Synthesis and Functionalization of Selenolopyrimidines S Hesse C Chenet D Thomae G Kirsch
1209 12-Disubstituted 4-Quinolones via Copper-Catalyzed Cyclization of 1-(2-Halophenyl)-2-en-3-amin-1-ones R Bernini S Cacchi G Fabrizi A Sferrazza
1220 A New Atom-Economical and Selective Synthesis of Secondary and Tertiary Alkylamines by Means of CpIridium Complex Catalyzed Multiple N-Alkylation of Ammonium Salts with Alcohols without Solvent R Yamaguchi Z Mingwen S Kawagoe C Asai K-i Fujita
1224 Synthesis of Regioisomerically Pure 5-Functionalized 27-Dichlorofluoresceins J C Castro A Malakhov K Burgess
XIII Forthcoming Articles
No 8 1227 Michael Additions to Activated Vinylphosphonates T Janecki J Kędzia
T Wąsek 1255 A Facile and General Synthesis of 2β-Aminosteroids X Ke H Hu
D Zhou W Xu Q Zhu N P Reddy X Hu 1261 Efficacious Preparation of Oppolzerrsquos Glycylsultam via the Deleacutepine
Reaction A Isleyen C Gonsky R C Ronald P Garner 1265 Synthesis of Masked Vicinal Amino Aldehydes of Pyrrolizine and Pyrrolo
[12-c]thiazole Series A V Tverdokhlebov A V Denisenko A A Tolmachev Y M Volovenko S V Shishkina O V Shishkin
1271 Preparation of 9-Substituted Pyridine-Stretched Adenines and Hypoxanthines J A Crawford W Fraser C A Ramsden
1279 A Versatile Synthesis of Heterocyclic Analogues of Neoflavonoids from Enamino Ketones V S Moskvina V P Khilya O V Turov U M Groth
1287 New Stereoselective Synthesis of Paeonilactone B F G Gatti S Serra 1291 The Use of NN-Dialkyltrimethylsilylamines in the Synthesis of
Pentamethinium Salts M Kořiacutenek M Rybaacutečkovaacute Boumlhm 1297 Synthesis of Triazoles via Regioselective Reactions of Aryl Azides with
Cyanoacetyl Pyrroles and Indoles N T Pokhodylo V S Matiychuk M D Obushak
1301 Gallium(III) Chloride Catalyzed Hydroarylation of Arylacetylenes with Naphthols and Phenols A Facile Synthesis of Vinylarenes J S Yadav B V S Reddy S Sengupta S K Biswas
1305 Electrophilic Bromination of meta-Substituted Anilines with N-Bromosuccinimide Regioselectivity and Solvent Effect S Bartoli A Cipollone A Squarcia A Madami D Fattori
1309 Cross-Coupling Reactions of Halopurines with Aryl- and Alkyltrifluoroborates The Scope and Limitations in the Synthesis of Modified Purines Z Hasniacutek R Pohl M Hocek
1318 A Convenient Method for Converting Hydroxyacetophenones into Their Ethylene or Trimethylene Acetals F Ono H Takenaka T Fujikawa M Mori T Sato
1323 γ-Chloromagnesio γ-Lactones and δ-Chloromagnesio δ-Lactones Generation Properties and Synthetic Uses H Shimizu S Fukuda S Sugiyama T Satoh
1336 Click Reactions with Nitroxides T Kaacutelai W L Hubbell K Hideg 1341 Synthesis of Novel 14-Benzoquinone-Containing 123-Triazoles An Entry
Into a New Library F Algi M Balci 1348 Efficient Synthesis of Two Sialylated Tetrasaccharides Found in Goat Milk
P K Mandal A K Misra 1355 Dendrimers of Vaccines Consisting of Tumor-Associated Glycopeptide
Antigens and T Cell Epitope Peptides S Keil A Kaiser F Syed H Kunz
1370 IBXTBAB-Mediated Oxidation of Primary Amines to Nitriles F Drouet P Fontaine G Masson J Zhu
1375 Chemoselectivity of Multicomponent Condensations of Barbituric Acids 5-Aminopyrazoles and Aldehydes E A Muravyova S V Shishkina V I Musatov I V Knyazeva O V Shishkin S M Desenko V A Chebanov
1386 Stereoselective Total Syntheses of Leiocarpin A and (ndash)-Galantinic Acid Starting from D-Mannitol K Nagaiah D Sreenu K V Purnima R S Rao J S Yadav
1393 A Facile Mild Deprotection Protocol for 13-Dithianes and 13-Dithiolanes with 30 Hydrogen Peroxide and Iodine Catalyst in Aqueous Micellar System N C Ganguly S K Barik
1400 Rhodium-Catalyzed Gram-Scale Synthesis of Highly Substituted Pyridine Derivatives K Parthasarathy C-H Cheng
1403 Enantioselective Synthesis of (R)-Propylene Carbonate from Ethyl (S)-Lactate J M Whitaker R C Ronald
XIII Forthcoming Articles
no 9 1405 Transition-Metal-Catalyzed Site-Selective Cross-Coupling of Di- and
Polyhalogenated Compounds J-R Wang K Manabe 1428 An Improved Synthesis of (4-4-Hydroxy-3-isopropyl-5-[(4-nitrophenyl)
ethynyl]benzyl-35-dimethylphenoxy)acetic Acid (NH-3) M B Gopinathan K S Rehder
1431 Copper-Catalyzed Tandem CndashN Bond Formation Reaction Selective Synthesis of 2-(Trifluoromethyl)benzimidazoles M-W Chen X-G Zhang P Zhong M-L Hu
1437 Synthesis and Thermochemical Properties of Stereoisomeric Dihydroxy- and Tetrahydroxyalkylammonium Salts M Thomas L Rothman J Hatcher P Agarkar R Ramkirath S Lall-Ramnarine R Engel
1445 Preparation of 5-Substituted 2-(2-Alkylaryl-1H-imidazol-4-yl)oxazoles and 5-Substituted 2-(2-Alkylarylthiazol-4-yl)oxazoles by Utilizing 5-Substituted 2-(2-Bromo-11-diethoxyethyl)oxazole as a Synthon D R St Laurent J L Romine
1459 Novel and Efficient Methods for the Synthesis of Symmetrical Trisulfides A Kertmen S Lach J Rachon D Witt
1463 An Environmentally Benign Electrochemical Process for the Reduction of Carboxylic Acid Hydrazides to Amides M Mentel M J Beier R Breinbauer
1469 Synthesis of 1-Chloroalkynes from Alkynylsilanes Using Trichloroisocyanuric Acid as Chlorinating Agent M H Vilhelmsen A S Andersson M B Nielsen
1473 A Convenient Approach to Enantioenriched Cyclopropanes Bearing Electron-Withdrawing Functionalities H Krawczyń K Wąsek J Kędzia
1477 Synthesis of Cyclopropenes via 12-Elimination of Bromocyclopropanes Catalyzed by Crown Ether W M Sherrill R Kim M Rubin
1485 A Base-Catalysed One-Pot Three-Component Coupling Reaction Leading to Nitrosubstituted Pyrroles I R Baxendale C D Buckle S V Ley L Tamborini
1494 Synthesis of 4-Alkylidene-4H-31-benzoxazine Derivatives by Acid-Catalyzed Cyclization of 2-Isocyanophenyl Ketones in the Presence of a Vinyl Ether K Kobayashi Y Okamura H Konishi
1499 Synthesis of Higher Helicenes via Olefin Metathesis and CndashH Activation J Cocircteacute S K Collins
1506 Azido- and Ethynyl-Substituted 2262-Terpyridines as Suitable Substrates for Click Reactions A Winter A Wild R Hoogenboom M W M Fijten M D Hager R-A Fallahpour U S Schubert
1513 Synthesis of 2-(Arylamino)ethanethiols via Lewis Acid Catalyzed Aminolysis of 22-Dimethylthiirane as Precursors of the 14-Benzothiazine Nucleus R Spogli S Sabatini G Manfroni O Tabarrini V Cecchetti
1520 Iron(III) Chloride A Versatile Catalyst for the Practical Synthesis of 3-Sulfenylindoles J S Yadav B V S Reddy Y J Reddy K Praneeth
1525 Organocatalytic Enantioselective Conjugate Addition of 2-Fluoromalonate to Nitroolefins Direct Synthesis of Chiral Fluorinated γ-Nitro Carboxylic Acid Derivatives H Li L Zu H Xie W Wang
1531 Asymmetric Transfer Hydrogenation of Ketimines with Trichlorosilane Structural Studies Z Zhang P Rooshenas H Hausmann P R Schreiner
1545 Prolinol Sulfinyl Ester Derivatives Organocatalytic Michael Addition of Ketones to Nitroolefins under Neat Conditions X Zeng G Zhong
1551 Asymmetric Oxidations of Electron-Poor Alkenes Promoted by the β-Amino AlcoholTBHP System A Russo A Lattanzi
1557 Enantioselectivity Switch in Direct Asymmetric Aminoxylation Catalyzed by Binaphthyl-Based Chiral Secondary Amines T Kano A Yamamoto F Shirozu K Maruoka
1564 Enantioselective Conjugate Addition of N-Heterocycles to αβ-Unsaturated Ketones Catalyzed by Chiral Primary Amines G Luo S Zhang W Duan W Wang
1573 Sulfonyl Hydrazine as New Functionality in Organocatalysis Camphorsulfonyl Hydrazine Catalyzed Enantioselective Aza-Michael Addition L-Y Chen H He B-J Pei W-H Chan A W M Lee
1578 Conversion of Primary Alcohols and Aldehydes into Methyl Esters by Ruthenium-Catalysed Hydrogen Transfer Reactions N A Owston T D Nixon A J Parker M K Whittlesey J M J Williams
1582 Addendum and Erratum XVII Forthcoming Articles
no 10 1583 Organocatalytic Formation of Quaternary Stereocenters M Bella
T Gasperi 1615 Regioselective Synthesis of 5H-Thiazolo[32-a]pyrimidin-5-ones from
MoritandashBaylisndashHillman Adduct Acetates under Solvent-Free and Base-Free Conditions W Zhong B Guo F Lin Y Liu W Su
1623 First Synthesis of 5-Cyanosalicylates by Formal [3+3] Cyclocondensations of 13-Bis(silyloxy)-13-butadienes A Riahi O Fatunsin M Shkoor R Dede H Reinke C Fischer P Langer
1635 Reaction of Isocyanides Dialkyl Acetylenedicarboxylates and a-Keto Lactones Unexpected Participation of an Ester Carbonyl Group in the Isocyanide-Based Three-Component Reaction A A Esmaeili H Vesalipoor
1639 An Efficient and Chemoselective Synthesis of 16-Naphthyridines and Pyrano[32-c]pyridines under Microwave Irradiation Z-G Han S-J Tu B Jiang S Yan X-H Zhang S-S Wu W-J Hao X-D Cao F Shi G Zhang N Ma
1647 N-Activation of N-Arylimidazoles Facile Syntheses of N-Alkyl-N-arylimidazolium Iodides from Less Expensive Chloro Substrates A M Oertel V Ritleng M J Chetcuti
1651 Synthesis of Polyhalogenated 2-(Phenylamino)pyridines by Thermal Amination Reactions S R Waldvogel A Faust W Barkmann R Froumlhlich O Wolff
1655 Cyanide Ion Promoted Addition of Acylphosphonates to Diethyl Cyanophosphonate Synthesis of Phosphonocyanohydrin O-Phosphates A S Demir A Aybey M Emrullahoglu
1659 Straightforward and Scalable Synthesis of Orthogonally Protected 37-Diazabicyclo[410]heptane H Schramm M Pavlova C Hoenke J Christoffers
1663 Hypervalent Iodine Mediated Oxidation of 12-Diaminobenzimidazole and Its Schiff Bases Efficient Synthesis of 3-Amino-124-benzotriazine and 2-Aryl-124-triazolo[15-a]benzimidazoles A Kumar M Parshad R K Gupta D Kumar
1667 Synthesis of the Reported Protoberberine Gusanlung D P B Wakchaure S Easwar N P Argade
1673 2-(Azidomethyl)arylboronic Acids in the Synthesis of Coumarin-Type Compounds M I Naumov A V Nuchev N S Sitnikov Y B Malysheva A S Shavyrin I P Beletskaya A E Gavryushin S Combes A Y Fedorov
1683 Asymmetric Synthesis of 12-anti-Disubstituted Taurine Derivatives D Enders D Iffland G Raabe
1689 A Novel One-Pot Three-Component Synthesis of 5-Imino-2358-tetrahydropyrazolo[12-a]pyridazin-1-one Derivatives B Qian M-J Fan Y-X Xie L-Y Wu Y Shi Y-M Liang
1694 One-Portion Synthesis of 2-Acetoxy Carbonyl Compounds from Aldehydes by Using an Acetylated Masked Acyl Cyanide H Nemoto T Kawamura K Kitasaki K Yatsuzuka M Kamiya Y Yoshioka
1703 Synthesis of 9-Anthryl Ethers from trans-910-Dihydro-910-dimethoxyanthracene by Acid-Catalyzed Transetherification K S Jang H Y Shin D Y Chi
1708 Efficient Synthesis of Azo Dye Labeled Terpenes Sugars and Steroids Using N-(4-Arylazobenzoyl)-1H-benzotriazoles A R Katritzky S R Tala N E Abo-Dya Z K Abdel-Samii
1715 Tandem CH-ActivationndashImine-Formation Reaction A New Route to Imidazo[21-a]phthalazines A Heim-Riether K R Gipson
1720 A Convenient and Efficient α-Sulfenylation of Carbonyl Compounds E Okragla S Demkowicz J Rachon D Witt
1725 Stereoselective Synthesis of β-Branched Phenylalanine Derivatives via Chelate-Claisen Rearrangement C Quirin U Kazmaier
1732 Catalyst-Free and Base-Free Water-Promoted SNAr Reaction of Heteroaryl Halides with Thiols B Sreedhar P S Reddy M A Reddy
1739 Convenient Methods for Synthesis of C2-Symmetric Diphenyltetrahydrothiophenes M Periasamy G Ramani G P Muthukumaragopal
1744 Highly Diastereoselective Conjugate AdditionndashElimination of Chiral Nickel(II) Glycinate with Activated Allylic Acetates for Asymmetric Synthesis of Glutamic Acid Derivatives J Wang J Shi X Zhang D Lin H Jiang H Liu
1753 Synthesis of 36-Dimethoxybenzene-12-diamine and of 47-Dimethoxy-2-methyl-1H-benzimidazole T Besset C Morin
1757 An Inexpensive Procedure for Reductive Aminations Using Dimethylamineborane on Millimolar and Molar Scale R Ortmann M Schlitzer
1760 Classics in Stereoselective Synthesis Edited by E M Carreira L Kvaerno Reviewed by Rolf Breinbauer
XV Forthcoming Articles
no 11 1761 Transition-Metal-Catalyzed Enantioselective Synthesis of Compounds with
Non-Centrochirality M Ogasawara S Watanabe 1786 One-Pot Synthesis of 3-Acyl-2-(alkylsulfanyl)indoles and 2-(Alkylsulfanyl)-
indole-3-carboxylates from (2-Isocyanophenyl)methyl Ketones or (2-Isocyanophenyl)acetates S Fukamachi H Konishi K Kobayashi
1791 Efficient and Recyclable Phthalocyanine-Based Sensitizers for Photooxygenation Reactions H Xu W-K Chan D K P Ng
1797 A Facile and Practical One-Pot Synthesis of β-Oxo Thioamides from β-Oxo Amides and Isothiocyanates P Huang D Xiang Y Zhou Y Liang T Na D Dong
1801 Microwave-Promoted Solid-Acid-Catalyzed One-Pot Synthesis of Phthalazinones V M Outerbridge S M Landge H Tamaki B Toumlroumlk
1807 Benzylic Brominations with N-Bromosuccinimide in (Trifluoromethyl)-benzene D Suarez G Laval S-M Tu D Jiang C L Robinson R Scott B T Golding
1811 Synthesis of Thioflavanone and Flavanone Derivatives by Cyclization of Chalcones W Konieczny M Konieczny
1815 A New and Expedient Total Synthesis of Ochratoxin A and d5-Ochratoxin A B Gabriele M Attya A Fazio L Di Donna P Plastina G Sindona
1821 Synthesis of Benzopyrrolizidinones by NorrishndashYang Cyclization of 3-(Acylmethyl)-2-alkylisoindol-1-ones J Wu W Zhang C Wang
1829 Reactions of MoritandashBaylisndashHillman Acetates with Huisgen Zwitterions A Novel Strategy for the Synthesis of β-Amino Acid Derivatives A Jose R R Paul R Mohan S C Mathew A T Biju E Suresh V Nair
1834 Peracetylated β-Allyl C-Glycosides of D-Ribofuranose and 2-Deoxy- D-ribofuranose in the Chemical Literature Until Now Mirages in the Literature H Otero Martinez H Reinke D Michalik C Vogel
1841 Core-Tetrasubstituted Naphthalene Diimides by Stille Cross-Coupling Reactions and Characterization of Their Optical and Redox Properties S-L Suraru F Wuumlrthner
1846 A Practical Synthesis of Indole-Based Heterocycles Using an Amidoaluminum-Mediated Strategy R Todd M M Hossain
1851 Synthesis of Fluorinated Pyrrolo[23-b]pyridine and Pyrrolo[23-d]pyrimidine Nucleosides V O Iaroshenko Y Wang D V Sevenard D M Volochnyuk
1858 Recyclization Reactions of 5-Formyl-13-dimethyluracil with Electron-Rich Amino Heterocycles A P Mityuk D M Volochnyuk S V Ryabukhin A S Plaskon A Shivanyuk A A Tolmachev
1865 Facile Synthesis of Fluorinated 1-Desazapurines V O Iaroshenko D V Sevenard D M Volochnyuk Y Wang A Martiloga A O Tolmachev
1876 A Practical Synthesis of 3-Diethoxyphosphoryl-12-pyridazine Derivatives J-C Monbaliu J Marchand-Brynaert
1881 Enantioselective Reduction of Prochiral Ketones Employing Sprouted Pisum sativa as Biocatalyst J S Yadav B V S Reddy C Sreelakshmi A B Rao
1886 Application of Phenolate Ion Mediated Intramolecular Epoxide Ring Opening in the Enantioselective Synthesis of Functionalized 23-Dihydrobenzofurans and 1-Benzopyrans S K Dinda S K Das G Panda
1897 Complementary Synthetic Approaches to Constitutionally Diverse N-Aminoalkylated Isoindolinones Application to the Synthesis of Falipamil and 5-HT1A Receptor Ligand Analogues M Lorion A Couture E Deniau P Grandclaudon
1904 Selective Deprotection of Silyl Ethers with Sodium Periodate J Li D Menche
1909 Micellar Solution of Sodium Dodecyl Sulfate (SDS) Catalyzes KabacknikndashFields Reaction in Aqueous Media S Sobhani A Vafaee
1916 Convenient Methods for the Synthesis of a Library of Hemilabile Phosphines M V Jimeacutenez J J Peacuterez-Torrente M I Bartolomeacute L A Oro
1923 Terminal Aziridines by Addition of Grignard Reagents or Organoceriums to an (α-Chloro)sulfinylimine D M Hodgson J Kloesges B Evans
1933 A Robust Synthesis of Nε-(Carboxymethyl)-L-lysine (CML) R Csuk S Stark A Barthel R Kluge D Stroumlhl
1935 One-Pot Curtius Rearrangement Processes from Carboxylic Acids O Leogane H Lebel
XV Forthcoming Articles
no 12 1941 The Chemistry of Deprotonated α-Aminonitriles T Opatz 1960 An Efficient Synthesis of Tetraalkyl 2345-Thiophenetetracarboxylate
Derivatives A Alizadeh R Hosseinpour 1963 Facile Deprotection of Bulky (Trialkylsilyl)acetylenes with Silver Fluoride
S Kim B Kim J In 1969 Highly Efficient and Reusable Ionic Liquids for the Catalyzed
Hydroamination of Alkenes with Sulfonamides Carbamates and Carboxamides L Yang L-W Xu C-G Xia
1975 Synthesis of 2391016172324-Octasubstituted Phthalocyaninatozinc(II) Complexes Mediated by Reductive Agents G A Gauna A C Monsalvo J Awruch
1979 A Short and Efficient Synthesis of 3-2-[2-(Bromomethyl)thiazol-4-yl]-ethynyl-5-fluorobenzonitrile A Precursor for PET Radioligand [18F]SP203 M B Gopinathan C Jin K S Rehder
1983 Synthesis of a Substituted Benzazepin-2-one Dihydrate S K Boini R K Vaid K P Moder D Mitchell
1987 Synthesis of Novel Trisubstituted Imidazolines F J Lakner M A Parker B Rogovoy A Khvat A Ivachtchenko
1991 A Novel Synthesis of N-But-3-enyl-α- and β-Amino Acids T T Van Nguyen R T C Brownlee A B Hughes
1999 Synthesis of Substituted 5-(3-Hydroxypropyl)pyrrolidin-2-ones and Pyrrolizidinones from Nitroethane via C3 Functionalized 56-Dihydro-4H-12-oxazines A Novel Approach to Some Analogues of the Antidepressant Rolipram A Yu Sukhorukov A V Lesiv Y A Khomutova S L Ioffe V A Tartakovsky
2009 Chiral Cyclobutanols and Cyclopentane Dimers via Samarium(II) Iodide Induced Keto-Olefin Cyclisations of Carbohydrate-Derived Unsaturated Ketones D B G Williams J Caddy K Blann J J C Groveacute C W Holzapfel
2015 Synthesis of Perfluoroalkylthio-Substituted Ferrocenes C Rhode J Lemke M Lieb N Metzler-Nolte
2019 Functionalization of Polyhedral Oligomeric Silsesquioxane (POSS) via Nucleophilic Substitution M Dutkiewicz H Maciejewski B Marciniec
2025 A Novel Synthesis of Aryl Mesylates via One-Pot DemethylationndashMesylation of Aryl Methyl Ethers Using a Mixture of Phosphorus Pentoxide in Methanesulfonic Acid B Kaboudin Y Abedi
2029 Anionic Cyclization of (NN-Dimethylamino)[2-(prop-2-yn-1-yloxy)aryl]-acetonitriles T Zdrojewski J Musielak A Jończyk
2035 Strecker-Type Reaction Catalyzed by Carboxylic Acids in Aqueous Media Z Xie G Li G Zhao J Wang
2040 Synthesis of Novel Structurally Simplified Estrogen Analogues with Electron-Donating Groups in Ring A L F Tietze C A Vock I K Krimmelbein L Nacke
2061 On the Resolution of Secondary Phosphine Oxides via Diastereomeric Complex Formation The Case of tert-Butylphenylphosphine Oxide J Holt A M Maj E P Schudde K M Pietrusiewicz L Sieroń W Wieczorek T Jerphagnon I W C E Arends U Hanefeld A J Minnaard
2066 Enantioselective Copper-Catalyzed Conjugate Addition of Dimethylzinc to 5-(1-Arylalkylidene) Meldrumrsquos Acids A Wilsily T Lou E Fillion
2073 SuzukindashMiyaura Coupling Reactions Using Phosphite Ligands M Jang Y Jo I-K Oh H M Jung S Lee
2076 Synthesis of 2-Methylindoline- and 2-Methyl-1234-tetrahydroquinoline-Derived Phosphoramidites and Their Applications in Iridium-Catalyzed Allylic Alkylation of Indoles W-B Liu H He L-X Dai S-L You
2083 Stereocontrolled Synthesis of 13-Amino Alcohols by Reduction of Substituted 2-1-[(tert-Butylsulfinyl)amino]alkylcyclohexanones J C Gonzaacutelez-Goacutemez F Foubelo M Yus
2089 Tunable Phosphoramidite Ligands for Asymmetric Hydrovinylation Ligands par excellence for Generation of All-Carbon Quaternary Centers C R Smith H J Lim A ZhangT V RajanBabu
2101 Copper-Catalyzed Asymmetric Ring-Opening Reaction of Oxabenzonorbornadienes with Grignard and Aluminum Reagents R Millet L Gremaud T Bernardez L Palais A Alexakis
2113 A Simplified Synthesis of Takemotorsquos Catalyst A Berkessel B Seelig 2116 Pharmaceutical Substances Syntheses Patents and Applications of the
Most Relevant AIPs Edited by Axel Kleeman Juumlrgen Engel Bernhard Kutscher Dietmar Reichert Reviewed by I Agranat
XV Forthcoming Articles
no 13 2117 Recent Advances in the Aza-Claisen Rearrangement K C Majumdar
T Bhattacharyya B Chattopadhyay B Sinha 2143 A Novel and Convenient Synthesis of lsquoReversedrsquo Diamidino 25-Aryl- and
25-Azaheterocycle-Substituted Furans L Hu D W Boykin 2146 Efficient and General Preparation of Pyranostilbenes First Total Synthesis
of Artocarbene and Pawhuskin B B H Park Y R Lee W S Lyoo 2155 Mild Oxidation of Diarylacetylenes to 12-Diketones Using Oxone in
Trifluoroacetic Acid J-H Chu Y-J Chen M-J Wu 2163 One-Pot Microwave-Assisted Selective Azido ReductionTandem Cyclization
in Condensed and Solid Phase with Nickel Boride N Shankaraiah N Markandeya M Espinoza-Moraga C Arancibia A Kamal L Silva Santos
2171 Pyrrolo[321-ij]quinolin-4-one and Pyrrolo[321-ij]quinolin-6-one H McNab D J Nelson E J Rozgowska
2175 Practical Synthesis of 5-Substituted Tetrazoles under Microwave Irradiation J Roh T V Artamonova K Vaacutevrovaacute G I Koldobskii A Hrabaacutelek
2179 A Simple Method for the Synthesis of 3-Arylthieno[23-b]pyridines via Iodine-Mediated Cyclization of 3-(1-Arylalkenyl)-2-[(1-phenylethyl)sulfanyl]pyridines K Kobayashi D Nakamura Y Shiroyama S Fukamachi H Konishi
2184 Synthesis of Four Lysine-Linked Cereulide Analogues Showing Ionophoric Activity Towards Potassium Cations as Lead Compounds for Emetic Toxin-Detection by Immunoassays A Makarasen T Nishikawa M Isobe
2205 Synthesis of α-Aliphatic and β-Aromatic Substituted Taurines via Regioselective Ring Opening of Thiiranes with Ammonia H Yu S Cao L Zhang G Liu J Xu
2210 Stability of 5(6)-Carboxyfluorescein in Microwave-Assisted Synthesis of Fluorescein-Labelled O-Dimannosylated Peptides R Kowalczyk P W R Harris R P Dunbar M A Brimble
2223 Diversity-Oriented Synthesis of Functionalized Diaryl Sulfones by Regioselective [3+3] Cyclizations of 13-Bis(siloxy)buta-13-dienes with 2-(Arylsulfonyl)-3-ethoxy-2-en-1-ones Scope and Limitations M Shkoor A Riahi O Fatunsin H Reinke C Fischer P Langer
2236 Synthesis of Functionalized Salicylates by Formal [3+3] Cyclocondensation of 13-Bis(silyloxy)buta-13-dienes with 3-Alkoxy-2-en-1-ones G Mroszlig S Ladzik H Reinke A Spannenberg C Fischer P Langer
2249 Synthetic Approach to Alkoxy-β-(trifluoromethyl)styrenes and Their Application in the Synthesis of New Trifluoromethylated Heterocycles V M Muzalevskiy V G Nenajdenko A V Shastin E S Balenkova G Haufe
2260 o-Benzenedisulfonimide as a Powerful and Recyclable Organocatalyst for the Nazarov Reaction M Barbero S Cadamuro A Deagostino S Dughera P Larini E G Occhiato C Prandi S Tabasso R Vulcano P Venturello
2267 The Catalytic Potential of 4-Guanidinylpyridines in Acylation Reactions I Held E Larionov C Bozler F Wagner H Zipse
2278 Iron(III) Chloride in EthanolndashWater Highly Efficient Catalytic System for the Synthesis of Garcia Gonzalez Polyhydroxyalkyl- and C-Glycosylfurans L Nagarapu M V Chary A Satyender B Supriya R Bantu
2283 Ruthenium-Catalyzed Addition of Primary Amides to Alkynes A Stereoselective Synthesis of Secondary Enamides L J Gooszligen M Blanchot K S M Salih K Gooszligen
2289 Binaphthyl-Modified Quaternary Phosphonium Salts as Chiral Phase Transfer Catalysts Application to Asymmetric Amination of β-Keto Esters R He K Maruoka
X Table of Contents XI Forthcoming Articles
no 14 2293 Direct Methods for Stereoselective Polypropionate Synthesis A Survey
J Li D Menche 2316 Synthesis of Symmetrical Ketones from Grignard Reagents and
11-Carbonyldiimidazole D Bottalico V Fiandanese G Marchese A Punzi
2319 Synthesis of 45-Substituted Imidazoles by a Fast Condensation of 12-Diketones and Urotropine in Heterogeneous Medium G Bratulescu
2321 (Arylsulfonyl)acetones and -acetonitriles New Activated Methylenic Building Blocks for Synthesis of 123-Triazoles N T Pokhodylo V S Matiychuk M D Obushak
2324 A Safe Convenient and Efficient One-Pot Synthesis of α-Chloroketone Acetals Directly from Ketones Using Iodobenzene Dichloride J Yu C Zhang
2329 An Efficient Oxidative Conversion of Aldehydes into 2-Substituted 2-Oxazolines Using 13-Diiodo-55-dimethylhydantoin S Takahashi H Togo
2333 A Novel Procedure for the Synthesis of Benzo[b][18]naphthyridine-3-carboxylate Derivatives from MoritandashBaylisndashHillman Adduct Acetates W Zhong F Lin R Chen W Su
2341 An Improved Synthesis of 147-Triazacyclononanes (tacns) and 14710-Tetraazacyclododecanes (cyclens) J Huang Z Zhou T H Chan
2345 The Ullmann Coupling between 2-Chlorobenzoic Acids and Amino Acids A Valuable Reaction for Preparing 2-Substituted 1-Acetyl-1H-indol-3-yl Acetates J C Rodriguez Dominguez X Gang G Kirsch
2349 gem-Dibromomethyl Aromatics Efficient Aldehyde Equivalents in the KnoevenagelndashDoebner Reaction J K Augustine Y A Naik S Poojari N Chowdappa B S Sherigara K Areppa
2357 Synthesis of Novel α-Aminophosphonates Containing Adamantyl Fragment M M Kabachnik L I Minaeva I P Beletskaya
2361 Efficient Fluoride-Mediated Synthesis of 5-Amino-Substituted Isothiazoles Y S Zubenko V I Potkin
2365 Phosphine-Catalyzed Reaction of Cyanohydrins with Activated Alkynes A Siby O Loreau F Taran
2371 Sulfanyl-Substituted [3]Cumulenes and Buta-13-dienes from a Tetrakis(pyridinium)-Substituted Butadiene A Schmidt A Rahimi M Gjikaj
2379 Efficient Synthesis of 2-Substituted Pyrido[32-d]pyrimidines Involving SNAr and Palladium-Catalyzed Cross-Coupling Reactions A Tikad S Routier M Akssira J-M Leacuteger C Jarry G Guillaumet
2385 Novel Synthesis of Medium-Sized Heterocycles by Palladium-Catalyzed Intramolecular Heck Reaction via 9-endo-trig Mode of Cyclization K C Majumdar B Chattopadhyay
2393 Facile Synthesis of Fluorinated Benzofuro- and Benzothieno[23-b]pyridines α-Carbolines and Nucleosides Containing the α-Carboline Framework V O Iaroshenko Y Wang B Zhang D Volochnyuk V Ya Sosnovskikh
2403 Synthesis of Functionalized N-Vinyl Nitrogen-Containing Heterocycles S M M Lopes A M Beja M Ramos Silva J A Paixatildeo F Palacios T M V D Pinho e Melo
2408 Kumada Cross-Coupling of Aryl Grignard Reagents with Aryl Halides Catalyzed by an Immobilized Nickel Catalyst X Chen L Wang J Liu
2413 Highly Enantioselective Synthesis of Heteroaromatic Alcohols Catalyzed by Chiral DiaminodiphosphinendashRuthenium(II) Complexes W-Y Shen Y-Y Li Z-R Dong J-X Gao
2418 Concise Total Synthesis of (+)-Disparlure and its trans-Isomer Using Asymmetric Organocatalysis S-G Kim
2423 Rhodium Carbenoid Induced [12]-Migration in an L-Lyxo-Configured α-Diazo β-Keto Ester Synthesis of a New Griseolic Acid Analogue N N Bhujbal K S A Kumar D D Dhavale
2430 Synthesis of 5-Arylthio-3-hydroxyphthalates by the First [4+2] Cycloadditions of 3-Arylthio-1-silyloxy-13-butadienes with Dimethyl Acetylenedicarboxylate I Iqbal M Imran P Langer
2435 Synthesis of Highly Functionalized Proline Derivatives via a One-Pot MichaelSN-AdditionCyclization Approach U Kazmaier C Schmidt
2440 RhodiumGraphite-Catalyzed Hydrogenation of Carbocyclic and Heterocyclic Aromatic Compounds G Falini A Gualandi D Savoia
2447 Potassium [1-(tert-Butoxycarbonyl)-1H-indol-2-yl]trifluoroborate as an Efficient Building Block in Palladium-Catalyzed SuzukindashMiyaura Cross Couplings P Kassis V Beacuteneacuteteau J-Y Meacuterour S Routier
2454 Syntheses of Substituted Furans and Pyrroles by Platinum-Catalyzed Cyclizations of Propargylic Oxiranes and Aziridines in Aqueous Media M Yoshida M Al-Amin K Shishido
2467 Transition-Metal-Free Oxidative Homocoupling of Aryl Alkenyl and Alkynyl Grignard Reagents with TEMPO M S Maji A Studer
XIII Forthcoming Articles
no 15 2471 Advances in Synthetic Approaches for the Preparation of Combretastatin-
Based Anti-Cancer Agents R Singh H Kaur 2492 Synthesis of Unsymmetrical Ureas by Sulfur-Assisted Carbonylation with
Carbon Monoxide and Oxidation with Molecular Oxygen under Mild Conditions T Mizuno T Nakai M Mihara
2497 Ring-OpeningRecyclization Reactions of (Dimethylamino)propenoyl-Substituted Cyclopropanes Facile Synthesis of Halogenated Pyridin-2(1H)-ones R Zhang Y Zhou Y Liang Z Jiang D Dong
2501 Facile and Efficient Total Synthesis of Taspine B Cheng S Zhang L Zhu J Zhang Q Li A Shan L He
2505 Oligomeric Iodosylbenzene Sulfate A Convenient Hypervalent Iodine Reagent for Oxidation of Organic Sulfides and Alkenes M S Yusubov R Y Yusubova T V Funk K-W Chi V V Zhdankin
2509 Pyrrolidine-Based Organocatalysts for Enantioselective Michael Addition of Cyclohexanone to trans-β-Nitrostyrene A P Carley S Dixon J D Kilburn
2517 CundashAl Hydrotalcite An Efficient and Reusable Ligand-Free Catalyst for the Coupling of Aryl Chlorides with Aliphatic Aromatic and N(H)-Heterocyclic Amines B Sreedhar R Arundhathi P L Reddy M A Reddy M L Kantam
2523 Highly Efficient Synthesis of trans-βγ-Unsaturated a-Keto Amides C Allais T Constantieux J Rodriguez
2531 Gas-Phase Synthesis of N-Unsubstituted 3-Hydroxypyrroles and 1H-Pyrrol-3(2H)-ones L Hill G A Hunter S H Imam H McNab W J OrsquoNeill
2535 3-Hydroxy-1H-pyrrole L Hill S H Imam H McNab W J OrsquoNeill 2539 123-Thiadiazoles with Unsaturated Side Chains Synthesis
Polymerization and Photocrosslinking M Al-Smadi N Hanold H Kalbitz H Meier
2547 Synthesis of 1112-Didehydrodibenzo[ae]cycloocten-5(6H)-one A Strained Eight-Membered Alkyne S C Kornmayer F Rominger R Gleiter
2553 Stannous Chloride Dihydrate A Novel and Efficient Catalyst for the Synthesis of gem-Dihydroperoxides from Ketones and Aldehydes D Azarifar K Khosravi F Soleimanei
2557 Synthesis of a Novel Class of Azacrown Macrocycles and Lariat Crown Ethers Containing Two 124-Triazole Rings as Subunits N Foroughifar A Mobinikhaledi S Ebrahimi
2561 Enantioselective Synthesis of the 3C-Protease Inhibitor (ndash)-Thysanone by a StauntonndashWeinreb Annulation Strategy J Sperry T Y Yuen M A Brimble
2570 Stereoselective Synthesis of Unnatural β-Amino Acids from Nitroethane via 56-Dihydro-4H-12-oxazin-3-ylacetates A Yu Sukhorukov A V Lesiv O L Eliseev Y A Khomutova S L Ioffe
2579 A Versatile Unexpected One-Pot Regioselective Synthesis of a New Class of 13-Diazepinoindolones by Reaction of Pyranoindolones with Monosubstituted Ureas D Livadiotou C A Tsoleridis J Stephanidou-Stephanatou
2584 Synthesis of a Trisaccharide and a Tetrasaccharide from the Cell-Wall Lipopolysaccharides of Azospirillum brasilense S17 S Pandey S Ghosh A K Misra
2591 Synthesis of Isoindoline Nitroxides by Electrocyclic Reactions T Kaacutelai J Jekı K Hideg
2596 Glycosylations of Tertiary Alcohols Synthesis of Fully Protected Disaccharides with Sterically Demanding Groups Attached to the Sugar Core A Holkenbrink J B Vicente D B Werz
2605 Copper-Catalyzed [13]-Dipolar Cycloaddition for the Synthesis of Macrocycles Containing Acyclic Aromatic and Steroidal Moieties G V Latyshev M S Baranom A V Kazantsev A D Averin N V Lukashev I P Beletskaya
2616 Aryl Ring Migration Reaction in the Synthesis of 24-Diaryl-4H-31-benzothiazines A V Butin F A Tsiunchik V T Abaev A V Gutnov D A Cheshkov
2627 Hydrogenation of β-N-Substituted and β-NN-Disubstituted Enamino Esters in the Presence of Iridium(I) Catalyst H Hebbache Z Hank C Bruneau J-L Renaud
2634 Stereoselective Olefination Reactions Promoted by Rieke Manganese J M Concelloacuten H Rodriacuteguez-Solla V del Amo P Diacuteaz
2646 Synthesis of Piperidinones through a Radical Cascade E Godineau Y Landais
2650 Asymmetric Organic Synthesis with Enzymes Edited by V Gotor I Alfonso E Garciacutea-Urdiales Reviewed by Steve Collier
XVII Forthcoming Articles
no 16 2651 Synthesis of Spirocyclic Ethers S Rosenberg R Leino 2674 Bimetallic PalladiumndashPlatinum-on-Carbon-Catalyzed HndashD Exchange
Reaction Synergistic Effect on Multiple Deuterium Incorporation T Maegawa N Ito K Oono Y Monguchi H Sajiki
2679 Efficient Copper-Catalyzed Synthesis of 2-Amino-4(3H)-quinazolinone and 2-Aminoquinazoline Derivatives X Huang H Yang H Fu R Qiao Y Zhao
2689 Synthesis and Chemoselective N- and O-Alkylation of Thiadiazolopyrimidine Nucleosides and Uridines A M L Hossion R Islam R K Kandahary T Nagamatsu
2697 Facile and Efficient Synthesis of a New Class of Indole-Substituted Pyridine Derivatives via One-Pot Multicomponent Reactions K Zhao X-P Xu S-L Zhu D-Q Shi Y Zhang S-J Ji
2709 Studies toward a Total Synthesis of Rhizoxin D Stereoselective Preparation of the C11ndashC19 Fragment S Padakanti C K Kumar E Ashok P Das
2715 A Short Synthesis of Enantiomeric Phytoprostanes B1 Type I W Perlikowska M Mikołajczyk
2719 Chemistry of Polyhalogenated Nitrobutadienes Part 7 A Novel Synthetic Access to Chlorinated Nitrile Oxides E Nutz V A Zapolrsquoskii D E Kaufmann
2725 Microwave-Assisted Silver(I)-Mediated Selective O-Alkylation of Aromatic Imidate Systems B K Singh C Cavalluzzo M De Maeyer Z Debyser V S Parmar E Van der Eycken
2729 Iodogen A Novel Reagent for the Oxidation of Urazoles under Heterogeneous Conditions A Khoramabadi A Shiri M A Zolfigol S Mallakpour
2733 An Unprecedented Synthesis of Eight-Membered-Ring Cyclic Thioimidic Esters by a Three-Component Reaction A Alizadeh R Hosseinpour
2737 A Novel Diastereoselective Synthesis of β-Phosphonato Unsaturated Thioimidates A Alizadeh N Zohreh
2741 Synthesis of 21-Benzisoxazoles by Nucleophilic Substitution of Hydrogen in Nitroarenes Activated by the Azole Ring N T Pokhodylo Y O Teslenko V S Matiychuk M D Obushak
2749 A Facile Synthesis of Two Series of Multifunctional Carbon Compounds from αα-Dihalo Ketones Using Allylsamarium Bromide X Liu S Zhang J Di
2756 Stereocontrolled Formation of Protected Aminodeoxyalditols from Simple Carbohydrate Precursors by Debenzylating Cycloetherification Y Jiang Z Fang Q Zheng H Jia J Cheng B Zheng
2761 trans-Stilbene as a Starting Material for the Synthesis of Tamoxifen Based on Palladium-Catalyzed Cross-Coupling Reactions C M Nunes J Limberger S Poersch M Seferin A L Monteiro
2766 Synthesis and Biological Evaluation of 6-Substituted Purinylcarbanucleosides with a Cyclopenta[b]thiophene Pseudosugar P Abeijoacuten J M Blanco O Caamantildeo F Fernaacutendez M D Garciacutea X Garciacutea-Mera J E Rodriacuteguez-Borges J Balzarini E De Clercq
2773 Synthesis and Electrochemical Signature of Novel Norbornyl-ferrocene Hybrids F A Khan S K Upadhyay
2778 A Regioselective TsujindashTrost Pentadienylation of 3-Allyltetronic Acid R Schobert B Barnickel
2785 Copper(I)-Catalyzed CarylndashCalkynyl Bond Formation of Aryl Iodides with Terminal Alkynes K G Thakur G Sekar
2790 Aminolysis of Epoxides Using Iridium Trichloride as an Efficient Catalyst J Agarwal A Duley R Rani R K Peddinti
2797 Preparation of Several Active N-Chloro Compounds from Trichloroisocyanuric Acid A Shiri A Khoramabadi-zad
2802 The First Mineral-Catalyzed One-Pot [3+1+2] Coupling Protocol for Multifunctionalized Fused-Ring Pyrimidines L D S Yadav A Rai
2809 Efficient Synthesis of Tetrahydro-β-carbolin-1-one and Dihydroisoquinolin-1-one Derivatives as Versatile Intermediates K E Judd M F Mahon L Caggiano
2818 A Concise Synthesis of ortho-Iodobenzyl Alcohols via Addition of ortho-Iodophenyl Grignard Reagent to Aldehydes and Ketones J Cvengroš D Stolz A Togni
XIII Forthcoming Articles
no 17 2825 Reactivity of Oxazol-5-(4H)-ones and Their Application toward Natural
Product Synthesis N M Hewlett C D Hupp J J Tepe 2840 Towards the Total Synthesis of 3-Hydroxyvibsanin E B D Schwartz
J R Denton P V Bernhardt H M L Davies C M Williams 2847 Structure Investigations of (ent)-Cladospolide D by De Novo Synthesis and
Kinetic and Thermodynamic Isomerization Y Xing J H Penn G A OrsquoDoherty
2855 New Applications of PhI(OAc)2 in Synthesis Total Synthesis and SAR Development of Potent Antitumor Natural Product PsymberinIrciniastatin A N Shao X Huang A Palani R Aslanian A Buevich J Piwinski R Huryk C Seidel-Dugan
2873 Total Synthesis of Largazole ndash Devolution of a Novel Synthetic Strategy B Wang C J Forsyth
2881 Formal Total Synthesis of Palmerolide A J Jaumlgel M E Maier 2893 Total Synthesis of Bongkrekic Acid via Sequential SuzukindashMiyaura Coupling
Reactions M Kanematsu M Shindo M Yoshida K Shishido 2905 Stereodivergent Approach to Both C28a-syn and C28a-anti Relative
Stereochemical Manifolds in the Lepadin Family via a TiCl4-Promoted G Li L J Carlson I K Sagamanova B W Slafer R P Hsung C Gilardi H M Sklenicka N Sydorenko
2915 Enantioselective Aldol Reaction of Tetrasubstituted Ketene Silyl Acetals with Achiral Aldehydes for the Construction of Asymmetric Tertiary Alcohols An Application for the Divergent Total Syntheses of Buergerinins F and G I Shiina T Iizumi Y-s Yamai Y-i Kawakita K Yokoyama Y-k Yamada
2927 Second-Generation Biomimetic Total Synthesis of Chaetominine A Coste G Karthikeyan F Couty G Evano
2935 Total Synthesis of (+)-Fostriecin and (+)-Phoslactomycin B S Shibahara M Fujino Y Tashiro N Okamoto T Esumi K Takahashi J Ishihara S Hatakeyama
2954 Stereochemical Assignments of the Chlorinated Residues in Victorin C A C Durow C Butts C L Willis
2963 Studies of the Asymmetric Total Synthesis of Clavilactone D by the lsquoLariatrsquo Cyclization Strategy T Yoshimitsu S Nojima M Hashimoto K Tsukamoto T Tanaka
2970 Total Synthesis of the Leucetta-Derived Alkaloid Calcaridine A P B Koswatta R Sivappa H V R Dias C J Lovely
2983 Formal Synthesis of Salinosporamide A Starting from D-Glucose T Momose Y Kaiya J-i Hasegawa T Sato N Chida
2992 Synthesis of Bioactive Natural Products by Asymmetric syn- and anti-Aldol Reactions A K Ghosh Z L Dawson
no 18 3003 Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural
Products B M Trost M K Brennan 3026 One-Pot Synthesis of Furo[34-b]pyridin-5(7H)-ones from 2-
Bromopyridine-3-carboxylic Acid and Carbonyl Compounds K Kobayashi T Kozuki H Konishi
3029 Iodocyclization of N-[2-(Methylthio)phenyl]propiolamides Selective Synthesis of 3-Iodo-15-benzothiazepin-4-ones T-S Jiang X-G Zhang J-H Li
3039 A Facile Synthetic Method for Fluorine-Containing 17-Phenanthrolines Pyridine-Ring Formation Reaction of N-Propargyl-68-bis(trifluoroacetyl)-quinolin-5-amine with Various Nucleophiles D Shibata E Okada M Hinoshita M Meacutedebielle
3047 Enantiotopic Discrimination in Palladium-Mediated Nucleophilic Substitutions on Achiral Substrates Chiral Ligand versus Chiral Nucleophile O Jacquet F Charnay J-C Fiaud J Ollivier
3051 Studies on the Chemistry of 2-[3-(2-Nitrophenyl)-2-oxopropyl]benzaldehydes Novel Syntheses of 5H-Benzo[b]carbazole-611-diones and Indolo[12-b]isoquinoline-611-diones M Fernaacutendez
3061 Studies on the C22ndashC23 Aldol Coupling of Spirangien M Lorenz N Bluhm M Kalesse
3067 One-Pot Synthesis of N-Alkyl Purine Pyrimidine and Azole Derivatives from Alcohols using Ph3PCCl4 A Rapid Route to Carboacyclic Nucleoside Synthesis M N Soltani Rad A Khalafi-Nezhad S Behrouz Z Asrari M Behrouz Z Amini
3077 Synthesis of 2-Amino-34-dihydroquinazolines and Imidazo[21-b]quinazoline-2-ones A Mishra S Batra
3089 Studies on the Reaction of Diimines with Thiourea Synthesis and Solvent-Induced cistrans-Isomerization of 135-Triazinane-2-thiones B Kaboudin T Ghasemi T Yokomatsu
3094 Suzuki Coupling of Heteroaromatic Chlorides Using Highly Electron-Donating ClickPhos Ligands S M Spinella Z-H Guan J Chen X Zhang
3099 Reaction of NN-Dioxyenamines with Anhydrides of Carboxylic and Sulfonic Acids A New Method for the Synthesis of a-Hydroxyoxime Derivatives A A Tabolin A V Lesiv S L Ioffe
3106 Directed ortho Metallation Chemistry and Phosphine Synthesis New Ligands for the SuzukindashMiyaura Reaction D B G Williams S J Evans H de Bod M S Mokhadinyana T Hughes
3113 New Functional Derivatives of 9-Phenylquinine P J Boratyński J SkarŜewski
3120 On the Synthesis of Asymmetric and Dissymmetric Amino Analogues of Troumlgerrsquos Base J Artacho K Waumlrnmark
3127 Synthesis of Polycyclic Sultams by Palladium-Catalyzed Intramolecular Cyclization K C Majumdar S Mondal N De
3136 Synthesis of Functionalized L-Cysteine and L-Methionine by Reaction with Electron-Deficient Acetylenes B A Trofimov A G Malrsquokina O A Shemyakina V V Nosyreva A P Borisova S S Khutsishvili L B Krivdin
3143 A lsquoClickrsquo Approach to the Synthesis of 3-[2-(1-Alkyltriazol-4-yl)ethyl]indoles M Petrini R R Shaikh
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
No 8 1227 Michael Additions to Activated Vinylphosphonates T Janecki J Kędzia
T Wąsek 1255 A Facile and General Synthesis of 2β-Aminosteroids X Ke H Hu
D Zhou W Xu Q Zhu N P Reddy X Hu 1261 Efficacious Preparation of Oppolzerrsquos Glycylsultam via the Deleacutepine
Reaction A Isleyen C Gonsky R C Ronald P Garner 1265 Synthesis of Masked Vicinal Amino Aldehydes of Pyrrolizine and Pyrrolo
[12-c]thiazole Series A V Tverdokhlebov A V Denisenko A A Tolmachev Y M Volovenko S V Shishkina O V Shishkin
1271 Preparation of 9-Substituted Pyridine-Stretched Adenines and Hypoxanthines J A Crawford W Fraser C A Ramsden
1279 A Versatile Synthesis of Heterocyclic Analogues of Neoflavonoids from Enamino Ketones V S Moskvina V P Khilya O V Turov U M Groth
1287 New Stereoselective Synthesis of Paeonilactone B F G Gatti S Serra 1291 The Use of NN-Dialkyltrimethylsilylamines in the Synthesis of
Pentamethinium Salts M Kořiacutenek M Rybaacutečkovaacute Boumlhm 1297 Synthesis of Triazoles via Regioselective Reactions of Aryl Azides with
Cyanoacetyl Pyrroles and Indoles N T Pokhodylo V S Matiychuk M D Obushak
1301 Gallium(III) Chloride Catalyzed Hydroarylation of Arylacetylenes with Naphthols and Phenols A Facile Synthesis of Vinylarenes J S Yadav B V S Reddy S Sengupta S K Biswas
1305 Electrophilic Bromination of meta-Substituted Anilines with N-Bromosuccinimide Regioselectivity and Solvent Effect S Bartoli A Cipollone A Squarcia A Madami D Fattori
1309 Cross-Coupling Reactions of Halopurines with Aryl- and Alkyltrifluoroborates The Scope and Limitations in the Synthesis of Modified Purines Z Hasniacutek R Pohl M Hocek
1318 A Convenient Method for Converting Hydroxyacetophenones into Their Ethylene or Trimethylene Acetals F Ono H Takenaka T Fujikawa M Mori T Sato
1323 γ-Chloromagnesio γ-Lactones and δ-Chloromagnesio δ-Lactones Generation Properties and Synthetic Uses H Shimizu S Fukuda S Sugiyama T Satoh
1336 Click Reactions with Nitroxides T Kaacutelai W L Hubbell K Hideg 1341 Synthesis of Novel 14-Benzoquinone-Containing 123-Triazoles An Entry
Into a New Library F Algi M Balci 1348 Efficient Synthesis of Two Sialylated Tetrasaccharides Found in Goat Milk
P K Mandal A K Misra 1355 Dendrimers of Vaccines Consisting of Tumor-Associated Glycopeptide
Antigens and T Cell Epitope Peptides S Keil A Kaiser F Syed H Kunz
1370 IBXTBAB-Mediated Oxidation of Primary Amines to Nitriles F Drouet P Fontaine G Masson J Zhu
1375 Chemoselectivity of Multicomponent Condensations of Barbituric Acids 5-Aminopyrazoles and Aldehydes E A Muravyova S V Shishkina V I Musatov I V Knyazeva O V Shishkin S M Desenko V A Chebanov
1386 Stereoselective Total Syntheses of Leiocarpin A and (ndash)-Galantinic Acid Starting from D-Mannitol K Nagaiah D Sreenu K V Purnima R S Rao J S Yadav
1393 A Facile Mild Deprotection Protocol for 13-Dithianes and 13-Dithiolanes with 30 Hydrogen Peroxide and Iodine Catalyst in Aqueous Micellar System N C Ganguly S K Barik
1400 Rhodium-Catalyzed Gram-Scale Synthesis of Highly Substituted Pyridine Derivatives K Parthasarathy C-H Cheng
1403 Enantioselective Synthesis of (R)-Propylene Carbonate from Ethyl (S)-Lactate J M Whitaker R C Ronald
XIII Forthcoming Articles
no 9 1405 Transition-Metal-Catalyzed Site-Selective Cross-Coupling of Di- and
Polyhalogenated Compounds J-R Wang K Manabe 1428 An Improved Synthesis of (4-4-Hydroxy-3-isopropyl-5-[(4-nitrophenyl)
ethynyl]benzyl-35-dimethylphenoxy)acetic Acid (NH-3) M B Gopinathan K S Rehder
1431 Copper-Catalyzed Tandem CndashN Bond Formation Reaction Selective Synthesis of 2-(Trifluoromethyl)benzimidazoles M-W Chen X-G Zhang P Zhong M-L Hu
1437 Synthesis and Thermochemical Properties of Stereoisomeric Dihydroxy- and Tetrahydroxyalkylammonium Salts M Thomas L Rothman J Hatcher P Agarkar R Ramkirath S Lall-Ramnarine R Engel
1445 Preparation of 5-Substituted 2-(2-Alkylaryl-1H-imidazol-4-yl)oxazoles and 5-Substituted 2-(2-Alkylarylthiazol-4-yl)oxazoles by Utilizing 5-Substituted 2-(2-Bromo-11-diethoxyethyl)oxazole as a Synthon D R St Laurent J L Romine
1459 Novel and Efficient Methods for the Synthesis of Symmetrical Trisulfides A Kertmen S Lach J Rachon D Witt
1463 An Environmentally Benign Electrochemical Process for the Reduction of Carboxylic Acid Hydrazides to Amides M Mentel M J Beier R Breinbauer
1469 Synthesis of 1-Chloroalkynes from Alkynylsilanes Using Trichloroisocyanuric Acid as Chlorinating Agent M H Vilhelmsen A S Andersson M B Nielsen
1473 A Convenient Approach to Enantioenriched Cyclopropanes Bearing Electron-Withdrawing Functionalities H Krawczyń K Wąsek J Kędzia
1477 Synthesis of Cyclopropenes via 12-Elimination of Bromocyclopropanes Catalyzed by Crown Ether W M Sherrill R Kim M Rubin
1485 A Base-Catalysed One-Pot Three-Component Coupling Reaction Leading to Nitrosubstituted Pyrroles I R Baxendale C D Buckle S V Ley L Tamborini
1494 Synthesis of 4-Alkylidene-4H-31-benzoxazine Derivatives by Acid-Catalyzed Cyclization of 2-Isocyanophenyl Ketones in the Presence of a Vinyl Ether K Kobayashi Y Okamura H Konishi
1499 Synthesis of Higher Helicenes via Olefin Metathesis and CndashH Activation J Cocircteacute S K Collins
1506 Azido- and Ethynyl-Substituted 2262-Terpyridines as Suitable Substrates for Click Reactions A Winter A Wild R Hoogenboom M W M Fijten M D Hager R-A Fallahpour U S Schubert
1513 Synthesis of 2-(Arylamino)ethanethiols via Lewis Acid Catalyzed Aminolysis of 22-Dimethylthiirane as Precursors of the 14-Benzothiazine Nucleus R Spogli S Sabatini G Manfroni O Tabarrini V Cecchetti
1520 Iron(III) Chloride A Versatile Catalyst for the Practical Synthesis of 3-Sulfenylindoles J S Yadav B V S Reddy Y J Reddy K Praneeth
1525 Organocatalytic Enantioselective Conjugate Addition of 2-Fluoromalonate to Nitroolefins Direct Synthesis of Chiral Fluorinated γ-Nitro Carboxylic Acid Derivatives H Li L Zu H Xie W Wang
1531 Asymmetric Transfer Hydrogenation of Ketimines with Trichlorosilane Structural Studies Z Zhang P Rooshenas H Hausmann P R Schreiner
1545 Prolinol Sulfinyl Ester Derivatives Organocatalytic Michael Addition of Ketones to Nitroolefins under Neat Conditions X Zeng G Zhong
1551 Asymmetric Oxidations of Electron-Poor Alkenes Promoted by the β-Amino AlcoholTBHP System A Russo A Lattanzi
1557 Enantioselectivity Switch in Direct Asymmetric Aminoxylation Catalyzed by Binaphthyl-Based Chiral Secondary Amines T Kano A Yamamoto F Shirozu K Maruoka
1564 Enantioselective Conjugate Addition of N-Heterocycles to αβ-Unsaturated Ketones Catalyzed by Chiral Primary Amines G Luo S Zhang W Duan W Wang
1573 Sulfonyl Hydrazine as New Functionality in Organocatalysis Camphorsulfonyl Hydrazine Catalyzed Enantioselective Aza-Michael Addition L-Y Chen H He B-J Pei W-H Chan A W M Lee
1578 Conversion of Primary Alcohols and Aldehydes into Methyl Esters by Ruthenium-Catalysed Hydrogen Transfer Reactions N A Owston T D Nixon A J Parker M K Whittlesey J M J Williams
1582 Addendum and Erratum XVII Forthcoming Articles
no 10 1583 Organocatalytic Formation of Quaternary Stereocenters M Bella
T Gasperi 1615 Regioselective Synthesis of 5H-Thiazolo[32-a]pyrimidin-5-ones from
MoritandashBaylisndashHillman Adduct Acetates under Solvent-Free and Base-Free Conditions W Zhong B Guo F Lin Y Liu W Su
1623 First Synthesis of 5-Cyanosalicylates by Formal [3+3] Cyclocondensations of 13-Bis(silyloxy)-13-butadienes A Riahi O Fatunsin M Shkoor R Dede H Reinke C Fischer P Langer
1635 Reaction of Isocyanides Dialkyl Acetylenedicarboxylates and a-Keto Lactones Unexpected Participation of an Ester Carbonyl Group in the Isocyanide-Based Three-Component Reaction A A Esmaeili H Vesalipoor
1639 An Efficient and Chemoselective Synthesis of 16-Naphthyridines and Pyrano[32-c]pyridines under Microwave Irradiation Z-G Han S-J Tu B Jiang S Yan X-H Zhang S-S Wu W-J Hao X-D Cao F Shi G Zhang N Ma
1647 N-Activation of N-Arylimidazoles Facile Syntheses of N-Alkyl-N-arylimidazolium Iodides from Less Expensive Chloro Substrates A M Oertel V Ritleng M J Chetcuti
1651 Synthesis of Polyhalogenated 2-(Phenylamino)pyridines by Thermal Amination Reactions S R Waldvogel A Faust W Barkmann R Froumlhlich O Wolff
1655 Cyanide Ion Promoted Addition of Acylphosphonates to Diethyl Cyanophosphonate Synthesis of Phosphonocyanohydrin O-Phosphates A S Demir A Aybey M Emrullahoglu
1659 Straightforward and Scalable Synthesis of Orthogonally Protected 37-Diazabicyclo[410]heptane H Schramm M Pavlova C Hoenke J Christoffers
1663 Hypervalent Iodine Mediated Oxidation of 12-Diaminobenzimidazole and Its Schiff Bases Efficient Synthesis of 3-Amino-124-benzotriazine and 2-Aryl-124-triazolo[15-a]benzimidazoles A Kumar M Parshad R K Gupta D Kumar
1667 Synthesis of the Reported Protoberberine Gusanlung D P B Wakchaure S Easwar N P Argade
1673 2-(Azidomethyl)arylboronic Acids in the Synthesis of Coumarin-Type Compounds M I Naumov A V Nuchev N S Sitnikov Y B Malysheva A S Shavyrin I P Beletskaya A E Gavryushin S Combes A Y Fedorov
1683 Asymmetric Synthesis of 12-anti-Disubstituted Taurine Derivatives D Enders D Iffland G Raabe
1689 A Novel One-Pot Three-Component Synthesis of 5-Imino-2358-tetrahydropyrazolo[12-a]pyridazin-1-one Derivatives B Qian M-J Fan Y-X Xie L-Y Wu Y Shi Y-M Liang
1694 One-Portion Synthesis of 2-Acetoxy Carbonyl Compounds from Aldehydes by Using an Acetylated Masked Acyl Cyanide H Nemoto T Kawamura K Kitasaki K Yatsuzuka M Kamiya Y Yoshioka
1703 Synthesis of 9-Anthryl Ethers from trans-910-Dihydro-910-dimethoxyanthracene by Acid-Catalyzed Transetherification K S Jang H Y Shin D Y Chi
1708 Efficient Synthesis of Azo Dye Labeled Terpenes Sugars and Steroids Using N-(4-Arylazobenzoyl)-1H-benzotriazoles A R Katritzky S R Tala N E Abo-Dya Z K Abdel-Samii
1715 Tandem CH-ActivationndashImine-Formation Reaction A New Route to Imidazo[21-a]phthalazines A Heim-Riether K R Gipson
1720 A Convenient and Efficient α-Sulfenylation of Carbonyl Compounds E Okragla S Demkowicz J Rachon D Witt
1725 Stereoselective Synthesis of β-Branched Phenylalanine Derivatives via Chelate-Claisen Rearrangement C Quirin U Kazmaier
1732 Catalyst-Free and Base-Free Water-Promoted SNAr Reaction of Heteroaryl Halides with Thiols B Sreedhar P S Reddy M A Reddy
1739 Convenient Methods for Synthesis of C2-Symmetric Diphenyltetrahydrothiophenes M Periasamy G Ramani G P Muthukumaragopal
1744 Highly Diastereoselective Conjugate AdditionndashElimination of Chiral Nickel(II) Glycinate with Activated Allylic Acetates for Asymmetric Synthesis of Glutamic Acid Derivatives J Wang J Shi X Zhang D Lin H Jiang H Liu
1753 Synthesis of 36-Dimethoxybenzene-12-diamine and of 47-Dimethoxy-2-methyl-1H-benzimidazole T Besset C Morin
1757 An Inexpensive Procedure for Reductive Aminations Using Dimethylamineborane on Millimolar and Molar Scale R Ortmann M Schlitzer
1760 Classics in Stereoselective Synthesis Edited by E M Carreira L Kvaerno Reviewed by Rolf Breinbauer
XV Forthcoming Articles
no 11 1761 Transition-Metal-Catalyzed Enantioselective Synthesis of Compounds with
Non-Centrochirality M Ogasawara S Watanabe 1786 One-Pot Synthesis of 3-Acyl-2-(alkylsulfanyl)indoles and 2-(Alkylsulfanyl)-
indole-3-carboxylates from (2-Isocyanophenyl)methyl Ketones or (2-Isocyanophenyl)acetates S Fukamachi H Konishi K Kobayashi
1791 Efficient and Recyclable Phthalocyanine-Based Sensitizers for Photooxygenation Reactions H Xu W-K Chan D K P Ng
1797 A Facile and Practical One-Pot Synthesis of β-Oxo Thioamides from β-Oxo Amides and Isothiocyanates P Huang D Xiang Y Zhou Y Liang T Na D Dong
1801 Microwave-Promoted Solid-Acid-Catalyzed One-Pot Synthesis of Phthalazinones V M Outerbridge S M Landge H Tamaki B Toumlroumlk
1807 Benzylic Brominations with N-Bromosuccinimide in (Trifluoromethyl)-benzene D Suarez G Laval S-M Tu D Jiang C L Robinson R Scott B T Golding
1811 Synthesis of Thioflavanone and Flavanone Derivatives by Cyclization of Chalcones W Konieczny M Konieczny
1815 A New and Expedient Total Synthesis of Ochratoxin A and d5-Ochratoxin A B Gabriele M Attya A Fazio L Di Donna P Plastina G Sindona
1821 Synthesis of Benzopyrrolizidinones by NorrishndashYang Cyclization of 3-(Acylmethyl)-2-alkylisoindol-1-ones J Wu W Zhang C Wang
1829 Reactions of MoritandashBaylisndashHillman Acetates with Huisgen Zwitterions A Novel Strategy for the Synthesis of β-Amino Acid Derivatives A Jose R R Paul R Mohan S C Mathew A T Biju E Suresh V Nair
1834 Peracetylated β-Allyl C-Glycosides of D-Ribofuranose and 2-Deoxy- D-ribofuranose in the Chemical Literature Until Now Mirages in the Literature H Otero Martinez H Reinke D Michalik C Vogel
1841 Core-Tetrasubstituted Naphthalene Diimides by Stille Cross-Coupling Reactions and Characterization of Their Optical and Redox Properties S-L Suraru F Wuumlrthner
1846 A Practical Synthesis of Indole-Based Heterocycles Using an Amidoaluminum-Mediated Strategy R Todd M M Hossain
1851 Synthesis of Fluorinated Pyrrolo[23-b]pyridine and Pyrrolo[23-d]pyrimidine Nucleosides V O Iaroshenko Y Wang D V Sevenard D M Volochnyuk
1858 Recyclization Reactions of 5-Formyl-13-dimethyluracil with Electron-Rich Amino Heterocycles A P Mityuk D M Volochnyuk S V Ryabukhin A S Plaskon A Shivanyuk A A Tolmachev
1865 Facile Synthesis of Fluorinated 1-Desazapurines V O Iaroshenko D V Sevenard D M Volochnyuk Y Wang A Martiloga A O Tolmachev
1876 A Practical Synthesis of 3-Diethoxyphosphoryl-12-pyridazine Derivatives J-C Monbaliu J Marchand-Brynaert
1881 Enantioselective Reduction of Prochiral Ketones Employing Sprouted Pisum sativa as Biocatalyst J S Yadav B V S Reddy C Sreelakshmi A B Rao
1886 Application of Phenolate Ion Mediated Intramolecular Epoxide Ring Opening in the Enantioselective Synthesis of Functionalized 23-Dihydrobenzofurans and 1-Benzopyrans S K Dinda S K Das G Panda
1897 Complementary Synthetic Approaches to Constitutionally Diverse N-Aminoalkylated Isoindolinones Application to the Synthesis of Falipamil and 5-HT1A Receptor Ligand Analogues M Lorion A Couture E Deniau P Grandclaudon
1904 Selective Deprotection of Silyl Ethers with Sodium Periodate J Li D Menche
1909 Micellar Solution of Sodium Dodecyl Sulfate (SDS) Catalyzes KabacknikndashFields Reaction in Aqueous Media S Sobhani A Vafaee
1916 Convenient Methods for the Synthesis of a Library of Hemilabile Phosphines M V Jimeacutenez J J Peacuterez-Torrente M I Bartolomeacute L A Oro
1923 Terminal Aziridines by Addition of Grignard Reagents or Organoceriums to an (α-Chloro)sulfinylimine D M Hodgson J Kloesges B Evans
1933 A Robust Synthesis of Nε-(Carboxymethyl)-L-lysine (CML) R Csuk S Stark A Barthel R Kluge D Stroumlhl
1935 One-Pot Curtius Rearrangement Processes from Carboxylic Acids O Leogane H Lebel
XV Forthcoming Articles
no 12 1941 The Chemistry of Deprotonated α-Aminonitriles T Opatz 1960 An Efficient Synthesis of Tetraalkyl 2345-Thiophenetetracarboxylate
Derivatives A Alizadeh R Hosseinpour 1963 Facile Deprotection of Bulky (Trialkylsilyl)acetylenes with Silver Fluoride
S Kim B Kim J In 1969 Highly Efficient and Reusable Ionic Liquids for the Catalyzed
Hydroamination of Alkenes with Sulfonamides Carbamates and Carboxamides L Yang L-W Xu C-G Xia
1975 Synthesis of 2391016172324-Octasubstituted Phthalocyaninatozinc(II) Complexes Mediated by Reductive Agents G A Gauna A C Monsalvo J Awruch
1979 A Short and Efficient Synthesis of 3-2-[2-(Bromomethyl)thiazol-4-yl]-ethynyl-5-fluorobenzonitrile A Precursor for PET Radioligand [18F]SP203 M B Gopinathan C Jin K S Rehder
1983 Synthesis of a Substituted Benzazepin-2-one Dihydrate S K Boini R K Vaid K P Moder D Mitchell
1987 Synthesis of Novel Trisubstituted Imidazolines F J Lakner M A Parker B Rogovoy A Khvat A Ivachtchenko
1991 A Novel Synthesis of N-But-3-enyl-α- and β-Amino Acids T T Van Nguyen R T C Brownlee A B Hughes
1999 Synthesis of Substituted 5-(3-Hydroxypropyl)pyrrolidin-2-ones and Pyrrolizidinones from Nitroethane via C3 Functionalized 56-Dihydro-4H-12-oxazines A Novel Approach to Some Analogues of the Antidepressant Rolipram A Yu Sukhorukov A V Lesiv Y A Khomutova S L Ioffe V A Tartakovsky
2009 Chiral Cyclobutanols and Cyclopentane Dimers via Samarium(II) Iodide Induced Keto-Olefin Cyclisations of Carbohydrate-Derived Unsaturated Ketones D B G Williams J Caddy K Blann J J C Groveacute C W Holzapfel
2015 Synthesis of Perfluoroalkylthio-Substituted Ferrocenes C Rhode J Lemke M Lieb N Metzler-Nolte
2019 Functionalization of Polyhedral Oligomeric Silsesquioxane (POSS) via Nucleophilic Substitution M Dutkiewicz H Maciejewski B Marciniec
2025 A Novel Synthesis of Aryl Mesylates via One-Pot DemethylationndashMesylation of Aryl Methyl Ethers Using a Mixture of Phosphorus Pentoxide in Methanesulfonic Acid B Kaboudin Y Abedi
2029 Anionic Cyclization of (NN-Dimethylamino)[2-(prop-2-yn-1-yloxy)aryl]-acetonitriles T Zdrojewski J Musielak A Jończyk
2035 Strecker-Type Reaction Catalyzed by Carboxylic Acids in Aqueous Media Z Xie G Li G Zhao J Wang
2040 Synthesis of Novel Structurally Simplified Estrogen Analogues with Electron-Donating Groups in Ring A L F Tietze C A Vock I K Krimmelbein L Nacke
2061 On the Resolution of Secondary Phosphine Oxides via Diastereomeric Complex Formation The Case of tert-Butylphenylphosphine Oxide J Holt A M Maj E P Schudde K M Pietrusiewicz L Sieroń W Wieczorek T Jerphagnon I W C E Arends U Hanefeld A J Minnaard
2066 Enantioselective Copper-Catalyzed Conjugate Addition of Dimethylzinc to 5-(1-Arylalkylidene) Meldrumrsquos Acids A Wilsily T Lou E Fillion
2073 SuzukindashMiyaura Coupling Reactions Using Phosphite Ligands M Jang Y Jo I-K Oh H M Jung S Lee
2076 Synthesis of 2-Methylindoline- and 2-Methyl-1234-tetrahydroquinoline-Derived Phosphoramidites and Their Applications in Iridium-Catalyzed Allylic Alkylation of Indoles W-B Liu H He L-X Dai S-L You
2083 Stereocontrolled Synthesis of 13-Amino Alcohols by Reduction of Substituted 2-1-[(tert-Butylsulfinyl)amino]alkylcyclohexanones J C Gonzaacutelez-Goacutemez F Foubelo M Yus
2089 Tunable Phosphoramidite Ligands for Asymmetric Hydrovinylation Ligands par excellence for Generation of All-Carbon Quaternary Centers C R Smith H J Lim A ZhangT V RajanBabu
2101 Copper-Catalyzed Asymmetric Ring-Opening Reaction of Oxabenzonorbornadienes with Grignard and Aluminum Reagents R Millet L Gremaud T Bernardez L Palais A Alexakis
2113 A Simplified Synthesis of Takemotorsquos Catalyst A Berkessel B Seelig 2116 Pharmaceutical Substances Syntheses Patents and Applications of the
Most Relevant AIPs Edited by Axel Kleeman Juumlrgen Engel Bernhard Kutscher Dietmar Reichert Reviewed by I Agranat
XV Forthcoming Articles
no 13 2117 Recent Advances in the Aza-Claisen Rearrangement K C Majumdar
T Bhattacharyya B Chattopadhyay B Sinha 2143 A Novel and Convenient Synthesis of lsquoReversedrsquo Diamidino 25-Aryl- and
25-Azaheterocycle-Substituted Furans L Hu D W Boykin 2146 Efficient and General Preparation of Pyranostilbenes First Total Synthesis
of Artocarbene and Pawhuskin B B H Park Y R Lee W S Lyoo 2155 Mild Oxidation of Diarylacetylenes to 12-Diketones Using Oxone in
Trifluoroacetic Acid J-H Chu Y-J Chen M-J Wu 2163 One-Pot Microwave-Assisted Selective Azido ReductionTandem Cyclization
in Condensed and Solid Phase with Nickel Boride N Shankaraiah N Markandeya M Espinoza-Moraga C Arancibia A Kamal L Silva Santos
2171 Pyrrolo[321-ij]quinolin-4-one and Pyrrolo[321-ij]quinolin-6-one H McNab D J Nelson E J Rozgowska
2175 Practical Synthesis of 5-Substituted Tetrazoles under Microwave Irradiation J Roh T V Artamonova K Vaacutevrovaacute G I Koldobskii A Hrabaacutelek
2179 A Simple Method for the Synthesis of 3-Arylthieno[23-b]pyridines via Iodine-Mediated Cyclization of 3-(1-Arylalkenyl)-2-[(1-phenylethyl)sulfanyl]pyridines K Kobayashi D Nakamura Y Shiroyama S Fukamachi H Konishi
2184 Synthesis of Four Lysine-Linked Cereulide Analogues Showing Ionophoric Activity Towards Potassium Cations as Lead Compounds for Emetic Toxin-Detection by Immunoassays A Makarasen T Nishikawa M Isobe
2205 Synthesis of α-Aliphatic and β-Aromatic Substituted Taurines via Regioselective Ring Opening of Thiiranes with Ammonia H Yu S Cao L Zhang G Liu J Xu
2210 Stability of 5(6)-Carboxyfluorescein in Microwave-Assisted Synthesis of Fluorescein-Labelled O-Dimannosylated Peptides R Kowalczyk P W R Harris R P Dunbar M A Brimble
2223 Diversity-Oriented Synthesis of Functionalized Diaryl Sulfones by Regioselective [3+3] Cyclizations of 13-Bis(siloxy)buta-13-dienes with 2-(Arylsulfonyl)-3-ethoxy-2-en-1-ones Scope and Limitations M Shkoor A Riahi O Fatunsin H Reinke C Fischer P Langer
2236 Synthesis of Functionalized Salicylates by Formal [3+3] Cyclocondensation of 13-Bis(silyloxy)buta-13-dienes with 3-Alkoxy-2-en-1-ones G Mroszlig S Ladzik H Reinke A Spannenberg C Fischer P Langer
2249 Synthetic Approach to Alkoxy-β-(trifluoromethyl)styrenes and Their Application in the Synthesis of New Trifluoromethylated Heterocycles V M Muzalevskiy V G Nenajdenko A V Shastin E S Balenkova G Haufe
2260 o-Benzenedisulfonimide as a Powerful and Recyclable Organocatalyst for the Nazarov Reaction M Barbero S Cadamuro A Deagostino S Dughera P Larini E G Occhiato C Prandi S Tabasso R Vulcano P Venturello
2267 The Catalytic Potential of 4-Guanidinylpyridines in Acylation Reactions I Held E Larionov C Bozler F Wagner H Zipse
2278 Iron(III) Chloride in EthanolndashWater Highly Efficient Catalytic System for the Synthesis of Garcia Gonzalez Polyhydroxyalkyl- and C-Glycosylfurans L Nagarapu M V Chary A Satyender B Supriya R Bantu
2283 Ruthenium-Catalyzed Addition of Primary Amides to Alkynes A Stereoselective Synthesis of Secondary Enamides L J Gooszligen M Blanchot K S M Salih K Gooszligen
2289 Binaphthyl-Modified Quaternary Phosphonium Salts as Chiral Phase Transfer Catalysts Application to Asymmetric Amination of β-Keto Esters R He K Maruoka
X Table of Contents XI Forthcoming Articles
no 14 2293 Direct Methods for Stereoselective Polypropionate Synthesis A Survey
J Li D Menche 2316 Synthesis of Symmetrical Ketones from Grignard Reagents and
11-Carbonyldiimidazole D Bottalico V Fiandanese G Marchese A Punzi
2319 Synthesis of 45-Substituted Imidazoles by a Fast Condensation of 12-Diketones and Urotropine in Heterogeneous Medium G Bratulescu
2321 (Arylsulfonyl)acetones and -acetonitriles New Activated Methylenic Building Blocks for Synthesis of 123-Triazoles N T Pokhodylo V S Matiychuk M D Obushak
2324 A Safe Convenient and Efficient One-Pot Synthesis of α-Chloroketone Acetals Directly from Ketones Using Iodobenzene Dichloride J Yu C Zhang
2329 An Efficient Oxidative Conversion of Aldehydes into 2-Substituted 2-Oxazolines Using 13-Diiodo-55-dimethylhydantoin S Takahashi H Togo
2333 A Novel Procedure for the Synthesis of Benzo[b][18]naphthyridine-3-carboxylate Derivatives from MoritandashBaylisndashHillman Adduct Acetates W Zhong F Lin R Chen W Su
2341 An Improved Synthesis of 147-Triazacyclononanes (tacns) and 14710-Tetraazacyclododecanes (cyclens) J Huang Z Zhou T H Chan
2345 The Ullmann Coupling between 2-Chlorobenzoic Acids and Amino Acids A Valuable Reaction for Preparing 2-Substituted 1-Acetyl-1H-indol-3-yl Acetates J C Rodriguez Dominguez X Gang G Kirsch
2349 gem-Dibromomethyl Aromatics Efficient Aldehyde Equivalents in the KnoevenagelndashDoebner Reaction J K Augustine Y A Naik S Poojari N Chowdappa B S Sherigara K Areppa
2357 Synthesis of Novel α-Aminophosphonates Containing Adamantyl Fragment M M Kabachnik L I Minaeva I P Beletskaya
2361 Efficient Fluoride-Mediated Synthesis of 5-Amino-Substituted Isothiazoles Y S Zubenko V I Potkin
2365 Phosphine-Catalyzed Reaction of Cyanohydrins with Activated Alkynes A Siby O Loreau F Taran
2371 Sulfanyl-Substituted [3]Cumulenes and Buta-13-dienes from a Tetrakis(pyridinium)-Substituted Butadiene A Schmidt A Rahimi M Gjikaj
2379 Efficient Synthesis of 2-Substituted Pyrido[32-d]pyrimidines Involving SNAr and Palladium-Catalyzed Cross-Coupling Reactions A Tikad S Routier M Akssira J-M Leacuteger C Jarry G Guillaumet
2385 Novel Synthesis of Medium-Sized Heterocycles by Palladium-Catalyzed Intramolecular Heck Reaction via 9-endo-trig Mode of Cyclization K C Majumdar B Chattopadhyay
2393 Facile Synthesis of Fluorinated Benzofuro- and Benzothieno[23-b]pyridines α-Carbolines and Nucleosides Containing the α-Carboline Framework V O Iaroshenko Y Wang B Zhang D Volochnyuk V Ya Sosnovskikh
2403 Synthesis of Functionalized N-Vinyl Nitrogen-Containing Heterocycles S M M Lopes A M Beja M Ramos Silva J A Paixatildeo F Palacios T M V D Pinho e Melo
2408 Kumada Cross-Coupling of Aryl Grignard Reagents with Aryl Halides Catalyzed by an Immobilized Nickel Catalyst X Chen L Wang J Liu
2413 Highly Enantioselective Synthesis of Heteroaromatic Alcohols Catalyzed by Chiral DiaminodiphosphinendashRuthenium(II) Complexes W-Y Shen Y-Y Li Z-R Dong J-X Gao
2418 Concise Total Synthesis of (+)-Disparlure and its trans-Isomer Using Asymmetric Organocatalysis S-G Kim
2423 Rhodium Carbenoid Induced [12]-Migration in an L-Lyxo-Configured α-Diazo β-Keto Ester Synthesis of a New Griseolic Acid Analogue N N Bhujbal K S A Kumar D D Dhavale
2430 Synthesis of 5-Arylthio-3-hydroxyphthalates by the First [4+2] Cycloadditions of 3-Arylthio-1-silyloxy-13-butadienes with Dimethyl Acetylenedicarboxylate I Iqbal M Imran P Langer
2435 Synthesis of Highly Functionalized Proline Derivatives via a One-Pot MichaelSN-AdditionCyclization Approach U Kazmaier C Schmidt
2440 RhodiumGraphite-Catalyzed Hydrogenation of Carbocyclic and Heterocyclic Aromatic Compounds G Falini A Gualandi D Savoia
2447 Potassium [1-(tert-Butoxycarbonyl)-1H-indol-2-yl]trifluoroborate as an Efficient Building Block in Palladium-Catalyzed SuzukindashMiyaura Cross Couplings P Kassis V Beacuteneacuteteau J-Y Meacuterour S Routier
2454 Syntheses of Substituted Furans and Pyrroles by Platinum-Catalyzed Cyclizations of Propargylic Oxiranes and Aziridines in Aqueous Media M Yoshida M Al-Amin K Shishido
2467 Transition-Metal-Free Oxidative Homocoupling of Aryl Alkenyl and Alkynyl Grignard Reagents with TEMPO M S Maji A Studer
XIII Forthcoming Articles
no 15 2471 Advances in Synthetic Approaches for the Preparation of Combretastatin-
Based Anti-Cancer Agents R Singh H Kaur 2492 Synthesis of Unsymmetrical Ureas by Sulfur-Assisted Carbonylation with
Carbon Monoxide and Oxidation with Molecular Oxygen under Mild Conditions T Mizuno T Nakai M Mihara
2497 Ring-OpeningRecyclization Reactions of (Dimethylamino)propenoyl-Substituted Cyclopropanes Facile Synthesis of Halogenated Pyridin-2(1H)-ones R Zhang Y Zhou Y Liang Z Jiang D Dong
2501 Facile and Efficient Total Synthesis of Taspine B Cheng S Zhang L Zhu J Zhang Q Li A Shan L He
2505 Oligomeric Iodosylbenzene Sulfate A Convenient Hypervalent Iodine Reagent for Oxidation of Organic Sulfides and Alkenes M S Yusubov R Y Yusubova T V Funk K-W Chi V V Zhdankin
2509 Pyrrolidine-Based Organocatalysts for Enantioselective Michael Addition of Cyclohexanone to trans-β-Nitrostyrene A P Carley S Dixon J D Kilburn
2517 CundashAl Hydrotalcite An Efficient and Reusable Ligand-Free Catalyst for the Coupling of Aryl Chlorides with Aliphatic Aromatic and N(H)-Heterocyclic Amines B Sreedhar R Arundhathi P L Reddy M A Reddy M L Kantam
2523 Highly Efficient Synthesis of trans-βγ-Unsaturated a-Keto Amides C Allais T Constantieux J Rodriguez
2531 Gas-Phase Synthesis of N-Unsubstituted 3-Hydroxypyrroles and 1H-Pyrrol-3(2H)-ones L Hill G A Hunter S H Imam H McNab W J OrsquoNeill
2535 3-Hydroxy-1H-pyrrole L Hill S H Imam H McNab W J OrsquoNeill 2539 123-Thiadiazoles with Unsaturated Side Chains Synthesis
Polymerization and Photocrosslinking M Al-Smadi N Hanold H Kalbitz H Meier
2547 Synthesis of 1112-Didehydrodibenzo[ae]cycloocten-5(6H)-one A Strained Eight-Membered Alkyne S C Kornmayer F Rominger R Gleiter
2553 Stannous Chloride Dihydrate A Novel and Efficient Catalyst for the Synthesis of gem-Dihydroperoxides from Ketones and Aldehydes D Azarifar K Khosravi F Soleimanei
2557 Synthesis of a Novel Class of Azacrown Macrocycles and Lariat Crown Ethers Containing Two 124-Triazole Rings as Subunits N Foroughifar A Mobinikhaledi S Ebrahimi
2561 Enantioselective Synthesis of the 3C-Protease Inhibitor (ndash)-Thysanone by a StauntonndashWeinreb Annulation Strategy J Sperry T Y Yuen M A Brimble
2570 Stereoselective Synthesis of Unnatural β-Amino Acids from Nitroethane via 56-Dihydro-4H-12-oxazin-3-ylacetates A Yu Sukhorukov A V Lesiv O L Eliseev Y A Khomutova S L Ioffe
2579 A Versatile Unexpected One-Pot Regioselective Synthesis of a New Class of 13-Diazepinoindolones by Reaction of Pyranoindolones with Monosubstituted Ureas D Livadiotou C A Tsoleridis J Stephanidou-Stephanatou
2584 Synthesis of a Trisaccharide and a Tetrasaccharide from the Cell-Wall Lipopolysaccharides of Azospirillum brasilense S17 S Pandey S Ghosh A K Misra
2591 Synthesis of Isoindoline Nitroxides by Electrocyclic Reactions T Kaacutelai J Jekı K Hideg
2596 Glycosylations of Tertiary Alcohols Synthesis of Fully Protected Disaccharides with Sterically Demanding Groups Attached to the Sugar Core A Holkenbrink J B Vicente D B Werz
2605 Copper-Catalyzed [13]-Dipolar Cycloaddition for the Synthesis of Macrocycles Containing Acyclic Aromatic and Steroidal Moieties G V Latyshev M S Baranom A V Kazantsev A D Averin N V Lukashev I P Beletskaya
2616 Aryl Ring Migration Reaction in the Synthesis of 24-Diaryl-4H-31-benzothiazines A V Butin F A Tsiunchik V T Abaev A V Gutnov D A Cheshkov
2627 Hydrogenation of β-N-Substituted and β-NN-Disubstituted Enamino Esters in the Presence of Iridium(I) Catalyst H Hebbache Z Hank C Bruneau J-L Renaud
2634 Stereoselective Olefination Reactions Promoted by Rieke Manganese J M Concelloacuten H Rodriacuteguez-Solla V del Amo P Diacuteaz
2646 Synthesis of Piperidinones through a Radical Cascade E Godineau Y Landais
2650 Asymmetric Organic Synthesis with Enzymes Edited by V Gotor I Alfonso E Garciacutea-Urdiales Reviewed by Steve Collier
XVII Forthcoming Articles
no 16 2651 Synthesis of Spirocyclic Ethers S Rosenberg R Leino 2674 Bimetallic PalladiumndashPlatinum-on-Carbon-Catalyzed HndashD Exchange
Reaction Synergistic Effect on Multiple Deuterium Incorporation T Maegawa N Ito K Oono Y Monguchi H Sajiki
2679 Efficient Copper-Catalyzed Synthesis of 2-Amino-4(3H)-quinazolinone and 2-Aminoquinazoline Derivatives X Huang H Yang H Fu R Qiao Y Zhao
2689 Synthesis and Chemoselective N- and O-Alkylation of Thiadiazolopyrimidine Nucleosides and Uridines A M L Hossion R Islam R K Kandahary T Nagamatsu
2697 Facile and Efficient Synthesis of a New Class of Indole-Substituted Pyridine Derivatives via One-Pot Multicomponent Reactions K Zhao X-P Xu S-L Zhu D-Q Shi Y Zhang S-J Ji
2709 Studies toward a Total Synthesis of Rhizoxin D Stereoselective Preparation of the C11ndashC19 Fragment S Padakanti C K Kumar E Ashok P Das
2715 A Short Synthesis of Enantiomeric Phytoprostanes B1 Type I W Perlikowska M Mikołajczyk
2719 Chemistry of Polyhalogenated Nitrobutadienes Part 7 A Novel Synthetic Access to Chlorinated Nitrile Oxides E Nutz V A Zapolrsquoskii D E Kaufmann
2725 Microwave-Assisted Silver(I)-Mediated Selective O-Alkylation of Aromatic Imidate Systems B K Singh C Cavalluzzo M De Maeyer Z Debyser V S Parmar E Van der Eycken
2729 Iodogen A Novel Reagent for the Oxidation of Urazoles under Heterogeneous Conditions A Khoramabadi A Shiri M A Zolfigol S Mallakpour
2733 An Unprecedented Synthesis of Eight-Membered-Ring Cyclic Thioimidic Esters by a Three-Component Reaction A Alizadeh R Hosseinpour
2737 A Novel Diastereoselective Synthesis of β-Phosphonato Unsaturated Thioimidates A Alizadeh N Zohreh
2741 Synthesis of 21-Benzisoxazoles by Nucleophilic Substitution of Hydrogen in Nitroarenes Activated by the Azole Ring N T Pokhodylo Y O Teslenko V S Matiychuk M D Obushak
2749 A Facile Synthesis of Two Series of Multifunctional Carbon Compounds from αα-Dihalo Ketones Using Allylsamarium Bromide X Liu S Zhang J Di
2756 Stereocontrolled Formation of Protected Aminodeoxyalditols from Simple Carbohydrate Precursors by Debenzylating Cycloetherification Y Jiang Z Fang Q Zheng H Jia J Cheng B Zheng
2761 trans-Stilbene as a Starting Material for the Synthesis of Tamoxifen Based on Palladium-Catalyzed Cross-Coupling Reactions C M Nunes J Limberger S Poersch M Seferin A L Monteiro
2766 Synthesis and Biological Evaluation of 6-Substituted Purinylcarbanucleosides with a Cyclopenta[b]thiophene Pseudosugar P Abeijoacuten J M Blanco O Caamantildeo F Fernaacutendez M D Garciacutea X Garciacutea-Mera J E Rodriacuteguez-Borges J Balzarini E De Clercq
2773 Synthesis and Electrochemical Signature of Novel Norbornyl-ferrocene Hybrids F A Khan S K Upadhyay
2778 A Regioselective TsujindashTrost Pentadienylation of 3-Allyltetronic Acid R Schobert B Barnickel
2785 Copper(I)-Catalyzed CarylndashCalkynyl Bond Formation of Aryl Iodides with Terminal Alkynes K G Thakur G Sekar
2790 Aminolysis of Epoxides Using Iridium Trichloride as an Efficient Catalyst J Agarwal A Duley R Rani R K Peddinti
2797 Preparation of Several Active N-Chloro Compounds from Trichloroisocyanuric Acid A Shiri A Khoramabadi-zad
2802 The First Mineral-Catalyzed One-Pot [3+1+2] Coupling Protocol for Multifunctionalized Fused-Ring Pyrimidines L D S Yadav A Rai
2809 Efficient Synthesis of Tetrahydro-β-carbolin-1-one and Dihydroisoquinolin-1-one Derivatives as Versatile Intermediates K E Judd M F Mahon L Caggiano
2818 A Concise Synthesis of ortho-Iodobenzyl Alcohols via Addition of ortho-Iodophenyl Grignard Reagent to Aldehydes and Ketones J Cvengroš D Stolz A Togni
XIII Forthcoming Articles
no 17 2825 Reactivity of Oxazol-5-(4H)-ones and Their Application toward Natural
Product Synthesis N M Hewlett C D Hupp J J Tepe 2840 Towards the Total Synthesis of 3-Hydroxyvibsanin E B D Schwartz
J R Denton P V Bernhardt H M L Davies C M Williams 2847 Structure Investigations of (ent)-Cladospolide D by De Novo Synthesis and
Kinetic and Thermodynamic Isomerization Y Xing J H Penn G A OrsquoDoherty
2855 New Applications of PhI(OAc)2 in Synthesis Total Synthesis and SAR Development of Potent Antitumor Natural Product PsymberinIrciniastatin A N Shao X Huang A Palani R Aslanian A Buevich J Piwinski R Huryk C Seidel-Dugan
2873 Total Synthesis of Largazole ndash Devolution of a Novel Synthetic Strategy B Wang C J Forsyth
2881 Formal Total Synthesis of Palmerolide A J Jaumlgel M E Maier 2893 Total Synthesis of Bongkrekic Acid via Sequential SuzukindashMiyaura Coupling
Reactions M Kanematsu M Shindo M Yoshida K Shishido 2905 Stereodivergent Approach to Both C28a-syn and C28a-anti Relative
Stereochemical Manifolds in the Lepadin Family via a TiCl4-Promoted G Li L J Carlson I K Sagamanova B W Slafer R P Hsung C Gilardi H M Sklenicka N Sydorenko
2915 Enantioselective Aldol Reaction of Tetrasubstituted Ketene Silyl Acetals with Achiral Aldehydes for the Construction of Asymmetric Tertiary Alcohols An Application for the Divergent Total Syntheses of Buergerinins F and G I Shiina T Iizumi Y-s Yamai Y-i Kawakita K Yokoyama Y-k Yamada
2927 Second-Generation Biomimetic Total Synthesis of Chaetominine A Coste G Karthikeyan F Couty G Evano
2935 Total Synthesis of (+)-Fostriecin and (+)-Phoslactomycin B S Shibahara M Fujino Y Tashiro N Okamoto T Esumi K Takahashi J Ishihara S Hatakeyama
2954 Stereochemical Assignments of the Chlorinated Residues in Victorin C A C Durow C Butts C L Willis
2963 Studies of the Asymmetric Total Synthesis of Clavilactone D by the lsquoLariatrsquo Cyclization Strategy T Yoshimitsu S Nojima M Hashimoto K Tsukamoto T Tanaka
2970 Total Synthesis of the Leucetta-Derived Alkaloid Calcaridine A P B Koswatta R Sivappa H V R Dias C J Lovely
2983 Formal Synthesis of Salinosporamide A Starting from D-Glucose T Momose Y Kaiya J-i Hasegawa T Sato N Chida
2992 Synthesis of Bioactive Natural Products by Asymmetric syn- and anti-Aldol Reactions A K Ghosh Z L Dawson
no 18 3003 Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural
Products B M Trost M K Brennan 3026 One-Pot Synthesis of Furo[34-b]pyridin-5(7H)-ones from 2-
Bromopyridine-3-carboxylic Acid and Carbonyl Compounds K Kobayashi T Kozuki H Konishi
3029 Iodocyclization of N-[2-(Methylthio)phenyl]propiolamides Selective Synthesis of 3-Iodo-15-benzothiazepin-4-ones T-S Jiang X-G Zhang J-H Li
3039 A Facile Synthetic Method for Fluorine-Containing 17-Phenanthrolines Pyridine-Ring Formation Reaction of N-Propargyl-68-bis(trifluoroacetyl)-quinolin-5-amine with Various Nucleophiles D Shibata E Okada M Hinoshita M Meacutedebielle
3047 Enantiotopic Discrimination in Palladium-Mediated Nucleophilic Substitutions on Achiral Substrates Chiral Ligand versus Chiral Nucleophile O Jacquet F Charnay J-C Fiaud J Ollivier
3051 Studies on the Chemistry of 2-[3-(2-Nitrophenyl)-2-oxopropyl]benzaldehydes Novel Syntheses of 5H-Benzo[b]carbazole-611-diones and Indolo[12-b]isoquinoline-611-diones M Fernaacutendez
3061 Studies on the C22ndashC23 Aldol Coupling of Spirangien M Lorenz N Bluhm M Kalesse
3067 One-Pot Synthesis of N-Alkyl Purine Pyrimidine and Azole Derivatives from Alcohols using Ph3PCCl4 A Rapid Route to Carboacyclic Nucleoside Synthesis M N Soltani Rad A Khalafi-Nezhad S Behrouz Z Asrari M Behrouz Z Amini
3077 Synthesis of 2-Amino-34-dihydroquinazolines and Imidazo[21-b]quinazoline-2-ones A Mishra S Batra
3089 Studies on the Reaction of Diimines with Thiourea Synthesis and Solvent-Induced cistrans-Isomerization of 135-Triazinane-2-thiones B Kaboudin T Ghasemi T Yokomatsu
3094 Suzuki Coupling of Heteroaromatic Chlorides Using Highly Electron-Donating ClickPhos Ligands S M Spinella Z-H Guan J Chen X Zhang
3099 Reaction of NN-Dioxyenamines with Anhydrides of Carboxylic and Sulfonic Acids A New Method for the Synthesis of a-Hydroxyoxime Derivatives A A Tabolin A V Lesiv S L Ioffe
3106 Directed ortho Metallation Chemistry and Phosphine Synthesis New Ligands for the SuzukindashMiyaura Reaction D B G Williams S J Evans H de Bod M S Mokhadinyana T Hughes
3113 New Functional Derivatives of 9-Phenylquinine P J Boratyński J SkarŜewski
3120 On the Synthesis of Asymmetric and Dissymmetric Amino Analogues of Troumlgerrsquos Base J Artacho K Waumlrnmark
3127 Synthesis of Polycyclic Sultams by Palladium-Catalyzed Intramolecular Cyclization K C Majumdar S Mondal N De
3136 Synthesis of Functionalized L-Cysteine and L-Methionine by Reaction with Electron-Deficient Acetylenes B A Trofimov A G Malrsquokina O A Shemyakina V V Nosyreva A P Borisova S S Khutsishvili L B Krivdin
3143 A lsquoClickrsquo Approach to the Synthesis of 3-[2-(1-Alkyltriazol-4-yl)ethyl]indoles M Petrini R R Shaikh
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
1386 Stereoselective Total Syntheses of Leiocarpin A and (ndash)-Galantinic Acid Starting from D-Mannitol K Nagaiah D Sreenu K V Purnima R S Rao J S Yadav
1393 A Facile Mild Deprotection Protocol for 13-Dithianes and 13-Dithiolanes with 30 Hydrogen Peroxide and Iodine Catalyst in Aqueous Micellar System N C Ganguly S K Barik
1400 Rhodium-Catalyzed Gram-Scale Synthesis of Highly Substituted Pyridine Derivatives K Parthasarathy C-H Cheng
1403 Enantioselective Synthesis of (R)-Propylene Carbonate from Ethyl (S)-Lactate J M Whitaker R C Ronald
XIII Forthcoming Articles
no 9 1405 Transition-Metal-Catalyzed Site-Selective Cross-Coupling of Di- and
Polyhalogenated Compounds J-R Wang K Manabe 1428 An Improved Synthesis of (4-4-Hydroxy-3-isopropyl-5-[(4-nitrophenyl)
ethynyl]benzyl-35-dimethylphenoxy)acetic Acid (NH-3) M B Gopinathan K S Rehder
1431 Copper-Catalyzed Tandem CndashN Bond Formation Reaction Selective Synthesis of 2-(Trifluoromethyl)benzimidazoles M-W Chen X-G Zhang P Zhong M-L Hu
1437 Synthesis and Thermochemical Properties of Stereoisomeric Dihydroxy- and Tetrahydroxyalkylammonium Salts M Thomas L Rothman J Hatcher P Agarkar R Ramkirath S Lall-Ramnarine R Engel
1445 Preparation of 5-Substituted 2-(2-Alkylaryl-1H-imidazol-4-yl)oxazoles and 5-Substituted 2-(2-Alkylarylthiazol-4-yl)oxazoles by Utilizing 5-Substituted 2-(2-Bromo-11-diethoxyethyl)oxazole as a Synthon D R St Laurent J L Romine
1459 Novel and Efficient Methods for the Synthesis of Symmetrical Trisulfides A Kertmen S Lach J Rachon D Witt
1463 An Environmentally Benign Electrochemical Process for the Reduction of Carboxylic Acid Hydrazides to Amides M Mentel M J Beier R Breinbauer
1469 Synthesis of 1-Chloroalkynes from Alkynylsilanes Using Trichloroisocyanuric Acid as Chlorinating Agent M H Vilhelmsen A S Andersson M B Nielsen
1473 A Convenient Approach to Enantioenriched Cyclopropanes Bearing Electron-Withdrawing Functionalities H Krawczyń K Wąsek J Kędzia
1477 Synthesis of Cyclopropenes via 12-Elimination of Bromocyclopropanes Catalyzed by Crown Ether W M Sherrill R Kim M Rubin
1485 A Base-Catalysed One-Pot Three-Component Coupling Reaction Leading to Nitrosubstituted Pyrroles I R Baxendale C D Buckle S V Ley L Tamborini
1494 Synthesis of 4-Alkylidene-4H-31-benzoxazine Derivatives by Acid-Catalyzed Cyclization of 2-Isocyanophenyl Ketones in the Presence of a Vinyl Ether K Kobayashi Y Okamura H Konishi
1499 Synthesis of Higher Helicenes via Olefin Metathesis and CndashH Activation J Cocircteacute S K Collins
1506 Azido- and Ethynyl-Substituted 2262-Terpyridines as Suitable Substrates for Click Reactions A Winter A Wild R Hoogenboom M W M Fijten M D Hager R-A Fallahpour U S Schubert
1513 Synthesis of 2-(Arylamino)ethanethiols via Lewis Acid Catalyzed Aminolysis of 22-Dimethylthiirane as Precursors of the 14-Benzothiazine Nucleus R Spogli S Sabatini G Manfroni O Tabarrini V Cecchetti
1520 Iron(III) Chloride A Versatile Catalyst for the Practical Synthesis of 3-Sulfenylindoles J S Yadav B V S Reddy Y J Reddy K Praneeth
1525 Organocatalytic Enantioselective Conjugate Addition of 2-Fluoromalonate to Nitroolefins Direct Synthesis of Chiral Fluorinated γ-Nitro Carboxylic Acid Derivatives H Li L Zu H Xie W Wang
1531 Asymmetric Transfer Hydrogenation of Ketimines with Trichlorosilane Structural Studies Z Zhang P Rooshenas H Hausmann P R Schreiner
1545 Prolinol Sulfinyl Ester Derivatives Organocatalytic Michael Addition of Ketones to Nitroolefins under Neat Conditions X Zeng G Zhong
1551 Asymmetric Oxidations of Electron-Poor Alkenes Promoted by the β-Amino AlcoholTBHP System A Russo A Lattanzi
1557 Enantioselectivity Switch in Direct Asymmetric Aminoxylation Catalyzed by Binaphthyl-Based Chiral Secondary Amines T Kano A Yamamoto F Shirozu K Maruoka
1564 Enantioselective Conjugate Addition of N-Heterocycles to αβ-Unsaturated Ketones Catalyzed by Chiral Primary Amines G Luo S Zhang W Duan W Wang
1573 Sulfonyl Hydrazine as New Functionality in Organocatalysis Camphorsulfonyl Hydrazine Catalyzed Enantioselective Aza-Michael Addition L-Y Chen H He B-J Pei W-H Chan A W M Lee
1578 Conversion of Primary Alcohols and Aldehydes into Methyl Esters by Ruthenium-Catalysed Hydrogen Transfer Reactions N A Owston T D Nixon A J Parker M K Whittlesey J M J Williams
1582 Addendum and Erratum XVII Forthcoming Articles
no 10 1583 Organocatalytic Formation of Quaternary Stereocenters M Bella
T Gasperi 1615 Regioselective Synthesis of 5H-Thiazolo[32-a]pyrimidin-5-ones from
MoritandashBaylisndashHillman Adduct Acetates under Solvent-Free and Base-Free Conditions W Zhong B Guo F Lin Y Liu W Su
1623 First Synthesis of 5-Cyanosalicylates by Formal [3+3] Cyclocondensations of 13-Bis(silyloxy)-13-butadienes A Riahi O Fatunsin M Shkoor R Dede H Reinke C Fischer P Langer
1635 Reaction of Isocyanides Dialkyl Acetylenedicarboxylates and a-Keto Lactones Unexpected Participation of an Ester Carbonyl Group in the Isocyanide-Based Three-Component Reaction A A Esmaeili H Vesalipoor
1639 An Efficient and Chemoselective Synthesis of 16-Naphthyridines and Pyrano[32-c]pyridines under Microwave Irradiation Z-G Han S-J Tu B Jiang S Yan X-H Zhang S-S Wu W-J Hao X-D Cao F Shi G Zhang N Ma
1647 N-Activation of N-Arylimidazoles Facile Syntheses of N-Alkyl-N-arylimidazolium Iodides from Less Expensive Chloro Substrates A M Oertel V Ritleng M J Chetcuti
1651 Synthesis of Polyhalogenated 2-(Phenylamino)pyridines by Thermal Amination Reactions S R Waldvogel A Faust W Barkmann R Froumlhlich O Wolff
1655 Cyanide Ion Promoted Addition of Acylphosphonates to Diethyl Cyanophosphonate Synthesis of Phosphonocyanohydrin O-Phosphates A S Demir A Aybey M Emrullahoglu
1659 Straightforward and Scalable Synthesis of Orthogonally Protected 37-Diazabicyclo[410]heptane H Schramm M Pavlova C Hoenke J Christoffers
1663 Hypervalent Iodine Mediated Oxidation of 12-Diaminobenzimidazole and Its Schiff Bases Efficient Synthesis of 3-Amino-124-benzotriazine and 2-Aryl-124-triazolo[15-a]benzimidazoles A Kumar M Parshad R K Gupta D Kumar
1667 Synthesis of the Reported Protoberberine Gusanlung D P B Wakchaure S Easwar N P Argade
1673 2-(Azidomethyl)arylboronic Acids in the Synthesis of Coumarin-Type Compounds M I Naumov A V Nuchev N S Sitnikov Y B Malysheva A S Shavyrin I P Beletskaya A E Gavryushin S Combes A Y Fedorov
1683 Asymmetric Synthesis of 12-anti-Disubstituted Taurine Derivatives D Enders D Iffland G Raabe
1689 A Novel One-Pot Three-Component Synthesis of 5-Imino-2358-tetrahydropyrazolo[12-a]pyridazin-1-one Derivatives B Qian M-J Fan Y-X Xie L-Y Wu Y Shi Y-M Liang
1694 One-Portion Synthesis of 2-Acetoxy Carbonyl Compounds from Aldehydes by Using an Acetylated Masked Acyl Cyanide H Nemoto T Kawamura K Kitasaki K Yatsuzuka M Kamiya Y Yoshioka
1703 Synthesis of 9-Anthryl Ethers from trans-910-Dihydro-910-dimethoxyanthracene by Acid-Catalyzed Transetherification K S Jang H Y Shin D Y Chi
1708 Efficient Synthesis of Azo Dye Labeled Terpenes Sugars and Steroids Using N-(4-Arylazobenzoyl)-1H-benzotriazoles A R Katritzky S R Tala N E Abo-Dya Z K Abdel-Samii
1715 Tandem CH-ActivationndashImine-Formation Reaction A New Route to Imidazo[21-a]phthalazines A Heim-Riether K R Gipson
1720 A Convenient and Efficient α-Sulfenylation of Carbonyl Compounds E Okragla S Demkowicz J Rachon D Witt
1725 Stereoselective Synthesis of β-Branched Phenylalanine Derivatives via Chelate-Claisen Rearrangement C Quirin U Kazmaier
1732 Catalyst-Free and Base-Free Water-Promoted SNAr Reaction of Heteroaryl Halides with Thiols B Sreedhar P S Reddy M A Reddy
1739 Convenient Methods for Synthesis of C2-Symmetric Diphenyltetrahydrothiophenes M Periasamy G Ramani G P Muthukumaragopal
1744 Highly Diastereoselective Conjugate AdditionndashElimination of Chiral Nickel(II) Glycinate with Activated Allylic Acetates for Asymmetric Synthesis of Glutamic Acid Derivatives J Wang J Shi X Zhang D Lin H Jiang H Liu
1753 Synthesis of 36-Dimethoxybenzene-12-diamine and of 47-Dimethoxy-2-methyl-1H-benzimidazole T Besset C Morin
1757 An Inexpensive Procedure for Reductive Aminations Using Dimethylamineborane on Millimolar and Molar Scale R Ortmann M Schlitzer
1760 Classics in Stereoselective Synthesis Edited by E M Carreira L Kvaerno Reviewed by Rolf Breinbauer
XV Forthcoming Articles
no 11 1761 Transition-Metal-Catalyzed Enantioselective Synthesis of Compounds with
Non-Centrochirality M Ogasawara S Watanabe 1786 One-Pot Synthesis of 3-Acyl-2-(alkylsulfanyl)indoles and 2-(Alkylsulfanyl)-
indole-3-carboxylates from (2-Isocyanophenyl)methyl Ketones or (2-Isocyanophenyl)acetates S Fukamachi H Konishi K Kobayashi
1791 Efficient and Recyclable Phthalocyanine-Based Sensitizers for Photooxygenation Reactions H Xu W-K Chan D K P Ng
1797 A Facile and Practical One-Pot Synthesis of β-Oxo Thioamides from β-Oxo Amides and Isothiocyanates P Huang D Xiang Y Zhou Y Liang T Na D Dong
1801 Microwave-Promoted Solid-Acid-Catalyzed One-Pot Synthesis of Phthalazinones V M Outerbridge S M Landge H Tamaki B Toumlroumlk
1807 Benzylic Brominations with N-Bromosuccinimide in (Trifluoromethyl)-benzene D Suarez G Laval S-M Tu D Jiang C L Robinson R Scott B T Golding
1811 Synthesis of Thioflavanone and Flavanone Derivatives by Cyclization of Chalcones W Konieczny M Konieczny
1815 A New and Expedient Total Synthesis of Ochratoxin A and d5-Ochratoxin A B Gabriele M Attya A Fazio L Di Donna P Plastina G Sindona
1821 Synthesis of Benzopyrrolizidinones by NorrishndashYang Cyclization of 3-(Acylmethyl)-2-alkylisoindol-1-ones J Wu W Zhang C Wang
1829 Reactions of MoritandashBaylisndashHillman Acetates with Huisgen Zwitterions A Novel Strategy for the Synthesis of β-Amino Acid Derivatives A Jose R R Paul R Mohan S C Mathew A T Biju E Suresh V Nair
1834 Peracetylated β-Allyl C-Glycosides of D-Ribofuranose and 2-Deoxy- D-ribofuranose in the Chemical Literature Until Now Mirages in the Literature H Otero Martinez H Reinke D Michalik C Vogel
1841 Core-Tetrasubstituted Naphthalene Diimides by Stille Cross-Coupling Reactions and Characterization of Their Optical and Redox Properties S-L Suraru F Wuumlrthner
1846 A Practical Synthesis of Indole-Based Heterocycles Using an Amidoaluminum-Mediated Strategy R Todd M M Hossain
1851 Synthesis of Fluorinated Pyrrolo[23-b]pyridine and Pyrrolo[23-d]pyrimidine Nucleosides V O Iaroshenko Y Wang D V Sevenard D M Volochnyuk
1858 Recyclization Reactions of 5-Formyl-13-dimethyluracil with Electron-Rich Amino Heterocycles A P Mityuk D M Volochnyuk S V Ryabukhin A S Plaskon A Shivanyuk A A Tolmachev
1865 Facile Synthesis of Fluorinated 1-Desazapurines V O Iaroshenko D V Sevenard D M Volochnyuk Y Wang A Martiloga A O Tolmachev
1876 A Practical Synthesis of 3-Diethoxyphosphoryl-12-pyridazine Derivatives J-C Monbaliu J Marchand-Brynaert
1881 Enantioselective Reduction of Prochiral Ketones Employing Sprouted Pisum sativa as Biocatalyst J S Yadav B V S Reddy C Sreelakshmi A B Rao
1886 Application of Phenolate Ion Mediated Intramolecular Epoxide Ring Opening in the Enantioselective Synthesis of Functionalized 23-Dihydrobenzofurans and 1-Benzopyrans S K Dinda S K Das G Panda
1897 Complementary Synthetic Approaches to Constitutionally Diverse N-Aminoalkylated Isoindolinones Application to the Synthesis of Falipamil and 5-HT1A Receptor Ligand Analogues M Lorion A Couture E Deniau P Grandclaudon
1904 Selective Deprotection of Silyl Ethers with Sodium Periodate J Li D Menche
1909 Micellar Solution of Sodium Dodecyl Sulfate (SDS) Catalyzes KabacknikndashFields Reaction in Aqueous Media S Sobhani A Vafaee
1916 Convenient Methods for the Synthesis of a Library of Hemilabile Phosphines M V Jimeacutenez J J Peacuterez-Torrente M I Bartolomeacute L A Oro
1923 Terminal Aziridines by Addition of Grignard Reagents or Organoceriums to an (α-Chloro)sulfinylimine D M Hodgson J Kloesges B Evans
1933 A Robust Synthesis of Nε-(Carboxymethyl)-L-lysine (CML) R Csuk S Stark A Barthel R Kluge D Stroumlhl
1935 One-Pot Curtius Rearrangement Processes from Carboxylic Acids O Leogane H Lebel
XV Forthcoming Articles
no 12 1941 The Chemistry of Deprotonated α-Aminonitriles T Opatz 1960 An Efficient Synthesis of Tetraalkyl 2345-Thiophenetetracarboxylate
Derivatives A Alizadeh R Hosseinpour 1963 Facile Deprotection of Bulky (Trialkylsilyl)acetylenes with Silver Fluoride
S Kim B Kim J In 1969 Highly Efficient and Reusable Ionic Liquids for the Catalyzed
Hydroamination of Alkenes with Sulfonamides Carbamates and Carboxamides L Yang L-W Xu C-G Xia
1975 Synthesis of 2391016172324-Octasubstituted Phthalocyaninatozinc(II) Complexes Mediated by Reductive Agents G A Gauna A C Monsalvo J Awruch
1979 A Short and Efficient Synthesis of 3-2-[2-(Bromomethyl)thiazol-4-yl]-ethynyl-5-fluorobenzonitrile A Precursor for PET Radioligand [18F]SP203 M B Gopinathan C Jin K S Rehder
1983 Synthesis of a Substituted Benzazepin-2-one Dihydrate S K Boini R K Vaid K P Moder D Mitchell
1987 Synthesis of Novel Trisubstituted Imidazolines F J Lakner M A Parker B Rogovoy A Khvat A Ivachtchenko
1991 A Novel Synthesis of N-But-3-enyl-α- and β-Amino Acids T T Van Nguyen R T C Brownlee A B Hughes
1999 Synthesis of Substituted 5-(3-Hydroxypropyl)pyrrolidin-2-ones and Pyrrolizidinones from Nitroethane via C3 Functionalized 56-Dihydro-4H-12-oxazines A Novel Approach to Some Analogues of the Antidepressant Rolipram A Yu Sukhorukov A V Lesiv Y A Khomutova S L Ioffe V A Tartakovsky
2009 Chiral Cyclobutanols and Cyclopentane Dimers via Samarium(II) Iodide Induced Keto-Olefin Cyclisations of Carbohydrate-Derived Unsaturated Ketones D B G Williams J Caddy K Blann J J C Groveacute C W Holzapfel
2015 Synthesis of Perfluoroalkylthio-Substituted Ferrocenes C Rhode J Lemke M Lieb N Metzler-Nolte
2019 Functionalization of Polyhedral Oligomeric Silsesquioxane (POSS) via Nucleophilic Substitution M Dutkiewicz H Maciejewski B Marciniec
2025 A Novel Synthesis of Aryl Mesylates via One-Pot DemethylationndashMesylation of Aryl Methyl Ethers Using a Mixture of Phosphorus Pentoxide in Methanesulfonic Acid B Kaboudin Y Abedi
2029 Anionic Cyclization of (NN-Dimethylamino)[2-(prop-2-yn-1-yloxy)aryl]-acetonitriles T Zdrojewski J Musielak A Jończyk
2035 Strecker-Type Reaction Catalyzed by Carboxylic Acids in Aqueous Media Z Xie G Li G Zhao J Wang
2040 Synthesis of Novel Structurally Simplified Estrogen Analogues with Electron-Donating Groups in Ring A L F Tietze C A Vock I K Krimmelbein L Nacke
2061 On the Resolution of Secondary Phosphine Oxides via Diastereomeric Complex Formation The Case of tert-Butylphenylphosphine Oxide J Holt A M Maj E P Schudde K M Pietrusiewicz L Sieroń W Wieczorek T Jerphagnon I W C E Arends U Hanefeld A J Minnaard
2066 Enantioselective Copper-Catalyzed Conjugate Addition of Dimethylzinc to 5-(1-Arylalkylidene) Meldrumrsquos Acids A Wilsily T Lou E Fillion
2073 SuzukindashMiyaura Coupling Reactions Using Phosphite Ligands M Jang Y Jo I-K Oh H M Jung S Lee
2076 Synthesis of 2-Methylindoline- and 2-Methyl-1234-tetrahydroquinoline-Derived Phosphoramidites and Their Applications in Iridium-Catalyzed Allylic Alkylation of Indoles W-B Liu H He L-X Dai S-L You
2083 Stereocontrolled Synthesis of 13-Amino Alcohols by Reduction of Substituted 2-1-[(tert-Butylsulfinyl)amino]alkylcyclohexanones J C Gonzaacutelez-Goacutemez F Foubelo M Yus
2089 Tunable Phosphoramidite Ligands for Asymmetric Hydrovinylation Ligands par excellence for Generation of All-Carbon Quaternary Centers C R Smith H J Lim A ZhangT V RajanBabu
2101 Copper-Catalyzed Asymmetric Ring-Opening Reaction of Oxabenzonorbornadienes with Grignard and Aluminum Reagents R Millet L Gremaud T Bernardez L Palais A Alexakis
2113 A Simplified Synthesis of Takemotorsquos Catalyst A Berkessel B Seelig 2116 Pharmaceutical Substances Syntheses Patents and Applications of the
Most Relevant AIPs Edited by Axel Kleeman Juumlrgen Engel Bernhard Kutscher Dietmar Reichert Reviewed by I Agranat
XV Forthcoming Articles
no 13 2117 Recent Advances in the Aza-Claisen Rearrangement K C Majumdar
T Bhattacharyya B Chattopadhyay B Sinha 2143 A Novel and Convenient Synthesis of lsquoReversedrsquo Diamidino 25-Aryl- and
25-Azaheterocycle-Substituted Furans L Hu D W Boykin 2146 Efficient and General Preparation of Pyranostilbenes First Total Synthesis
of Artocarbene and Pawhuskin B B H Park Y R Lee W S Lyoo 2155 Mild Oxidation of Diarylacetylenes to 12-Diketones Using Oxone in
Trifluoroacetic Acid J-H Chu Y-J Chen M-J Wu 2163 One-Pot Microwave-Assisted Selective Azido ReductionTandem Cyclization
in Condensed and Solid Phase with Nickel Boride N Shankaraiah N Markandeya M Espinoza-Moraga C Arancibia A Kamal L Silva Santos
2171 Pyrrolo[321-ij]quinolin-4-one and Pyrrolo[321-ij]quinolin-6-one H McNab D J Nelson E J Rozgowska
2175 Practical Synthesis of 5-Substituted Tetrazoles under Microwave Irradiation J Roh T V Artamonova K Vaacutevrovaacute G I Koldobskii A Hrabaacutelek
2179 A Simple Method for the Synthesis of 3-Arylthieno[23-b]pyridines via Iodine-Mediated Cyclization of 3-(1-Arylalkenyl)-2-[(1-phenylethyl)sulfanyl]pyridines K Kobayashi D Nakamura Y Shiroyama S Fukamachi H Konishi
2184 Synthesis of Four Lysine-Linked Cereulide Analogues Showing Ionophoric Activity Towards Potassium Cations as Lead Compounds for Emetic Toxin-Detection by Immunoassays A Makarasen T Nishikawa M Isobe
2205 Synthesis of α-Aliphatic and β-Aromatic Substituted Taurines via Regioselective Ring Opening of Thiiranes with Ammonia H Yu S Cao L Zhang G Liu J Xu
2210 Stability of 5(6)-Carboxyfluorescein in Microwave-Assisted Synthesis of Fluorescein-Labelled O-Dimannosylated Peptides R Kowalczyk P W R Harris R P Dunbar M A Brimble
2223 Diversity-Oriented Synthesis of Functionalized Diaryl Sulfones by Regioselective [3+3] Cyclizations of 13-Bis(siloxy)buta-13-dienes with 2-(Arylsulfonyl)-3-ethoxy-2-en-1-ones Scope and Limitations M Shkoor A Riahi O Fatunsin H Reinke C Fischer P Langer
2236 Synthesis of Functionalized Salicylates by Formal [3+3] Cyclocondensation of 13-Bis(silyloxy)buta-13-dienes with 3-Alkoxy-2-en-1-ones G Mroszlig S Ladzik H Reinke A Spannenberg C Fischer P Langer
2249 Synthetic Approach to Alkoxy-β-(trifluoromethyl)styrenes and Their Application in the Synthesis of New Trifluoromethylated Heterocycles V M Muzalevskiy V G Nenajdenko A V Shastin E S Balenkova G Haufe
2260 o-Benzenedisulfonimide as a Powerful and Recyclable Organocatalyst for the Nazarov Reaction M Barbero S Cadamuro A Deagostino S Dughera P Larini E G Occhiato C Prandi S Tabasso R Vulcano P Venturello
2267 The Catalytic Potential of 4-Guanidinylpyridines in Acylation Reactions I Held E Larionov C Bozler F Wagner H Zipse
2278 Iron(III) Chloride in EthanolndashWater Highly Efficient Catalytic System for the Synthesis of Garcia Gonzalez Polyhydroxyalkyl- and C-Glycosylfurans L Nagarapu M V Chary A Satyender B Supriya R Bantu
2283 Ruthenium-Catalyzed Addition of Primary Amides to Alkynes A Stereoselective Synthesis of Secondary Enamides L J Gooszligen M Blanchot K S M Salih K Gooszligen
2289 Binaphthyl-Modified Quaternary Phosphonium Salts as Chiral Phase Transfer Catalysts Application to Asymmetric Amination of β-Keto Esters R He K Maruoka
X Table of Contents XI Forthcoming Articles
no 14 2293 Direct Methods for Stereoselective Polypropionate Synthesis A Survey
J Li D Menche 2316 Synthesis of Symmetrical Ketones from Grignard Reagents and
11-Carbonyldiimidazole D Bottalico V Fiandanese G Marchese A Punzi
2319 Synthesis of 45-Substituted Imidazoles by a Fast Condensation of 12-Diketones and Urotropine in Heterogeneous Medium G Bratulescu
2321 (Arylsulfonyl)acetones and -acetonitriles New Activated Methylenic Building Blocks for Synthesis of 123-Triazoles N T Pokhodylo V S Matiychuk M D Obushak
2324 A Safe Convenient and Efficient One-Pot Synthesis of α-Chloroketone Acetals Directly from Ketones Using Iodobenzene Dichloride J Yu C Zhang
2329 An Efficient Oxidative Conversion of Aldehydes into 2-Substituted 2-Oxazolines Using 13-Diiodo-55-dimethylhydantoin S Takahashi H Togo
2333 A Novel Procedure for the Synthesis of Benzo[b][18]naphthyridine-3-carboxylate Derivatives from MoritandashBaylisndashHillman Adduct Acetates W Zhong F Lin R Chen W Su
2341 An Improved Synthesis of 147-Triazacyclononanes (tacns) and 14710-Tetraazacyclododecanes (cyclens) J Huang Z Zhou T H Chan
2345 The Ullmann Coupling between 2-Chlorobenzoic Acids and Amino Acids A Valuable Reaction for Preparing 2-Substituted 1-Acetyl-1H-indol-3-yl Acetates J C Rodriguez Dominguez X Gang G Kirsch
2349 gem-Dibromomethyl Aromatics Efficient Aldehyde Equivalents in the KnoevenagelndashDoebner Reaction J K Augustine Y A Naik S Poojari N Chowdappa B S Sherigara K Areppa
2357 Synthesis of Novel α-Aminophosphonates Containing Adamantyl Fragment M M Kabachnik L I Minaeva I P Beletskaya
2361 Efficient Fluoride-Mediated Synthesis of 5-Amino-Substituted Isothiazoles Y S Zubenko V I Potkin
2365 Phosphine-Catalyzed Reaction of Cyanohydrins with Activated Alkynes A Siby O Loreau F Taran
2371 Sulfanyl-Substituted [3]Cumulenes and Buta-13-dienes from a Tetrakis(pyridinium)-Substituted Butadiene A Schmidt A Rahimi M Gjikaj
2379 Efficient Synthesis of 2-Substituted Pyrido[32-d]pyrimidines Involving SNAr and Palladium-Catalyzed Cross-Coupling Reactions A Tikad S Routier M Akssira J-M Leacuteger C Jarry G Guillaumet
2385 Novel Synthesis of Medium-Sized Heterocycles by Palladium-Catalyzed Intramolecular Heck Reaction via 9-endo-trig Mode of Cyclization K C Majumdar B Chattopadhyay
2393 Facile Synthesis of Fluorinated Benzofuro- and Benzothieno[23-b]pyridines α-Carbolines and Nucleosides Containing the α-Carboline Framework V O Iaroshenko Y Wang B Zhang D Volochnyuk V Ya Sosnovskikh
2403 Synthesis of Functionalized N-Vinyl Nitrogen-Containing Heterocycles S M M Lopes A M Beja M Ramos Silva J A Paixatildeo F Palacios T M V D Pinho e Melo
2408 Kumada Cross-Coupling of Aryl Grignard Reagents with Aryl Halides Catalyzed by an Immobilized Nickel Catalyst X Chen L Wang J Liu
2413 Highly Enantioselective Synthesis of Heteroaromatic Alcohols Catalyzed by Chiral DiaminodiphosphinendashRuthenium(II) Complexes W-Y Shen Y-Y Li Z-R Dong J-X Gao
2418 Concise Total Synthesis of (+)-Disparlure and its trans-Isomer Using Asymmetric Organocatalysis S-G Kim
2423 Rhodium Carbenoid Induced [12]-Migration in an L-Lyxo-Configured α-Diazo β-Keto Ester Synthesis of a New Griseolic Acid Analogue N N Bhujbal K S A Kumar D D Dhavale
2430 Synthesis of 5-Arylthio-3-hydroxyphthalates by the First [4+2] Cycloadditions of 3-Arylthio-1-silyloxy-13-butadienes with Dimethyl Acetylenedicarboxylate I Iqbal M Imran P Langer
2435 Synthesis of Highly Functionalized Proline Derivatives via a One-Pot MichaelSN-AdditionCyclization Approach U Kazmaier C Schmidt
2440 RhodiumGraphite-Catalyzed Hydrogenation of Carbocyclic and Heterocyclic Aromatic Compounds G Falini A Gualandi D Savoia
2447 Potassium [1-(tert-Butoxycarbonyl)-1H-indol-2-yl]trifluoroborate as an Efficient Building Block in Palladium-Catalyzed SuzukindashMiyaura Cross Couplings P Kassis V Beacuteneacuteteau J-Y Meacuterour S Routier
2454 Syntheses of Substituted Furans and Pyrroles by Platinum-Catalyzed Cyclizations of Propargylic Oxiranes and Aziridines in Aqueous Media M Yoshida M Al-Amin K Shishido
2467 Transition-Metal-Free Oxidative Homocoupling of Aryl Alkenyl and Alkynyl Grignard Reagents with TEMPO M S Maji A Studer
XIII Forthcoming Articles
no 15 2471 Advances in Synthetic Approaches for the Preparation of Combretastatin-
Based Anti-Cancer Agents R Singh H Kaur 2492 Synthesis of Unsymmetrical Ureas by Sulfur-Assisted Carbonylation with
Carbon Monoxide and Oxidation with Molecular Oxygen under Mild Conditions T Mizuno T Nakai M Mihara
2497 Ring-OpeningRecyclization Reactions of (Dimethylamino)propenoyl-Substituted Cyclopropanes Facile Synthesis of Halogenated Pyridin-2(1H)-ones R Zhang Y Zhou Y Liang Z Jiang D Dong
2501 Facile and Efficient Total Synthesis of Taspine B Cheng S Zhang L Zhu J Zhang Q Li A Shan L He
2505 Oligomeric Iodosylbenzene Sulfate A Convenient Hypervalent Iodine Reagent for Oxidation of Organic Sulfides and Alkenes M S Yusubov R Y Yusubova T V Funk K-W Chi V V Zhdankin
2509 Pyrrolidine-Based Organocatalysts for Enantioselective Michael Addition of Cyclohexanone to trans-β-Nitrostyrene A P Carley S Dixon J D Kilburn
2517 CundashAl Hydrotalcite An Efficient and Reusable Ligand-Free Catalyst for the Coupling of Aryl Chlorides with Aliphatic Aromatic and N(H)-Heterocyclic Amines B Sreedhar R Arundhathi P L Reddy M A Reddy M L Kantam
2523 Highly Efficient Synthesis of trans-βγ-Unsaturated a-Keto Amides C Allais T Constantieux J Rodriguez
2531 Gas-Phase Synthesis of N-Unsubstituted 3-Hydroxypyrroles and 1H-Pyrrol-3(2H)-ones L Hill G A Hunter S H Imam H McNab W J OrsquoNeill
2535 3-Hydroxy-1H-pyrrole L Hill S H Imam H McNab W J OrsquoNeill 2539 123-Thiadiazoles with Unsaturated Side Chains Synthesis
Polymerization and Photocrosslinking M Al-Smadi N Hanold H Kalbitz H Meier
2547 Synthesis of 1112-Didehydrodibenzo[ae]cycloocten-5(6H)-one A Strained Eight-Membered Alkyne S C Kornmayer F Rominger R Gleiter
2553 Stannous Chloride Dihydrate A Novel and Efficient Catalyst for the Synthesis of gem-Dihydroperoxides from Ketones and Aldehydes D Azarifar K Khosravi F Soleimanei
2557 Synthesis of a Novel Class of Azacrown Macrocycles and Lariat Crown Ethers Containing Two 124-Triazole Rings as Subunits N Foroughifar A Mobinikhaledi S Ebrahimi
2561 Enantioselective Synthesis of the 3C-Protease Inhibitor (ndash)-Thysanone by a StauntonndashWeinreb Annulation Strategy J Sperry T Y Yuen M A Brimble
2570 Stereoselective Synthesis of Unnatural β-Amino Acids from Nitroethane via 56-Dihydro-4H-12-oxazin-3-ylacetates A Yu Sukhorukov A V Lesiv O L Eliseev Y A Khomutova S L Ioffe
2579 A Versatile Unexpected One-Pot Regioselective Synthesis of a New Class of 13-Diazepinoindolones by Reaction of Pyranoindolones with Monosubstituted Ureas D Livadiotou C A Tsoleridis J Stephanidou-Stephanatou
2584 Synthesis of a Trisaccharide and a Tetrasaccharide from the Cell-Wall Lipopolysaccharides of Azospirillum brasilense S17 S Pandey S Ghosh A K Misra
2591 Synthesis of Isoindoline Nitroxides by Electrocyclic Reactions T Kaacutelai J Jekı K Hideg
2596 Glycosylations of Tertiary Alcohols Synthesis of Fully Protected Disaccharides with Sterically Demanding Groups Attached to the Sugar Core A Holkenbrink J B Vicente D B Werz
2605 Copper-Catalyzed [13]-Dipolar Cycloaddition for the Synthesis of Macrocycles Containing Acyclic Aromatic and Steroidal Moieties G V Latyshev M S Baranom A V Kazantsev A D Averin N V Lukashev I P Beletskaya
2616 Aryl Ring Migration Reaction in the Synthesis of 24-Diaryl-4H-31-benzothiazines A V Butin F A Tsiunchik V T Abaev A V Gutnov D A Cheshkov
2627 Hydrogenation of β-N-Substituted and β-NN-Disubstituted Enamino Esters in the Presence of Iridium(I) Catalyst H Hebbache Z Hank C Bruneau J-L Renaud
2634 Stereoselective Olefination Reactions Promoted by Rieke Manganese J M Concelloacuten H Rodriacuteguez-Solla V del Amo P Diacuteaz
2646 Synthesis of Piperidinones through a Radical Cascade E Godineau Y Landais
2650 Asymmetric Organic Synthesis with Enzymes Edited by V Gotor I Alfonso E Garciacutea-Urdiales Reviewed by Steve Collier
XVII Forthcoming Articles
no 16 2651 Synthesis of Spirocyclic Ethers S Rosenberg R Leino 2674 Bimetallic PalladiumndashPlatinum-on-Carbon-Catalyzed HndashD Exchange
Reaction Synergistic Effect on Multiple Deuterium Incorporation T Maegawa N Ito K Oono Y Monguchi H Sajiki
2679 Efficient Copper-Catalyzed Synthesis of 2-Amino-4(3H)-quinazolinone and 2-Aminoquinazoline Derivatives X Huang H Yang H Fu R Qiao Y Zhao
2689 Synthesis and Chemoselective N- and O-Alkylation of Thiadiazolopyrimidine Nucleosides and Uridines A M L Hossion R Islam R K Kandahary T Nagamatsu
2697 Facile and Efficient Synthesis of a New Class of Indole-Substituted Pyridine Derivatives via One-Pot Multicomponent Reactions K Zhao X-P Xu S-L Zhu D-Q Shi Y Zhang S-J Ji
2709 Studies toward a Total Synthesis of Rhizoxin D Stereoselective Preparation of the C11ndashC19 Fragment S Padakanti C K Kumar E Ashok P Das
2715 A Short Synthesis of Enantiomeric Phytoprostanes B1 Type I W Perlikowska M Mikołajczyk
2719 Chemistry of Polyhalogenated Nitrobutadienes Part 7 A Novel Synthetic Access to Chlorinated Nitrile Oxides E Nutz V A Zapolrsquoskii D E Kaufmann
2725 Microwave-Assisted Silver(I)-Mediated Selective O-Alkylation of Aromatic Imidate Systems B K Singh C Cavalluzzo M De Maeyer Z Debyser V S Parmar E Van der Eycken
2729 Iodogen A Novel Reagent for the Oxidation of Urazoles under Heterogeneous Conditions A Khoramabadi A Shiri M A Zolfigol S Mallakpour
2733 An Unprecedented Synthesis of Eight-Membered-Ring Cyclic Thioimidic Esters by a Three-Component Reaction A Alizadeh R Hosseinpour
2737 A Novel Diastereoselective Synthesis of β-Phosphonato Unsaturated Thioimidates A Alizadeh N Zohreh
2741 Synthesis of 21-Benzisoxazoles by Nucleophilic Substitution of Hydrogen in Nitroarenes Activated by the Azole Ring N T Pokhodylo Y O Teslenko V S Matiychuk M D Obushak
2749 A Facile Synthesis of Two Series of Multifunctional Carbon Compounds from αα-Dihalo Ketones Using Allylsamarium Bromide X Liu S Zhang J Di
2756 Stereocontrolled Formation of Protected Aminodeoxyalditols from Simple Carbohydrate Precursors by Debenzylating Cycloetherification Y Jiang Z Fang Q Zheng H Jia J Cheng B Zheng
2761 trans-Stilbene as a Starting Material for the Synthesis of Tamoxifen Based on Palladium-Catalyzed Cross-Coupling Reactions C M Nunes J Limberger S Poersch M Seferin A L Monteiro
2766 Synthesis and Biological Evaluation of 6-Substituted Purinylcarbanucleosides with a Cyclopenta[b]thiophene Pseudosugar P Abeijoacuten J M Blanco O Caamantildeo F Fernaacutendez M D Garciacutea X Garciacutea-Mera J E Rodriacuteguez-Borges J Balzarini E De Clercq
2773 Synthesis and Electrochemical Signature of Novel Norbornyl-ferrocene Hybrids F A Khan S K Upadhyay
2778 A Regioselective TsujindashTrost Pentadienylation of 3-Allyltetronic Acid R Schobert B Barnickel
2785 Copper(I)-Catalyzed CarylndashCalkynyl Bond Formation of Aryl Iodides with Terminal Alkynes K G Thakur G Sekar
2790 Aminolysis of Epoxides Using Iridium Trichloride as an Efficient Catalyst J Agarwal A Duley R Rani R K Peddinti
2797 Preparation of Several Active N-Chloro Compounds from Trichloroisocyanuric Acid A Shiri A Khoramabadi-zad
2802 The First Mineral-Catalyzed One-Pot [3+1+2] Coupling Protocol for Multifunctionalized Fused-Ring Pyrimidines L D S Yadav A Rai
2809 Efficient Synthesis of Tetrahydro-β-carbolin-1-one and Dihydroisoquinolin-1-one Derivatives as Versatile Intermediates K E Judd M F Mahon L Caggiano
2818 A Concise Synthesis of ortho-Iodobenzyl Alcohols via Addition of ortho-Iodophenyl Grignard Reagent to Aldehydes and Ketones J Cvengroš D Stolz A Togni
XIII Forthcoming Articles
no 17 2825 Reactivity of Oxazol-5-(4H)-ones and Their Application toward Natural
Product Synthesis N M Hewlett C D Hupp J J Tepe 2840 Towards the Total Synthesis of 3-Hydroxyvibsanin E B D Schwartz
J R Denton P V Bernhardt H M L Davies C M Williams 2847 Structure Investigations of (ent)-Cladospolide D by De Novo Synthesis and
Kinetic and Thermodynamic Isomerization Y Xing J H Penn G A OrsquoDoherty
2855 New Applications of PhI(OAc)2 in Synthesis Total Synthesis and SAR Development of Potent Antitumor Natural Product PsymberinIrciniastatin A N Shao X Huang A Palani R Aslanian A Buevich J Piwinski R Huryk C Seidel-Dugan
2873 Total Synthesis of Largazole ndash Devolution of a Novel Synthetic Strategy B Wang C J Forsyth
2881 Formal Total Synthesis of Palmerolide A J Jaumlgel M E Maier 2893 Total Synthesis of Bongkrekic Acid via Sequential SuzukindashMiyaura Coupling
Reactions M Kanematsu M Shindo M Yoshida K Shishido 2905 Stereodivergent Approach to Both C28a-syn and C28a-anti Relative
Stereochemical Manifolds in the Lepadin Family via a TiCl4-Promoted G Li L J Carlson I K Sagamanova B W Slafer R P Hsung C Gilardi H M Sklenicka N Sydorenko
2915 Enantioselective Aldol Reaction of Tetrasubstituted Ketene Silyl Acetals with Achiral Aldehydes for the Construction of Asymmetric Tertiary Alcohols An Application for the Divergent Total Syntheses of Buergerinins F and G I Shiina T Iizumi Y-s Yamai Y-i Kawakita K Yokoyama Y-k Yamada
2927 Second-Generation Biomimetic Total Synthesis of Chaetominine A Coste G Karthikeyan F Couty G Evano
2935 Total Synthesis of (+)-Fostriecin and (+)-Phoslactomycin B S Shibahara M Fujino Y Tashiro N Okamoto T Esumi K Takahashi J Ishihara S Hatakeyama
2954 Stereochemical Assignments of the Chlorinated Residues in Victorin C A C Durow C Butts C L Willis
2963 Studies of the Asymmetric Total Synthesis of Clavilactone D by the lsquoLariatrsquo Cyclization Strategy T Yoshimitsu S Nojima M Hashimoto K Tsukamoto T Tanaka
2970 Total Synthesis of the Leucetta-Derived Alkaloid Calcaridine A P B Koswatta R Sivappa H V R Dias C J Lovely
2983 Formal Synthesis of Salinosporamide A Starting from D-Glucose T Momose Y Kaiya J-i Hasegawa T Sato N Chida
2992 Synthesis of Bioactive Natural Products by Asymmetric syn- and anti-Aldol Reactions A K Ghosh Z L Dawson
no 18 3003 Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural
Products B M Trost M K Brennan 3026 One-Pot Synthesis of Furo[34-b]pyridin-5(7H)-ones from 2-
Bromopyridine-3-carboxylic Acid and Carbonyl Compounds K Kobayashi T Kozuki H Konishi
3029 Iodocyclization of N-[2-(Methylthio)phenyl]propiolamides Selective Synthesis of 3-Iodo-15-benzothiazepin-4-ones T-S Jiang X-G Zhang J-H Li
3039 A Facile Synthetic Method for Fluorine-Containing 17-Phenanthrolines Pyridine-Ring Formation Reaction of N-Propargyl-68-bis(trifluoroacetyl)-quinolin-5-amine with Various Nucleophiles D Shibata E Okada M Hinoshita M Meacutedebielle
3047 Enantiotopic Discrimination in Palladium-Mediated Nucleophilic Substitutions on Achiral Substrates Chiral Ligand versus Chiral Nucleophile O Jacquet F Charnay J-C Fiaud J Ollivier
3051 Studies on the Chemistry of 2-[3-(2-Nitrophenyl)-2-oxopropyl]benzaldehydes Novel Syntheses of 5H-Benzo[b]carbazole-611-diones and Indolo[12-b]isoquinoline-611-diones M Fernaacutendez
3061 Studies on the C22ndashC23 Aldol Coupling of Spirangien M Lorenz N Bluhm M Kalesse
3067 One-Pot Synthesis of N-Alkyl Purine Pyrimidine and Azole Derivatives from Alcohols using Ph3PCCl4 A Rapid Route to Carboacyclic Nucleoside Synthesis M N Soltani Rad A Khalafi-Nezhad S Behrouz Z Asrari M Behrouz Z Amini
3077 Synthesis of 2-Amino-34-dihydroquinazolines and Imidazo[21-b]quinazoline-2-ones A Mishra S Batra
3089 Studies on the Reaction of Diimines with Thiourea Synthesis and Solvent-Induced cistrans-Isomerization of 135-Triazinane-2-thiones B Kaboudin T Ghasemi T Yokomatsu
3094 Suzuki Coupling of Heteroaromatic Chlorides Using Highly Electron-Donating ClickPhos Ligands S M Spinella Z-H Guan J Chen X Zhang
3099 Reaction of NN-Dioxyenamines with Anhydrides of Carboxylic and Sulfonic Acids A New Method for the Synthesis of a-Hydroxyoxime Derivatives A A Tabolin A V Lesiv S L Ioffe
3106 Directed ortho Metallation Chemistry and Phosphine Synthesis New Ligands for the SuzukindashMiyaura Reaction D B G Williams S J Evans H de Bod M S Mokhadinyana T Hughes
3113 New Functional Derivatives of 9-Phenylquinine P J Boratyński J SkarŜewski
3120 On the Synthesis of Asymmetric and Dissymmetric Amino Analogues of Troumlgerrsquos Base J Artacho K Waumlrnmark
3127 Synthesis of Polycyclic Sultams by Palladium-Catalyzed Intramolecular Cyclization K C Majumdar S Mondal N De
3136 Synthesis of Functionalized L-Cysteine and L-Methionine by Reaction with Electron-Deficient Acetylenes B A Trofimov A G Malrsquokina O A Shemyakina V V Nosyreva A P Borisova S S Khutsishvili L B Krivdin
3143 A lsquoClickrsquo Approach to the Synthesis of 3-[2-(1-Alkyltriazol-4-yl)ethyl]indoles M Petrini R R Shaikh
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
no 9 1405 Transition-Metal-Catalyzed Site-Selective Cross-Coupling of Di- and
Polyhalogenated Compounds J-R Wang K Manabe 1428 An Improved Synthesis of (4-4-Hydroxy-3-isopropyl-5-[(4-nitrophenyl)
ethynyl]benzyl-35-dimethylphenoxy)acetic Acid (NH-3) M B Gopinathan K S Rehder
1431 Copper-Catalyzed Tandem CndashN Bond Formation Reaction Selective Synthesis of 2-(Trifluoromethyl)benzimidazoles M-W Chen X-G Zhang P Zhong M-L Hu
1437 Synthesis and Thermochemical Properties of Stereoisomeric Dihydroxy- and Tetrahydroxyalkylammonium Salts M Thomas L Rothman J Hatcher P Agarkar R Ramkirath S Lall-Ramnarine R Engel
1445 Preparation of 5-Substituted 2-(2-Alkylaryl-1H-imidazol-4-yl)oxazoles and 5-Substituted 2-(2-Alkylarylthiazol-4-yl)oxazoles by Utilizing 5-Substituted 2-(2-Bromo-11-diethoxyethyl)oxazole as a Synthon D R St Laurent J L Romine
1459 Novel and Efficient Methods for the Synthesis of Symmetrical Trisulfides A Kertmen S Lach J Rachon D Witt
1463 An Environmentally Benign Electrochemical Process for the Reduction of Carboxylic Acid Hydrazides to Amides M Mentel M J Beier R Breinbauer
1469 Synthesis of 1-Chloroalkynes from Alkynylsilanes Using Trichloroisocyanuric Acid as Chlorinating Agent M H Vilhelmsen A S Andersson M B Nielsen
1473 A Convenient Approach to Enantioenriched Cyclopropanes Bearing Electron-Withdrawing Functionalities H Krawczyń K Wąsek J Kędzia
1477 Synthesis of Cyclopropenes via 12-Elimination of Bromocyclopropanes Catalyzed by Crown Ether W M Sherrill R Kim M Rubin
1485 A Base-Catalysed One-Pot Three-Component Coupling Reaction Leading to Nitrosubstituted Pyrroles I R Baxendale C D Buckle S V Ley L Tamborini
1494 Synthesis of 4-Alkylidene-4H-31-benzoxazine Derivatives by Acid-Catalyzed Cyclization of 2-Isocyanophenyl Ketones in the Presence of a Vinyl Ether K Kobayashi Y Okamura H Konishi
1499 Synthesis of Higher Helicenes via Olefin Metathesis and CndashH Activation J Cocircteacute S K Collins
1506 Azido- and Ethynyl-Substituted 2262-Terpyridines as Suitable Substrates for Click Reactions A Winter A Wild R Hoogenboom M W M Fijten M D Hager R-A Fallahpour U S Schubert
1513 Synthesis of 2-(Arylamino)ethanethiols via Lewis Acid Catalyzed Aminolysis of 22-Dimethylthiirane as Precursors of the 14-Benzothiazine Nucleus R Spogli S Sabatini G Manfroni O Tabarrini V Cecchetti
1520 Iron(III) Chloride A Versatile Catalyst for the Practical Synthesis of 3-Sulfenylindoles J S Yadav B V S Reddy Y J Reddy K Praneeth
1525 Organocatalytic Enantioselective Conjugate Addition of 2-Fluoromalonate to Nitroolefins Direct Synthesis of Chiral Fluorinated γ-Nitro Carboxylic Acid Derivatives H Li L Zu H Xie W Wang
1531 Asymmetric Transfer Hydrogenation of Ketimines with Trichlorosilane Structural Studies Z Zhang P Rooshenas H Hausmann P R Schreiner
1545 Prolinol Sulfinyl Ester Derivatives Organocatalytic Michael Addition of Ketones to Nitroolefins under Neat Conditions X Zeng G Zhong
1551 Asymmetric Oxidations of Electron-Poor Alkenes Promoted by the β-Amino AlcoholTBHP System A Russo A Lattanzi
1557 Enantioselectivity Switch in Direct Asymmetric Aminoxylation Catalyzed by Binaphthyl-Based Chiral Secondary Amines T Kano A Yamamoto F Shirozu K Maruoka
1564 Enantioselective Conjugate Addition of N-Heterocycles to αβ-Unsaturated Ketones Catalyzed by Chiral Primary Amines G Luo S Zhang W Duan W Wang
1573 Sulfonyl Hydrazine as New Functionality in Organocatalysis Camphorsulfonyl Hydrazine Catalyzed Enantioselective Aza-Michael Addition L-Y Chen H He B-J Pei W-H Chan A W M Lee
1578 Conversion of Primary Alcohols and Aldehydes into Methyl Esters by Ruthenium-Catalysed Hydrogen Transfer Reactions N A Owston T D Nixon A J Parker M K Whittlesey J M J Williams
1582 Addendum and Erratum XVII Forthcoming Articles
no 10 1583 Organocatalytic Formation of Quaternary Stereocenters M Bella
T Gasperi 1615 Regioselective Synthesis of 5H-Thiazolo[32-a]pyrimidin-5-ones from
MoritandashBaylisndashHillman Adduct Acetates under Solvent-Free and Base-Free Conditions W Zhong B Guo F Lin Y Liu W Su
1623 First Synthesis of 5-Cyanosalicylates by Formal [3+3] Cyclocondensations of 13-Bis(silyloxy)-13-butadienes A Riahi O Fatunsin M Shkoor R Dede H Reinke C Fischer P Langer
1635 Reaction of Isocyanides Dialkyl Acetylenedicarboxylates and a-Keto Lactones Unexpected Participation of an Ester Carbonyl Group in the Isocyanide-Based Three-Component Reaction A A Esmaeili H Vesalipoor
1639 An Efficient and Chemoselective Synthesis of 16-Naphthyridines and Pyrano[32-c]pyridines under Microwave Irradiation Z-G Han S-J Tu B Jiang S Yan X-H Zhang S-S Wu W-J Hao X-D Cao F Shi G Zhang N Ma
1647 N-Activation of N-Arylimidazoles Facile Syntheses of N-Alkyl-N-arylimidazolium Iodides from Less Expensive Chloro Substrates A M Oertel V Ritleng M J Chetcuti
1651 Synthesis of Polyhalogenated 2-(Phenylamino)pyridines by Thermal Amination Reactions S R Waldvogel A Faust W Barkmann R Froumlhlich O Wolff
1655 Cyanide Ion Promoted Addition of Acylphosphonates to Diethyl Cyanophosphonate Synthesis of Phosphonocyanohydrin O-Phosphates A S Demir A Aybey M Emrullahoglu
1659 Straightforward and Scalable Synthesis of Orthogonally Protected 37-Diazabicyclo[410]heptane H Schramm M Pavlova C Hoenke J Christoffers
1663 Hypervalent Iodine Mediated Oxidation of 12-Diaminobenzimidazole and Its Schiff Bases Efficient Synthesis of 3-Amino-124-benzotriazine and 2-Aryl-124-triazolo[15-a]benzimidazoles A Kumar M Parshad R K Gupta D Kumar
1667 Synthesis of the Reported Protoberberine Gusanlung D P B Wakchaure S Easwar N P Argade
1673 2-(Azidomethyl)arylboronic Acids in the Synthesis of Coumarin-Type Compounds M I Naumov A V Nuchev N S Sitnikov Y B Malysheva A S Shavyrin I P Beletskaya A E Gavryushin S Combes A Y Fedorov
1683 Asymmetric Synthesis of 12-anti-Disubstituted Taurine Derivatives D Enders D Iffland G Raabe
1689 A Novel One-Pot Three-Component Synthesis of 5-Imino-2358-tetrahydropyrazolo[12-a]pyridazin-1-one Derivatives B Qian M-J Fan Y-X Xie L-Y Wu Y Shi Y-M Liang
1694 One-Portion Synthesis of 2-Acetoxy Carbonyl Compounds from Aldehydes by Using an Acetylated Masked Acyl Cyanide H Nemoto T Kawamura K Kitasaki K Yatsuzuka M Kamiya Y Yoshioka
1703 Synthesis of 9-Anthryl Ethers from trans-910-Dihydro-910-dimethoxyanthracene by Acid-Catalyzed Transetherification K S Jang H Y Shin D Y Chi
1708 Efficient Synthesis of Azo Dye Labeled Terpenes Sugars and Steroids Using N-(4-Arylazobenzoyl)-1H-benzotriazoles A R Katritzky S R Tala N E Abo-Dya Z K Abdel-Samii
1715 Tandem CH-ActivationndashImine-Formation Reaction A New Route to Imidazo[21-a]phthalazines A Heim-Riether K R Gipson
1720 A Convenient and Efficient α-Sulfenylation of Carbonyl Compounds E Okragla S Demkowicz J Rachon D Witt
1725 Stereoselective Synthesis of β-Branched Phenylalanine Derivatives via Chelate-Claisen Rearrangement C Quirin U Kazmaier
1732 Catalyst-Free and Base-Free Water-Promoted SNAr Reaction of Heteroaryl Halides with Thiols B Sreedhar P S Reddy M A Reddy
1739 Convenient Methods for Synthesis of C2-Symmetric Diphenyltetrahydrothiophenes M Periasamy G Ramani G P Muthukumaragopal
1744 Highly Diastereoselective Conjugate AdditionndashElimination of Chiral Nickel(II) Glycinate with Activated Allylic Acetates for Asymmetric Synthesis of Glutamic Acid Derivatives J Wang J Shi X Zhang D Lin H Jiang H Liu
1753 Synthesis of 36-Dimethoxybenzene-12-diamine and of 47-Dimethoxy-2-methyl-1H-benzimidazole T Besset C Morin
1757 An Inexpensive Procedure for Reductive Aminations Using Dimethylamineborane on Millimolar and Molar Scale R Ortmann M Schlitzer
1760 Classics in Stereoselective Synthesis Edited by E M Carreira L Kvaerno Reviewed by Rolf Breinbauer
XV Forthcoming Articles
no 11 1761 Transition-Metal-Catalyzed Enantioselective Synthesis of Compounds with
Non-Centrochirality M Ogasawara S Watanabe 1786 One-Pot Synthesis of 3-Acyl-2-(alkylsulfanyl)indoles and 2-(Alkylsulfanyl)-
indole-3-carboxylates from (2-Isocyanophenyl)methyl Ketones or (2-Isocyanophenyl)acetates S Fukamachi H Konishi K Kobayashi
1791 Efficient and Recyclable Phthalocyanine-Based Sensitizers for Photooxygenation Reactions H Xu W-K Chan D K P Ng
1797 A Facile and Practical One-Pot Synthesis of β-Oxo Thioamides from β-Oxo Amides and Isothiocyanates P Huang D Xiang Y Zhou Y Liang T Na D Dong
1801 Microwave-Promoted Solid-Acid-Catalyzed One-Pot Synthesis of Phthalazinones V M Outerbridge S M Landge H Tamaki B Toumlroumlk
1807 Benzylic Brominations with N-Bromosuccinimide in (Trifluoromethyl)-benzene D Suarez G Laval S-M Tu D Jiang C L Robinson R Scott B T Golding
1811 Synthesis of Thioflavanone and Flavanone Derivatives by Cyclization of Chalcones W Konieczny M Konieczny
1815 A New and Expedient Total Synthesis of Ochratoxin A and d5-Ochratoxin A B Gabriele M Attya A Fazio L Di Donna P Plastina G Sindona
1821 Synthesis of Benzopyrrolizidinones by NorrishndashYang Cyclization of 3-(Acylmethyl)-2-alkylisoindol-1-ones J Wu W Zhang C Wang
1829 Reactions of MoritandashBaylisndashHillman Acetates with Huisgen Zwitterions A Novel Strategy for the Synthesis of β-Amino Acid Derivatives A Jose R R Paul R Mohan S C Mathew A T Biju E Suresh V Nair
1834 Peracetylated β-Allyl C-Glycosides of D-Ribofuranose and 2-Deoxy- D-ribofuranose in the Chemical Literature Until Now Mirages in the Literature H Otero Martinez H Reinke D Michalik C Vogel
1841 Core-Tetrasubstituted Naphthalene Diimides by Stille Cross-Coupling Reactions and Characterization of Their Optical and Redox Properties S-L Suraru F Wuumlrthner
1846 A Practical Synthesis of Indole-Based Heterocycles Using an Amidoaluminum-Mediated Strategy R Todd M M Hossain
1851 Synthesis of Fluorinated Pyrrolo[23-b]pyridine and Pyrrolo[23-d]pyrimidine Nucleosides V O Iaroshenko Y Wang D V Sevenard D M Volochnyuk
1858 Recyclization Reactions of 5-Formyl-13-dimethyluracil with Electron-Rich Amino Heterocycles A P Mityuk D M Volochnyuk S V Ryabukhin A S Plaskon A Shivanyuk A A Tolmachev
1865 Facile Synthesis of Fluorinated 1-Desazapurines V O Iaroshenko D V Sevenard D M Volochnyuk Y Wang A Martiloga A O Tolmachev
1876 A Practical Synthesis of 3-Diethoxyphosphoryl-12-pyridazine Derivatives J-C Monbaliu J Marchand-Brynaert
1881 Enantioselective Reduction of Prochiral Ketones Employing Sprouted Pisum sativa as Biocatalyst J S Yadav B V S Reddy C Sreelakshmi A B Rao
1886 Application of Phenolate Ion Mediated Intramolecular Epoxide Ring Opening in the Enantioselective Synthesis of Functionalized 23-Dihydrobenzofurans and 1-Benzopyrans S K Dinda S K Das G Panda
1897 Complementary Synthetic Approaches to Constitutionally Diverse N-Aminoalkylated Isoindolinones Application to the Synthesis of Falipamil and 5-HT1A Receptor Ligand Analogues M Lorion A Couture E Deniau P Grandclaudon
1904 Selective Deprotection of Silyl Ethers with Sodium Periodate J Li D Menche
1909 Micellar Solution of Sodium Dodecyl Sulfate (SDS) Catalyzes KabacknikndashFields Reaction in Aqueous Media S Sobhani A Vafaee
1916 Convenient Methods for the Synthesis of a Library of Hemilabile Phosphines M V Jimeacutenez J J Peacuterez-Torrente M I Bartolomeacute L A Oro
1923 Terminal Aziridines by Addition of Grignard Reagents or Organoceriums to an (α-Chloro)sulfinylimine D M Hodgson J Kloesges B Evans
1933 A Robust Synthesis of Nε-(Carboxymethyl)-L-lysine (CML) R Csuk S Stark A Barthel R Kluge D Stroumlhl
1935 One-Pot Curtius Rearrangement Processes from Carboxylic Acids O Leogane H Lebel
XV Forthcoming Articles
no 12 1941 The Chemistry of Deprotonated α-Aminonitriles T Opatz 1960 An Efficient Synthesis of Tetraalkyl 2345-Thiophenetetracarboxylate
Derivatives A Alizadeh R Hosseinpour 1963 Facile Deprotection of Bulky (Trialkylsilyl)acetylenes with Silver Fluoride
S Kim B Kim J In 1969 Highly Efficient and Reusable Ionic Liquids for the Catalyzed
Hydroamination of Alkenes with Sulfonamides Carbamates and Carboxamides L Yang L-W Xu C-G Xia
1975 Synthesis of 2391016172324-Octasubstituted Phthalocyaninatozinc(II) Complexes Mediated by Reductive Agents G A Gauna A C Monsalvo J Awruch
1979 A Short and Efficient Synthesis of 3-2-[2-(Bromomethyl)thiazol-4-yl]-ethynyl-5-fluorobenzonitrile A Precursor for PET Radioligand [18F]SP203 M B Gopinathan C Jin K S Rehder
1983 Synthesis of a Substituted Benzazepin-2-one Dihydrate S K Boini R K Vaid K P Moder D Mitchell
1987 Synthesis of Novel Trisubstituted Imidazolines F J Lakner M A Parker B Rogovoy A Khvat A Ivachtchenko
1991 A Novel Synthesis of N-But-3-enyl-α- and β-Amino Acids T T Van Nguyen R T C Brownlee A B Hughes
1999 Synthesis of Substituted 5-(3-Hydroxypropyl)pyrrolidin-2-ones and Pyrrolizidinones from Nitroethane via C3 Functionalized 56-Dihydro-4H-12-oxazines A Novel Approach to Some Analogues of the Antidepressant Rolipram A Yu Sukhorukov A V Lesiv Y A Khomutova S L Ioffe V A Tartakovsky
2009 Chiral Cyclobutanols and Cyclopentane Dimers via Samarium(II) Iodide Induced Keto-Olefin Cyclisations of Carbohydrate-Derived Unsaturated Ketones D B G Williams J Caddy K Blann J J C Groveacute C W Holzapfel
2015 Synthesis of Perfluoroalkylthio-Substituted Ferrocenes C Rhode J Lemke M Lieb N Metzler-Nolte
2019 Functionalization of Polyhedral Oligomeric Silsesquioxane (POSS) via Nucleophilic Substitution M Dutkiewicz H Maciejewski B Marciniec
2025 A Novel Synthesis of Aryl Mesylates via One-Pot DemethylationndashMesylation of Aryl Methyl Ethers Using a Mixture of Phosphorus Pentoxide in Methanesulfonic Acid B Kaboudin Y Abedi
2029 Anionic Cyclization of (NN-Dimethylamino)[2-(prop-2-yn-1-yloxy)aryl]-acetonitriles T Zdrojewski J Musielak A Jończyk
2035 Strecker-Type Reaction Catalyzed by Carboxylic Acids in Aqueous Media Z Xie G Li G Zhao J Wang
2040 Synthesis of Novel Structurally Simplified Estrogen Analogues with Electron-Donating Groups in Ring A L F Tietze C A Vock I K Krimmelbein L Nacke
2061 On the Resolution of Secondary Phosphine Oxides via Diastereomeric Complex Formation The Case of tert-Butylphenylphosphine Oxide J Holt A M Maj E P Schudde K M Pietrusiewicz L Sieroń W Wieczorek T Jerphagnon I W C E Arends U Hanefeld A J Minnaard
2066 Enantioselective Copper-Catalyzed Conjugate Addition of Dimethylzinc to 5-(1-Arylalkylidene) Meldrumrsquos Acids A Wilsily T Lou E Fillion
2073 SuzukindashMiyaura Coupling Reactions Using Phosphite Ligands M Jang Y Jo I-K Oh H M Jung S Lee
2076 Synthesis of 2-Methylindoline- and 2-Methyl-1234-tetrahydroquinoline-Derived Phosphoramidites and Their Applications in Iridium-Catalyzed Allylic Alkylation of Indoles W-B Liu H He L-X Dai S-L You
2083 Stereocontrolled Synthesis of 13-Amino Alcohols by Reduction of Substituted 2-1-[(tert-Butylsulfinyl)amino]alkylcyclohexanones J C Gonzaacutelez-Goacutemez F Foubelo M Yus
2089 Tunable Phosphoramidite Ligands for Asymmetric Hydrovinylation Ligands par excellence for Generation of All-Carbon Quaternary Centers C R Smith H J Lim A ZhangT V RajanBabu
2101 Copper-Catalyzed Asymmetric Ring-Opening Reaction of Oxabenzonorbornadienes with Grignard and Aluminum Reagents R Millet L Gremaud T Bernardez L Palais A Alexakis
2113 A Simplified Synthesis of Takemotorsquos Catalyst A Berkessel B Seelig 2116 Pharmaceutical Substances Syntheses Patents and Applications of the
Most Relevant AIPs Edited by Axel Kleeman Juumlrgen Engel Bernhard Kutscher Dietmar Reichert Reviewed by I Agranat
XV Forthcoming Articles
no 13 2117 Recent Advances in the Aza-Claisen Rearrangement K C Majumdar
T Bhattacharyya B Chattopadhyay B Sinha 2143 A Novel and Convenient Synthesis of lsquoReversedrsquo Diamidino 25-Aryl- and
25-Azaheterocycle-Substituted Furans L Hu D W Boykin 2146 Efficient and General Preparation of Pyranostilbenes First Total Synthesis
of Artocarbene and Pawhuskin B B H Park Y R Lee W S Lyoo 2155 Mild Oxidation of Diarylacetylenes to 12-Diketones Using Oxone in
Trifluoroacetic Acid J-H Chu Y-J Chen M-J Wu 2163 One-Pot Microwave-Assisted Selective Azido ReductionTandem Cyclization
in Condensed and Solid Phase with Nickel Boride N Shankaraiah N Markandeya M Espinoza-Moraga C Arancibia A Kamal L Silva Santos
2171 Pyrrolo[321-ij]quinolin-4-one and Pyrrolo[321-ij]quinolin-6-one H McNab D J Nelson E J Rozgowska
2175 Practical Synthesis of 5-Substituted Tetrazoles under Microwave Irradiation J Roh T V Artamonova K Vaacutevrovaacute G I Koldobskii A Hrabaacutelek
2179 A Simple Method for the Synthesis of 3-Arylthieno[23-b]pyridines via Iodine-Mediated Cyclization of 3-(1-Arylalkenyl)-2-[(1-phenylethyl)sulfanyl]pyridines K Kobayashi D Nakamura Y Shiroyama S Fukamachi H Konishi
2184 Synthesis of Four Lysine-Linked Cereulide Analogues Showing Ionophoric Activity Towards Potassium Cations as Lead Compounds for Emetic Toxin-Detection by Immunoassays A Makarasen T Nishikawa M Isobe
2205 Synthesis of α-Aliphatic and β-Aromatic Substituted Taurines via Regioselective Ring Opening of Thiiranes with Ammonia H Yu S Cao L Zhang G Liu J Xu
2210 Stability of 5(6)-Carboxyfluorescein in Microwave-Assisted Synthesis of Fluorescein-Labelled O-Dimannosylated Peptides R Kowalczyk P W R Harris R P Dunbar M A Brimble
2223 Diversity-Oriented Synthesis of Functionalized Diaryl Sulfones by Regioselective [3+3] Cyclizations of 13-Bis(siloxy)buta-13-dienes with 2-(Arylsulfonyl)-3-ethoxy-2-en-1-ones Scope and Limitations M Shkoor A Riahi O Fatunsin H Reinke C Fischer P Langer
2236 Synthesis of Functionalized Salicylates by Formal [3+3] Cyclocondensation of 13-Bis(silyloxy)buta-13-dienes with 3-Alkoxy-2-en-1-ones G Mroszlig S Ladzik H Reinke A Spannenberg C Fischer P Langer
2249 Synthetic Approach to Alkoxy-β-(trifluoromethyl)styrenes and Their Application in the Synthesis of New Trifluoromethylated Heterocycles V M Muzalevskiy V G Nenajdenko A V Shastin E S Balenkova G Haufe
2260 o-Benzenedisulfonimide as a Powerful and Recyclable Organocatalyst for the Nazarov Reaction M Barbero S Cadamuro A Deagostino S Dughera P Larini E G Occhiato C Prandi S Tabasso R Vulcano P Venturello
2267 The Catalytic Potential of 4-Guanidinylpyridines in Acylation Reactions I Held E Larionov C Bozler F Wagner H Zipse
2278 Iron(III) Chloride in EthanolndashWater Highly Efficient Catalytic System for the Synthesis of Garcia Gonzalez Polyhydroxyalkyl- and C-Glycosylfurans L Nagarapu M V Chary A Satyender B Supriya R Bantu
2283 Ruthenium-Catalyzed Addition of Primary Amides to Alkynes A Stereoselective Synthesis of Secondary Enamides L J Gooszligen M Blanchot K S M Salih K Gooszligen
2289 Binaphthyl-Modified Quaternary Phosphonium Salts as Chiral Phase Transfer Catalysts Application to Asymmetric Amination of β-Keto Esters R He K Maruoka
X Table of Contents XI Forthcoming Articles
no 14 2293 Direct Methods for Stereoselective Polypropionate Synthesis A Survey
J Li D Menche 2316 Synthesis of Symmetrical Ketones from Grignard Reagents and
11-Carbonyldiimidazole D Bottalico V Fiandanese G Marchese A Punzi
2319 Synthesis of 45-Substituted Imidazoles by a Fast Condensation of 12-Diketones and Urotropine in Heterogeneous Medium G Bratulescu
2321 (Arylsulfonyl)acetones and -acetonitriles New Activated Methylenic Building Blocks for Synthesis of 123-Triazoles N T Pokhodylo V S Matiychuk M D Obushak
2324 A Safe Convenient and Efficient One-Pot Synthesis of α-Chloroketone Acetals Directly from Ketones Using Iodobenzene Dichloride J Yu C Zhang
2329 An Efficient Oxidative Conversion of Aldehydes into 2-Substituted 2-Oxazolines Using 13-Diiodo-55-dimethylhydantoin S Takahashi H Togo
2333 A Novel Procedure for the Synthesis of Benzo[b][18]naphthyridine-3-carboxylate Derivatives from MoritandashBaylisndashHillman Adduct Acetates W Zhong F Lin R Chen W Su
2341 An Improved Synthesis of 147-Triazacyclononanes (tacns) and 14710-Tetraazacyclododecanes (cyclens) J Huang Z Zhou T H Chan
2345 The Ullmann Coupling between 2-Chlorobenzoic Acids and Amino Acids A Valuable Reaction for Preparing 2-Substituted 1-Acetyl-1H-indol-3-yl Acetates J C Rodriguez Dominguez X Gang G Kirsch
2349 gem-Dibromomethyl Aromatics Efficient Aldehyde Equivalents in the KnoevenagelndashDoebner Reaction J K Augustine Y A Naik S Poojari N Chowdappa B S Sherigara K Areppa
2357 Synthesis of Novel α-Aminophosphonates Containing Adamantyl Fragment M M Kabachnik L I Minaeva I P Beletskaya
2361 Efficient Fluoride-Mediated Synthesis of 5-Amino-Substituted Isothiazoles Y S Zubenko V I Potkin
2365 Phosphine-Catalyzed Reaction of Cyanohydrins with Activated Alkynes A Siby O Loreau F Taran
2371 Sulfanyl-Substituted [3]Cumulenes and Buta-13-dienes from a Tetrakis(pyridinium)-Substituted Butadiene A Schmidt A Rahimi M Gjikaj
2379 Efficient Synthesis of 2-Substituted Pyrido[32-d]pyrimidines Involving SNAr and Palladium-Catalyzed Cross-Coupling Reactions A Tikad S Routier M Akssira J-M Leacuteger C Jarry G Guillaumet
2385 Novel Synthesis of Medium-Sized Heterocycles by Palladium-Catalyzed Intramolecular Heck Reaction via 9-endo-trig Mode of Cyclization K C Majumdar B Chattopadhyay
2393 Facile Synthesis of Fluorinated Benzofuro- and Benzothieno[23-b]pyridines α-Carbolines and Nucleosides Containing the α-Carboline Framework V O Iaroshenko Y Wang B Zhang D Volochnyuk V Ya Sosnovskikh
2403 Synthesis of Functionalized N-Vinyl Nitrogen-Containing Heterocycles S M M Lopes A M Beja M Ramos Silva J A Paixatildeo F Palacios T M V D Pinho e Melo
2408 Kumada Cross-Coupling of Aryl Grignard Reagents with Aryl Halides Catalyzed by an Immobilized Nickel Catalyst X Chen L Wang J Liu
2413 Highly Enantioselective Synthesis of Heteroaromatic Alcohols Catalyzed by Chiral DiaminodiphosphinendashRuthenium(II) Complexes W-Y Shen Y-Y Li Z-R Dong J-X Gao
2418 Concise Total Synthesis of (+)-Disparlure and its trans-Isomer Using Asymmetric Organocatalysis S-G Kim
2423 Rhodium Carbenoid Induced [12]-Migration in an L-Lyxo-Configured α-Diazo β-Keto Ester Synthesis of a New Griseolic Acid Analogue N N Bhujbal K S A Kumar D D Dhavale
2430 Synthesis of 5-Arylthio-3-hydroxyphthalates by the First [4+2] Cycloadditions of 3-Arylthio-1-silyloxy-13-butadienes with Dimethyl Acetylenedicarboxylate I Iqbal M Imran P Langer
2435 Synthesis of Highly Functionalized Proline Derivatives via a One-Pot MichaelSN-AdditionCyclization Approach U Kazmaier C Schmidt
2440 RhodiumGraphite-Catalyzed Hydrogenation of Carbocyclic and Heterocyclic Aromatic Compounds G Falini A Gualandi D Savoia
2447 Potassium [1-(tert-Butoxycarbonyl)-1H-indol-2-yl]trifluoroborate as an Efficient Building Block in Palladium-Catalyzed SuzukindashMiyaura Cross Couplings P Kassis V Beacuteneacuteteau J-Y Meacuterour S Routier
2454 Syntheses of Substituted Furans and Pyrroles by Platinum-Catalyzed Cyclizations of Propargylic Oxiranes and Aziridines in Aqueous Media M Yoshida M Al-Amin K Shishido
2467 Transition-Metal-Free Oxidative Homocoupling of Aryl Alkenyl and Alkynyl Grignard Reagents with TEMPO M S Maji A Studer
XIII Forthcoming Articles
no 15 2471 Advances in Synthetic Approaches for the Preparation of Combretastatin-
Based Anti-Cancer Agents R Singh H Kaur 2492 Synthesis of Unsymmetrical Ureas by Sulfur-Assisted Carbonylation with
Carbon Monoxide and Oxidation with Molecular Oxygen under Mild Conditions T Mizuno T Nakai M Mihara
2497 Ring-OpeningRecyclization Reactions of (Dimethylamino)propenoyl-Substituted Cyclopropanes Facile Synthesis of Halogenated Pyridin-2(1H)-ones R Zhang Y Zhou Y Liang Z Jiang D Dong
2501 Facile and Efficient Total Synthesis of Taspine B Cheng S Zhang L Zhu J Zhang Q Li A Shan L He
2505 Oligomeric Iodosylbenzene Sulfate A Convenient Hypervalent Iodine Reagent for Oxidation of Organic Sulfides and Alkenes M S Yusubov R Y Yusubova T V Funk K-W Chi V V Zhdankin
2509 Pyrrolidine-Based Organocatalysts for Enantioselective Michael Addition of Cyclohexanone to trans-β-Nitrostyrene A P Carley S Dixon J D Kilburn
2517 CundashAl Hydrotalcite An Efficient and Reusable Ligand-Free Catalyst for the Coupling of Aryl Chlorides with Aliphatic Aromatic and N(H)-Heterocyclic Amines B Sreedhar R Arundhathi P L Reddy M A Reddy M L Kantam
2523 Highly Efficient Synthesis of trans-βγ-Unsaturated a-Keto Amides C Allais T Constantieux J Rodriguez
2531 Gas-Phase Synthesis of N-Unsubstituted 3-Hydroxypyrroles and 1H-Pyrrol-3(2H)-ones L Hill G A Hunter S H Imam H McNab W J OrsquoNeill
2535 3-Hydroxy-1H-pyrrole L Hill S H Imam H McNab W J OrsquoNeill 2539 123-Thiadiazoles with Unsaturated Side Chains Synthesis
Polymerization and Photocrosslinking M Al-Smadi N Hanold H Kalbitz H Meier
2547 Synthesis of 1112-Didehydrodibenzo[ae]cycloocten-5(6H)-one A Strained Eight-Membered Alkyne S C Kornmayer F Rominger R Gleiter
2553 Stannous Chloride Dihydrate A Novel and Efficient Catalyst for the Synthesis of gem-Dihydroperoxides from Ketones and Aldehydes D Azarifar K Khosravi F Soleimanei
2557 Synthesis of a Novel Class of Azacrown Macrocycles and Lariat Crown Ethers Containing Two 124-Triazole Rings as Subunits N Foroughifar A Mobinikhaledi S Ebrahimi
2561 Enantioselective Synthesis of the 3C-Protease Inhibitor (ndash)-Thysanone by a StauntonndashWeinreb Annulation Strategy J Sperry T Y Yuen M A Brimble
2570 Stereoselective Synthesis of Unnatural β-Amino Acids from Nitroethane via 56-Dihydro-4H-12-oxazin-3-ylacetates A Yu Sukhorukov A V Lesiv O L Eliseev Y A Khomutova S L Ioffe
2579 A Versatile Unexpected One-Pot Regioselective Synthesis of a New Class of 13-Diazepinoindolones by Reaction of Pyranoindolones with Monosubstituted Ureas D Livadiotou C A Tsoleridis J Stephanidou-Stephanatou
2584 Synthesis of a Trisaccharide and a Tetrasaccharide from the Cell-Wall Lipopolysaccharides of Azospirillum brasilense S17 S Pandey S Ghosh A K Misra
2591 Synthesis of Isoindoline Nitroxides by Electrocyclic Reactions T Kaacutelai J Jekı K Hideg
2596 Glycosylations of Tertiary Alcohols Synthesis of Fully Protected Disaccharides with Sterically Demanding Groups Attached to the Sugar Core A Holkenbrink J B Vicente D B Werz
2605 Copper-Catalyzed [13]-Dipolar Cycloaddition for the Synthesis of Macrocycles Containing Acyclic Aromatic and Steroidal Moieties G V Latyshev M S Baranom A V Kazantsev A D Averin N V Lukashev I P Beletskaya
2616 Aryl Ring Migration Reaction in the Synthesis of 24-Diaryl-4H-31-benzothiazines A V Butin F A Tsiunchik V T Abaev A V Gutnov D A Cheshkov
2627 Hydrogenation of β-N-Substituted and β-NN-Disubstituted Enamino Esters in the Presence of Iridium(I) Catalyst H Hebbache Z Hank C Bruneau J-L Renaud
2634 Stereoselective Olefination Reactions Promoted by Rieke Manganese J M Concelloacuten H Rodriacuteguez-Solla V del Amo P Diacuteaz
2646 Synthesis of Piperidinones through a Radical Cascade E Godineau Y Landais
2650 Asymmetric Organic Synthesis with Enzymes Edited by V Gotor I Alfonso E Garciacutea-Urdiales Reviewed by Steve Collier
XVII Forthcoming Articles
no 16 2651 Synthesis of Spirocyclic Ethers S Rosenberg R Leino 2674 Bimetallic PalladiumndashPlatinum-on-Carbon-Catalyzed HndashD Exchange
Reaction Synergistic Effect on Multiple Deuterium Incorporation T Maegawa N Ito K Oono Y Monguchi H Sajiki
2679 Efficient Copper-Catalyzed Synthesis of 2-Amino-4(3H)-quinazolinone and 2-Aminoquinazoline Derivatives X Huang H Yang H Fu R Qiao Y Zhao
2689 Synthesis and Chemoselective N- and O-Alkylation of Thiadiazolopyrimidine Nucleosides and Uridines A M L Hossion R Islam R K Kandahary T Nagamatsu
2697 Facile and Efficient Synthesis of a New Class of Indole-Substituted Pyridine Derivatives via One-Pot Multicomponent Reactions K Zhao X-P Xu S-L Zhu D-Q Shi Y Zhang S-J Ji
2709 Studies toward a Total Synthesis of Rhizoxin D Stereoselective Preparation of the C11ndashC19 Fragment S Padakanti C K Kumar E Ashok P Das
2715 A Short Synthesis of Enantiomeric Phytoprostanes B1 Type I W Perlikowska M Mikołajczyk
2719 Chemistry of Polyhalogenated Nitrobutadienes Part 7 A Novel Synthetic Access to Chlorinated Nitrile Oxides E Nutz V A Zapolrsquoskii D E Kaufmann
2725 Microwave-Assisted Silver(I)-Mediated Selective O-Alkylation of Aromatic Imidate Systems B K Singh C Cavalluzzo M De Maeyer Z Debyser V S Parmar E Van der Eycken
2729 Iodogen A Novel Reagent for the Oxidation of Urazoles under Heterogeneous Conditions A Khoramabadi A Shiri M A Zolfigol S Mallakpour
2733 An Unprecedented Synthesis of Eight-Membered-Ring Cyclic Thioimidic Esters by a Three-Component Reaction A Alizadeh R Hosseinpour
2737 A Novel Diastereoselective Synthesis of β-Phosphonato Unsaturated Thioimidates A Alizadeh N Zohreh
2741 Synthesis of 21-Benzisoxazoles by Nucleophilic Substitution of Hydrogen in Nitroarenes Activated by the Azole Ring N T Pokhodylo Y O Teslenko V S Matiychuk M D Obushak
2749 A Facile Synthesis of Two Series of Multifunctional Carbon Compounds from αα-Dihalo Ketones Using Allylsamarium Bromide X Liu S Zhang J Di
2756 Stereocontrolled Formation of Protected Aminodeoxyalditols from Simple Carbohydrate Precursors by Debenzylating Cycloetherification Y Jiang Z Fang Q Zheng H Jia J Cheng B Zheng
2761 trans-Stilbene as a Starting Material for the Synthesis of Tamoxifen Based on Palladium-Catalyzed Cross-Coupling Reactions C M Nunes J Limberger S Poersch M Seferin A L Monteiro
2766 Synthesis and Biological Evaluation of 6-Substituted Purinylcarbanucleosides with a Cyclopenta[b]thiophene Pseudosugar P Abeijoacuten J M Blanco O Caamantildeo F Fernaacutendez M D Garciacutea X Garciacutea-Mera J E Rodriacuteguez-Borges J Balzarini E De Clercq
2773 Synthesis and Electrochemical Signature of Novel Norbornyl-ferrocene Hybrids F A Khan S K Upadhyay
2778 A Regioselective TsujindashTrost Pentadienylation of 3-Allyltetronic Acid R Schobert B Barnickel
2785 Copper(I)-Catalyzed CarylndashCalkynyl Bond Formation of Aryl Iodides with Terminal Alkynes K G Thakur G Sekar
2790 Aminolysis of Epoxides Using Iridium Trichloride as an Efficient Catalyst J Agarwal A Duley R Rani R K Peddinti
2797 Preparation of Several Active N-Chloro Compounds from Trichloroisocyanuric Acid A Shiri A Khoramabadi-zad
2802 The First Mineral-Catalyzed One-Pot [3+1+2] Coupling Protocol for Multifunctionalized Fused-Ring Pyrimidines L D S Yadav A Rai
2809 Efficient Synthesis of Tetrahydro-β-carbolin-1-one and Dihydroisoquinolin-1-one Derivatives as Versatile Intermediates K E Judd M F Mahon L Caggiano
2818 A Concise Synthesis of ortho-Iodobenzyl Alcohols via Addition of ortho-Iodophenyl Grignard Reagent to Aldehydes and Ketones J Cvengroš D Stolz A Togni
XIII Forthcoming Articles
no 17 2825 Reactivity of Oxazol-5-(4H)-ones and Their Application toward Natural
Product Synthesis N M Hewlett C D Hupp J J Tepe 2840 Towards the Total Synthesis of 3-Hydroxyvibsanin E B D Schwartz
J R Denton P V Bernhardt H M L Davies C M Williams 2847 Structure Investigations of (ent)-Cladospolide D by De Novo Synthesis and
Kinetic and Thermodynamic Isomerization Y Xing J H Penn G A OrsquoDoherty
2855 New Applications of PhI(OAc)2 in Synthesis Total Synthesis and SAR Development of Potent Antitumor Natural Product PsymberinIrciniastatin A N Shao X Huang A Palani R Aslanian A Buevich J Piwinski R Huryk C Seidel-Dugan
2873 Total Synthesis of Largazole ndash Devolution of a Novel Synthetic Strategy B Wang C J Forsyth
2881 Formal Total Synthesis of Palmerolide A J Jaumlgel M E Maier 2893 Total Synthesis of Bongkrekic Acid via Sequential SuzukindashMiyaura Coupling
Reactions M Kanematsu M Shindo M Yoshida K Shishido 2905 Stereodivergent Approach to Both C28a-syn and C28a-anti Relative
Stereochemical Manifolds in the Lepadin Family via a TiCl4-Promoted G Li L J Carlson I K Sagamanova B W Slafer R P Hsung C Gilardi H M Sklenicka N Sydorenko
2915 Enantioselective Aldol Reaction of Tetrasubstituted Ketene Silyl Acetals with Achiral Aldehydes for the Construction of Asymmetric Tertiary Alcohols An Application for the Divergent Total Syntheses of Buergerinins F and G I Shiina T Iizumi Y-s Yamai Y-i Kawakita K Yokoyama Y-k Yamada
2927 Second-Generation Biomimetic Total Synthesis of Chaetominine A Coste G Karthikeyan F Couty G Evano
2935 Total Synthesis of (+)-Fostriecin and (+)-Phoslactomycin B S Shibahara M Fujino Y Tashiro N Okamoto T Esumi K Takahashi J Ishihara S Hatakeyama
2954 Stereochemical Assignments of the Chlorinated Residues in Victorin C A C Durow C Butts C L Willis
2963 Studies of the Asymmetric Total Synthesis of Clavilactone D by the lsquoLariatrsquo Cyclization Strategy T Yoshimitsu S Nojima M Hashimoto K Tsukamoto T Tanaka
2970 Total Synthesis of the Leucetta-Derived Alkaloid Calcaridine A P B Koswatta R Sivappa H V R Dias C J Lovely
2983 Formal Synthesis of Salinosporamide A Starting from D-Glucose T Momose Y Kaiya J-i Hasegawa T Sato N Chida
2992 Synthesis of Bioactive Natural Products by Asymmetric syn- and anti-Aldol Reactions A K Ghosh Z L Dawson
no 18 3003 Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural
Products B M Trost M K Brennan 3026 One-Pot Synthesis of Furo[34-b]pyridin-5(7H)-ones from 2-
Bromopyridine-3-carboxylic Acid and Carbonyl Compounds K Kobayashi T Kozuki H Konishi
3029 Iodocyclization of N-[2-(Methylthio)phenyl]propiolamides Selective Synthesis of 3-Iodo-15-benzothiazepin-4-ones T-S Jiang X-G Zhang J-H Li
3039 A Facile Synthetic Method for Fluorine-Containing 17-Phenanthrolines Pyridine-Ring Formation Reaction of N-Propargyl-68-bis(trifluoroacetyl)-quinolin-5-amine with Various Nucleophiles D Shibata E Okada M Hinoshita M Meacutedebielle
3047 Enantiotopic Discrimination in Palladium-Mediated Nucleophilic Substitutions on Achiral Substrates Chiral Ligand versus Chiral Nucleophile O Jacquet F Charnay J-C Fiaud J Ollivier
3051 Studies on the Chemistry of 2-[3-(2-Nitrophenyl)-2-oxopropyl]benzaldehydes Novel Syntheses of 5H-Benzo[b]carbazole-611-diones and Indolo[12-b]isoquinoline-611-diones M Fernaacutendez
3061 Studies on the C22ndashC23 Aldol Coupling of Spirangien M Lorenz N Bluhm M Kalesse
3067 One-Pot Synthesis of N-Alkyl Purine Pyrimidine and Azole Derivatives from Alcohols using Ph3PCCl4 A Rapid Route to Carboacyclic Nucleoside Synthesis M N Soltani Rad A Khalafi-Nezhad S Behrouz Z Asrari M Behrouz Z Amini
3077 Synthesis of 2-Amino-34-dihydroquinazolines and Imidazo[21-b]quinazoline-2-ones A Mishra S Batra
3089 Studies on the Reaction of Diimines with Thiourea Synthesis and Solvent-Induced cistrans-Isomerization of 135-Triazinane-2-thiones B Kaboudin T Ghasemi T Yokomatsu
3094 Suzuki Coupling of Heteroaromatic Chlorides Using Highly Electron-Donating ClickPhos Ligands S M Spinella Z-H Guan J Chen X Zhang
3099 Reaction of NN-Dioxyenamines with Anhydrides of Carboxylic and Sulfonic Acids A New Method for the Synthesis of a-Hydroxyoxime Derivatives A A Tabolin A V Lesiv S L Ioffe
3106 Directed ortho Metallation Chemistry and Phosphine Synthesis New Ligands for the SuzukindashMiyaura Reaction D B G Williams S J Evans H de Bod M S Mokhadinyana T Hughes
3113 New Functional Derivatives of 9-Phenylquinine P J Boratyński J SkarŜewski
3120 On the Synthesis of Asymmetric and Dissymmetric Amino Analogues of Troumlgerrsquos Base J Artacho K Waumlrnmark
3127 Synthesis of Polycyclic Sultams by Palladium-Catalyzed Intramolecular Cyclization K C Majumdar S Mondal N De
3136 Synthesis of Functionalized L-Cysteine and L-Methionine by Reaction with Electron-Deficient Acetylenes B A Trofimov A G Malrsquokina O A Shemyakina V V Nosyreva A P Borisova S S Khutsishvili L B Krivdin
3143 A lsquoClickrsquo Approach to the Synthesis of 3-[2-(1-Alkyltriazol-4-yl)ethyl]indoles M Petrini R R Shaikh
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
1531 Asymmetric Transfer Hydrogenation of Ketimines with Trichlorosilane Structural Studies Z Zhang P Rooshenas H Hausmann P R Schreiner
1545 Prolinol Sulfinyl Ester Derivatives Organocatalytic Michael Addition of Ketones to Nitroolefins under Neat Conditions X Zeng G Zhong
1551 Asymmetric Oxidations of Electron-Poor Alkenes Promoted by the β-Amino AlcoholTBHP System A Russo A Lattanzi
1557 Enantioselectivity Switch in Direct Asymmetric Aminoxylation Catalyzed by Binaphthyl-Based Chiral Secondary Amines T Kano A Yamamoto F Shirozu K Maruoka
1564 Enantioselective Conjugate Addition of N-Heterocycles to αβ-Unsaturated Ketones Catalyzed by Chiral Primary Amines G Luo S Zhang W Duan W Wang
1573 Sulfonyl Hydrazine as New Functionality in Organocatalysis Camphorsulfonyl Hydrazine Catalyzed Enantioselective Aza-Michael Addition L-Y Chen H He B-J Pei W-H Chan A W M Lee
1578 Conversion of Primary Alcohols and Aldehydes into Methyl Esters by Ruthenium-Catalysed Hydrogen Transfer Reactions N A Owston T D Nixon A J Parker M K Whittlesey J M J Williams
1582 Addendum and Erratum XVII Forthcoming Articles
no 10 1583 Organocatalytic Formation of Quaternary Stereocenters M Bella
T Gasperi 1615 Regioselective Synthesis of 5H-Thiazolo[32-a]pyrimidin-5-ones from
MoritandashBaylisndashHillman Adduct Acetates under Solvent-Free and Base-Free Conditions W Zhong B Guo F Lin Y Liu W Su
1623 First Synthesis of 5-Cyanosalicylates by Formal [3+3] Cyclocondensations of 13-Bis(silyloxy)-13-butadienes A Riahi O Fatunsin M Shkoor R Dede H Reinke C Fischer P Langer
1635 Reaction of Isocyanides Dialkyl Acetylenedicarboxylates and a-Keto Lactones Unexpected Participation of an Ester Carbonyl Group in the Isocyanide-Based Three-Component Reaction A A Esmaeili H Vesalipoor
1639 An Efficient and Chemoselective Synthesis of 16-Naphthyridines and Pyrano[32-c]pyridines under Microwave Irradiation Z-G Han S-J Tu B Jiang S Yan X-H Zhang S-S Wu W-J Hao X-D Cao F Shi G Zhang N Ma
1647 N-Activation of N-Arylimidazoles Facile Syntheses of N-Alkyl-N-arylimidazolium Iodides from Less Expensive Chloro Substrates A M Oertel V Ritleng M J Chetcuti
1651 Synthesis of Polyhalogenated 2-(Phenylamino)pyridines by Thermal Amination Reactions S R Waldvogel A Faust W Barkmann R Froumlhlich O Wolff
1655 Cyanide Ion Promoted Addition of Acylphosphonates to Diethyl Cyanophosphonate Synthesis of Phosphonocyanohydrin O-Phosphates A S Demir A Aybey M Emrullahoglu
1659 Straightforward and Scalable Synthesis of Orthogonally Protected 37-Diazabicyclo[410]heptane H Schramm M Pavlova C Hoenke J Christoffers
1663 Hypervalent Iodine Mediated Oxidation of 12-Diaminobenzimidazole and Its Schiff Bases Efficient Synthesis of 3-Amino-124-benzotriazine and 2-Aryl-124-triazolo[15-a]benzimidazoles A Kumar M Parshad R K Gupta D Kumar
1667 Synthesis of the Reported Protoberberine Gusanlung D P B Wakchaure S Easwar N P Argade
1673 2-(Azidomethyl)arylboronic Acids in the Synthesis of Coumarin-Type Compounds M I Naumov A V Nuchev N S Sitnikov Y B Malysheva A S Shavyrin I P Beletskaya A E Gavryushin S Combes A Y Fedorov
1683 Asymmetric Synthesis of 12-anti-Disubstituted Taurine Derivatives D Enders D Iffland G Raabe
1689 A Novel One-Pot Three-Component Synthesis of 5-Imino-2358-tetrahydropyrazolo[12-a]pyridazin-1-one Derivatives B Qian M-J Fan Y-X Xie L-Y Wu Y Shi Y-M Liang
1694 One-Portion Synthesis of 2-Acetoxy Carbonyl Compounds from Aldehydes by Using an Acetylated Masked Acyl Cyanide H Nemoto T Kawamura K Kitasaki K Yatsuzuka M Kamiya Y Yoshioka
1703 Synthesis of 9-Anthryl Ethers from trans-910-Dihydro-910-dimethoxyanthracene by Acid-Catalyzed Transetherification K S Jang H Y Shin D Y Chi
1708 Efficient Synthesis of Azo Dye Labeled Terpenes Sugars and Steroids Using N-(4-Arylazobenzoyl)-1H-benzotriazoles A R Katritzky S R Tala N E Abo-Dya Z K Abdel-Samii
1715 Tandem CH-ActivationndashImine-Formation Reaction A New Route to Imidazo[21-a]phthalazines A Heim-Riether K R Gipson
1720 A Convenient and Efficient α-Sulfenylation of Carbonyl Compounds E Okragla S Demkowicz J Rachon D Witt
1725 Stereoselective Synthesis of β-Branched Phenylalanine Derivatives via Chelate-Claisen Rearrangement C Quirin U Kazmaier
1732 Catalyst-Free and Base-Free Water-Promoted SNAr Reaction of Heteroaryl Halides with Thiols B Sreedhar P S Reddy M A Reddy
1739 Convenient Methods for Synthesis of C2-Symmetric Diphenyltetrahydrothiophenes M Periasamy G Ramani G P Muthukumaragopal
1744 Highly Diastereoselective Conjugate AdditionndashElimination of Chiral Nickel(II) Glycinate with Activated Allylic Acetates for Asymmetric Synthesis of Glutamic Acid Derivatives J Wang J Shi X Zhang D Lin H Jiang H Liu
1753 Synthesis of 36-Dimethoxybenzene-12-diamine and of 47-Dimethoxy-2-methyl-1H-benzimidazole T Besset C Morin
1757 An Inexpensive Procedure for Reductive Aminations Using Dimethylamineborane on Millimolar and Molar Scale R Ortmann M Schlitzer
1760 Classics in Stereoselective Synthesis Edited by E M Carreira L Kvaerno Reviewed by Rolf Breinbauer
XV Forthcoming Articles
no 11 1761 Transition-Metal-Catalyzed Enantioselective Synthesis of Compounds with
Non-Centrochirality M Ogasawara S Watanabe 1786 One-Pot Synthesis of 3-Acyl-2-(alkylsulfanyl)indoles and 2-(Alkylsulfanyl)-
indole-3-carboxylates from (2-Isocyanophenyl)methyl Ketones or (2-Isocyanophenyl)acetates S Fukamachi H Konishi K Kobayashi
1791 Efficient and Recyclable Phthalocyanine-Based Sensitizers for Photooxygenation Reactions H Xu W-K Chan D K P Ng
1797 A Facile and Practical One-Pot Synthesis of β-Oxo Thioamides from β-Oxo Amides and Isothiocyanates P Huang D Xiang Y Zhou Y Liang T Na D Dong
1801 Microwave-Promoted Solid-Acid-Catalyzed One-Pot Synthesis of Phthalazinones V M Outerbridge S M Landge H Tamaki B Toumlroumlk
1807 Benzylic Brominations with N-Bromosuccinimide in (Trifluoromethyl)-benzene D Suarez G Laval S-M Tu D Jiang C L Robinson R Scott B T Golding
1811 Synthesis of Thioflavanone and Flavanone Derivatives by Cyclization of Chalcones W Konieczny M Konieczny
1815 A New and Expedient Total Synthesis of Ochratoxin A and d5-Ochratoxin A B Gabriele M Attya A Fazio L Di Donna P Plastina G Sindona
1821 Synthesis of Benzopyrrolizidinones by NorrishndashYang Cyclization of 3-(Acylmethyl)-2-alkylisoindol-1-ones J Wu W Zhang C Wang
1829 Reactions of MoritandashBaylisndashHillman Acetates with Huisgen Zwitterions A Novel Strategy for the Synthesis of β-Amino Acid Derivatives A Jose R R Paul R Mohan S C Mathew A T Biju E Suresh V Nair
1834 Peracetylated β-Allyl C-Glycosides of D-Ribofuranose and 2-Deoxy- D-ribofuranose in the Chemical Literature Until Now Mirages in the Literature H Otero Martinez H Reinke D Michalik C Vogel
1841 Core-Tetrasubstituted Naphthalene Diimides by Stille Cross-Coupling Reactions and Characterization of Their Optical and Redox Properties S-L Suraru F Wuumlrthner
1846 A Practical Synthesis of Indole-Based Heterocycles Using an Amidoaluminum-Mediated Strategy R Todd M M Hossain
1851 Synthesis of Fluorinated Pyrrolo[23-b]pyridine and Pyrrolo[23-d]pyrimidine Nucleosides V O Iaroshenko Y Wang D V Sevenard D M Volochnyuk
1858 Recyclization Reactions of 5-Formyl-13-dimethyluracil with Electron-Rich Amino Heterocycles A P Mityuk D M Volochnyuk S V Ryabukhin A S Plaskon A Shivanyuk A A Tolmachev
1865 Facile Synthesis of Fluorinated 1-Desazapurines V O Iaroshenko D V Sevenard D M Volochnyuk Y Wang A Martiloga A O Tolmachev
1876 A Practical Synthesis of 3-Diethoxyphosphoryl-12-pyridazine Derivatives J-C Monbaliu J Marchand-Brynaert
1881 Enantioselective Reduction of Prochiral Ketones Employing Sprouted Pisum sativa as Biocatalyst J S Yadav B V S Reddy C Sreelakshmi A B Rao
1886 Application of Phenolate Ion Mediated Intramolecular Epoxide Ring Opening in the Enantioselective Synthesis of Functionalized 23-Dihydrobenzofurans and 1-Benzopyrans S K Dinda S K Das G Panda
1897 Complementary Synthetic Approaches to Constitutionally Diverse N-Aminoalkylated Isoindolinones Application to the Synthesis of Falipamil and 5-HT1A Receptor Ligand Analogues M Lorion A Couture E Deniau P Grandclaudon
1904 Selective Deprotection of Silyl Ethers with Sodium Periodate J Li D Menche
1909 Micellar Solution of Sodium Dodecyl Sulfate (SDS) Catalyzes KabacknikndashFields Reaction in Aqueous Media S Sobhani A Vafaee
1916 Convenient Methods for the Synthesis of a Library of Hemilabile Phosphines M V Jimeacutenez J J Peacuterez-Torrente M I Bartolomeacute L A Oro
1923 Terminal Aziridines by Addition of Grignard Reagents or Organoceriums to an (α-Chloro)sulfinylimine D M Hodgson J Kloesges B Evans
1933 A Robust Synthesis of Nε-(Carboxymethyl)-L-lysine (CML) R Csuk S Stark A Barthel R Kluge D Stroumlhl
1935 One-Pot Curtius Rearrangement Processes from Carboxylic Acids O Leogane H Lebel
XV Forthcoming Articles
no 12 1941 The Chemistry of Deprotonated α-Aminonitriles T Opatz 1960 An Efficient Synthesis of Tetraalkyl 2345-Thiophenetetracarboxylate
Derivatives A Alizadeh R Hosseinpour 1963 Facile Deprotection of Bulky (Trialkylsilyl)acetylenes with Silver Fluoride
S Kim B Kim J In 1969 Highly Efficient and Reusable Ionic Liquids for the Catalyzed
Hydroamination of Alkenes with Sulfonamides Carbamates and Carboxamides L Yang L-W Xu C-G Xia
1975 Synthesis of 2391016172324-Octasubstituted Phthalocyaninatozinc(II) Complexes Mediated by Reductive Agents G A Gauna A C Monsalvo J Awruch
1979 A Short and Efficient Synthesis of 3-2-[2-(Bromomethyl)thiazol-4-yl]-ethynyl-5-fluorobenzonitrile A Precursor for PET Radioligand [18F]SP203 M B Gopinathan C Jin K S Rehder
1983 Synthesis of a Substituted Benzazepin-2-one Dihydrate S K Boini R K Vaid K P Moder D Mitchell
1987 Synthesis of Novel Trisubstituted Imidazolines F J Lakner M A Parker B Rogovoy A Khvat A Ivachtchenko
1991 A Novel Synthesis of N-But-3-enyl-α- and β-Amino Acids T T Van Nguyen R T C Brownlee A B Hughes
1999 Synthesis of Substituted 5-(3-Hydroxypropyl)pyrrolidin-2-ones and Pyrrolizidinones from Nitroethane via C3 Functionalized 56-Dihydro-4H-12-oxazines A Novel Approach to Some Analogues of the Antidepressant Rolipram A Yu Sukhorukov A V Lesiv Y A Khomutova S L Ioffe V A Tartakovsky
2009 Chiral Cyclobutanols and Cyclopentane Dimers via Samarium(II) Iodide Induced Keto-Olefin Cyclisations of Carbohydrate-Derived Unsaturated Ketones D B G Williams J Caddy K Blann J J C Groveacute C W Holzapfel
2015 Synthesis of Perfluoroalkylthio-Substituted Ferrocenes C Rhode J Lemke M Lieb N Metzler-Nolte
2019 Functionalization of Polyhedral Oligomeric Silsesquioxane (POSS) via Nucleophilic Substitution M Dutkiewicz H Maciejewski B Marciniec
2025 A Novel Synthesis of Aryl Mesylates via One-Pot DemethylationndashMesylation of Aryl Methyl Ethers Using a Mixture of Phosphorus Pentoxide in Methanesulfonic Acid B Kaboudin Y Abedi
2029 Anionic Cyclization of (NN-Dimethylamino)[2-(prop-2-yn-1-yloxy)aryl]-acetonitriles T Zdrojewski J Musielak A Jończyk
2035 Strecker-Type Reaction Catalyzed by Carboxylic Acids in Aqueous Media Z Xie G Li G Zhao J Wang
2040 Synthesis of Novel Structurally Simplified Estrogen Analogues with Electron-Donating Groups in Ring A L F Tietze C A Vock I K Krimmelbein L Nacke
2061 On the Resolution of Secondary Phosphine Oxides via Diastereomeric Complex Formation The Case of tert-Butylphenylphosphine Oxide J Holt A M Maj E P Schudde K M Pietrusiewicz L Sieroń W Wieczorek T Jerphagnon I W C E Arends U Hanefeld A J Minnaard
2066 Enantioselective Copper-Catalyzed Conjugate Addition of Dimethylzinc to 5-(1-Arylalkylidene) Meldrumrsquos Acids A Wilsily T Lou E Fillion
2073 SuzukindashMiyaura Coupling Reactions Using Phosphite Ligands M Jang Y Jo I-K Oh H M Jung S Lee
2076 Synthesis of 2-Methylindoline- and 2-Methyl-1234-tetrahydroquinoline-Derived Phosphoramidites and Their Applications in Iridium-Catalyzed Allylic Alkylation of Indoles W-B Liu H He L-X Dai S-L You
2083 Stereocontrolled Synthesis of 13-Amino Alcohols by Reduction of Substituted 2-1-[(tert-Butylsulfinyl)amino]alkylcyclohexanones J C Gonzaacutelez-Goacutemez F Foubelo M Yus
2089 Tunable Phosphoramidite Ligands for Asymmetric Hydrovinylation Ligands par excellence for Generation of All-Carbon Quaternary Centers C R Smith H J Lim A ZhangT V RajanBabu
2101 Copper-Catalyzed Asymmetric Ring-Opening Reaction of Oxabenzonorbornadienes with Grignard and Aluminum Reagents R Millet L Gremaud T Bernardez L Palais A Alexakis
2113 A Simplified Synthesis of Takemotorsquos Catalyst A Berkessel B Seelig 2116 Pharmaceutical Substances Syntheses Patents and Applications of the
Most Relevant AIPs Edited by Axel Kleeman Juumlrgen Engel Bernhard Kutscher Dietmar Reichert Reviewed by I Agranat
XV Forthcoming Articles
no 13 2117 Recent Advances in the Aza-Claisen Rearrangement K C Majumdar
T Bhattacharyya B Chattopadhyay B Sinha 2143 A Novel and Convenient Synthesis of lsquoReversedrsquo Diamidino 25-Aryl- and
25-Azaheterocycle-Substituted Furans L Hu D W Boykin 2146 Efficient and General Preparation of Pyranostilbenes First Total Synthesis
of Artocarbene and Pawhuskin B B H Park Y R Lee W S Lyoo 2155 Mild Oxidation of Diarylacetylenes to 12-Diketones Using Oxone in
Trifluoroacetic Acid J-H Chu Y-J Chen M-J Wu 2163 One-Pot Microwave-Assisted Selective Azido ReductionTandem Cyclization
in Condensed and Solid Phase with Nickel Boride N Shankaraiah N Markandeya M Espinoza-Moraga C Arancibia A Kamal L Silva Santos
2171 Pyrrolo[321-ij]quinolin-4-one and Pyrrolo[321-ij]quinolin-6-one H McNab D J Nelson E J Rozgowska
2175 Practical Synthesis of 5-Substituted Tetrazoles under Microwave Irradiation J Roh T V Artamonova K Vaacutevrovaacute G I Koldobskii A Hrabaacutelek
2179 A Simple Method for the Synthesis of 3-Arylthieno[23-b]pyridines via Iodine-Mediated Cyclization of 3-(1-Arylalkenyl)-2-[(1-phenylethyl)sulfanyl]pyridines K Kobayashi D Nakamura Y Shiroyama S Fukamachi H Konishi
2184 Synthesis of Four Lysine-Linked Cereulide Analogues Showing Ionophoric Activity Towards Potassium Cations as Lead Compounds for Emetic Toxin-Detection by Immunoassays A Makarasen T Nishikawa M Isobe
2205 Synthesis of α-Aliphatic and β-Aromatic Substituted Taurines via Regioselective Ring Opening of Thiiranes with Ammonia H Yu S Cao L Zhang G Liu J Xu
2210 Stability of 5(6)-Carboxyfluorescein in Microwave-Assisted Synthesis of Fluorescein-Labelled O-Dimannosylated Peptides R Kowalczyk P W R Harris R P Dunbar M A Brimble
2223 Diversity-Oriented Synthesis of Functionalized Diaryl Sulfones by Regioselective [3+3] Cyclizations of 13-Bis(siloxy)buta-13-dienes with 2-(Arylsulfonyl)-3-ethoxy-2-en-1-ones Scope and Limitations M Shkoor A Riahi O Fatunsin H Reinke C Fischer P Langer
2236 Synthesis of Functionalized Salicylates by Formal [3+3] Cyclocondensation of 13-Bis(silyloxy)buta-13-dienes with 3-Alkoxy-2-en-1-ones G Mroszlig S Ladzik H Reinke A Spannenberg C Fischer P Langer
2249 Synthetic Approach to Alkoxy-β-(trifluoromethyl)styrenes and Their Application in the Synthesis of New Trifluoromethylated Heterocycles V M Muzalevskiy V G Nenajdenko A V Shastin E S Balenkova G Haufe
2260 o-Benzenedisulfonimide as a Powerful and Recyclable Organocatalyst for the Nazarov Reaction M Barbero S Cadamuro A Deagostino S Dughera P Larini E G Occhiato C Prandi S Tabasso R Vulcano P Venturello
2267 The Catalytic Potential of 4-Guanidinylpyridines in Acylation Reactions I Held E Larionov C Bozler F Wagner H Zipse
2278 Iron(III) Chloride in EthanolndashWater Highly Efficient Catalytic System for the Synthesis of Garcia Gonzalez Polyhydroxyalkyl- and C-Glycosylfurans L Nagarapu M V Chary A Satyender B Supriya R Bantu
2283 Ruthenium-Catalyzed Addition of Primary Amides to Alkynes A Stereoselective Synthesis of Secondary Enamides L J Gooszligen M Blanchot K S M Salih K Gooszligen
2289 Binaphthyl-Modified Quaternary Phosphonium Salts as Chiral Phase Transfer Catalysts Application to Asymmetric Amination of β-Keto Esters R He K Maruoka
X Table of Contents XI Forthcoming Articles
no 14 2293 Direct Methods for Stereoselective Polypropionate Synthesis A Survey
J Li D Menche 2316 Synthesis of Symmetrical Ketones from Grignard Reagents and
11-Carbonyldiimidazole D Bottalico V Fiandanese G Marchese A Punzi
2319 Synthesis of 45-Substituted Imidazoles by a Fast Condensation of 12-Diketones and Urotropine in Heterogeneous Medium G Bratulescu
2321 (Arylsulfonyl)acetones and -acetonitriles New Activated Methylenic Building Blocks for Synthesis of 123-Triazoles N T Pokhodylo V S Matiychuk M D Obushak
2324 A Safe Convenient and Efficient One-Pot Synthesis of α-Chloroketone Acetals Directly from Ketones Using Iodobenzene Dichloride J Yu C Zhang
2329 An Efficient Oxidative Conversion of Aldehydes into 2-Substituted 2-Oxazolines Using 13-Diiodo-55-dimethylhydantoin S Takahashi H Togo
2333 A Novel Procedure for the Synthesis of Benzo[b][18]naphthyridine-3-carboxylate Derivatives from MoritandashBaylisndashHillman Adduct Acetates W Zhong F Lin R Chen W Su
2341 An Improved Synthesis of 147-Triazacyclononanes (tacns) and 14710-Tetraazacyclododecanes (cyclens) J Huang Z Zhou T H Chan
2345 The Ullmann Coupling between 2-Chlorobenzoic Acids and Amino Acids A Valuable Reaction for Preparing 2-Substituted 1-Acetyl-1H-indol-3-yl Acetates J C Rodriguez Dominguez X Gang G Kirsch
2349 gem-Dibromomethyl Aromatics Efficient Aldehyde Equivalents in the KnoevenagelndashDoebner Reaction J K Augustine Y A Naik S Poojari N Chowdappa B S Sherigara K Areppa
2357 Synthesis of Novel α-Aminophosphonates Containing Adamantyl Fragment M M Kabachnik L I Minaeva I P Beletskaya
2361 Efficient Fluoride-Mediated Synthesis of 5-Amino-Substituted Isothiazoles Y S Zubenko V I Potkin
2365 Phosphine-Catalyzed Reaction of Cyanohydrins with Activated Alkynes A Siby O Loreau F Taran
2371 Sulfanyl-Substituted [3]Cumulenes and Buta-13-dienes from a Tetrakis(pyridinium)-Substituted Butadiene A Schmidt A Rahimi M Gjikaj
2379 Efficient Synthesis of 2-Substituted Pyrido[32-d]pyrimidines Involving SNAr and Palladium-Catalyzed Cross-Coupling Reactions A Tikad S Routier M Akssira J-M Leacuteger C Jarry G Guillaumet
2385 Novel Synthesis of Medium-Sized Heterocycles by Palladium-Catalyzed Intramolecular Heck Reaction via 9-endo-trig Mode of Cyclization K C Majumdar B Chattopadhyay
2393 Facile Synthesis of Fluorinated Benzofuro- and Benzothieno[23-b]pyridines α-Carbolines and Nucleosides Containing the α-Carboline Framework V O Iaroshenko Y Wang B Zhang D Volochnyuk V Ya Sosnovskikh
2403 Synthesis of Functionalized N-Vinyl Nitrogen-Containing Heterocycles S M M Lopes A M Beja M Ramos Silva J A Paixatildeo F Palacios T M V D Pinho e Melo
2408 Kumada Cross-Coupling of Aryl Grignard Reagents with Aryl Halides Catalyzed by an Immobilized Nickel Catalyst X Chen L Wang J Liu
2413 Highly Enantioselective Synthesis of Heteroaromatic Alcohols Catalyzed by Chiral DiaminodiphosphinendashRuthenium(II) Complexes W-Y Shen Y-Y Li Z-R Dong J-X Gao
2418 Concise Total Synthesis of (+)-Disparlure and its trans-Isomer Using Asymmetric Organocatalysis S-G Kim
2423 Rhodium Carbenoid Induced [12]-Migration in an L-Lyxo-Configured α-Diazo β-Keto Ester Synthesis of a New Griseolic Acid Analogue N N Bhujbal K S A Kumar D D Dhavale
2430 Synthesis of 5-Arylthio-3-hydroxyphthalates by the First [4+2] Cycloadditions of 3-Arylthio-1-silyloxy-13-butadienes with Dimethyl Acetylenedicarboxylate I Iqbal M Imran P Langer
2435 Synthesis of Highly Functionalized Proline Derivatives via a One-Pot MichaelSN-AdditionCyclization Approach U Kazmaier C Schmidt
2440 RhodiumGraphite-Catalyzed Hydrogenation of Carbocyclic and Heterocyclic Aromatic Compounds G Falini A Gualandi D Savoia
2447 Potassium [1-(tert-Butoxycarbonyl)-1H-indol-2-yl]trifluoroborate as an Efficient Building Block in Palladium-Catalyzed SuzukindashMiyaura Cross Couplings P Kassis V Beacuteneacuteteau J-Y Meacuterour S Routier
2454 Syntheses of Substituted Furans and Pyrroles by Platinum-Catalyzed Cyclizations of Propargylic Oxiranes and Aziridines in Aqueous Media M Yoshida M Al-Amin K Shishido
2467 Transition-Metal-Free Oxidative Homocoupling of Aryl Alkenyl and Alkynyl Grignard Reagents with TEMPO M S Maji A Studer
XIII Forthcoming Articles
no 15 2471 Advances in Synthetic Approaches for the Preparation of Combretastatin-
Based Anti-Cancer Agents R Singh H Kaur 2492 Synthesis of Unsymmetrical Ureas by Sulfur-Assisted Carbonylation with
Carbon Monoxide and Oxidation with Molecular Oxygen under Mild Conditions T Mizuno T Nakai M Mihara
2497 Ring-OpeningRecyclization Reactions of (Dimethylamino)propenoyl-Substituted Cyclopropanes Facile Synthesis of Halogenated Pyridin-2(1H)-ones R Zhang Y Zhou Y Liang Z Jiang D Dong
2501 Facile and Efficient Total Synthesis of Taspine B Cheng S Zhang L Zhu J Zhang Q Li A Shan L He
2505 Oligomeric Iodosylbenzene Sulfate A Convenient Hypervalent Iodine Reagent for Oxidation of Organic Sulfides and Alkenes M S Yusubov R Y Yusubova T V Funk K-W Chi V V Zhdankin
2509 Pyrrolidine-Based Organocatalysts for Enantioselective Michael Addition of Cyclohexanone to trans-β-Nitrostyrene A P Carley S Dixon J D Kilburn
2517 CundashAl Hydrotalcite An Efficient and Reusable Ligand-Free Catalyst for the Coupling of Aryl Chlorides with Aliphatic Aromatic and N(H)-Heterocyclic Amines B Sreedhar R Arundhathi P L Reddy M A Reddy M L Kantam
2523 Highly Efficient Synthesis of trans-βγ-Unsaturated a-Keto Amides C Allais T Constantieux J Rodriguez
2531 Gas-Phase Synthesis of N-Unsubstituted 3-Hydroxypyrroles and 1H-Pyrrol-3(2H)-ones L Hill G A Hunter S H Imam H McNab W J OrsquoNeill
2535 3-Hydroxy-1H-pyrrole L Hill S H Imam H McNab W J OrsquoNeill 2539 123-Thiadiazoles with Unsaturated Side Chains Synthesis
Polymerization and Photocrosslinking M Al-Smadi N Hanold H Kalbitz H Meier
2547 Synthesis of 1112-Didehydrodibenzo[ae]cycloocten-5(6H)-one A Strained Eight-Membered Alkyne S C Kornmayer F Rominger R Gleiter
2553 Stannous Chloride Dihydrate A Novel and Efficient Catalyst for the Synthesis of gem-Dihydroperoxides from Ketones and Aldehydes D Azarifar K Khosravi F Soleimanei
2557 Synthesis of a Novel Class of Azacrown Macrocycles and Lariat Crown Ethers Containing Two 124-Triazole Rings as Subunits N Foroughifar A Mobinikhaledi S Ebrahimi
2561 Enantioselective Synthesis of the 3C-Protease Inhibitor (ndash)-Thysanone by a StauntonndashWeinreb Annulation Strategy J Sperry T Y Yuen M A Brimble
2570 Stereoselective Synthesis of Unnatural β-Amino Acids from Nitroethane via 56-Dihydro-4H-12-oxazin-3-ylacetates A Yu Sukhorukov A V Lesiv O L Eliseev Y A Khomutova S L Ioffe
2579 A Versatile Unexpected One-Pot Regioselective Synthesis of a New Class of 13-Diazepinoindolones by Reaction of Pyranoindolones with Monosubstituted Ureas D Livadiotou C A Tsoleridis J Stephanidou-Stephanatou
2584 Synthesis of a Trisaccharide and a Tetrasaccharide from the Cell-Wall Lipopolysaccharides of Azospirillum brasilense S17 S Pandey S Ghosh A K Misra
2591 Synthesis of Isoindoline Nitroxides by Electrocyclic Reactions T Kaacutelai J Jekı K Hideg
2596 Glycosylations of Tertiary Alcohols Synthesis of Fully Protected Disaccharides with Sterically Demanding Groups Attached to the Sugar Core A Holkenbrink J B Vicente D B Werz
2605 Copper-Catalyzed [13]-Dipolar Cycloaddition for the Synthesis of Macrocycles Containing Acyclic Aromatic and Steroidal Moieties G V Latyshev M S Baranom A V Kazantsev A D Averin N V Lukashev I P Beletskaya
2616 Aryl Ring Migration Reaction in the Synthesis of 24-Diaryl-4H-31-benzothiazines A V Butin F A Tsiunchik V T Abaev A V Gutnov D A Cheshkov
2627 Hydrogenation of β-N-Substituted and β-NN-Disubstituted Enamino Esters in the Presence of Iridium(I) Catalyst H Hebbache Z Hank C Bruneau J-L Renaud
2634 Stereoselective Olefination Reactions Promoted by Rieke Manganese J M Concelloacuten H Rodriacuteguez-Solla V del Amo P Diacuteaz
2646 Synthesis of Piperidinones through a Radical Cascade E Godineau Y Landais
2650 Asymmetric Organic Synthesis with Enzymes Edited by V Gotor I Alfonso E Garciacutea-Urdiales Reviewed by Steve Collier
XVII Forthcoming Articles
no 16 2651 Synthesis of Spirocyclic Ethers S Rosenberg R Leino 2674 Bimetallic PalladiumndashPlatinum-on-Carbon-Catalyzed HndashD Exchange
Reaction Synergistic Effect on Multiple Deuterium Incorporation T Maegawa N Ito K Oono Y Monguchi H Sajiki
2679 Efficient Copper-Catalyzed Synthesis of 2-Amino-4(3H)-quinazolinone and 2-Aminoquinazoline Derivatives X Huang H Yang H Fu R Qiao Y Zhao
2689 Synthesis and Chemoselective N- and O-Alkylation of Thiadiazolopyrimidine Nucleosides and Uridines A M L Hossion R Islam R K Kandahary T Nagamatsu
2697 Facile and Efficient Synthesis of a New Class of Indole-Substituted Pyridine Derivatives via One-Pot Multicomponent Reactions K Zhao X-P Xu S-L Zhu D-Q Shi Y Zhang S-J Ji
2709 Studies toward a Total Synthesis of Rhizoxin D Stereoselective Preparation of the C11ndashC19 Fragment S Padakanti C K Kumar E Ashok P Das
2715 A Short Synthesis of Enantiomeric Phytoprostanes B1 Type I W Perlikowska M Mikołajczyk
2719 Chemistry of Polyhalogenated Nitrobutadienes Part 7 A Novel Synthetic Access to Chlorinated Nitrile Oxides E Nutz V A Zapolrsquoskii D E Kaufmann
2725 Microwave-Assisted Silver(I)-Mediated Selective O-Alkylation of Aromatic Imidate Systems B K Singh C Cavalluzzo M De Maeyer Z Debyser V S Parmar E Van der Eycken
2729 Iodogen A Novel Reagent for the Oxidation of Urazoles under Heterogeneous Conditions A Khoramabadi A Shiri M A Zolfigol S Mallakpour
2733 An Unprecedented Synthesis of Eight-Membered-Ring Cyclic Thioimidic Esters by a Three-Component Reaction A Alizadeh R Hosseinpour
2737 A Novel Diastereoselective Synthesis of β-Phosphonato Unsaturated Thioimidates A Alizadeh N Zohreh
2741 Synthesis of 21-Benzisoxazoles by Nucleophilic Substitution of Hydrogen in Nitroarenes Activated by the Azole Ring N T Pokhodylo Y O Teslenko V S Matiychuk M D Obushak
2749 A Facile Synthesis of Two Series of Multifunctional Carbon Compounds from αα-Dihalo Ketones Using Allylsamarium Bromide X Liu S Zhang J Di
2756 Stereocontrolled Formation of Protected Aminodeoxyalditols from Simple Carbohydrate Precursors by Debenzylating Cycloetherification Y Jiang Z Fang Q Zheng H Jia J Cheng B Zheng
2761 trans-Stilbene as a Starting Material for the Synthesis of Tamoxifen Based on Palladium-Catalyzed Cross-Coupling Reactions C M Nunes J Limberger S Poersch M Seferin A L Monteiro
2766 Synthesis and Biological Evaluation of 6-Substituted Purinylcarbanucleosides with a Cyclopenta[b]thiophene Pseudosugar P Abeijoacuten J M Blanco O Caamantildeo F Fernaacutendez M D Garciacutea X Garciacutea-Mera J E Rodriacuteguez-Borges J Balzarini E De Clercq
2773 Synthesis and Electrochemical Signature of Novel Norbornyl-ferrocene Hybrids F A Khan S K Upadhyay
2778 A Regioselective TsujindashTrost Pentadienylation of 3-Allyltetronic Acid R Schobert B Barnickel
2785 Copper(I)-Catalyzed CarylndashCalkynyl Bond Formation of Aryl Iodides with Terminal Alkynes K G Thakur G Sekar
2790 Aminolysis of Epoxides Using Iridium Trichloride as an Efficient Catalyst J Agarwal A Duley R Rani R K Peddinti
2797 Preparation of Several Active N-Chloro Compounds from Trichloroisocyanuric Acid A Shiri A Khoramabadi-zad
2802 The First Mineral-Catalyzed One-Pot [3+1+2] Coupling Protocol for Multifunctionalized Fused-Ring Pyrimidines L D S Yadav A Rai
2809 Efficient Synthesis of Tetrahydro-β-carbolin-1-one and Dihydroisoquinolin-1-one Derivatives as Versatile Intermediates K E Judd M F Mahon L Caggiano
2818 A Concise Synthesis of ortho-Iodobenzyl Alcohols via Addition of ortho-Iodophenyl Grignard Reagent to Aldehydes and Ketones J Cvengroš D Stolz A Togni
XIII Forthcoming Articles
no 17 2825 Reactivity of Oxazol-5-(4H)-ones and Their Application toward Natural
Product Synthesis N M Hewlett C D Hupp J J Tepe 2840 Towards the Total Synthesis of 3-Hydroxyvibsanin E B D Schwartz
J R Denton P V Bernhardt H M L Davies C M Williams 2847 Structure Investigations of (ent)-Cladospolide D by De Novo Synthesis and
Kinetic and Thermodynamic Isomerization Y Xing J H Penn G A OrsquoDoherty
2855 New Applications of PhI(OAc)2 in Synthesis Total Synthesis and SAR Development of Potent Antitumor Natural Product PsymberinIrciniastatin A N Shao X Huang A Palani R Aslanian A Buevich J Piwinski R Huryk C Seidel-Dugan
2873 Total Synthesis of Largazole ndash Devolution of a Novel Synthetic Strategy B Wang C J Forsyth
2881 Formal Total Synthesis of Palmerolide A J Jaumlgel M E Maier 2893 Total Synthesis of Bongkrekic Acid via Sequential SuzukindashMiyaura Coupling
Reactions M Kanematsu M Shindo M Yoshida K Shishido 2905 Stereodivergent Approach to Both C28a-syn and C28a-anti Relative
Stereochemical Manifolds in the Lepadin Family via a TiCl4-Promoted G Li L J Carlson I K Sagamanova B W Slafer R P Hsung C Gilardi H M Sklenicka N Sydorenko
2915 Enantioselective Aldol Reaction of Tetrasubstituted Ketene Silyl Acetals with Achiral Aldehydes for the Construction of Asymmetric Tertiary Alcohols An Application for the Divergent Total Syntheses of Buergerinins F and G I Shiina T Iizumi Y-s Yamai Y-i Kawakita K Yokoyama Y-k Yamada
2927 Second-Generation Biomimetic Total Synthesis of Chaetominine A Coste G Karthikeyan F Couty G Evano
2935 Total Synthesis of (+)-Fostriecin and (+)-Phoslactomycin B S Shibahara M Fujino Y Tashiro N Okamoto T Esumi K Takahashi J Ishihara S Hatakeyama
2954 Stereochemical Assignments of the Chlorinated Residues in Victorin C A C Durow C Butts C L Willis
2963 Studies of the Asymmetric Total Synthesis of Clavilactone D by the lsquoLariatrsquo Cyclization Strategy T Yoshimitsu S Nojima M Hashimoto K Tsukamoto T Tanaka
2970 Total Synthesis of the Leucetta-Derived Alkaloid Calcaridine A P B Koswatta R Sivappa H V R Dias C J Lovely
2983 Formal Synthesis of Salinosporamide A Starting from D-Glucose T Momose Y Kaiya J-i Hasegawa T Sato N Chida
2992 Synthesis of Bioactive Natural Products by Asymmetric syn- and anti-Aldol Reactions A K Ghosh Z L Dawson
no 18 3003 Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural
Products B M Trost M K Brennan 3026 One-Pot Synthesis of Furo[34-b]pyridin-5(7H)-ones from 2-
Bromopyridine-3-carboxylic Acid and Carbonyl Compounds K Kobayashi T Kozuki H Konishi
3029 Iodocyclization of N-[2-(Methylthio)phenyl]propiolamides Selective Synthesis of 3-Iodo-15-benzothiazepin-4-ones T-S Jiang X-G Zhang J-H Li
3039 A Facile Synthetic Method for Fluorine-Containing 17-Phenanthrolines Pyridine-Ring Formation Reaction of N-Propargyl-68-bis(trifluoroacetyl)-quinolin-5-amine with Various Nucleophiles D Shibata E Okada M Hinoshita M Meacutedebielle
3047 Enantiotopic Discrimination in Palladium-Mediated Nucleophilic Substitutions on Achiral Substrates Chiral Ligand versus Chiral Nucleophile O Jacquet F Charnay J-C Fiaud J Ollivier
3051 Studies on the Chemistry of 2-[3-(2-Nitrophenyl)-2-oxopropyl]benzaldehydes Novel Syntheses of 5H-Benzo[b]carbazole-611-diones and Indolo[12-b]isoquinoline-611-diones M Fernaacutendez
3061 Studies on the C22ndashC23 Aldol Coupling of Spirangien M Lorenz N Bluhm M Kalesse
3067 One-Pot Synthesis of N-Alkyl Purine Pyrimidine and Azole Derivatives from Alcohols using Ph3PCCl4 A Rapid Route to Carboacyclic Nucleoside Synthesis M N Soltani Rad A Khalafi-Nezhad S Behrouz Z Asrari M Behrouz Z Amini
3077 Synthesis of 2-Amino-34-dihydroquinazolines and Imidazo[21-b]quinazoline-2-ones A Mishra S Batra
3089 Studies on the Reaction of Diimines with Thiourea Synthesis and Solvent-Induced cistrans-Isomerization of 135-Triazinane-2-thiones B Kaboudin T Ghasemi T Yokomatsu
3094 Suzuki Coupling of Heteroaromatic Chlorides Using Highly Electron-Donating ClickPhos Ligands S M Spinella Z-H Guan J Chen X Zhang
3099 Reaction of NN-Dioxyenamines with Anhydrides of Carboxylic and Sulfonic Acids A New Method for the Synthesis of a-Hydroxyoxime Derivatives A A Tabolin A V Lesiv S L Ioffe
3106 Directed ortho Metallation Chemistry and Phosphine Synthesis New Ligands for the SuzukindashMiyaura Reaction D B G Williams S J Evans H de Bod M S Mokhadinyana T Hughes
3113 New Functional Derivatives of 9-Phenylquinine P J Boratyński J SkarŜewski
3120 On the Synthesis of Asymmetric and Dissymmetric Amino Analogues of Troumlgerrsquos Base J Artacho K Waumlrnmark
3127 Synthesis of Polycyclic Sultams by Palladium-Catalyzed Intramolecular Cyclization K C Majumdar S Mondal N De
3136 Synthesis of Functionalized L-Cysteine and L-Methionine by Reaction with Electron-Deficient Acetylenes B A Trofimov A G Malrsquokina O A Shemyakina V V Nosyreva A P Borisova S S Khutsishvili L B Krivdin
3143 A lsquoClickrsquo Approach to the Synthesis of 3-[2-(1-Alkyltriazol-4-yl)ethyl]indoles M Petrini R R Shaikh
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
no 10 1583 Organocatalytic Formation of Quaternary Stereocenters M Bella
T Gasperi 1615 Regioselective Synthesis of 5H-Thiazolo[32-a]pyrimidin-5-ones from
MoritandashBaylisndashHillman Adduct Acetates under Solvent-Free and Base-Free Conditions W Zhong B Guo F Lin Y Liu W Su
1623 First Synthesis of 5-Cyanosalicylates by Formal [3+3] Cyclocondensations of 13-Bis(silyloxy)-13-butadienes A Riahi O Fatunsin M Shkoor R Dede H Reinke C Fischer P Langer
1635 Reaction of Isocyanides Dialkyl Acetylenedicarboxylates and a-Keto Lactones Unexpected Participation of an Ester Carbonyl Group in the Isocyanide-Based Three-Component Reaction A A Esmaeili H Vesalipoor
1639 An Efficient and Chemoselective Synthesis of 16-Naphthyridines and Pyrano[32-c]pyridines under Microwave Irradiation Z-G Han S-J Tu B Jiang S Yan X-H Zhang S-S Wu W-J Hao X-D Cao F Shi G Zhang N Ma
1647 N-Activation of N-Arylimidazoles Facile Syntheses of N-Alkyl-N-arylimidazolium Iodides from Less Expensive Chloro Substrates A M Oertel V Ritleng M J Chetcuti
1651 Synthesis of Polyhalogenated 2-(Phenylamino)pyridines by Thermal Amination Reactions S R Waldvogel A Faust W Barkmann R Froumlhlich O Wolff
1655 Cyanide Ion Promoted Addition of Acylphosphonates to Diethyl Cyanophosphonate Synthesis of Phosphonocyanohydrin O-Phosphates A S Demir A Aybey M Emrullahoglu
1659 Straightforward and Scalable Synthesis of Orthogonally Protected 37-Diazabicyclo[410]heptane H Schramm M Pavlova C Hoenke J Christoffers
1663 Hypervalent Iodine Mediated Oxidation of 12-Diaminobenzimidazole and Its Schiff Bases Efficient Synthesis of 3-Amino-124-benzotriazine and 2-Aryl-124-triazolo[15-a]benzimidazoles A Kumar M Parshad R K Gupta D Kumar
1667 Synthesis of the Reported Protoberberine Gusanlung D P B Wakchaure S Easwar N P Argade
1673 2-(Azidomethyl)arylboronic Acids in the Synthesis of Coumarin-Type Compounds M I Naumov A V Nuchev N S Sitnikov Y B Malysheva A S Shavyrin I P Beletskaya A E Gavryushin S Combes A Y Fedorov
1683 Asymmetric Synthesis of 12-anti-Disubstituted Taurine Derivatives D Enders D Iffland G Raabe
1689 A Novel One-Pot Three-Component Synthesis of 5-Imino-2358-tetrahydropyrazolo[12-a]pyridazin-1-one Derivatives B Qian M-J Fan Y-X Xie L-Y Wu Y Shi Y-M Liang
1694 One-Portion Synthesis of 2-Acetoxy Carbonyl Compounds from Aldehydes by Using an Acetylated Masked Acyl Cyanide H Nemoto T Kawamura K Kitasaki K Yatsuzuka M Kamiya Y Yoshioka
1703 Synthesis of 9-Anthryl Ethers from trans-910-Dihydro-910-dimethoxyanthracene by Acid-Catalyzed Transetherification K S Jang H Y Shin D Y Chi
1708 Efficient Synthesis of Azo Dye Labeled Terpenes Sugars and Steroids Using N-(4-Arylazobenzoyl)-1H-benzotriazoles A R Katritzky S R Tala N E Abo-Dya Z K Abdel-Samii
1715 Tandem CH-ActivationndashImine-Formation Reaction A New Route to Imidazo[21-a]phthalazines A Heim-Riether K R Gipson
1720 A Convenient and Efficient α-Sulfenylation of Carbonyl Compounds E Okragla S Demkowicz J Rachon D Witt
1725 Stereoselective Synthesis of β-Branched Phenylalanine Derivatives via Chelate-Claisen Rearrangement C Quirin U Kazmaier
1732 Catalyst-Free and Base-Free Water-Promoted SNAr Reaction of Heteroaryl Halides with Thiols B Sreedhar P S Reddy M A Reddy
1739 Convenient Methods for Synthesis of C2-Symmetric Diphenyltetrahydrothiophenes M Periasamy G Ramani G P Muthukumaragopal
1744 Highly Diastereoselective Conjugate AdditionndashElimination of Chiral Nickel(II) Glycinate with Activated Allylic Acetates for Asymmetric Synthesis of Glutamic Acid Derivatives J Wang J Shi X Zhang D Lin H Jiang H Liu
1753 Synthesis of 36-Dimethoxybenzene-12-diamine and of 47-Dimethoxy-2-methyl-1H-benzimidazole T Besset C Morin
1757 An Inexpensive Procedure for Reductive Aminations Using Dimethylamineborane on Millimolar and Molar Scale R Ortmann M Schlitzer
1760 Classics in Stereoselective Synthesis Edited by E M Carreira L Kvaerno Reviewed by Rolf Breinbauer
XV Forthcoming Articles
no 11 1761 Transition-Metal-Catalyzed Enantioselective Synthesis of Compounds with
Non-Centrochirality M Ogasawara S Watanabe 1786 One-Pot Synthesis of 3-Acyl-2-(alkylsulfanyl)indoles and 2-(Alkylsulfanyl)-
indole-3-carboxylates from (2-Isocyanophenyl)methyl Ketones or (2-Isocyanophenyl)acetates S Fukamachi H Konishi K Kobayashi
1791 Efficient and Recyclable Phthalocyanine-Based Sensitizers for Photooxygenation Reactions H Xu W-K Chan D K P Ng
1797 A Facile and Practical One-Pot Synthesis of β-Oxo Thioamides from β-Oxo Amides and Isothiocyanates P Huang D Xiang Y Zhou Y Liang T Na D Dong
1801 Microwave-Promoted Solid-Acid-Catalyzed One-Pot Synthesis of Phthalazinones V M Outerbridge S M Landge H Tamaki B Toumlroumlk
1807 Benzylic Brominations with N-Bromosuccinimide in (Trifluoromethyl)-benzene D Suarez G Laval S-M Tu D Jiang C L Robinson R Scott B T Golding
1811 Synthesis of Thioflavanone and Flavanone Derivatives by Cyclization of Chalcones W Konieczny M Konieczny
1815 A New and Expedient Total Synthesis of Ochratoxin A and d5-Ochratoxin A B Gabriele M Attya A Fazio L Di Donna P Plastina G Sindona
1821 Synthesis of Benzopyrrolizidinones by NorrishndashYang Cyclization of 3-(Acylmethyl)-2-alkylisoindol-1-ones J Wu W Zhang C Wang
1829 Reactions of MoritandashBaylisndashHillman Acetates with Huisgen Zwitterions A Novel Strategy for the Synthesis of β-Amino Acid Derivatives A Jose R R Paul R Mohan S C Mathew A T Biju E Suresh V Nair
1834 Peracetylated β-Allyl C-Glycosides of D-Ribofuranose and 2-Deoxy- D-ribofuranose in the Chemical Literature Until Now Mirages in the Literature H Otero Martinez H Reinke D Michalik C Vogel
1841 Core-Tetrasubstituted Naphthalene Diimides by Stille Cross-Coupling Reactions and Characterization of Their Optical and Redox Properties S-L Suraru F Wuumlrthner
1846 A Practical Synthesis of Indole-Based Heterocycles Using an Amidoaluminum-Mediated Strategy R Todd M M Hossain
1851 Synthesis of Fluorinated Pyrrolo[23-b]pyridine and Pyrrolo[23-d]pyrimidine Nucleosides V O Iaroshenko Y Wang D V Sevenard D M Volochnyuk
1858 Recyclization Reactions of 5-Formyl-13-dimethyluracil with Electron-Rich Amino Heterocycles A P Mityuk D M Volochnyuk S V Ryabukhin A S Plaskon A Shivanyuk A A Tolmachev
1865 Facile Synthesis of Fluorinated 1-Desazapurines V O Iaroshenko D V Sevenard D M Volochnyuk Y Wang A Martiloga A O Tolmachev
1876 A Practical Synthesis of 3-Diethoxyphosphoryl-12-pyridazine Derivatives J-C Monbaliu J Marchand-Brynaert
1881 Enantioselective Reduction of Prochiral Ketones Employing Sprouted Pisum sativa as Biocatalyst J S Yadav B V S Reddy C Sreelakshmi A B Rao
1886 Application of Phenolate Ion Mediated Intramolecular Epoxide Ring Opening in the Enantioselective Synthesis of Functionalized 23-Dihydrobenzofurans and 1-Benzopyrans S K Dinda S K Das G Panda
1897 Complementary Synthetic Approaches to Constitutionally Diverse N-Aminoalkylated Isoindolinones Application to the Synthesis of Falipamil and 5-HT1A Receptor Ligand Analogues M Lorion A Couture E Deniau P Grandclaudon
1904 Selective Deprotection of Silyl Ethers with Sodium Periodate J Li D Menche
1909 Micellar Solution of Sodium Dodecyl Sulfate (SDS) Catalyzes KabacknikndashFields Reaction in Aqueous Media S Sobhani A Vafaee
1916 Convenient Methods for the Synthesis of a Library of Hemilabile Phosphines M V Jimeacutenez J J Peacuterez-Torrente M I Bartolomeacute L A Oro
1923 Terminal Aziridines by Addition of Grignard Reagents or Organoceriums to an (α-Chloro)sulfinylimine D M Hodgson J Kloesges B Evans
1933 A Robust Synthesis of Nε-(Carboxymethyl)-L-lysine (CML) R Csuk S Stark A Barthel R Kluge D Stroumlhl
1935 One-Pot Curtius Rearrangement Processes from Carboxylic Acids O Leogane H Lebel
XV Forthcoming Articles
no 12 1941 The Chemistry of Deprotonated α-Aminonitriles T Opatz 1960 An Efficient Synthesis of Tetraalkyl 2345-Thiophenetetracarboxylate
Derivatives A Alizadeh R Hosseinpour 1963 Facile Deprotection of Bulky (Trialkylsilyl)acetylenes with Silver Fluoride
S Kim B Kim J In 1969 Highly Efficient and Reusable Ionic Liquids for the Catalyzed
Hydroamination of Alkenes with Sulfonamides Carbamates and Carboxamides L Yang L-W Xu C-G Xia
1975 Synthesis of 2391016172324-Octasubstituted Phthalocyaninatozinc(II) Complexes Mediated by Reductive Agents G A Gauna A C Monsalvo J Awruch
1979 A Short and Efficient Synthesis of 3-2-[2-(Bromomethyl)thiazol-4-yl]-ethynyl-5-fluorobenzonitrile A Precursor for PET Radioligand [18F]SP203 M B Gopinathan C Jin K S Rehder
1983 Synthesis of a Substituted Benzazepin-2-one Dihydrate S K Boini R K Vaid K P Moder D Mitchell
1987 Synthesis of Novel Trisubstituted Imidazolines F J Lakner M A Parker B Rogovoy A Khvat A Ivachtchenko
1991 A Novel Synthesis of N-But-3-enyl-α- and β-Amino Acids T T Van Nguyen R T C Brownlee A B Hughes
1999 Synthesis of Substituted 5-(3-Hydroxypropyl)pyrrolidin-2-ones and Pyrrolizidinones from Nitroethane via C3 Functionalized 56-Dihydro-4H-12-oxazines A Novel Approach to Some Analogues of the Antidepressant Rolipram A Yu Sukhorukov A V Lesiv Y A Khomutova S L Ioffe V A Tartakovsky
2009 Chiral Cyclobutanols and Cyclopentane Dimers via Samarium(II) Iodide Induced Keto-Olefin Cyclisations of Carbohydrate-Derived Unsaturated Ketones D B G Williams J Caddy K Blann J J C Groveacute C W Holzapfel
2015 Synthesis of Perfluoroalkylthio-Substituted Ferrocenes C Rhode J Lemke M Lieb N Metzler-Nolte
2019 Functionalization of Polyhedral Oligomeric Silsesquioxane (POSS) via Nucleophilic Substitution M Dutkiewicz H Maciejewski B Marciniec
2025 A Novel Synthesis of Aryl Mesylates via One-Pot DemethylationndashMesylation of Aryl Methyl Ethers Using a Mixture of Phosphorus Pentoxide in Methanesulfonic Acid B Kaboudin Y Abedi
2029 Anionic Cyclization of (NN-Dimethylamino)[2-(prop-2-yn-1-yloxy)aryl]-acetonitriles T Zdrojewski J Musielak A Jończyk
2035 Strecker-Type Reaction Catalyzed by Carboxylic Acids in Aqueous Media Z Xie G Li G Zhao J Wang
2040 Synthesis of Novel Structurally Simplified Estrogen Analogues with Electron-Donating Groups in Ring A L F Tietze C A Vock I K Krimmelbein L Nacke
2061 On the Resolution of Secondary Phosphine Oxides via Diastereomeric Complex Formation The Case of tert-Butylphenylphosphine Oxide J Holt A M Maj E P Schudde K M Pietrusiewicz L Sieroń W Wieczorek T Jerphagnon I W C E Arends U Hanefeld A J Minnaard
2066 Enantioselective Copper-Catalyzed Conjugate Addition of Dimethylzinc to 5-(1-Arylalkylidene) Meldrumrsquos Acids A Wilsily T Lou E Fillion
2073 SuzukindashMiyaura Coupling Reactions Using Phosphite Ligands M Jang Y Jo I-K Oh H M Jung S Lee
2076 Synthesis of 2-Methylindoline- and 2-Methyl-1234-tetrahydroquinoline-Derived Phosphoramidites and Their Applications in Iridium-Catalyzed Allylic Alkylation of Indoles W-B Liu H He L-X Dai S-L You
2083 Stereocontrolled Synthesis of 13-Amino Alcohols by Reduction of Substituted 2-1-[(tert-Butylsulfinyl)amino]alkylcyclohexanones J C Gonzaacutelez-Goacutemez F Foubelo M Yus
2089 Tunable Phosphoramidite Ligands for Asymmetric Hydrovinylation Ligands par excellence for Generation of All-Carbon Quaternary Centers C R Smith H J Lim A ZhangT V RajanBabu
2101 Copper-Catalyzed Asymmetric Ring-Opening Reaction of Oxabenzonorbornadienes with Grignard and Aluminum Reagents R Millet L Gremaud T Bernardez L Palais A Alexakis
2113 A Simplified Synthesis of Takemotorsquos Catalyst A Berkessel B Seelig 2116 Pharmaceutical Substances Syntheses Patents and Applications of the
Most Relevant AIPs Edited by Axel Kleeman Juumlrgen Engel Bernhard Kutscher Dietmar Reichert Reviewed by I Agranat
XV Forthcoming Articles
no 13 2117 Recent Advances in the Aza-Claisen Rearrangement K C Majumdar
T Bhattacharyya B Chattopadhyay B Sinha 2143 A Novel and Convenient Synthesis of lsquoReversedrsquo Diamidino 25-Aryl- and
25-Azaheterocycle-Substituted Furans L Hu D W Boykin 2146 Efficient and General Preparation of Pyranostilbenes First Total Synthesis
of Artocarbene and Pawhuskin B B H Park Y R Lee W S Lyoo 2155 Mild Oxidation of Diarylacetylenes to 12-Diketones Using Oxone in
Trifluoroacetic Acid J-H Chu Y-J Chen M-J Wu 2163 One-Pot Microwave-Assisted Selective Azido ReductionTandem Cyclization
in Condensed and Solid Phase with Nickel Boride N Shankaraiah N Markandeya M Espinoza-Moraga C Arancibia A Kamal L Silva Santos
2171 Pyrrolo[321-ij]quinolin-4-one and Pyrrolo[321-ij]quinolin-6-one H McNab D J Nelson E J Rozgowska
2175 Practical Synthesis of 5-Substituted Tetrazoles under Microwave Irradiation J Roh T V Artamonova K Vaacutevrovaacute G I Koldobskii A Hrabaacutelek
2179 A Simple Method for the Synthesis of 3-Arylthieno[23-b]pyridines via Iodine-Mediated Cyclization of 3-(1-Arylalkenyl)-2-[(1-phenylethyl)sulfanyl]pyridines K Kobayashi D Nakamura Y Shiroyama S Fukamachi H Konishi
2184 Synthesis of Four Lysine-Linked Cereulide Analogues Showing Ionophoric Activity Towards Potassium Cations as Lead Compounds for Emetic Toxin-Detection by Immunoassays A Makarasen T Nishikawa M Isobe
2205 Synthesis of α-Aliphatic and β-Aromatic Substituted Taurines via Regioselective Ring Opening of Thiiranes with Ammonia H Yu S Cao L Zhang G Liu J Xu
2210 Stability of 5(6)-Carboxyfluorescein in Microwave-Assisted Synthesis of Fluorescein-Labelled O-Dimannosylated Peptides R Kowalczyk P W R Harris R P Dunbar M A Brimble
2223 Diversity-Oriented Synthesis of Functionalized Diaryl Sulfones by Regioselective [3+3] Cyclizations of 13-Bis(siloxy)buta-13-dienes with 2-(Arylsulfonyl)-3-ethoxy-2-en-1-ones Scope and Limitations M Shkoor A Riahi O Fatunsin H Reinke C Fischer P Langer
2236 Synthesis of Functionalized Salicylates by Formal [3+3] Cyclocondensation of 13-Bis(silyloxy)buta-13-dienes with 3-Alkoxy-2-en-1-ones G Mroszlig S Ladzik H Reinke A Spannenberg C Fischer P Langer
2249 Synthetic Approach to Alkoxy-β-(trifluoromethyl)styrenes and Their Application in the Synthesis of New Trifluoromethylated Heterocycles V M Muzalevskiy V G Nenajdenko A V Shastin E S Balenkova G Haufe
2260 o-Benzenedisulfonimide as a Powerful and Recyclable Organocatalyst for the Nazarov Reaction M Barbero S Cadamuro A Deagostino S Dughera P Larini E G Occhiato C Prandi S Tabasso R Vulcano P Venturello
2267 The Catalytic Potential of 4-Guanidinylpyridines in Acylation Reactions I Held E Larionov C Bozler F Wagner H Zipse
2278 Iron(III) Chloride in EthanolndashWater Highly Efficient Catalytic System for the Synthesis of Garcia Gonzalez Polyhydroxyalkyl- and C-Glycosylfurans L Nagarapu M V Chary A Satyender B Supriya R Bantu
2283 Ruthenium-Catalyzed Addition of Primary Amides to Alkynes A Stereoselective Synthesis of Secondary Enamides L J Gooszligen M Blanchot K S M Salih K Gooszligen
2289 Binaphthyl-Modified Quaternary Phosphonium Salts as Chiral Phase Transfer Catalysts Application to Asymmetric Amination of β-Keto Esters R He K Maruoka
X Table of Contents XI Forthcoming Articles
no 14 2293 Direct Methods for Stereoselective Polypropionate Synthesis A Survey
J Li D Menche 2316 Synthesis of Symmetrical Ketones from Grignard Reagents and
11-Carbonyldiimidazole D Bottalico V Fiandanese G Marchese A Punzi
2319 Synthesis of 45-Substituted Imidazoles by a Fast Condensation of 12-Diketones and Urotropine in Heterogeneous Medium G Bratulescu
2321 (Arylsulfonyl)acetones and -acetonitriles New Activated Methylenic Building Blocks for Synthesis of 123-Triazoles N T Pokhodylo V S Matiychuk M D Obushak
2324 A Safe Convenient and Efficient One-Pot Synthesis of α-Chloroketone Acetals Directly from Ketones Using Iodobenzene Dichloride J Yu C Zhang
2329 An Efficient Oxidative Conversion of Aldehydes into 2-Substituted 2-Oxazolines Using 13-Diiodo-55-dimethylhydantoin S Takahashi H Togo
2333 A Novel Procedure for the Synthesis of Benzo[b][18]naphthyridine-3-carboxylate Derivatives from MoritandashBaylisndashHillman Adduct Acetates W Zhong F Lin R Chen W Su
2341 An Improved Synthesis of 147-Triazacyclononanes (tacns) and 14710-Tetraazacyclododecanes (cyclens) J Huang Z Zhou T H Chan
2345 The Ullmann Coupling between 2-Chlorobenzoic Acids and Amino Acids A Valuable Reaction for Preparing 2-Substituted 1-Acetyl-1H-indol-3-yl Acetates J C Rodriguez Dominguez X Gang G Kirsch
2349 gem-Dibromomethyl Aromatics Efficient Aldehyde Equivalents in the KnoevenagelndashDoebner Reaction J K Augustine Y A Naik S Poojari N Chowdappa B S Sherigara K Areppa
2357 Synthesis of Novel α-Aminophosphonates Containing Adamantyl Fragment M M Kabachnik L I Minaeva I P Beletskaya
2361 Efficient Fluoride-Mediated Synthesis of 5-Amino-Substituted Isothiazoles Y S Zubenko V I Potkin
2365 Phosphine-Catalyzed Reaction of Cyanohydrins with Activated Alkynes A Siby O Loreau F Taran
2371 Sulfanyl-Substituted [3]Cumulenes and Buta-13-dienes from a Tetrakis(pyridinium)-Substituted Butadiene A Schmidt A Rahimi M Gjikaj
2379 Efficient Synthesis of 2-Substituted Pyrido[32-d]pyrimidines Involving SNAr and Palladium-Catalyzed Cross-Coupling Reactions A Tikad S Routier M Akssira J-M Leacuteger C Jarry G Guillaumet
2385 Novel Synthesis of Medium-Sized Heterocycles by Palladium-Catalyzed Intramolecular Heck Reaction via 9-endo-trig Mode of Cyclization K C Majumdar B Chattopadhyay
2393 Facile Synthesis of Fluorinated Benzofuro- and Benzothieno[23-b]pyridines α-Carbolines and Nucleosides Containing the α-Carboline Framework V O Iaroshenko Y Wang B Zhang D Volochnyuk V Ya Sosnovskikh
2403 Synthesis of Functionalized N-Vinyl Nitrogen-Containing Heterocycles S M M Lopes A M Beja M Ramos Silva J A Paixatildeo F Palacios T M V D Pinho e Melo
2408 Kumada Cross-Coupling of Aryl Grignard Reagents with Aryl Halides Catalyzed by an Immobilized Nickel Catalyst X Chen L Wang J Liu
2413 Highly Enantioselective Synthesis of Heteroaromatic Alcohols Catalyzed by Chiral DiaminodiphosphinendashRuthenium(II) Complexes W-Y Shen Y-Y Li Z-R Dong J-X Gao
2418 Concise Total Synthesis of (+)-Disparlure and its trans-Isomer Using Asymmetric Organocatalysis S-G Kim
2423 Rhodium Carbenoid Induced [12]-Migration in an L-Lyxo-Configured α-Diazo β-Keto Ester Synthesis of a New Griseolic Acid Analogue N N Bhujbal K S A Kumar D D Dhavale
2430 Synthesis of 5-Arylthio-3-hydroxyphthalates by the First [4+2] Cycloadditions of 3-Arylthio-1-silyloxy-13-butadienes with Dimethyl Acetylenedicarboxylate I Iqbal M Imran P Langer
2435 Synthesis of Highly Functionalized Proline Derivatives via a One-Pot MichaelSN-AdditionCyclization Approach U Kazmaier C Schmidt
2440 RhodiumGraphite-Catalyzed Hydrogenation of Carbocyclic and Heterocyclic Aromatic Compounds G Falini A Gualandi D Savoia
2447 Potassium [1-(tert-Butoxycarbonyl)-1H-indol-2-yl]trifluoroborate as an Efficient Building Block in Palladium-Catalyzed SuzukindashMiyaura Cross Couplings P Kassis V Beacuteneacuteteau J-Y Meacuterour S Routier
2454 Syntheses of Substituted Furans and Pyrroles by Platinum-Catalyzed Cyclizations of Propargylic Oxiranes and Aziridines in Aqueous Media M Yoshida M Al-Amin K Shishido
2467 Transition-Metal-Free Oxidative Homocoupling of Aryl Alkenyl and Alkynyl Grignard Reagents with TEMPO M S Maji A Studer
XIII Forthcoming Articles
no 15 2471 Advances in Synthetic Approaches for the Preparation of Combretastatin-
Based Anti-Cancer Agents R Singh H Kaur 2492 Synthesis of Unsymmetrical Ureas by Sulfur-Assisted Carbonylation with
Carbon Monoxide and Oxidation with Molecular Oxygen under Mild Conditions T Mizuno T Nakai M Mihara
2497 Ring-OpeningRecyclization Reactions of (Dimethylamino)propenoyl-Substituted Cyclopropanes Facile Synthesis of Halogenated Pyridin-2(1H)-ones R Zhang Y Zhou Y Liang Z Jiang D Dong
2501 Facile and Efficient Total Synthesis of Taspine B Cheng S Zhang L Zhu J Zhang Q Li A Shan L He
2505 Oligomeric Iodosylbenzene Sulfate A Convenient Hypervalent Iodine Reagent for Oxidation of Organic Sulfides and Alkenes M S Yusubov R Y Yusubova T V Funk K-W Chi V V Zhdankin
2509 Pyrrolidine-Based Organocatalysts for Enantioselective Michael Addition of Cyclohexanone to trans-β-Nitrostyrene A P Carley S Dixon J D Kilburn
2517 CundashAl Hydrotalcite An Efficient and Reusable Ligand-Free Catalyst for the Coupling of Aryl Chlorides with Aliphatic Aromatic and N(H)-Heterocyclic Amines B Sreedhar R Arundhathi P L Reddy M A Reddy M L Kantam
2523 Highly Efficient Synthesis of trans-βγ-Unsaturated a-Keto Amides C Allais T Constantieux J Rodriguez
2531 Gas-Phase Synthesis of N-Unsubstituted 3-Hydroxypyrroles and 1H-Pyrrol-3(2H)-ones L Hill G A Hunter S H Imam H McNab W J OrsquoNeill
2535 3-Hydroxy-1H-pyrrole L Hill S H Imam H McNab W J OrsquoNeill 2539 123-Thiadiazoles with Unsaturated Side Chains Synthesis
Polymerization and Photocrosslinking M Al-Smadi N Hanold H Kalbitz H Meier
2547 Synthesis of 1112-Didehydrodibenzo[ae]cycloocten-5(6H)-one A Strained Eight-Membered Alkyne S C Kornmayer F Rominger R Gleiter
2553 Stannous Chloride Dihydrate A Novel and Efficient Catalyst for the Synthesis of gem-Dihydroperoxides from Ketones and Aldehydes D Azarifar K Khosravi F Soleimanei
2557 Synthesis of a Novel Class of Azacrown Macrocycles and Lariat Crown Ethers Containing Two 124-Triazole Rings as Subunits N Foroughifar A Mobinikhaledi S Ebrahimi
2561 Enantioselective Synthesis of the 3C-Protease Inhibitor (ndash)-Thysanone by a StauntonndashWeinreb Annulation Strategy J Sperry T Y Yuen M A Brimble
2570 Stereoselective Synthesis of Unnatural β-Amino Acids from Nitroethane via 56-Dihydro-4H-12-oxazin-3-ylacetates A Yu Sukhorukov A V Lesiv O L Eliseev Y A Khomutova S L Ioffe
2579 A Versatile Unexpected One-Pot Regioselective Synthesis of a New Class of 13-Diazepinoindolones by Reaction of Pyranoindolones with Monosubstituted Ureas D Livadiotou C A Tsoleridis J Stephanidou-Stephanatou
2584 Synthesis of a Trisaccharide and a Tetrasaccharide from the Cell-Wall Lipopolysaccharides of Azospirillum brasilense S17 S Pandey S Ghosh A K Misra
2591 Synthesis of Isoindoline Nitroxides by Electrocyclic Reactions T Kaacutelai J Jekı K Hideg
2596 Glycosylations of Tertiary Alcohols Synthesis of Fully Protected Disaccharides with Sterically Demanding Groups Attached to the Sugar Core A Holkenbrink J B Vicente D B Werz
2605 Copper-Catalyzed [13]-Dipolar Cycloaddition for the Synthesis of Macrocycles Containing Acyclic Aromatic and Steroidal Moieties G V Latyshev M S Baranom A V Kazantsev A D Averin N V Lukashev I P Beletskaya
2616 Aryl Ring Migration Reaction in the Synthesis of 24-Diaryl-4H-31-benzothiazines A V Butin F A Tsiunchik V T Abaev A V Gutnov D A Cheshkov
2627 Hydrogenation of β-N-Substituted and β-NN-Disubstituted Enamino Esters in the Presence of Iridium(I) Catalyst H Hebbache Z Hank C Bruneau J-L Renaud
2634 Stereoselective Olefination Reactions Promoted by Rieke Manganese J M Concelloacuten H Rodriacuteguez-Solla V del Amo P Diacuteaz
2646 Synthesis of Piperidinones through a Radical Cascade E Godineau Y Landais
2650 Asymmetric Organic Synthesis with Enzymes Edited by V Gotor I Alfonso E Garciacutea-Urdiales Reviewed by Steve Collier
XVII Forthcoming Articles
no 16 2651 Synthesis of Spirocyclic Ethers S Rosenberg R Leino 2674 Bimetallic PalladiumndashPlatinum-on-Carbon-Catalyzed HndashD Exchange
Reaction Synergistic Effect on Multiple Deuterium Incorporation T Maegawa N Ito K Oono Y Monguchi H Sajiki
2679 Efficient Copper-Catalyzed Synthesis of 2-Amino-4(3H)-quinazolinone and 2-Aminoquinazoline Derivatives X Huang H Yang H Fu R Qiao Y Zhao
2689 Synthesis and Chemoselective N- and O-Alkylation of Thiadiazolopyrimidine Nucleosides and Uridines A M L Hossion R Islam R K Kandahary T Nagamatsu
2697 Facile and Efficient Synthesis of a New Class of Indole-Substituted Pyridine Derivatives via One-Pot Multicomponent Reactions K Zhao X-P Xu S-L Zhu D-Q Shi Y Zhang S-J Ji
2709 Studies toward a Total Synthesis of Rhizoxin D Stereoselective Preparation of the C11ndashC19 Fragment S Padakanti C K Kumar E Ashok P Das
2715 A Short Synthesis of Enantiomeric Phytoprostanes B1 Type I W Perlikowska M Mikołajczyk
2719 Chemistry of Polyhalogenated Nitrobutadienes Part 7 A Novel Synthetic Access to Chlorinated Nitrile Oxides E Nutz V A Zapolrsquoskii D E Kaufmann
2725 Microwave-Assisted Silver(I)-Mediated Selective O-Alkylation of Aromatic Imidate Systems B K Singh C Cavalluzzo M De Maeyer Z Debyser V S Parmar E Van der Eycken
2729 Iodogen A Novel Reagent for the Oxidation of Urazoles under Heterogeneous Conditions A Khoramabadi A Shiri M A Zolfigol S Mallakpour
2733 An Unprecedented Synthesis of Eight-Membered-Ring Cyclic Thioimidic Esters by a Three-Component Reaction A Alizadeh R Hosseinpour
2737 A Novel Diastereoselective Synthesis of β-Phosphonato Unsaturated Thioimidates A Alizadeh N Zohreh
2741 Synthesis of 21-Benzisoxazoles by Nucleophilic Substitution of Hydrogen in Nitroarenes Activated by the Azole Ring N T Pokhodylo Y O Teslenko V S Matiychuk M D Obushak
2749 A Facile Synthesis of Two Series of Multifunctional Carbon Compounds from αα-Dihalo Ketones Using Allylsamarium Bromide X Liu S Zhang J Di
2756 Stereocontrolled Formation of Protected Aminodeoxyalditols from Simple Carbohydrate Precursors by Debenzylating Cycloetherification Y Jiang Z Fang Q Zheng H Jia J Cheng B Zheng
2761 trans-Stilbene as a Starting Material for the Synthesis of Tamoxifen Based on Palladium-Catalyzed Cross-Coupling Reactions C M Nunes J Limberger S Poersch M Seferin A L Monteiro
2766 Synthesis and Biological Evaluation of 6-Substituted Purinylcarbanucleosides with a Cyclopenta[b]thiophene Pseudosugar P Abeijoacuten J M Blanco O Caamantildeo F Fernaacutendez M D Garciacutea X Garciacutea-Mera J E Rodriacuteguez-Borges J Balzarini E De Clercq
2773 Synthesis and Electrochemical Signature of Novel Norbornyl-ferrocene Hybrids F A Khan S K Upadhyay
2778 A Regioselective TsujindashTrost Pentadienylation of 3-Allyltetronic Acid R Schobert B Barnickel
2785 Copper(I)-Catalyzed CarylndashCalkynyl Bond Formation of Aryl Iodides with Terminal Alkynes K G Thakur G Sekar
2790 Aminolysis of Epoxides Using Iridium Trichloride as an Efficient Catalyst J Agarwal A Duley R Rani R K Peddinti
2797 Preparation of Several Active N-Chloro Compounds from Trichloroisocyanuric Acid A Shiri A Khoramabadi-zad
2802 The First Mineral-Catalyzed One-Pot [3+1+2] Coupling Protocol for Multifunctionalized Fused-Ring Pyrimidines L D S Yadav A Rai
2809 Efficient Synthesis of Tetrahydro-β-carbolin-1-one and Dihydroisoquinolin-1-one Derivatives as Versatile Intermediates K E Judd M F Mahon L Caggiano
2818 A Concise Synthesis of ortho-Iodobenzyl Alcohols via Addition of ortho-Iodophenyl Grignard Reagent to Aldehydes and Ketones J Cvengroš D Stolz A Togni
XIII Forthcoming Articles
no 17 2825 Reactivity of Oxazol-5-(4H)-ones and Their Application toward Natural
Product Synthesis N M Hewlett C D Hupp J J Tepe 2840 Towards the Total Synthesis of 3-Hydroxyvibsanin E B D Schwartz
J R Denton P V Bernhardt H M L Davies C M Williams 2847 Structure Investigations of (ent)-Cladospolide D by De Novo Synthesis and
Kinetic and Thermodynamic Isomerization Y Xing J H Penn G A OrsquoDoherty
2855 New Applications of PhI(OAc)2 in Synthesis Total Synthesis and SAR Development of Potent Antitumor Natural Product PsymberinIrciniastatin A N Shao X Huang A Palani R Aslanian A Buevich J Piwinski R Huryk C Seidel-Dugan
2873 Total Synthesis of Largazole ndash Devolution of a Novel Synthetic Strategy B Wang C J Forsyth
2881 Formal Total Synthesis of Palmerolide A J Jaumlgel M E Maier 2893 Total Synthesis of Bongkrekic Acid via Sequential SuzukindashMiyaura Coupling
Reactions M Kanematsu M Shindo M Yoshida K Shishido 2905 Stereodivergent Approach to Both C28a-syn and C28a-anti Relative
Stereochemical Manifolds in the Lepadin Family via a TiCl4-Promoted G Li L J Carlson I K Sagamanova B W Slafer R P Hsung C Gilardi H M Sklenicka N Sydorenko
2915 Enantioselective Aldol Reaction of Tetrasubstituted Ketene Silyl Acetals with Achiral Aldehydes for the Construction of Asymmetric Tertiary Alcohols An Application for the Divergent Total Syntheses of Buergerinins F and G I Shiina T Iizumi Y-s Yamai Y-i Kawakita K Yokoyama Y-k Yamada
2927 Second-Generation Biomimetic Total Synthesis of Chaetominine A Coste G Karthikeyan F Couty G Evano
2935 Total Synthesis of (+)-Fostriecin and (+)-Phoslactomycin B S Shibahara M Fujino Y Tashiro N Okamoto T Esumi K Takahashi J Ishihara S Hatakeyama
2954 Stereochemical Assignments of the Chlorinated Residues in Victorin C A C Durow C Butts C L Willis
2963 Studies of the Asymmetric Total Synthesis of Clavilactone D by the lsquoLariatrsquo Cyclization Strategy T Yoshimitsu S Nojima M Hashimoto K Tsukamoto T Tanaka
2970 Total Synthesis of the Leucetta-Derived Alkaloid Calcaridine A P B Koswatta R Sivappa H V R Dias C J Lovely
2983 Formal Synthesis of Salinosporamide A Starting from D-Glucose T Momose Y Kaiya J-i Hasegawa T Sato N Chida
2992 Synthesis of Bioactive Natural Products by Asymmetric syn- and anti-Aldol Reactions A K Ghosh Z L Dawson
no 18 3003 Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural
Products B M Trost M K Brennan 3026 One-Pot Synthesis of Furo[34-b]pyridin-5(7H)-ones from 2-
Bromopyridine-3-carboxylic Acid and Carbonyl Compounds K Kobayashi T Kozuki H Konishi
3029 Iodocyclization of N-[2-(Methylthio)phenyl]propiolamides Selective Synthesis of 3-Iodo-15-benzothiazepin-4-ones T-S Jiang X-G Zhang J-H Li
3039 A Facile Synthetic Method for Fluorine-Containing 17-Phenanthrolines Pyridine-Ring Formation Reaction of N-Propargyl-68-bis(trifluoroacetyl)-quinolin-5-amine with Various Nucleophiles D Shibata E Okada M Hinoshita M Meacutedebielle
3047 Enantiotopic Discrimination in Palladium-Mediated Nucleophilic Substitutions on Achiral Substrates Chiral Ligand versus Chiral Nucleophile O Jacquet F Charnay J-C Fiaud J Ollivier
3051 Studies on the Chemistry of 2-[3-(2-Nitrophenyl)-2-oxopropyl]benzaldehydes Novel Syntheses of 5H-Benzo[b]carbazole-611-diones and Indolo[12-b]isoquinoline-611-diones M Fernaacutendez
3061 Studies on the C22ndashC23 Aldol Coupling of Spirangien M Lorenz N Bluhm M Kalesse
3067 One-Pot Synthesis of N-Alkyl Purine Pyrimidine and Azole Derivatives from Alcohols using Ph3PCCl4 A Rapid Route to Carboacyclic Nucleoside Synthesis M N Soltani Rad A Khalafi-Nezhad S Behrouz Z Asrari M Behrouz Z Amini
3077 Synthesis of 2-Amino-34-dihydroquinazolines and Imidazo[21-b]quinazoline-2-ones A Mishra S Batra
3089 Studies on the Reaction of Diimines with Thiourea Synthesis and Solvent-Induced cistrans-Isomerization of 135-Triazinane-2-thiones B Kaboudin T Ghasemi T Yokomatsu
3094 Suzuki Coupling of Heteroaromatic Chlorides Using Highly Electron-Donating ClickPhos Ligands S M Spinella Z-H Guan J Chen X Zhang
3099 Reaction of NN-Dioxyenamines with Anhydrides of Carboxylic and Sulfonic Acids A New Method for the Synthesis of a-Hydroxyoxime Derivatives A A Tabolin A V Lesiv S L Ioffe
3106 Directed ortho Metallation Chemistry and Phosphine Synthesis New Ligands for the SuzukindashMiyaura Reaction D B G Williams S J Evans H de Bod M S Mokhadinyana T Hughes
3113 New Functional Derivatives of 9-Phenylquinine P J Boratyński J SkarŜewski
3120 On the Synthesis of Asymmetric and Dissymmetric Amino Analogues of Troumlgerrsquos Base J Artacho K Waumlrnmark
3127 Synthesis of Polycyclic Sultams by Palladium-Catalyzed Intramolecular Cyclization K C Majumdar S Mondal N De
3136 Synthesis of Functionalized L-Cysteine and L-Methionine by Reaction with Electron-Deficient Acetylenes B A Trofimov A G Malrsquokina O A Shemyakina V V Nosyreva A P Borisova S S Khutsishvili L B Krivdin
3143 A lsquoClickrsquo Approach to the Synthesis of 3-[2-(1-Alkyltriazol-4-yl)ethyl]indoles M Petrini R R Shaikh
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
1708 Efficient Synthesis of Azo Dye Labeled Terpenes Sugars and Steroids Using N-(4-Arylazobenzoyl)-1H-benzotriazoles A R Katritzky S R Tala N E Abo-Dya Z K Abdel-Samii
1715 Tandem CH-ActivationndashImine-Formation Reaction A New Route to Imidazo[21-a]phthalazines A Heim-Riether K R Gipson
1720 A Convenient and Efficient α-Sulfenylation of Carbonyl Compounds E Okragla S Demkowicz J Rachon D Witt
1725 Stereoselective Synthesis of β-Branched Phenylalanine Derivatives via Chelate-Claisen Rearrangement C Quirin U Kazmaier
1732 Catalyst-Free and Base-Free Water-Promoted SNAr Reaction of Heteroaryl Halides with Thiols B Sreedhar P S Reddy M A Reddy
1739 Convenient Methods for Synthesis of C2-Symmetric Diphenyltetrahydrothiophenes M Periasamy G Ramani G P Muthukumaragopal
1744 Highly Diastereoselective Conjugate AdditionndashElimination of Chiral Nickel(II) Glycinate with Activated Allylic Acetates for Asymmetric Synthesis of Glutamic Acid Derivatives J Wang J Shi X Zhang D Lin H Jiang H Liu
1753 Synthesis of 36-Dimethoxybenzene-12-diamine and of 47-Dimethoxy-2-methyl-1H-benzimidazole T Besset C Morin
1757 An Inexpensive Procedure for Reductive Aminations Using Dimethylamineborane on Millimolar and Molar Scale R Ortmann M Schlitzer
1760 Classics in Stereoselective Synthesis Edited by E M Carreira L Kvaerno Reviewed by Rolf Breinbauer
XV Forthcoming Articles
no 11 1761 Transition-Metal-Catalyzed Enantioselective Synthesis of Compounds with
Non-Centrochirality M Ogasawara S Watanabe 1786 One-Pot Synthesis of 3-Acyl-2-(alkylsulfanyl)indoles and 2-(Alkylsulfanyl)-
indole-3-carboxylates from (2-Isocyanophenyl)methyl Ketones or (2-Isocyanophenyl)acetates S Fukamachi H Konishi K Kobayashi
1791 Efficient and Recyclable Phthalocyanine-Based Sensitizers for Photooxygenation Reactions H Xu W-K Chan D K P Ng
1797 A Facile and Practical One-Pot Synthesis of β-Oxo Thioamides from β-Oxo Amides and Isothiocyanates P Huang D Xiang Y Zhou Y Liang T Na D Dong
1801 Microwave-Promoted Solid-Acid-Catalyzed One-Pot Synthesis of Phthalazinones V M Outerbridge S M Landge H Tamaki B Toumlroumlk
1807 Benzylic Brominations with N-Bromosuccinimide in (Trifluoromethyl)-benzene D Suarez G Laval S-M Tu D Jiang C L Robinson R Scott B T Golding
1811 Synthesis of Thioflavanone and Flavanone Derivatives by Cyclization of Chalcones W Konieczny M Konieczny
1815 A New and Expedient Total Synthesis of Ochratoxin A and d5-Ochratoxin A B Gabriele M Attya A Fazio L Di Donna P Plastina G Sindona
1821 Synthesis of Benzopyrrolizidinones by NorrishndashYang Cyclization of 3-(Acylmethyl)-2-alkylisoindol-1-ones J Wu W Zhang C Wang
1829 Reactions of MoritandashBaylisndashHillman Acetates with Huisgen Zwitterions A Novel Strategy for the Synthesis of β-Amino Acid Derivatives A Jose R R Paul R Mohan S C Mathew A T Biju E Suresh V Nair
1834 Peracetylated β-Allyl C-Glycosides of D-Ribofuranose and 2-Deoxy- D-ribofuranose in the Chemical Literature Until Now Mirages in the Literature H Otero Martinez H Reinke D Michalik C Vogel
1841 Core-Tetrasubstituted Naphthalene Diimides by Stille Cross-Coupling Reactions and Characterization of Their Optical and Redox Properties S-L Suraru F Wuumlrthner
1846 A Practical Synthesis of Indole-Based Heterocycles Using an Amidoaluminum-Mediated Strategy R Todd M M Hossain
1851 Synthesis of Fluorinated Pyrrolo[23-b]pyridine and Pyrrolo[23-d]pyrimidine Nucleosides V O Iaroshenko Y Wang D V Sevenard D M Volochnyuk
1858 Recyclization Reactions of 5-Formyl-13-dimethyluracil with Electron-Rich Amino Heterocycles A P Mityuk D M Volochnyuk S V Ryabukhin A S Plaskon A Shivanyuk A A Tolmachev
1865 Facile Synthesis of Fluorinated 1-Desazapurines V O Iaroshenko D V Sevenard D M Volochnyuk Y Wang A Martiloga A O Tolmachev
1876 A Practical Synthesis of 3-Diethoxyphosphoryl-12-pyridazine Derivatives J-C Monbaliu J Marchand-Brynaert
1881 Enantioselective Reduction of Prochiral Ketones Employing Sprouted Pisum sativa as Biocatalyst J S Yadav B V S Reddy C Sreelakshmi A B Rao
1886 Application of Phenolate Ion Mediated Intramolecular Epoxide Ring Opening in the Enantioselective Synthesis of Functionalized 23-Dihydrobenzofurans and 1-Benzopyrans S K Dinda S K Das G Panda
1897 Complementary Synthetic Approaches to Constitutionally Diverse N-Aminoalkylated Isoindolinones Application to the Synthesis of Falipamil and 5-HT1A Receptor Ligand Analogues M Lorion A Couture E Deniau P Grandclaudon
1904 Selective Deprotection of Silyl Ethers with Sodium Periodate J Li D Menche
1909 Micellar Solution of Sodium Dodecyl Sulfate (SDS) Catalyzes KabacknikndashFields Reaction in Aqueous Media S Sobhani A Vafaee
1916 Convenient Methods for the Synthesis of a Library of Hemilabile Phosphines M V Jimeacutenez J J Peacuterez-Torrente M I Bartolomeacute L A Oro
1923 Terminal Aziridines by Addition of Grignard Reagents or Organoceriums to an (α-Chloro)sulfinylimine D M Hodgson J Kloesges B Evans
1933 A Robust Synthesis of Nε-(Carboxymethyl)-L-lysine (CML) R Csuk S Stark A Barthel R Kluge D Stroumlhl
1935 One-Pot Curtius Rearrangement Processes from Carboxylic Acids O Leogane H Lebel
XV Forthcoming Articles
no 12 1941 The Chemistry of Deprotonated α-Aminonitriles T Opatz 1960 An Efficient Synthesis of Tetraalkyl 2345-Thiophenetetracarboxylate
Derivatives A Alizadeh R Hosseinpour 1963 Facile Deprotection of Bulky (Trialkylsilyl)acetylenes with Silver Fluoride
S Kim B Kim J In 1969 Highly Efficient and Reusable Ionic Liquids for the Catalyzed
Hydroamination of Alkenes with Sulfonamides Carbamates and Carboxamides L Yang L-W Xu C-G Xia
1975 Synthesis of 2391016172324-Octasubstituted Phthalocyaninatozinc(II) Complexes Mediated by Reductive Agents G A Gauna A C Monsalvo J Awruch
1979 A Short and Efficient Synthesis of 3-2-[2-(Bromomethyl)thiazol-4-yl]-ethynyl-5-fluorobenzonitrile A Precursor for PET Radioligand [18F]SP203 M B Gopinathan C Jin K S Rehder
1983 Synthesis of a Substituted Benzazepin-2-one Dihydrate S K Boini R K Vaid K P Moder D Mitchell
1987 Synthesis of Novel Trisubstituted Imidazolines F J Lakner M A Parker B Rogovoy A Khvat A Ivachtchenko
1991 A Novel Synthesis of N-But-3-enyl-α- and β-Amino Acids T T Van Nguyen R T C Brownlee A B Hughes
1999 Synthesis of Substituted 5-(3-Hydroxypropyl)pyrrolidin-2-ones and Pyrrolizidinones from Nitroethane via C3 Functionalized 56-Dihydro-4H-12-oxazines A Novel Approach to Some Analogues of the Antidepressant Rolipram A Yu Sukhorukov A V Lesiv Y A Khomutova S L Ioffe V A Tartakovsky
2009 Chiral Cyclobutanols and Cyclopentane Dimers via Samarium(II) Iodide Induced Keto-Olefin Cyclisations of Carbohydrate-Derived Unsaturated Ketones D B G Williams J Caddy K Blann J J C Groveacute C W Holzapfel
2015 Synthesis of Perfluoroalkylthio-Substituted Ferrocenes C Rhode J Lemke M Lieb N Metzler-Nolte
2019 Functionalization of Polyhedral Oligomeric Silsesquioxane (POSS) via Nucleophilic Substitution M Dutkiewicz H Maciejewski B Marciniec
2025 A Novel Synthesis of Aryl Mesylates via One-Pot DemethylationndashMesylation of Aryl Methyl Ethers Using a Mixture of Phosphorus Pentoxide in Methanesulfonic Acid B Kaboudin Y Abedi
2029 Anionic Cyclization of (NN-Dimethylamino)[2-(prop-2-yn-1-yloxy)aryl]-acetonitriles T Zdrojewski J Musielak A Jończyk
2035 Strecker-Type Reaction Catalyzed by Carboxylic Acids in Aqueous Media Z Xie G Li G Zhao J Wang
2040 Synthesis of Novel Structurally Simplified Estrogen Analogues with Electron-Donating Groups in Ring A L F Tietze C A Vock I K Krimmelbein L Nacke
2061 On the Resolution of Secondary Phosphine Oxides via Diastereomeric Complex Formation The Case of tert-Butylphenylphosphine Oxide J Holt A M Maj E P Schudde K M Pietrusiewicz L Sieroń W Wieczorek T Jerphagnon I W C E Arends U Hanefeld A J Minnaard
2066 Enantioselective Copper-Catalyzed Conjugate Addition of Dimethylzinc to 5-(1-Arylalkylidene) Meldrumrsquos Acids A Wilsily T Lou E Fillion
2073 SuzukindashMiyaura Coupling Reactions Using Phosphite Ligands M Jang Y Jo I-K Oh H M Jung S Lee
2076 Synthesis of 2-Methylindoline- and 2-Methyl-1234-tetrahydroquinoline-Derived Phosphoramidites and Their Applications in Iridium-Catalyzed Allylic Alkylation of Indoles W-B Liu H He L-X Dai S-L You
2083 Stereocontrolled Synthesis of 13-Amino Alcohols by Reduction of Substituted 2-1-[(tert-Butylsulfinyl)amino]alkylcyclohexanones J C Gonzaacutelez-Goacutemez F Foubelo M Yus
2089 Tunable Phosphoramidite Ligands for Asymmetric Hydrovinylation Ligands par excellence for Generation of All-Carbon Quaternary Centers C R Smith H J Lim A ZhangT V RajanBabu
2101 Copper-Catalyzed Asymmetric Ring-Opening Reaction of Oxabenzonorbornadienes with Grignard and Aluminum Reagents R Millet L Gremaud T Bernardez L Palais A Alexakis
2113 A Simplified Synthesis of Takemotorsquos Catalyst A Berkessel B Seelig 2116 Pharmaceutical Substances Syntheses Patents and Applications of the
Most Relevant AIPs Edited by Axel Kleeman Juumlrgen Engel Bernhard Kutscher Dietmar Reichert Reviewed by I Agranat
XV Forthcoming Articles
no 13 2117 Recent Advances in the Aza-Claisen Rearrangement K C Majumdar
T Bhattacharyya B Chattopadhyay B Sinha 2143 A Novel and Convenient Synthesis of lsquoReversedrsquo Diamidino 25-Aryl- and
25-Azaheterocycle-Substituted Furans L Hu D W Boykin 2146 Efficient and General Preparation of Pyranostilbenes First Total Synthesis
of Artocarbene and Pawhuskin B B H Park Y R Lee W S Lyoo 2155 Mild Oxidation of Diarylacetylenes to 12-Diketones Using Oxone in
Trifluoroacetic Acid J-H Chu Y-J Chen M-J Wu 2163 One-Pot Microwave-Assisted Selective Azido ReductionTandem Cyclization
in Condensed and Solid Phase with Nickel Boride N Shankaraiah N Markandeya M Espinoza-Moraga C Arancibia A Kamal L Silva Santos
2171 Pyrrolo[321-ij]quinolin-4-one and Pyrrolo[321-ij]quinolin-6-one H McNab D J Nelson E J Rozgowska
2175 Practical Synthesis of 5-Substituted Tetrazoles under Microwave Irradiation J Roh T V Artamonova K Vaacutevrovaacute G I Koldobskii A Hrabaacutelek
2179 A Simple Method for the Synthesis of 3-Arylthieno[23-b]pyridines via Iodine-Mediated Cyclization of 3-(1-Arylalkenyl)-2-[(1-phenylethyl)sulfanyl]pyridines K Kobayashi D Nakamura Y Shiroyama S Fukamachi H Konishi
2184 Synthesis of Four Lysine-Linked Cereulide Analogues Showing Ionophoric Activity Towards Potassium Cations as Lead Compounds for Emetic Toxin-Detection by Immunoassays A Makarasen T Nishikawa M Isobe
2205 Synthesis of α-Aliphatic and β-Aromatic Substituted Taurines via Regioselective Ring Opening of Thiiranes with Ammonia H Yu S Cao L Zhang G Liu J Xu
2210 Stability of 5(6)-Carboxyfluorescein in Microwave-Assisted Synthesis of Fluorescein-Labelled O-Dimannosylated Peptides R Kowalczyk P W R Harris R P Dunbar M A Brimble
2223 Diversity-Oriented Synthesis of Functionalized Diaryl Sulfones by Regioselective [3+3] Cyclizations of 13-Bis(siloxy)buta-13-dienes with 2-(Arylsulfonyl)-3-ethoxy-2-en-1-ones Scope and Limitations M Shkoor A Riahi O Fatunsin H Reinke C Fischer P Langer
2236 Synthesis of Functionalized Salicylates by Formal [3+3] Cyclocondensation of 13-Bis(silyloxy)buta-13-dienes with 3-Alkoxy-2-en-1-ones G Mroszlig S Ladzik H Reinke A Spannenberg C Fischer P Langer
2249 Synthetic Approach to Alkoxy-β-(trifluoromethyl)styrenes and Their Application in the Synthesis of New Trifluoromethylated Heterocycles V M Muzalevskiy V G Nenajdenko A V Shastin E S Balenkova G Haufe
2260 o-Benzenedisulfonimide as a Powerful and Recyclable Organocatalyst for the Nazarov Reaction M Barbero S Cadamuro A Deagostino S Dughera P Larini E G Occhiato C Prandi S Tabasso R Vulcano P Venturello
2267 The Catalytic Potential of 4-Guanidinylpyridines in Acylation Reactions I Held E Larionov C Bozler F Wagner H Zipse
2278 Iron(III) Chloride in EthanolndashWater Highly Efficient Catalytic System for the Synthesis of Garcia Gonzalez Polyhydroxyalkyl- and C-Glycosylfurans L Nagarapu M V Chary A Satyender B Supriya R Bantu
2283 Ruthenium-Catalyzed Addition of Primary Amides to Alkynes A Stereoselective Synthesis of Secondary Enamides L J Gooszligen M Blanchot K S M Salih K Gooszligen
2289 Binaphthyl-Modified Quaternary Phosphonium Salts as Chiral Phase Transfer Catalysts Application to Asymmetric Amination of β-Keto Esters R He K Maruoka
X Table of Contents XI Forthcoming Articles
no 14 2293 Direct Methods for Stereoselective Polypropionate Synthesis A Survey
J Li D Menche 2316 Synthesis of Symmetrical Ketones from Grignard Reagents and
11-Carbonyldiimidazole D Bottalico V Fiandanese G Marchese A Punzi
2319 Synthesis of 45-Substituted Imidazoles by a Fast Condensation of 12-Diketones and Urotropine in Heterogeneous Medium G Bratulescu
2321 (Arylsulfonyl)acetones and -acetonitriles New Activated Methylenic Building Blocks for Synthesis of 123-Triazoles N T Pokhodylo V S Matiychuk M D Obushak
2324 A Safe Convenient and Efficient One-Pot Synthesis of α-Chloroketone Acetals Directly from Ketones Using Iodobenzene Dichloride J Yu C Zhang
2329 An Efficient Oxidative Conversion of Aldehydes into 2-Substituted 2-Oxazolines Using 13-Diiodo-55-dimethylhydantoin S Takahashi H Togo
2333 A Novel Procedure for the Synthesis of Benzo[b][18]naphthyridine-3-carboxylate Derivatives from MoritandashBaylisndashHillman Adduct Acetates W Zhong F Lin R Chen W Su
2341 An Improved Synthesis of 147-Triazacyclononanes (tacns) and 14710-Tetraazacyclododecanes (cyclens) J Huang Z Zhou T H Chan
2345 The Ullmann Coupling between 2-Chlorobenzoic Acids and Amino Acids A Valuable Reaction for Preparing 2-Substituted 1-Acetyl-1H-indol-3-yl Acetates J C Rodriguez Dominguez X Gang G Kirsch
2349 gem-Dibromomethyl Aromatics Efficient Aldehyde Equivalents in the KnoevenagelndashDoebner Reaction J K Augustine Y A Naik S Poojari N Chowdappa B S Sherigara K Areppa
2357 Synthesis of Novel α-Aminophosphonates Containing Adamantyl Fragment M M Kabachnik L I Minaeva I P Beletskaya
2361 Efficient Fluoride-Mediated Synthesis of 5-Amino-Substituted Isothiazoles Y S Zubenko V I Potkin
2365 Phosphine-Catalyzed Reaction of Cyanohydrins with Activated Alkynes A Siby O Loreau F Taran
2371 Sulfanyl-Substituted [3]Cumulenes and Buta-13-dienes from a Tetrakis(pyridinium)-Substituted Butadiene A Schmidt A Rahimi M Gjikaj
2379 Efficient Synthesis of 2-Substituted Pyrido[32-d]pyrimidines Involving SNAr and Palladium-Catalyzed Cross-Coupling Reactions A Tikad S Routier M Akssira J-M Leacuteger C Jarry G Guillaumet
2385 Novel Synthesis of Medium-Sized Heterocycles by Palladium-Catalyzed Intramolecular Heck Reaction via 9-endo-trig Mode of Cyclization K C Majumdar B Chattopadhyay
2393 Facile Synthesis of Fluorinated Benzofuro- and Benzothieno[23-b]pyridines α-Carbolines and Nucleosides Containing the α-Carboline Framework V O Iaroshenko Y Wang B Zhang D Volochnyuk V Ya Sosnovskikh
2403 Synthesis of Functionalized N-Vinyl Nitrogen-Containing Heterocycles S M M Lopes A M Beja M Ramos Silva J A Paixatildeo F Palacios T M V D Pinho e Melo
2408 Kumada Cross-Coupling of Aryl Grignard Reagents with Aryl Halides Catalyzed by an Immobilized Nickel Catalyst X Chen L Wang J Liu
2413 Highly Enantioselective Synthesis of Heteroaromatic Alcohols Catalyzed by Chiral DiaminodiphosphinendashRuthenium(II) Complexes W-Y Shen Y-Y Li Z-R Dong J-X Gao
2418 Concise Total Synthesis of (+)-Disparlure and its trans-Isomer Using Asymmetric Organocatalysis S-G Kim
2423 Rhodium Carbenoid Induced [12]-Migration in an L-Lyxo-Configured α-Diazo β-Keto Ester Synthesis of a New Griseolic Acid Analogue N N Bhujbal K S A Kumar D D Dhavale
2430 Synthesis of 5-Arylthio-3-hydroxyphthalates by the First [4+2] Cycloadditions of 3-Arylthio-1-silyloxy-13-butadienes with Dimethyl Acetylenedicarboxylate I Iqbal M Imran P Langer
2435 Synthesis of Highly Functionalized Proline Derivatives via a One-Pot MichaelSN-AdditionCyclization Approach U Kazmaier C Schmidt
2440 RhodiumGraphite-Catalyzed Hydrogenation of Carbocyclic and Heterocyclic Aromatic Compounds G Falini A Gualandi D Savoia
2447 Potassium [1-(tert-Butoxycarbonyl)-1H-indol-2-yl]trifluoroborate as an Efficient Building Block in Palladium-Catalyzed SuzukindashMiyaura Cross Couplings P Kassis V Beacuteneacuteteau J-Y Meacuterour S Routier
2454 Syntheses of Substituted Furans and Pyrroles by Platinum-Catalyzed Cyclizations of Propargylic Oxiranes and Aziridines in Aqueous Media M Yoshida M Al-Amin K Shishido
2467 Transition-Metal-Free Oxidative Homocoupling of Aryl Alkenyl and Alkynyl Grignard Reagents with TEMPO M S Maji A Studer
XIII Forthcoming Articles
no 15 2471 Advances in Synthetic Approaches for the Preparation of Combretastatin-
Based Anti-Cancer Agents R Singh H Kaur 2492 Synthesis of Unsymmetrical Ureas by Sulfur-Assisted Carbonylation with
Carbon Monoxide and Oxidation with Molecular Oxygen under Mild Conditions T Mizuno T Nakai M Mihara
2497 Ring-OpeningRecyclization Reactions of (Dimethylamino)propenoyl-Substituted Cyclopropanes Facile Synthesis of Halogenated Pyridin-2(1H)-ones R Zhang Y Zhou Y Liang Z Jiang D Dong
2501 Facile and Efficient Total Synthesis of Taspine B Cheng S Zhang L Zhu J Zhang Q Li A Shan L He
2505 Oligomeric Iodosylbenzene Sulfate A Convenient Hypervalent Iodine Reagent for Oxidation of Organic Sulfides and Alkenes M S Yusubov R Y Yusubova T V Funk K-W Chi V V Zhdankin
2509 Pyrrolidine-Based Organocatalysts for Enantioselective Michael Addition of Cyclohexanone to trans-β-Nitrostyrene A P Carley S Dixon J D Kilburn
2517 CundashAl Hydrotalcite An Efficient and Reusable Ligand-Free Catalyst for the Coupling of Aryl Chlorides with Aliphatic Aromatic and N(H)-Heterocyclic Amines B Sreedhar R Arundhathi P L Reddy M A Reddy M L Kantam
2523 Highly Efficient Synthesis of trans-βγ-Unsaturated a-Keto Amides C Allais T Constantieux J Rodriguez
2531 Gas-Phase Synthesis of N-Unsubstituted 3-Hydroxypyrroles and 1H-Pyrrol-3(2H)-ones L Hill G A Hunter S H Imam H McNab W J OrsquoNeill
2535 3-Hydroxy-1H-pyrrole L Hill S H Imam H McNab W J OrsquoNeill 2539 123-Thiadiazoles with Unsaturated Side Chains Synthesis
Polymerization and Photocrosslinking M Al-Smadi N Hanold H Kalbitz H Meier
2547 Synthesis of 1112-Didehydrodibenzo[ae]cycloocten-5(6H)-one A Strained Eight-Membered Alkyne S C Kornmayer F Rominger R Gleiter
2553 Stannous Chloride Dihydrate A Novel and Efficient Catalyst for the Synthesis of gem-Dihydroperoxides from Ketones and Aldehydes D Azarifar K Khosravi F Soleimanei
2557 Synthesis of a Novel Class of Azacrown Macrocycles and Lariat Crown Ethers Containing Two 124-Triazole Rings as Subunits N Foroughifar A Mobinikhaledi S Ebrahimi
2561 Enantioselective Synthesis of the 3C-Protease Inhibitor (ndash)-Thysanone by a StauntonndashWeinreb Annulation Strategy J Sperry T Y Yuen M A Brimble
2570 Stereoselective Synthesis of Unnatural β-Amino Acids from Nitroethane via 56-Dihydro-4H-12-oxazin-3-ylacetates A Yu Sukhorukov A V Lesiv O L Eliseev Y A Khomutova S L Ioffe
2579 A Versatile Unexpected One-Pot Regioselective Synthesis of a New Class of 13-Diazepinoindolones by Reaction of Pyranoindolones with Monosubstituted Ureas D Livadiotou C A Tsoleridis J Stephanidou-Stephanatou
2584 Synthesis of a Trisaccharide and a Tetrasaccharide from the Cell-Wall Lipopolysaccharides of Azospirillum brasilense S17 S Pandey S Ghosh A K Misra
2591 Synthesis of Isoindoline Nitroxides by Electrocyclic Reactions T Kaacutelai J Jekı K Hideg
2596 Glycosylations of Tertiary Alcohols Synthesis of Fully Protected Disaccharides with Sterically Demanding Groups Attached to the Sugar Core A Holkenbrink J B Vicente D B Werz
2605 Copper-Catalyzed [13]-Dipolar Cycloaddition for the Synthesis of Macrocycles Containing Acyclic Aromatic and Steroidal Moieties G V Latyshev M S Baranom A V Kazantsev A D Averin N V Lukashev I P Beletskaya
2616 Aryl Ring Migration Reaction in the Synthesis of 24-Diaryl-4H-31-benzothiazines A V Butin F A Tsiunchik V T Abaev A V Gutnov D A Cheshkov
2627 Hydrogenation of β-N-Substituted and β-NN-Disubstituted Enamino Esters in the Presence of Iridium(I) Catalyst H Hebbache Z Hank C Bruneau J-L Renaud
2634 Stereoselective Olefination Reactions Promoted by Rieke Manganese J M Concelloacuten H Rodriacuteguez-Solla V del Amo P Diacuteaz
2646 Synthesis of Piperidinones through a Radical Cascade E Godineau Y Landais
2650 Asymmetric Organic Synthesis with Enzymes Edited by V Gotor I Alfonso E Garciacutea-Urdiales Reviewed by Steve Collier
XVII Forthcoming Articles
no 16 2651 Synthesis of Spirocyclic Ethers S Rosenberg R Leino 2674 Bimetallic PalladiumndashPlatinum-on-Carbon-Catalyzed HndashD Exchange
Reaction Synergistic Effect on Multiple Deuterium Incorporation T Maegawa N Ito K Oono Y Monguchi H Sajiki
2679 Efficient Copper-Catalyzed Synthesis of 2-Amino-4(3H)-quinazolinone and 2-Aminoquinazoline Derivatives X Huang H Yang H Fu R Qiao Y Zhao
2689 Synthesis and Chemoselective N- and O-Alkylation of Thiadiazolopyrimidine Nucleosides and Uridines A M L Hossion R Islam R K Kandahary T Nagamatsu
2697 Facile and Efficient Synthesis of a New Class of Indole-Substituted Pyridine Derivatives via One-Pot Multicomponent Reactions K Zhao X-P Xu S-L Zhu D-Q Shi Y Zhang S-J Ji
2709 Studies toward a Total Synthesis of Rhizoxin D Stereoselective Preparation of the C11ndashC19 Fragment S Padakanti C K Kumar E Ashok P Das
2715 A Short Synthesis of Enantiomeric Phytoprostanes B1 Type I W Perlikowska M Mikołajczyk
2719 Chemistry of Polyhalogenated Nitrobutadienes Part 7 A Novel Synthetic Access to Chlorinated Nitrile Oxides E Nutz V A Zapolrsquoskii D E Kaufmann
2725 Microwave-Assisted Silver(I)-Mediated Selective O-Alkylation of Aromatic Imidate Systems B K Singh C Cavalluzzo M De Maeyer Z Debyser V S Parmar E Van der Eycken
2729 Iodogen A Novel Reagent for the Oxidation of Urazoles under Heterogeneous Conditions A Khoramabadi A Shiri M A Zolfigol S Mallakpour
2733 An Unprecedented Synthesis of Eight-Membered-Ring Cyclic Thioimidic Esters by a Three-Component Reaction A Alizadeh R Hosseinpour
2737 A Novel Diastereoselective Synthesis of β-Phosphonato Unsaturated Thioimidates A Alizadeh N Zohreh
2741 Synthesis of 21-Benzisoxazoles by Nucleophilic Substitution of Hydrogen in Nitroarenes Activated by the Azole Ring N T Pokhodylo Y O Teslenko V S Matiychuk M D Obushak
2749 A Facile Synthesis of Two Series of Multifunctional Carbon Compounds from αα-Dihalo Ketones Using Allylsamarium Bromide X Liu S Zhang J Di
2756 Stereocontrolled Formation of Protected Aminodeoxyalditols from Simple Carbohydrate Precursors by Debenzylating Cycloetherification Y Jiang Z Fang Q Zheng H Jia J Cheng B Zheng
2761 trans-Stilbene as a Starting Material for the Synthesis of Tamoxifen Based on Palladium-Catalyzed Cross-Coupling Reactions C M Nunes J Limberger S Poersch M Seferin A L Monteiro
2766 Synthesis and Biological Evaluation of 6-Substituted Purinylcarbanucleosides with a Cyclopenta[b]thiophene Pseudosugar P Abeijoacuten J M Blanco O Caamantildeo F Fernaacutendez M D Garciacutea X Garciacutea-Mera J E Rodriacuteguez-Borges J Balzarini E De Clercq
2773 Synthesis and Electrochemical Signature of Novel Norbornyl-ferrocene Hybrids F A Khan S K Upadhyay
2778 A Regioselective TsujindashTrost Pentadienylation of 3-Allyltetronic Acid R Schobert B Barnickel
2785 Copper(I)-Catalyzed CarylndashCalkynyl Bond Formation of Aryl Iodides with Terminal Alkynes K G Thakur G Sekar
2790 Aminolysis of Epoxides Using Iridium Trichloride as an Efficient Catalyst J Agarwal A Duley R Rani R K Peddinti
2797 Preparation of Several Active N-Chloro Compounds from Trichloroisocyanuric Acid A Shiri A Khoramabadi-zad
2802 The First Mineral-Catalyzed One-Pot [3+1+2] Coupling Protocol for Multifunctionalized Fused-Ring Pyrimidines L D S Yadav A Rai
2809 Efficient Synthesis of Tetrahydro-β-carbolin-1-one and Dihydroisoquinolin-1-one Derivatives as Versatile Intermediates K E Judd M F Mahon L Caggiano
2818 A Concise Synthesis of ortho-Iodobenzyl Alcohols via Addition of ortho-Iodophenyl Grignard Reagent to Aldehydes and Ketones J Cvengroš D Stolz A Togni
XIII Forthcoming Articles
no 17 2825 Reactivity of Oxazol-5-(4H)-ones and Their Application toward Natural
Product Synthesis N M Hewlett C D Hupp J J Tepe 2840 Towards the Total Synthesis of 3-Hydroxyvibsanin E B D Schwartz
J R Denton P V Bernhardt H M L Davies C M Williams 2847 Structure Investigations of (ent)-Cladospolide D by De Novo Synthesis and
Kinetic and Thermodynamic Isomerization Y Xing J H Penn G A OrsquoDoherty
2855 New Applications of PhI(OAc)2 in Synthesis Total Synthesis and SAR Development of Potent Antitumor Natural Product PsymberinIrciniastatin A N Shao X Huang A Palani R Aslanian A Buevich J Piwinski R Huryk C Seidel-Dugan
2873 Total Synthesis of Largazole ndash Devolution of a Novel Synthetic Strategy B Wang C J Forsyth
2881 Formal Total Synthesis of Palmerolide A J Jaumlgel M E Maier 2893 Total Synthesis of Bongkrekic Acid via Sequential SuzukindashMiyaura Coupling
Reactions M Kanematsu M Shindo M Yoshida K Shishido 2905 Stereodivergent Approach to Both C28a-syn and C28a-anti Relative
Stereochemical Manifolds in the Lepadin Family via a TiCl4-Promoted G Li L J Carlson I K Sagamanova B W Slafer R P Hsung C Gilardi H M Sklenicka N Sydorenko
2915 Enantioselective Aldol Reaction of Tetrasubstituted Ketene Silyl Acetals with Achiral Aldehydes for the Construction of Asymmetric Tertiary Alcohols An Application for the Divergent Total Syntheses of Buergerinins F and G I Shiina T Iizumi Y-s Yamai Y-i Kawakita K Yokoyama Y-k Yamada
2927 Second-Generation Biomimetic Total Synthesis of Chaetominine A Coste G Karthikeyan F Couty G Evano
2935 Total Synthesis of (+)-Fostriecin and (+)-Phoslactomycin B S Shibahara M Fujino Y Tashiro N Okamoto T Esumi K Takahashi J Ishihara S Hatakeyama
2954 Stereochemical Assignments of the Chlorinated Residues in Victorin C A C Durow C Butts C L Willis
2963 Studies of the Asymmetric Total Synthesis of Clavilactone D by the lsquoLariatrsquo Cyclization Strategy T Yoshimitsu S Nojima M Hashimoto K Tsukamoto T Tanaka
2970 Total Synthesis of the Leucetta-Derived Alkaloid Calcaridine A P B Koswatta R Sivappa H V R Dias C J Lovely
2983 Formal Synthesis of Salinosporamide A Starting from D-Glucose T Momose Y Kaiya J-i Hasegawa T Sato N Chida
2992 Synthesis of Bioactive Natural Products by Asymmetric syn- and anti-Aldol Reactions A K Ghosh Z L Dawson
no 18 3003 Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural
Products B M Trost M K Brennan 3026 One-Pot Synthesis of Furo[34-b]pyridin-5(7H)-ones from 2-
Bromopyridine-3-carboxylic Acid and Carbonyl Compounds K Kobayashi T Kozuki H Konishi
3029 Iodocyclization of N-[2-(Methylthio)phenyl]propiolamides Selective Synthesis of 3-Iodo-15-benzothiazepin-4-ones T-S Jiang X-G Zhang J-H Li
3039 A Facile Synthetic Method for Fluorine-Containing 17-Phenanthrolines Pyridine-Ring Formation Reaction of N-Propargyl-68-bis(trifluoroacetyl)-quinolin-5-amine with Various Nucleophiles D Shibata E Okada M Hinoshita M Meacutedebielle
3047 Enantiotopic Discrimination in Palladium-Mediated Nucleophilic Substitutions on Achiral Substrates Chiral Ligand versus Chiral Nucleophile O Jacquet F Charnay J-C Fiaud J Ollivier
3051 Studies on the Chemistry of 2-[3-(2-Nitrophenyl)-2-oxopropyl]benzaldehydes Novel Syntheses of 5H-Benzo[b]carbazole-611-diones and Indolo[12-b]isoquinoline-611-diones M Fernaacutendez
3061 Studies on the C22ndashC23 Aldol Coupling of Spirangien M Lorenz N Bluhm M Kalesse
3067 One-Pot Synthesis of N-Alkyl Purine Pyrimidine and Azole Derivatives from Alcohols using Ph3PCCl4 A Rapid Route to Carboacyclic Nucleoside Synthesis M N Soltani Rad A Khalafi-Nezhad S Behrouz Z Asrari M Behrouz Z Amini
3077 Synthesis of 2-Amino-34-dihydroquinazolines and Imidazo[21-b]quinazoline-2-ones A Mishra S Batra
3089 Studies on the Reaction of Diimines with Thiourea Synthesis and Solvent-Induced cistrans-Isomerization of 135-Triazinane-2-thiones B Kaboudin T Ghasemi T Yokomatsu
3094 Suzuki Coupling of Heteroaromatic Chlorides Using Highly Electron-Donating ClickPhos Ligands S M Spinella Z-H Guan J Chen X Zhang
3099 Reaction of NN-Dioxyenamines with Anhydrides of Carboxylic and Sulfonic Acids A New Method for the Synthesis of a-Hydroxyoxime Derivatives A A Tabolin A V Lesiv S L Ioffe
3106 Directed ortho Metallation Chemistry and Phosphine Synthesis New Ligands for the SuzukindashMiyaura Reaction D B G Williams S J Evans H de Bod M S Mokhadinyana T Hughes
3113 New Functional Derivatives of 9-Phenylquinine P J Boratyński J SkarŜewski
3120 On the Synthesis of Asymmetric and Dissymmetric Amino Analogues of Troumlgerrsquos Base J Artacho K Waumlrnmark
3127 Synthesis of Polycyclic Sultams by Palladium-Catalyzed Intramolecular Cyclization K C Majumdar S Mondal N De
3136 Synthesis of Functionalized L-Cysteine and L-Methionine by Reaction with Electron-Deficient Acetylenes B A Trofimov A G Malrsquokina O A Shemyakina V V Nosyreva A P Borisova S S Khutsishvili L B Krivdin
3143 A lsquoClickrsquo Approach to the Synthesis of 3-[2-(1-Alkyltriazol-4-yl)ethyl]indoles M Petrini R R Shaikh
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
no 11 1761 Transition-Metal-Catalyzed Enantioselective Synthesis of Compounds with
Non-Centrochirality M Ogasawara S Watanabe 1786 One-Pot Synthesis of 3-Acyl-2-(alkylsulfanyl)indoles and 2-(Alkylsulfanyl)-
indole-3-carboxylates from (2-Isocyanophenyl)methyl Ketones or (2-Isocyanophenyl)acetates S Fukamachi H Konishi K Kobayashi
1791 Efficient and Recyclable Phthalocyanine-Based Sensitizers for Photooxygenation Reactions H Xu W-K Chan D K P Ng
1797 A Facile and Practical One-Pot Synthesis of β-Oxo Thioamides from β-Oxo Amides and Isothiocyanates P Huang D Xiang Y Zhou Y Liang T Na D Dong
1801 Microwave-Promoted Solid-Acid-Catalyzed One-Pot Synthesis of Phthalazinones V M Outerbridge S M Landge H Tamaki B Toumlroumlk
1807 Benzylic Brominations with N-Bromosuccinimide in (Trifluoromethyl)-benzene D Suarez G Laval S-M Tu D Jiang C L Robinson R Scott B T Golding
1811 Synthesis of Thioflavanone and Flavanone Derivatives by Cyclization of Chalcones W Konieczny M Konieczny
1815 A New and Expedient Total Synthesis of Ochratoxin A and d5-Ochratoxin A B Gabriele M Attya A Fazio L Di Donna P Plastina G Sindona
1821 Synthesis of Benzopyrrolizidinones by NorrishndashYang Cyclization of 3-(Acylmethyl)-2-alkylisoindol-1-ones J Wu W Zhang C Wang
1829 Reactions of MoritandashBaylisndashHillman Acetates with Huisgen Zwitterions A Novel Strategy for the Synthesis of β-Amino Acid Derivatives A Jose R R Paul R Mohan S C Mathew A T Biju E Suresh V Nair
1834 Peracetylated β-Allyl C-Glycosides of D-Ribofuranose and 2-Deoxy- D-ribofuranose in the Chemical Literature Until Now Mirages in the Literature H Otero Martinez H Reinke D Michalik C Vogel
1841 Core-Tetrasubstituted Naphthalene Diimides by Stille Cross-Coupling Reactions and Characterization of Their Optical and Redox Properties S-L Suraru F Wuumlrthner
1846 A Practical Synthesis of Indole-Based Heterocycles Using an Amidoaluminum-Mediated Strategy R Todd M M Hossain
1851 Synthesis of Fluorinated Pyrrolo[23-b]pyridine and Pyrrolo[23-d]pyrimidine Nucleosides V O Iaroshenko Y Wang D V Sevenard D M Volochnyuk
1858 Recyclization Reactions of 5-Formyl-13-dimethyluracil with Electron-Rich Amino Heterocycles A P Mityuk D M Volochnyuk S V Ryabukhin A S Plaskon A Shivanyuk A A Tolmachev
1865 Facile Synthesis of Fluorinated 1-Desazapurines V O Iaroshenko D V Sevenard D M Volochnyuk Y Wang A Martiloga A O Tolmachev
1876 A Practical Synthesis of 3-Diethoxyphosphoryl-12-pyridazine Derivatives J-C Monbaliu J Marchand-Brynaert
1881 Enantioselective Reduction of Prochiral Ketones Employing Sprouted Pisum sativa as Biocatalyst J S Yadav B V S Reddy C Sreelakshmi A B Rao
1886 Application of Phenolate Ion Mediated Intramolecular Epoxide Ring Opening in the Enantioselective Synthesis of Functionalized 23-Dihydrobenzofurans and 1-Benzopyrans S K Dinda S K Das G Panda
1897 Complementary Synthetic Approaches to Constitutionally Diverse N-Aminoalkylated Isoindolinones Application to the Synthesis of Falipamil and 5-HT1A Receptor Ligand Analogues M Lorion A Couture E Deniau P Grandclaudon
1904 Selective Deprotection of Silyl Ethers with Sodium Periodate J Li D Menche
1909 Micellar Solution of Sodium Dodecyl Sulfate (SDS) Catalyzes KabacknikndashFields Reaction in Aqueous Media S Sobhani A Vafaee
1916 Convenient Methods for the Synthesis of a Library of Hemilabile Phosphines M V Jimeacutenez J J Peacuterez-Torrente M I Bartolomeacute L A Oro
1923 Terminal Aziridines by Addition of Grignard Reagents or Organoceriums to an (α-Chloro)sulfinylimine D M Hodgson J Kloesges B Evans
1933 A Robust Synthesis of Nε-(Carboxymethyl)-L-lysine (CML) R Csuk S Stark A Barthel R Kluge D Stroumlhl
1935 One-Pot Curtius Rearrangement Processes from Carboxylic Acids O Leogane H Lebel
XV Forthcoming Articles
no 12 1941 The Chemistry of Deprotonated α-Aminonitriles T Opatz 1960 An Efficient Synthesis of Tetraalkyl 2345-Thiophenetetracarboxylate
Derivatives A Alizadeh R Hosseinpour 1963 Facile Deprotection of Bulky (Trialkylsilyl)acetylenes with Silver Fluoride
S Kim B Kim J In 1969 Highly Efficient and Reusable Ionic Liquids for the Catalyzed
Hydroamination of Alkenes with Sulfonamides Carbamates and Carboxamides L Yang L-W Xu C-G Xia
1975 Synthesis of 2391016172324-Octasubstituted Phthalocyaninatozinc(II) Complexes Mediated by Reductive Agents G A Gauna A C Monsalvo J Awruch
1979 A Short and Efficient Synthesis of 3-2-[2-(Bromomethyl)thiazol-4-yl]-ethynyl-5-fluorobenzonitrile A Precursor for PET Radioligand [18F]SP203 M B Gopinathan C Jin K S Rehder
1983 Synthesis of a Substituted Benzazepin-2-one Dihydrate S K Boini R K Vaid K P Moder D Mitchell
1987 Synthesis of Novel Trisubstituted Imidazolines F J Lakner M A Parker B Rogovoy A Khvat A Ivachtchenko
1991 A Novel Synthesis of N-But-3-enyl-α- and β-Amino Acids T T Van Nguyen R T C Brownlee A B Hughes
1999 Synthesis of Substituted 5-(3-Hydroxypropyl)pyrrolidin-2-ones and Pyrrolizidinones from Nitroethane via C3 Functionalized 56-Dihydro-4H-12-oxazines A Novel Approach to Some Analogues of the Antidepressant Rolipram A Yu Sukhorukov A V Lesiv Y A Khomutova S L Ioffe V A Tartakovsky
2009 Chiral Cyclobutanols and Cyclopentane Dimers via Samarium(II) Iodide Induced Keto-Olefin Cyclisations of Carbohydrate-Derived Unsaturated Ketones D B G Williams J Caddy K Blann J J C Groveacute C W Holzapfel
2015 Synthesis of Perfluoroalkylthio-Substituted Ferrocenes C Rhode J Lemke M Lieb N Metzler-Nolte
2019 Functionalization of Polyhedral Oligomeric Silsesquioxane (POSS) via Nucleophilic Substitution M Dutkiewicz H Maciejewski B Marciniec
2025 A Novel Synthesis of Aryl Mesylates via One-Pot DemethylationndashMesylation of Aryl Methyl Ethers Using a Mixture of Phosphorus Pentoxide in Methanesulfonic Acid B Kaboudin Y Abedi
2029 Anionic Cyclization of (NN-Dimethylamino)[2-(prop-2-yn-1-yloxy)aryl]-acetonitriles T Zdrojewski J Musielak A Jończyk
2035 Strecker-Type Reaction Catalyzed by Carboxylic Acids in Aqueous Media Z Xie G Li G Zhao J Wang
2040 Synthesis of Novel Structurally Simplified Estrogen Analogues with Electron-Donating Groups in Ring A L F Tietze C A Vock I K Krimmelbein L Nacke
2061 On the Resolution of Secondary Phosphine Oxides via Diastereomeric Complex Formation The Case of tert-Butylphenylphosphine Oxide J Holt A M Maj E P Schudde K M Pietrusiewicz L Sieroń W Wieczorek T Jerphagnon I W C E Arends U Hanefeld A J Minnaard
2066 Enantioselective Copper-Catalyzed Conjugate Addition of Dimethylzinc to 5-(1-Arylalkylidene) Meldrumrsquos Acids A Wilsily T Lou E Fillion
2073 SuzukindashMiyaura Coupling Reactions Using Phosphite Ligands M Jang Y Jo I-K Oh H M Jung S Lee
2076 Synthesis of 2-Methylindoline- and 2-Methyl-1234-tetrahydroquinoline-Derived Phosphoramidites and Their Applications in Iridium-Catalyzed Allylic Alkylation of Indoles W-B Liu H He L-X Dai S-L You
2083 Stereocontrolled Synthesis of 13-Amino Alcohols by Reduction of Substituted 2-1-[(tert-Butylsulfinyl)amino]alkylcyclohexanones J C Gonzaacutelez-Goacutemez F Foubelo M Yus
2089 Tunable Phosphoramidite Ligands for Asymmetric Hydrovinylation Ligands par excellence for Generation of All-Carbon Quaternary Centers C R Smith H J Lim A ZhangT V RajanBabu
2101 Copper-Catalyzed Asymmetric Ring-Opening Reaction of Oxabenzonorbornadienes with Grignard and Aluminum Reagents R Millet L Gremaud T Bernardez L Palais A Alexakis
2113 A Simplified Synthesis of Takemotorsquos Catalyst A Berkessel B Seelig 2116 Pharmaceutical Substances Syntheses Patents and Applications of the
Most Relevant AIPs Edited by Axel Kleeman Juumlrgen Engel Bernhard Kutscher Dietmar Reichert Reviewed by I Agranat
XV Forthcoming Articles
no 13 2117 Recent Advances in the Aza-Claisen Rearrangement K C Majumdar
T Bhattacharyya B Chattopadhyay B Sinha 2143 A Novel and Convenient Synthesis of lsquoReversedrsquo Diamidino 25-Aryl- and
25-Azaheterocycle-Substituted Furans L Hu D W Boykin 2146 Efficient and General Preparation of Pyranostilbenes First Total Synthesis
of Artocarbene and Pawhuskin B B H Park Y R Lee W S Lyoo 2155 Mild Oxidation of Diarylacetylenes to 12-Diketones Using Oxone in
Trifluoroacetic Acid J-H Chu Y-J Chen M-J Wu 2163 One-Pot Microwave-Assisted Selective Azido ReductionTandem Cyclization
in Condensed and Solid Phase with Nickel Boride N Shankaraiah N Markandeya M Espinoza-Moraga C Arancibia A Kamal L Silva Santos
2171 Pyrrolo[321-ij]quinolin-4-one and Pyrrolo[321-ij]quinolin-6-one H McNab D J Nelson E J Rozgowska
2175 Practical Synthesis of 5-Substituted Tetrazoles under Microwave Irradiation J Roh T V Artamonova K Vaacutevrovaacute G I Koldobskii A Hrabaacutelek
2179 A Simple Method for the Synthesis of 3-Arylthieno[23-b]pyridines via Iodine-Mediated Cyclization of 3-(1-Arylalkenyl)-2-[(1-phenylethyl)sulfanyl]pyridines K Kobayashi D Nakamura Y Shiroyama S Fukamachi H Konishi
2184 Synthesis of Four Lysine-Linked Cereulide Analogues Showing Ionophoric Activity Towards Potassium Cations as Lead Compounds for Emetic Toxin-Detection by Immunoassays A Makarasen T Nishikawa M Isobe
2205 Synthesis of α-Aliphatic and β-Aromatic Substituted Taurines via Regioselective Ring Opening of Thiiranes with Ammonia H Yu S Cao L Zhang G Liu J Xu
2210 Stability of 5(6)-Carboxyfluorescein in Microwave-Assisted Synthesis of Fluorescein-Labelled O-Dimannosylated Peptides R Kowalczyk P W R Harris R P Dunbar M A Brimble
2223 Diversity-Oriented Synthesis of Functionalized Diaryl Sulfones by Regioselective [3+3] Cyclizations of 13-Bis(siloxy)buta-13-dienes with 2-(Arylsulfonyl)-3-ethoxy-2-en-1-ones Scope and Limitations M Shkoor A Riahi O Fatunsin H Reinke C Fischer P Langer
2236 Synthesis of Functionalized Salicylates by Formal [3+3] Cyclocondensation of 13-Bis(silyloxy)buta-13-dienes with 3-Alkoxy-2-en-1-ones G Mroszlig S Ladzik H Reinke A Spannenberg C Fischer P Langer
2249 Synthetic Approach to Alkoxy-β-(trifluoromethyl)styrenes and Their Application in the Synthesis of New Trifluoromethylated Heterocycles V M Muzalevskiy V G Nenajdenko A V Shastin E S Balenkova G Haufe
2260 o-Benzenedisulfonimide as a Powerful and Recyclable Organocatalyst for the Nazarov Reaction M Barbero S Cadamuro A Deagostino S Dughera P Larini E G Occhiato C Prandi S Tabasso R Vulcano P Venturello
2267 The Catalytic Potential of 4-Guanidinylpyridines in Acylation Reactions I Held E Larionov C Bozler F Wagner H Zipse
2278 Iron(III) Chloride in EthanolndashWater Highly Efficient Catalytic System for the Synthesis of Garcia Gonzalez Polyhydroxyalkyl- and C-Glycosylfurans L Nagarapu M V Chary A Satyender B Supriya R Bantu
2283 Ruthenium-Catalyzed Addition of Primary Amides to Alkynes A Stereoselective Synthesis of Secondary Enamides L J Gooszligen M Blanchot K S M Salih K Gooszligen
2289 Binaphthyl-Modified Quaternary Phosphonium Salts as Chiral Phase Transfer Catalysts Application to Asymmetric Amination of β-Keto Esters R He K Maruoka
X Table of Contents XI Forthcoming Articles
no 14 2293 Direct Methods for Stereoselective Polypropionate Synthesis A Survey
J Li D Menche 2316 Synthesis of Symmetrical Ketones from Grignard Reagents and
11-Carbonyldiimidazole D Bottalico V Fiandanese G Marchese A Punzi
2319 Synthesis of 45-Substituted Imidazoles by a Fast Condensation of 12-Diketones and Urotropine in Heterogeneous Medium G Bratulescu
2321 (Arylsulfonyl)acetones and -acetonitriles New Activated Methylenic Building Blocks for Synthesis of 123-Triazoles N T Pokhodylo V S Matiychuk M D Obushak
2324 A Safe Convenient and Efficient One-Pot Synthesis of α-Chloroketone Acetals Directly from Ketones Using Iodobenzene Dichloride J Yu C Zhang
2329 An Efficient Oxidative Conversion of Aldehydes into 2-Substituted 2-Oxazolines Using 13-Diiodo-55-dimethylhydantoin S Takahashi H Togo
2333 A Novel Procedure for the Synthesis of Benzo[b][18]naphthyridine-3-carboxylate Derivatives from MoritandashBaylisndashHillman Adduct Acetates W Zhong F Lin R Chen W Su
2341 An Improved Synthesis of 147-Triazacyclononanes (tacns) and 14710-Tetraazacyclododecanes (cyclens) J Huang Z Zhou T H Chan
2345 The Ullmann Coupling between 2-Chlorobenzoic Acids and Amino Acids A Valuable Reaction for Preparing 2-Substituted 1-Acetyl-1H-indol-3-yl Acetates J C Rodriguez Dominguez X Gang G Kirsch
2349 gem-Dibromomethyl Aromatics Efficient Aldehyde Equivalents in the KnoevenagelndashDoebner Reaction J K Augustine Y A Naik S Poojari N Chowdappa B S Sherigara K Areppa
2357 Synthesis of Novel α-Aminophosphonates Containing Adamantyl Fragment M M Kabachnik L I Minaeva I P Beletskaya
2361 Efficient Fluoride-Mediated Synthesis of 5-Amino-Substituted Isothiazoles Y S Zubenko V I Potkin
2365 Phosphine-Catalyzed Reaction of Cyanohydrins with Activated Alkynes A Siby O Loreau F Taran
2371 Sulfanyl-Substituted [3]Cumulenes and Buta-13-dienes from a Tetrakis(pyridinium)-Substituted Butadiene A Schmidt A Rahimi M Gjikaj
2379 Efficient Synthesis of 2-Substituted Pyrido[32-d]pyrimidines Involving SNAr and Palladium-Catalyzed Cross-Coupling Reactions A Tikad S Routier M Akssira J-M Leacuteger C Jarry G Guillaumet
2385 Novel Synthesis of Medium-Sized Heterocycles by Palladium-Catalyzed Intramolecular Heck Reaction via 9-endo-trig Mode of Cyclization K C Majumdar B Chattopadhyay
2393 Facile Synthesis of Fluorinated Benzofuro- and Benzothieno[23-b]pyridines α-Carbolines and Nucleosides Containing the α-Carboline Framework V O Iaroshenko Y Wang B Zhang D Volochnyuk V Ya Sosnovskikh
2403 Synthesis of Functionalized N-Vinyl Nitrogen-Containing Heterocycles S M M Lopes A M Beja M Ramos Silva J A Paixatildeo F Palacios T M V D Pinho e Melo
2408 Kumada Cross-Coupling of Aryl Grignard Reagents with Aryl Halides Catalyzed by an Immobilized Nickel Catalyst X Chen L Wang J Liu
2413 Highly Enantioselective Synthesis of Heteroaromatic Alcohols Catalyzed by Chiral DiaminodiphosphinendashRuthenium(II) Complexes W-Y Shen Y-Y Li Z-R Dong J-X Gao
2418 Concise Total Synthesis of (+)-Disparlure and its trans-Isomer Using Asymmetric Organocatalysis S-G Kim
2423 Rhodium Carbenoid Induced [12]-Migration in an L-Lyxo-Configured α-Diazo β-Keto Ester Synthesis of a New Griseolic Acid Analogue N N Bhujbal K S A Kumar D D Dhavale
2430 Synthesis of 5-Arylthio-3-hydroxyphthalates by the First [4+2] Cycloadditions of 3-Arylthio-1-silyloxy-13-butadienes with Dimethyl Acetylenedicarboxylate I Iqbal M Imran P Langer
2435 Synthesis of Highly Functionalized Proline Derivatives via a One-Pot MichaelSN-AdditionCyclization Approach U Kazmaier C Schmidt
2440 RhodiumGraphite-Catalyzed Hydrogenation of Carbocyclic and Heterocyclic Aromatic Compounds G Falini A Gualandi D Savoia
2447 Potassium [1-(tert-Butoxycarbonyl)-1H-indol-2-yl]trifluoroborate as an Efficient Building Block in Palladium-Catalyzed SuzukindashMiyaura Cross Couplings P Kassis V Beacuteneacuteteau J-Y Meacuterour S Routier
2454 Syntheses of Substituted Furans and Pyrroles by Platinum-Catalyzed Cyclizations of Propargylic Oxiranes and Aziridines in Aqueous Media M Yoshida M Al-Amin K Shishido
2467 Transition-Metal-Free Oxidative Homocoupling of Aryl Alkenyl and Alkynyl Grignard Reagents with TEMPO M S Maji A Studer
XIII Forthcoming Articles
no 15 2471 Advances in Synthetic Approaches for the Preparation of Combretastatin-
Based Anti-Cancer Agents R Singh H Kaur 2492 Synthesis of Unsymmetrical Ureas by Sulfur-Assisted Carbonylation with
Carbon Monoxide and Oxidation with Molecular Oxygen under Mild Conditions T Mizuno T Nakai M Mihara
2497 Ring-OpeningRecyclization Reactions of (Dimethylamino)propenoyl-Substituted Cyclopropanes Facile Synthesis of Halogenated Pyridin-2(1H)-ones R Zhang Y Zhou Y Liang Z Jiang D Dong
2501 Facile and Efficient Total Synthesis of Taspine B Cheng S Zhang L Zhu J Zhang Q Li A Shan L He
2505 Oligomeric Iodosylbenzene Sulfate A Convenient Hypervalent Iodine Reagent for Oxidation of Organic Sulfides and Alkenes M S Yusubov R Y Yusubova T V Funk K-W Chi V V Zhdankin
2509 Pyrrolidine-Based Organocatalysts for Enantioselective Michael Addition of Cyclohexanone to trans-β-Nitrostyrene A P Carley S Dixon J D Kilburn
2517 CundashAl Hydrotalcite An Efficient and Reusable Ligand-Free Catalyst for the Coupling of Aryl Chlorides with Aliphatic Aromatic and N(H)-Heterocyclic Amines B Sreedhar R Arundhathi P L Reddy M A Reddy M L Kantam
2523 Highly Efficient Synthesis of trans-βγ-Unsaturated a-Keto Amides C Allais T Constantieux J Rodriguez
2531 Gas-Phase Synthesis of N-Unsubstituted 3-Hydroxypyrroles and 1H-Pyrrol-3(2H)-ones L Hill G A Hunter S H Imam H McNab W J OrsquoNeill
2535 3-Hydroxy-1H-pyrrole L Hill S H Imam H McNab W J OrsquoNeill 2539 123-Thiadiazoles with Unsaturated Side Chains Synthesis
Polymerization and Photocrosslinking M Al-Smadi N Hanold H Kalbitz H Meier
2547 Synthesis of 1112-Didehydrodibenzo[ae]cycloocten-5(6H)-one A Strained Eight-Membered Alkyne S C Kornmayer F Rominger R Gleiter
2553 Stannous Chloride Dihydrate A Novel and Efficient Catalyst for the Synthesis of gem-Dihydroperoxides from Ketones and Aldehydes D Azarifar K Khosravi F Soleimanei
2557 Synthesis of a Novel Class of Azacrown Macrocycles and Lariat Crown Ethers Containing Two 124-Triazole Rings as Subunits N Foroughifar A Mobinikhaledi S Ebrahimi
2561 Enantioselective Synthesis of the 3C-Protease Inhibitor (ndash)-Thysanone by a StauntonndashWeinreb Annulation Strategy J Sperry T Y Yuen M A Brimble
2570 Stereoselective Synthesis of Unnatural β-Amino Acids from Nitroethane via 56-Dihydro-4H-12-oxazin-3-ylacetates A Yu Sukhorukov A V Lesiv O L Eliseev Y A Khomutova S L Ioffe
2579 A Versatile Unexpected One-Pot Regioselective Synthesis of a New Class of 13-Diazepinoindolones by Reaction of Pyranoindolones with Monosubstituted Ureas D Livadiotou C A Tsoleridis J Stephanidou-Stephanatou
2584 Synthesis of a Trisaccharide and a Tetrasaccharide from the Cell-Wall Lipopolysaccharides of Azospirillum brasilense S17 S Pandey S Ghosh A K Misra
2591 Synthesis of Isoindoline Nitroxides by Electrocyclic Reactions T Kaacutelai J Jekı K Hideg
2596 Glycosylations of Tertiary Alcohols Synthesis of Fully Protected Disaccharides with Sterically Demanding Groups Attached to the Sugar Core A Holkenbrink J B Vicente D B Werz
2605 Copper-Catalyzed [13]-Dipolar Cycloaddition for the Synthesis of Macrocycles Containing Acyclic Aromatic and Steroidal Moieties G V Latyshev M S Baranom A V Kazantsev A D Averin N V Lukashev I P Beletskaya
2616 Aryl Ring Migration Reaction in the Synthesis of 24-Diaryl-4H-31-benzothiazines A V Butin F A Tsiunchik V T Abaev A V Gutnov D A Cheshkov
2627 Hydrogenation of β-N-Substituted and β-NN-Disubstituted Enamino Esters in the Presence of Iridium(I) Catalyst H Hebbache Z Hank C Bruneau J-L Renaud
2634 Stereoselective Olefination Reactions Promoted by Rieke Manganese J M Concelloacuten H Rodriacuteguez-Solla V del Amo P Diacuteaz
2646 Synthesis of Piperidinones through a Radical Cascade E Godineau Y Landais
2650 Asymmetric Organic Synthesis with Enzymes Edited by V Gotor I Alfonso E Garciacutea-Urdiales Reviewed by Steve Collier
XVII Forthcoming Articles
no 16 2651 Synthesis of Spirocyclic Ethers S Rosenberg R Leino 2674 Bimetallic PalladiumndashPlatinum-on-Carbon-Catalyzed HndashD Exchange
Reaction Synergistic Effect on Multiple Deuterium Incorporation T Maegawa N Ito K Oono Y Monguchi H Sajiki
2679 Efficient Copper-Catalyzed Synthesis of 2-Amino-4(3H)-quinazolinone and 2-Aminoquinazoline Derivatives X Huang H Yang H Fu R Qiao Y Zhao
2689 Synthesis and Chemoselective N- and O-Alkylation of Thiadiazolopyrimidine Nucleosides and Uridines A M L Hossion R Islam R K Kandahary T Nagamatsu
2697 Facile and Efficient Synthesis of a New Class of Indole-Substituted Pyridine Derivatives via One-Pot Multicomponent Reactions K Zhao X-P Xu S-L Zhu D-Q Shi Y Zhang S-J Ji
2709 Studies toward a Total Synthesis of Rhizoxin D Stereoselective Preparation of the C11ndashC19 Fragment S Padakanti C K Kumar E Ashok P Das
2715 A Short Synthesis of Enantiomeric Phytoprostanes B1 Type I W Perlikowska M Mikołajczyk
2719 Chemistry of Polyhalogenated Nitrobutadienes Part 7 A Novel Synthetic Access to Chlorinated Nitrile Oxides E Nutz V A Zapolrsquoskii D E Kaufmann
2725 Microwave-Assisted Silver(I)-Mediated Selective O-Alkylation of Aromatic Imidate Systems B K Singh C Cavalluzzo M De Maeyer Z Debyser V S Parmar E Van der Eycken
2729 Iodogen A Novel Reagent for the Oxidation of Urazoles under Heterogeneous Conditions A Khoramabadi A Shiri M A Zolfigol S Mallakpour
2733 An Unprecedented Synthesis of Eight-Membered-Ring Cyclic Thioimidic Esters by a Three-Component Reaction A Alizadeh R Hosseinpour
2737 A Novel Diastereoselective Synthesis of β-Phosphonato Unsaturated Thioimidates A Alizadeh N Zohreh
2741 Synthesis of 21-Benzisoxazoles by Nucleophilic Substitution of Hydrogen in Nitroarenes Activated by the Azole Ring N T Pokhodylo Y O Teslenko V S Matiychuk M D Obushak
2749 A Facile Synthesis of Two Series of Multifunctional Carbon Compounds from αα-Dihalo Ketones Using Allylsamarium Bromide X Liu S Zhang J Di
2756 Stereocontrolled Formation of Protected Aminodeoxyalditols from Simple Carbohydrate Precursors by Debenzylating Cycloetherification Y Jiang Z Fang Q Zheng H Jia J Cheng B Zheng
2761 trans-Stilbene as a Starting Material for the Synthesis of Tamoxifen Based on Palladium-Catalyzed Cross-Coupling Reactions C M Nunes J Limberger S Poersch M Seferin A L Monteiro
2766 Synthesis and Biological Evaluation of 6-Substituted Purinylcarbanucleosides with a Cyclopenta[b]thiophene Pseudosugar P Abeijoacuten J M Blanco O Caamantildeo F Fernaacutendez M D Garciacutea X Garciacutea-Mera J E Rodriacuteguez-Borges J Balzarini E De Clercq
2773 Synthesis and Electrochemical Signature of Novel Norbornyl-ferrocene Hybrids F A Khan S K Upadhyay
2778 A Regioselective TsujindashTrost Pentadienylation of 3-Allyltetronic Acid R Schobert B Barnickel
2785 Copper(I)-Catalyzed CarylndashCalkynyl Bond Formation of Aryl Iodides with Terminal Alkynes K G Thakur G Sekar
2790 Aminolysis of Epoxides Using Iridium Trichloride as an Efficient Catalyst J Agarwal A Duley R Rani R K Peddinti
2797 Preparation of Several Active N-Chloro Compounds from Trichloroisocyanuric Acid A Shiri A Khoramabadi-zad
2802 The First Mineral-Catalyzed One-Pot [3+1+2] Coupling Protocol for Multifunctionalized Fused-Ring Pyrimidines L D S Yadav A Rai
2809 Efficient Synthesis of Tetrahydro-β-carbolin-1-one and Dihydroisoquinolin-1-one Derivatives as Versatile Intermediates K E Judd M F Mahon L Caggiano
2818 A Concise Synthesis of ortho-Iodobenzyl Alcohols via Addition of ortho-Iodophenyl Grignard Reagent to Aldehydes and Ketones J Cvengroš D Stolz A Togni
XIII Forthcoming Articles
no 17 2825 Reactivity of Oxazol-5-(4H)-ones and Their Application toward Natural
Product Synthesis N M Hewlett C D Hupp J J Tepe 2840 Towards the Total Synthesis of 3-Hydroxyvibsanin E B D Schwartz
J R Denton P V Bernhardt H M L Davies C M Williams 2847 Structure Investigations of (ent)-Cladospolide D by De Novo Synthesis and
Kinetic and Thermodynamic Isomerization Y Xing J H Penn G A OrsquoDoherty
2855 New Applications of PhI(OAc)2 in Synthesis Total Synthesis and SAR Development of Potent Antitumor Natural Product PsymberinIrciniastatin A N Shao X Huang A Palani R Aslanian A Buevich J Piwinski R Huryk C Seidel-Dugan
2873 Total Synthesis of Largazole ndash Devolution of a Novel Synthetic Strategy B Wang C J Forsyth
2881 Formal Total Synthesis of Palmerolide A J Jaumlgel M E Maier 2893 Total Synthesis of Bongkrekic Acid via Sequential SuzukindashMiyaura Coupling
Reactions M Kanematsu M Shindo M Yoshida K Shishido 2905 Stereodivergent Approach to Both C28a-syn and C28a-anti Relative
Stereochemical Manifolds in the Lepadin Family via a TiCl4-Promoted G Li L J Carlson I K Sagamanova B W Slafer R P Hsung C Gilardi H M Sklenicka N Sydorenko
2915 Enantioselective Aldol Reaction of Tetrasubstituted Ketene Silyl Acetals with Achiral Aldehydes for the Construction of Asymmetric Tertiary Alcohols An Application for the Divergent Total Syntheses of Buergerinins F and G I Shiina T Iizumi Y-s Yamai Y-i Kawakita K Yokoyama Y-k Yamada
2927 Second-Generation Biomimetic Total Synthesis of Chaetominine A Coste G Karthikeyan F Couty G Evano
2935 Total Synthesis of (+)-Fostriecin and (+)-Phoslactomycin B S Shibahara M Fujino Y Tashiro N Okamoto T Esumi K Takahashi J Ishihara S Hatakeyama
2954 Stereochemical Assignments of the Chlorinated Residues in Victorin C A C Durow C Butts C L Willis
2963 Studies of the Asymmetric Total Synthesis of Clavilactone D by the lsquoLariatrsquo Cyclization Strategy T Yoshimitsu S Nojima M Hashimoto K Tsukamoto T Tanaka
2970 Total Synthesis of the Leucetta-Derived Alkaloid Calcaridine A P B Koswatta R Sivappa H V R Dias C J Lovely
2983 Formal Synthesis of Salinosporamide A Starting from D-Glucose T Momose Y Kaiya J-i Hasegawa T Sato N Chida
2992 Synthesis of Bioactive Natural Products by Asymmetric syn- and anti-Aldol Reactions A K Ghosh Z L Dawson
no 18 3003 Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural
Products B M Trost M K Brennan 3026 One-Pot Synthesis of Furo[34-b]pyridin-5(7H)-ones from 2-
Bromopyridine-3-carboxylic Acid and Carbonyl Compounds K Kobayashi T Kozuki H Konishi
3029 Iodocyclization of N-[2-(Methylthio)phenyl]propiolamides Selective Synthesis of 3-Iodo-15-benzothiazepin-4-ones T-S Jiang X-G Zhang J-H Li
3039 A Facile Synthetic Method for Fluorine-Containing 17-Phenanthrolines Pyridine-Ring Formation Reaction of N-Propargyl-68-bis(trifluoroacetyl)-quinolin-5-amine with Various Nucleophiles D Shibata E Okada M Hinoshita M Meacutedebielle
3047 Enantiotopic Discrimination in Palladium-Mediated Nucleophilic Substitutions on Achiral Substrates Chiral Ligand versus Chiral Nucleophile O Jacquet F Charnay J-C Fiaud J Ollivier
3051 Studies on the Chemistry of 2-[3-(2-Nitrophenyl)-2-oxopropyl]benzaldehydes Novel Syntheses of 5H-Benzo[b]carbazole-611-diones and Indolo[12-b]isoquinoline-611-diones M Fernaacutendez
3061 Studies on the C22ndashC23 Aldol Coupling of Spirangien M Lorenz N Bluhm M Kalesse
3067 One-Pot Synthesis of N-Alkyl Purine Pyrimidine and Azole Derivatives from Alcohols using Ph3PCCl4 A Rapid Route to Carboacyclic Nucleoside Synthesis M N Soltani Rad A Khalafi-Nezhad S Behrouz Z Asrari M Behrouz Z Amini
3077 Synthesis of 2-Amino-34-dihydroquinazolines and Imidazo[21-b]quinazoline-2-ones A Mishra S Batra
3089 Studies on the Reaction of Diimines with Thiourea Synthesis and Solvent-Induced cistrans-Isomerization of 135-Triazinane-2-thiones B Kaboudin T Ghasemi T Yokomatsu
3094 Suzuki Coupling of Heteroaromatic Chlorides Using Highly Electron-Donating ClickPhos Ligands S M Spinella Z-H Guan J Chen X Zhang
3099 Reaction of NN-Dioxyenamines with Anhydrides of Carboxylic and Sulfonic Acids A New Method for the Synthesis of a-Hydroxyoxime Derivatives A A Tabolin A V Lesiv S L Ioffe
3106 Directed ortho Metallation Chemistry and Phosphine Synthesis New Ligands for the SuzukindashMiyaura Reaction D B G Williams S J Evans H de Bod M S Mokhadinyana T Hughes
3113 New Functional Derivatives of 9-Phenylquinine P J Boratyński J SkarŜewski
3120 On the Synthesis of Asymmetric and Dissymmetric Amino Analogues of Troumlgerrsquos Base J Artacho K Waumlrnmark
3127 Synthesis of Polycyclic Sultams by Palladium-Catalyzed Intramolecular Cyclization K C Majumdar S Mondal N De
3136 Synthesis of Functionalized L-Cysteine and L-Methionine by Reaction with Electron-Deficient Acetylenes B A Trofimov A G Malrsquokina O A Shemyakina V V Nosyreva A P Borisova S S Khutsishvili L B Krivdin
3143 A lsquoClickrsquo Approach to the Synthesis of 3-[2-(1-Alkyltriazol-4-yl)ethyl]indoles M Petrini R R Shaikh
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
1886 Application of Phenolate Ion Mediated Intramolecular Epoxide Ring Opening in the Enantioselective Synthesis of Functionalized 23-Dihydrobenzofurans and 1-Benzopyrans S K Dinda S K Das G Panda
1897 Complementary Synthetic Approaches to Constitutionally Diverse N-Aminoalkylated Isoindolinones Application to the Synthesis of Falipamil and 5-HT1A Receptor Ligand Analogues M Lorion A Couture E Deniau P Grandclaudon
1904 Selective Deprotection of Silyl Ethers with Sodium Periodate J Li D Menche
1909 Micellar Solution of Sodium Dodecyl Sulfate (SDS) Catalyzes KabacknikndashFields Reaction in Aqueous Media S Sobhani A Vafaee
1916 Convenient Methods for the Synthesis of a Library of Hemilabile Phosphines M V Jimeacutenez J J Peacuterez-Torrente M I Bartolomeacute L A Oro
1923 Terminal Aziridines by Addition of Grignard Reagents or Organoceriums to an (α-Chloro)sulfinylimine D M Hodgson J Kloesges B Evans
1933 A Robust Synthesis of Nε-(Carboxymethyl)-L-lysine (CML) R Csuk S Stark A Barthel R Kluge D Stroumlhl
1935 One-Pot Curtius Rearrangement Processes from Carboxylic Acids O Leogane H Lebel
XV Forthcoming Articles
no 12 1941 The Chemistry of Deprotonated α-Aminonitriles T Opatz 1960 An Efficient Synthesis of Tetraalkyl 2345-Thiophenetetracarboxylate
Derivatives A Alizadeh R Hosseinpour 1963 Facile Deprotection of Bulky (Trialkylsilyl)acetylenes with Silver Fluoride
S Kim B Kim J In 1969 Highly Efficient and Reusable Ionic Liquids for the Catalyzed
Hydroamination of Alkenes with Sulfonamides Carbamates and Carboxamides L Yang L-W Xu C-G Xia
1975 Synthesis of 2391016172324-Octasubstituted Phthalocyaninatozinc(II) Complexes Mediated by Reductive Agents G A Gauna A C Monsalvo J Awruch
1979 A Short and Efficient Synthesis of 3-2-[2-(Bromomethyl)thiazol-4-yl]-ethynyl-5-fluorobenzonitrile A Precursor for PET Radioligand [18F]SP203 M B Gopinathan C Jin K S Rehder
1983 Synthesis of a Substituted Benzazepin-2-one Dihydrate S K Boini R K Vaid K P Moder D Mitchell
1987 Synthesis of Novel Trisubstituted Imidazolines F J Lakner M A Parker B Rogovoy A Khvat A Ivachtchenko
1991 A Novel Synthesis of N-But-3-enyl-α- and β-Amino Acids T T Van Nguyen R T C Brownlee A B Hughes
1999 Synthesis of Substituted 5-(3-Hydroxypropyl)pyrrolidin-2-ones and Pyrrolizidinones from Nitroethane via C3 Functionalized 56-Dihydro-4H-12-oxazines A Novel Approach to Some Analogues of the Antidepressant Rolipram A Yu Sukhorukov A V Lesiv Y A Khomutova S L Ioffe V A Tartakovsky
2009 Chiral Cyclobutanols and Cyclopentane Dimers via Samarium(II) Iodide Induced Keto-Olefin Cyclisations of Carbohydrate-Derived Unsaturated Ketones D B G Williams J Caddy K Blann J J C Groveacute C W Holzapfel
2015 Synthesis of Perfluoroalkylthio-Substituted Ferrocenes C Rhode J Lemke M Lieb N Metzler-Nolte
2019 Functionalization of Polyhedral Oligomeric Silsesquioxane (POSS) via Nucleophilic Substitution M Dutkiewicz H Maciejewski B Marciniec
2025 A Novel Synthesis of Aryl Mesylates via One-Pot DemethylationndashMesylation of Aryl Methyl Ethers Using a Mixture of Phosphorus Pentoxide in Methanesulfonic Acid B Kaboudin Y Abedi
2029 Anionic Cyclization of (NN-Dimethylamino)[2-(prop-2-yn-1-yloxy)aryl]-acetonitriles T Zdrojewski J Musielak A Jończyk
2035 Strecker-Type Reaction Catalyzed by Carboxylic Acids in Aqueous Media Z Xie G Li G Zhao J Wang
2040 Synthesis of Novel Structurally Simplified Estrogen Analogues with Electron-Donating Groups in Ring A L F Tietze C A Vock I K Krimmelbein L Nacke
2061 On the Resolution of Secondary Phosphine Oxides via Diastereomeric Complex Formation The Case of tert-Butylphenylphosphine Oxide J Holt A M Maj E P Schudde K M Pietrusiewicz L Sieroń W Wieczorek T Jerphagnon I W C E Arends U Hanefeld A J Minnaard
2066 Enantioselective Copper-Catalyzed Conjugate Addition of Dimethylzinc to 5-(1-Arylalkylidene) Meldrumrsquos Acids A Wilsily T Lou E Fillion
2073 SuzukindashMiyaura Coupling Reactions Using Phosphite Ligands M Jang Y Jo I-K Oh H M Jung S Lee
2076 Synthesis of 2-Methylindoline- and 2-Methyl-1234-tetrahydroquinoline-Derived Phosphoramidites and Their Applications in Iridium-Catalyzed Allylic Alkylation of Indoles W-B Liu H He L-X Dai S-L You
2083 Stereocontrolled Synthesis of 13-Amino Alcohols by Reduction of Substituted 2-1-[(tert-Butylsulfinyl)amino]alkylcyclohexanones J C Gonzaacutelez-Goacutemez F Foubelo M Yus
2089 Tunable Phosphoramidite Ligands for Asymmetric Hydrovinylation Ligands par excellence for Generation of All-Carbon Quaternary Centers C R Smith H J Lim A ZhangT V RajanBabu
2101 Copper-Catalyzed Asymmetric Ring-Opening Reaction of Oxabenzonorbornadienes with Grignard and Aluminum Reagents R Millet L Gremaud T Bernardez L Palais A Alexakis
2113 A Simplified Synthesis of Takemotorsquos Catalyst A Berkessel B Seelig 2116 Pharmaceutical Substances Syntheses Patents and Applications of the
Most Relevant AIPs Edited by Axel Kleeman Juumlrgen Engel Bernhard Kutscher Dietmar Reichert Reviewed by I Agranat
XV Forthcoming Articles
no 13 2117 Recent Advances in the Aza-Claisen Rearrangement K C Majumdar
T Bhattacharyya B Chattopadhyay B Sinha 2143 A Novel and Convenient Synthesis of lsquoReversedrsquo Diamidino 25-Aryl- and
25-Azaheterocycle-Substituted Furans L Hu D W Boykin 2146 Efficient and General Preparation of Pyranostilbenes First Total Synthesis
of Artocarbene and Pawhuskin B B H Park Y R Lee W S Lyoo 2155 Mild Oxidation of Diarylacetylenes to 12-Diketones Using Oxone in
Trifluoroacetic Acid J-H Chu Y-J Chen M-J Wu 2163 One-Pot Microwave-Assisted Selective Azido ReductionTandem Cyclization
in Condensed and Solid Phase with Nickel Boride N Shankaraiah N Markandeya M Espinoza-Moraga C Arancibia A Kamal L Silva Santos
2171 Pyrrolo[321-ij]quinolin-4-one and Pyrrolo[321-ij]quinolin-6-one H McNab D J Nelson E J Rozgowska
2175 Practical Synthesis of 5-Substituted Tetrazoles under Microwave Irradiation J Roh T V Artamonova K Vaacutevrovaacute G I Koldobskii A Hrabaacutelek
2179 A Simple Method for the Synthesis of 3-Arylthieno[23-b]pyridines via Iodine-Mediated Cyclization of 3-(1-Arylalkenyl)-2-[(1-phenylethyl)sulfanyl]pyridines K Kobayashi D Nakamura Y Shiroyama S Fukamachi H Konishi
2184 Synthesis of Four Lysine-Linked Cereulide Analogues Showing Ionophoric Activity Towards Potassium Cations as Lead Compounds for Emetic Toxin-Detection by Immunoassays A Makarasen T Nishikawa M Isobe
2205 Synthesis of α-Aliphatic and β-Aromatic Substituted Taurines via Regioselective Ring Opening of Thiiranes with Ammonia H Yu S Cao L Zhang G Liu J Xu
2210 Stability of 5(6)-Carboxyfluorescein in Microwave-Assisted Synthesis of Fluorescein-Labelled O-Dimannosylated Peptides R Kowalczyk P W R Harris R P Dunbar M A Brimble
2223 Diversity-Oriented Synthesis of Functionalized Diaryl Sulfones by Regioselective [3+3] Cyclizations of 13-Bis(siloxy)buta-13-dienes with 2-(Arylsulfonyl)-3-ethoxy-2-en-1-ones Scope and Limitations M Shkoor A Riahi O Fatunsin H Reinke C Fischer P Langer
2236 Synthesis of Functionalized Salicylates by Formal [3+3] Cyclocondensation of 13-Bis(silyloxy)buta-13-dienes with 3-Alkoxy-2-en-1-ones G Mroszlig S Ladzik H Reinke A Spannenberg C Fischer P Langer
2249 Synthetic Approach to Alkoxy-β-(trifluoromethyl)styrenes and Their Application in the Synthesis of New Trifluoromethylated Heterocycles V M Muzalevskiy V G Nenajdenko A V Shastin E S Balenkova G Haufe
2260 o-Benzenedisulfonimide as a Powerful and Recyclable Organocatalyst for the Nazarov Reaction M Barbero S Cadamuro A Deagostino S Dughera P Larini E G Occhiato C Prandi S Tabasso R Vulcano P Venturello
2267 The Catalytic Potential of 4-Guanidinylpyridines in Acylation Reactions I Held E Larionov C Bozler F Wagner H Zipse
2278 Iron(III) Chloride in EthanolndashWater Highly Efficient Catalytic System for the Synthesis of Garcia Gonzalez Polyhydroxyalkyl- and C-Glycosylfurans L Nagarapu M V Chary A Satyender B Supriya R Bantu
2283 Ruthenium-Catalyzed Addition of Primary Amides to Alkynes A Stereoselective Synthesis of Secondary Enamides L J Gooszligen M Blanchot K S M Salih K Gooszligen
2289 Binaphthyl-Modified Quaternary Phosphonium Salts as Chiral Phase Transfer Catalysts Application to Asymmetric Amination of β-Keto Esters R He K Maruoka
X Table of Contents XI Forthcoming Articles
no 14 2293 Direct Methods for Stereoselective Polypropionate Synthesis A Survey
J Li D Menche 2316 Synthesis of Symmetrical Ketones from Grignard Reagents and
11-Carbonyldiimidazole D Bottalico V Fiandanese G Marchese A Punzi
2319 Synthesis of 45-Substituted Imidazoles by a Fast Condensation of 12-Diketones and Urotropine in Heterogeneous Medium G Bratulescu
2321 (Arylsulfonyl)acetones and -acetonitriles New Activated Methylenic Building Blocks for Synthesis of 123-Triazoles N T Pokhodylo V S Matiychuk M D Obushak
2324 A Safe Convenient and Efficient One-Pot Synthesis of α-Chloroketone Acetals Directly from Ketones Using Iodobenzene Dichloride J Yu C Zhang
2329 An Efficient Oxidative Conversion of Aldehydes into 2-Substituted 2-Oxazolines Using 13-Diiodo-55-dimethylhydantoin S Takahashi H Togo
2333 A Novel Procedure for the Synthesis of Benzo[b][18]naphthyridine-3-carboxylate Derivatives from MoritandashBaylisndashHillman Adduct Acetates W Zhong F Lin R Chen W Su
2341 An Improved Synthesis of 147-Triazacyclononanes (tacns) and 14710-Tetraazacyclododecanes (cyclens) J Huang Z Zhou T H Chan
2345 The Ullmann Coupling between 2-Chlorobenzoic Acids and Amino Acids A Valuable Reaction for Preparing 2-Substituted 1-Acetyl-1H-indol-3-yl Acetates J C Rodriguez Dominguez X Gang G Kirsch
2349 gem-Dibromomethyl Aromatics Efficient Aldehyde Equivalents in the KnoevenagelndashDoebner Reaction J K Augustine Y A Naik S Poojari N Chowdappa B S Sherigara K Areppa
2357 Synthesis of Novel α-Aminophosphonates Containing Adamantyl Fragment M M Kabachnik L I Minaeva I P Beletskaya
2361 Efficient Fluoride-Mediated Synthesis of 5-Amino-Substituted Isothiazoles Y S Zubenko V I Potkin
2365 Phosphine-Catalyzed Reaction of Cyanohydrins with Activated Alkynes A Siby O Loreau F Taran
2371 Sulfanyl-Substituted [3]Cumulenes and Buta-13-dienes from a Tetrakis(pyridinium)-Substituted Butadiene A Schmidt A Rahimi M Gjikaj
2379 Efficient Synthesis of 2-Substituted Pyrido[32-d]pyrimidines Involving SNAr and Palladium-Catalyzed Cross-Coupling Reactions A Tikad S Routier M Akssira J-M Leacuteger C Jarry G Guillaumet
2385 Novel Synthesis of Medium-Sized Heterocycles by Palladium-Catalyzed Intramolecular Heck Reaction via 9-endo-trig Mode of Cyclization K C Majumdar B Chattopadhyay
2393 Facile Synthesis of Fluorinated Benzofuro- and Benzothieno[23-b]pyridines α-Carbolines and Nucleosides Containing the α-Carboline Framework V O Iaroshenko Y Wang B Zhang D Volochnyuk V Ya Sosnovskikh
2403 Synthesis of Functionalized N-Vinyl Nitrogen-Containing Heterocycles S M M Lopes A M Beja M Ramos Silva J A Paixatildeo F Palacios T M V D Pinho e Melo
2408 Kumada Cross-Coupling of Aryl Grignard Reagents with Aryl Halides Catalyzed by an Immobilized Nickel Catalyst X Chen L Wang J Liu
2413 Highly Enantioselective Synthesis of Heteroaromatic Alcohols Catalyzed by Chiral DiaminodiphosphinendashRuthenium(II) Complexes W-Y Shen Y-Y Li Z-R Dong J-X Gao
2418 Concise Total Synthesis of (+)-Disparlure and its trans-Isomer Using Asymmetric Organocatalysis S-G Kim
2423 Rhodium Carbenoid Induced [12]-Migration in an L-Lyxo-Configured α-Diazo β-Keto Ester Synthesis of a New Griseolic Acid Analogue N N Bhujbal K S A Kumar D D Dhavale
2430 Synthesis of 5-Arylthio-3-hydroxyphthalates by the First [4+2] Cycloadditions of 3-Arylthio-1-silyloxy-13-butadienes with Dimethyl Acetylenedicarboxylate I Iqbal M Imran P Langer
2435 Synthesis of Highly Functionalized Proline Derivatives via a One-Pot MichaelSN-AdditionCyclization Approach U Kazmaier C Schmidt
2440 RhodiumGraphite-Catalyzed Hydrogenation of Carbocyclic and Heterocyclic Aromatic Compounds G Falini A Gualandi D Savoia
2447 Potassium [1-(tert-Butoxycarbonyl)-1H-indol-2-yl]trifluoroborate as an Efficient Building Block in Palladium-Catalyzed SuzukindashMiyaura Cross Couplings P Kassis V Beacuteneacuteteau J-Y Meacuterour S Routier
2454 Syntheses of Substituted Furans and Pyrroles by Platinum-Catalyzed Cyclizations of Propargylic Oxiranes and Aziridines in Aqueous Media M Yoshida M Al-Amin K Shishido
2467 Transition-Metal-Free Oxidative Homocoupling of Aryl Alkenyl and Alkynyl Grignard Reagents with TEMPO M S Maji A Studer
XIII Forthcoming Articles
no 15 2471 Advances in Synthetic Approaches for the Preparation of Combretastatin-
Based Anti-Cancer Agents R Singh H Kaur 2492 Synthesis of Unsymmetrical Ureas by Sulfur-Assisted Carbonylation with
Carbon Monoxide and Oxidation with Molecular Oxygen under Mild Conditions T Mizuno T Nakai M Mihara
2497 Ring-OpeningRecyclization Reactions of (Dimethylamino)propenoyl-Substituted Cyclopropanes Facile Synthesis of Halogenated Pyridin-2(1H)-ones R Zhang Y Zhou Y Liang Z Jiang D Dong
2501 Facile and Efficient Total Synthesis of Taspine B Cheng S Zhang L Zhu J Zhang Q Li A Shan L He
2505 Oligomeric Iodosylbenzene Sulfate A Convenient Hypervalent Iodine Reagent for Oxidation of Organic Sulfides and Alkenes M S Yusubov R Y Yusubova T V Funk K-W Chi V V Zhdankin
2509 Pyrrolidine-Based Organocatalysts for Enantioselective Michael Addition of Cyclohexanone to trans-β-Nitrostyrene A P Carley S Dixon J D Kilburn
2517 CundashAl Hydrotalcite An Efficient and Reusable Ligand-Free Catalyst for the Coupling of Aryl Chlorides with Aliphatic Aromatic and N(H)-Heterocyclic Amines B Sreedhar R Arundhathi P L Reddy M A Reddy M L Kantam
2523 Highly Efficient Synthesis of trans-βγ-Unsaturated a-Keto Amides C Allais T Constantieux J Rodriguez
2531 Gas-Phase Synthesis of N-Unsubstituted 3-Hydroxypyrroles and 1H-Pyrrol-3(2H)-ones L Hill G A Hunter S H Imam H McNab W J OrsquoNeill
2535 3-Hydroxy-1H-pyrrole L Hill S H Imam H McNab W J OrsquoNeill 2539 123-Thiadiazoles with Unsaturated Side Chains Synthesis
Polymerization and Photocrosslinking M Al-Smadi N Hanold H Kalbitz H Meier
2547 Synthesis of 1112-Didehydrodibenzo[ae]cycloocten-5(6H)-one A Strained Eight-Membered Alkyne S C Kornmayer F Rominger R Gleiter
2553 Stannous Chloride Dihydrate A Novel and Efficient Catalyst for the Synthesis of gem-Dihydroperoxides from Ketones and Aldehydes D Azarifar K Khosravi F Soleimanei
2557 Synthesis of a Novel Class of Azacrown Macrocycles and Lariat Crown Ethers Containing Two 124-Triazole Rings as Subunits N Foroughifar A Mobinikhaledi S Ebrahimi
2561 Enantioselective Synthesis of the 3C-Protease Inhibitor (ndash)-Thysanone by a StauntonndashWeinreb Annulation Strategy J Sperry T Y Yuen M A Brimble
2570 Stereoselective Synthesis of Unnatural β-Amino Acids from Nitroethane via 56-Dihydro-4H-12-oxazin-3-ylacetates A Yu Sukhorukov A V Lesiv O L Eliseev Y A Khomutova S L Ioffe
2579 A Versatile Unexpected One-Pot Regioselective Synthesis of a New Class of 13-Diazepinoindolones by Reaction of Pyranoindolones with Monosubstituted Ureas D Livadiotou C A Tsoleridis J Stephanidou-Stephanatou
2584 Synthesis of a Trisaccharide and a Tetrasaccharide from the Cell-Wall Lipopolysaccharides of Azospirillum brasilense S17 S Pandey S Ghosh A K Misra
2591 Synthesis of Isoindoline Nitroxides by Electrocyclic Reactions T Kaacutelai J Jekı K Hideg
2596 Glycosylations of Tertiary Alcohols Synthesis of Fully Protected Disaccharides with Sterically Demanding Groups Attached to the Sugar Core A Holkenbrink J B Vicente D B Werz
2605 Copper-Catalyzed [13]-Dipolar Cycloaddition for the Synthesis of Macrocycles Containing Acyclic Aromatic and Steroidal Moieties G V Latyshev M S Baranom A V Kazantsev A D Averin N V Lukashev I P Beletskaya
2616 Aryl Ring Migration Reaction in the Synthesis of 24-Diaryl-4H-31-benzothiazines A V Butin F A Tsiunchik V T Abaev A V Gutnov D A Cheshkov
2627 Hydrogenation of β-N-Substituted and β-NN-Disubstituted Enamino Esters in the Presence of Iridium(I) Catalyst H Hebbache Z Hank C Bruneau J-L Renaud
2634 Stereoselective Olefination Reactions Promoted by Rieke Manganese J M Concelloacuten H Rodriacuteguez-Solla V del Amo P Diacuteaz
2646 Synthesis of Piperidinones through a Radical Cascade E Godineau Y Landais
2650 Asymmetric Organic Synthesis with Enzymes Edited by V Gotor I Alfonso E Garciacutea-Urdiales Reviewed by Steve Collier
XVII Forthcoming Articles
no 16 2651 Synthesis of Spirocyclic Ethers S Rosenberg R Leino 2674 Bimetallic PalladiumndashPlatinum-on-Carbon-Catalyzed HndashD Exchange
Reaction Synergistic Effect on Multiple Deuterium Incorporation T Maegawa N Ito K Oono Y Monguchi H Sajiki
2679 Efficient Copper-Catalyzed Synthesis of 2-Amino-4(3H)-quinazolinone and 2-Aminoquinazoline Derivatives X Huang H Yang H Fu R Qiao Y Zhao
2689 Synthesis and Chemoselective N- and O-Alkylation of Thiadiazolopyrimidine Nucleosides and Uridines A M L Hossion R Islam R K Kandahary T Nagamatsu
2697 Facile and Efficient Synthesis of a New Class of Indole-Substituted Pyridine Derivatives via One-Pot Multicomponent Reactions K Zhao X-P Xu S-L Zhu D-Q Shi Y Zhang S-J Ji
2709 Studies toward a Total Synthesis of Rhizoxin D Stereoselective Preparation of the C11ndashC19 Fragment S Padakanti C K Kumar E Ashok P Das
2715 A Short Synthesis of Enantiomeric Phytoprostanes B1 Type I W Perlikowska M Mikołajczyk
2719 Chemistry of Polyhalogenated Nitrobutadienes Part 7 A Novel Synthetic Access to Chlorinated Nitrile Oxides E Nutz V A Zapolrsquoskii D E Kaufmann
2725 Microwave-Assisted Silver(I)-Mediated Selective O-Alkylation of Aromatic Imidate Systems B K Singh C Cavalluzzo M De Maeyer Z Debyser V S Parmar E Van der Eycken
2729 Iodogen A Novel Reagent for the Oxidation of Urazoles under Heterogeneous Conditions A Khoramabadi A Shiri M A Zolfigol S Mallakpour
2733 An Unprecedented Synthesis of Eight-Membered-Ring Cyclic Thioimidic Esters by a Three-Component Reaction A Alizadeh R Hosseinpour
2737 A Novel Diastereoselective Synthesis of β-Phosphonato Unsaturated Thioimidates A Alizadeh N Zohreh
2741 Synthesis of 21-Benzisoxazoles by Nucleophilic Substitution of Hydrogen in Nitroarenes Activated by the Azole Ring N T Pokhodylo Y O Teslenko V S Matiychuk M D Obushak
2749 A Facile Synthesis of Two Series of Multifunctional Carbon Compounds from αα-Dihalo Ketones Using Allylsamarium Bromide X Liu S Zhang J Di
2756 Stereocontrolled Formation of Protected Aminodeoxyalditols from Simple Carbohydrate Precursors by Debenzylating Cycloetherification Y Jiang Z Fang Q Zheng H Jia J Cheng B Zheng
2761 trans-Stilbene as a Starting Material for the Synthesis of Tamoxifen Based on Palladium-Catalyzed Cross-Coupling Reactions C M Nunes J Limberger S Poersch M Seferin A L Monteiro
2766 Synthesis and Biological Evaluation of 6-Substituted Purinylcarbanucleosides with a Cyclopenta[b]thiophene Pseudosugar P Abeijoacuten J M Blanco O Caamantildeo F Fernaacutendez M D Garciacutea X Garciacutea-Mera J E Rodriacuteguez-Borges J Balzarini E De Clercq
2773 Synthesis and Electrochemical Signature of Novel Norbornyl-ferrocene Hybrids F A Khan S K Upadhyay
2778 A Regioselective TsujindashTrost Pentadienylation of 3-Allyltetronic Acid R Schobert B Barnickel
2785 Copper(I)-Catalyzed CarylndashCalkynyl Bond Formation of Aryl Iodides with Terminal Alkynes K G Thakur G Sekar
2790 Aminolysis of Epoxides Using Iridium Trichloride as an Efficient Catalyst J Agarwal A Duley R Rani R K Peddinti
2797 Preparation of Several Active N-Chloro Compounds from Trichloroisocyanuric Acid A Shiri A Khoramabadi-zad
2802 The First Mineral-Catalyzed One-Pot [3+1+2] Coupling Protocol for Multifunctionalized Fused-Ring Pyrimidines L D S Yadav A Rai
2809 Efficient Synthesis of Tetrahydro-β-carbolin-1-one and Dihydroisoquinolin-1-one Derivatives as Versatile Intermediates K E Judd M F Mahon L Caggiano
2818 A Concise Synthesis of ortho-Iodobenzyl Alcohols via Addition of ortho-Iodophenyl Grignard Reagent to Aldehydes and Ketones J Cvengroš D Stolz A Togni
XIII Forthcoming Articles
no 17 2825 Reactivity of Oxazol-5-(4H)-ones and Their Application toward Natural
Product Synthesis N M Hewlett C D Hupp J J Tepe 2840 Towards the Total Synthesis of 3-Hydroxyvibsanin E B D Schwartz
J R Denton P V Bernhardt H M L Davies C M Williams 2847 Structure Investigations of (ent)-Cladospolide D by De Novo Synthesis and
Kinetic and Thermodynamic Isomerization Y Xing J H Penn G A OrsquoDoherty
2855 New Applications of PhI(OAc)2 in Synthesis Total Synthesis and SAR Development of Potent Antitumor Natural Product PsymberinIrciniastatin A N Shao X Huang A Palani R Aslanian A Buevich J Piwinski R Huryk C Seidel-Dugan
2873 Total Synthesis of Largazole ndash Devolution of a Novel Synthetic Strategy B Wang C J Forsyth
2881 Formal Total Synthesis of Palmerolide A J Jaumlgel M E Maier 2893 Total Synthesis of Bongkrekic Acid via Sequential SuzukindashMiyaura Coupling
Reactions M Kanematsu M Shindo M Yoshida K Shishido 2905 Stereodivergent Approach to Both C28a-syn and C28a-anti Relative
Stereochemical Manifolds in the Lepadin Family via a TiCl4-Promoted G Li L J Carlson I K Sagamanova B W Slafer R P Hsung C Gilardi H M Sklenicka N Sydorenko
2915 Enantioselective Aldol Reaction of Tetrasubstituted Ketene Silyl Acetals with Achiral Aldehydes for the Construction of Asymmetric Tertiary Alcohols An Application for the Divergent Total Syntheses of Buergerinins F and G I Shiina T Iizumi Y-s Yamai Y-i Kawakita K Yokoyama Y-k Yamada
2927 Second-Generation Biomimetic Total Synthesis of Chaetominine A Coste G Karthikeyan F Couty G Evano
2935 Total Synthesis of (+)-Fostriecin and (+)-Phoslactomycin B S Shibahara M Fujino Y Tashiro N Okamoto T Esumi K Takahashi J Ishihara S Hatakeyama
2954 Stereochemical Assignments of the Chlorinated Residues in Victorin C A C Durow C Butts C L Willis
2963 Studies of the Asymmetric Total Synthesis of Clavilactone D by the lsquoLariatrsquo Cyclization Strategy T Yoshimitsu S Nojima M Hashimoto K Tsukamoto T Tanaka
2970 Total Synthesis of the Leucetta-Derived Alkaloid Calcaridine A P B Koswatta R Sivappa H V R Dias C J Lovely
2983 Formal Synthesis of Salinosporamide A Starting from D-Glucose T Momose Y Kaiya J-i Hasegawa T Sato N Chida
2992 Synthesis of Bioactive Natural Products by Asymmetric syn- and anti-Aldol Reactions A K Ghosh Z L Dawson
no 18 3003 Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural
Products B M Trost M K Brennan 3026 One-Pot Synthesis of Furo[34-b]pyridin-5(7H)-ones from 2-
Bromopyridine-3-carboxylic Acid and Carbonyl Compounds K Kobayashi T Kozuki H Konishi
3029 Iodocyclization of N-[2-(Methylthio)phenyl]propiolamides Selective Synthesis of 3-Iodo-15-benzothiazepin-4-ones T-S Jiang X-G Zhang J-H Li
3039 A Facile Synthetic Method for Fluorine-Containing 17-Phenanthrolines Pyridine-Ring Formation Reaction of N-Propargyl-68-bis(trifluoroacetyl)-quinolin-5-amine with Various Nucleophiles D Shibata E Okada M Hinoshita M Meacutedebielle
3047 Enantiotopic Discrimination in Palladium-Mediated Nucleophilic Substitutions on Achiral Substrates Chiral Ligand versus Chiral Nucleophile O Jacquet F Charnay J-C Fiaud J Ollivier
3051 Studies on the Chemistry of 2-[3-(2-Nitrophenyl)-2-oxopropyl]benzaldehydes Novel Syntheses of 5H-Benzo[b]carbazole-611-diones and Indolo[12-b]isoquinoline-611-diones M Fernaacutendez
3061 Studies on the C22ndashC23 Aldol Coupling of Spirangien M Lorenz N Bluhm M Kalesse
3067 One-Pot Synthesis of N-Alkyl Purine Pyrimidine and Azole Derivatives from Alcohols using Ph3PCCl4 A Rapid Route to Carboacyclic Nucleoside Synthesis M N Soltani Rad A Khalafi-Nezhad S Behrouz Z Asrari M Behrouz Z Amini
3077 Synthesis of 2-Amino-34-dihydroquinazolines and Imidazo[21-b]quinazoline-2-ones A Mishra S Batra
3089 Studies on the Reaction of Diimines with Thiourea Synthesis and Solvent-Induced cistrans-Isomerization of 135-Triazinane-2-thiones B Kaboudin T Ghasemi T Yokomatsu
3094 Suzuki Coupling of Heteroaromatic Chlorides Using Highly Electron-Donating ClickPhos Ligands S M Spinella Z-H Guan J Chen X Zhang
3099 Reaction of NN-Dioxyenamines with Anhydrides of Carboxylic and Sulfonic Acids A New Method for the Synthesis of a-Hydroxyoxime Derivatives A A Tabolin A V Lesiv S L Ioffe
3106 Directed ortho Metallation Chemistry and Phosphine Synthesis New Ligands for the SuzukindashMiyaura Reaction D B G Williams S J Evans H de Bod M S Mokhadinyana T Hughes
3113 New Functional Derivatives of 9-Phenylquinine P J Boratyński J SkarŜewski
3120 On the Synthesis of Asymmetric and Dissymmetric Amino Analogues of Troumlgerrsquos Base J Artacho K Waumlrnmark
3127 Synthesis of Polycyclic Sultams by Palladium-Catalyzed Intramolecular Cyclization K C Majumdar S Mondal N De
3136 Synthesis of Functionalized L-Cysteine and L-Methionine by Reaction with Electron-Deficient Acetylenes B A Trofimov A G Malrsquokina O A Shemyakina V V Nosyreva A P Borisova S S Khutsishvili L B Krivdin
3143 A lsquoClickrsquo Approach to the Synthesis of 3-[2-(1-Alkyltriazol-4-yl)ethyl]indoles M Petrini R R Shaikh
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
no 12 1941 The Chemistry of Deprotonated α-Aminonitriles T Opatz 1960 An Efficient Synthesis of Tetraalkyl 2345-Thiophenetetracarboxylate
Derivatives A Alizadeh R Hosseinpour 1963 Facile Deprotection of Bulky (Trialkylsilyl)acetylenes with Silver Fluoride
S Kim B Kim J In 1969 Highly Efficient and Reusable Ionic Liquids for the Catalyzed
Hydroamination of Alkenes with Sulfonamides Carbamates and Carboxamides L Yang L-W Xu C-G Xia
1975 Synthesis of 2391016172324-Octasubstituted Phthalocyaninatozinc(II) Complexes Mediated by Reductive Agents G A Gauna A C Monsalvo J Awruch
1979 A Short and Efficient Synthesis of 3-2-[2-(Bromomethyl)thiazol-4-yl]-ethynyl-5-fluorobenzonitrile A Precursor for PET Radioligand [18F]SP203 M B Gopinathan C Jin K S Rehder
1983 Synthesis of a Substituted Benzazepin-2-one Dihydrate S K Boini R K Vaid K P Moder D Mitchell
1987 Synthesis of Novel Trisubstituted Imidazolines F J Lakner M A Parker B Rogovoy A Khvat A Ivachtchenko
1991 A Novel Synthesis of N-But-3-enyl-α- and β-Amino Acids T T Van Nguyen R T C Brownlee A B Hughes
1999 Synthesis of Substituted 5-(3-Hydroxypropyl)pyrrolidin-2-ones and Pyrrolizidinones from Nitroethane via C3 Functionalized 56-Dihydro-4H-12-oxazines A Novel Approach to Some Analogues of the Antidepressant Rolipram A Yu Sukhorukov A V Lesiv Y A Khomutova S L Ioffe V A Tartakovsky
2009 Chiral Cyclobutanols and Cyclopentane Dimers via Samarium(II) Iodide Induced Keto-Olefin Cyclisations of Carbohydrate-Derived Unsaturated Ketones D B G Williams J Caddy K Blann J J C Groveacute C W Holzapfel
2015 Synthesis of Perfluoroalkylthio-Substituted Ferrocenes C Rhode J Lemke M Lieb N Metzler-Nolte
2019 Functionalization of Polyhedral Oligomeric Silsesquioxane (POSS) via Nucleophilic Substitution M Dutkiewicz H Maciejewski B Marciniec
2025 A Novel Synthesis of Aryl Mesylates via One-Pot DemethylationndashMesylation of Aryl Methyl Ethers Using a Mixture of Phosphorus Pentoxide in Methanesulfonic Acid B Kaboudin Y Abedi
2029 Anionic Cyclization of (NN-Dimethylamino)[2-(prop-2-yn-1-yloxy)aryl]-acetonitriles T Zdrojewski J Musielak A Jończyk
2035 Strecker-Type Reaction Catalyzed by Carboxylic Acids in Aqueous Media Z Xie G Li G Zhao J Wang
2040 Synthesis of Novel Structurally Simplified Estrogen Analogues with Electron-Donating Groups in Ring A L F Tietze C A Vock I K Krimmelbein L Nacke
2061 On the Resolution of Secondary Phosphine Oxides via Diastereomeric Complex Formation The Case of tert-Butylphenylphosphine Oxide J Holt A M Maj E P Schudde K M Pietrusiewicz L Sieroń W Wieczorek T Jerphagnon I W C E Arends U Hanefeld A J Minnaard
2066 Enantioselective Copper-Catalyzed Conjugate Addition of Dimethylzinc to 5-(1-Arylalkylidene) Meldrumrsquos Acids A Wilsily T Lou E Fillion
2073 SuzukindashMiyaura Coupling Reactions Using Phosphite Ligands M Jang Y Jo I-K Oh H M Jung S Lee
2076 Synthesis of 2-Methylindoline- and 2-Methyl-1234-tetrahydroquinoline-Derived Phosphoramidites and Their Applications in Iridium-Catalyzed Allylic Alkylation of Indoles W-B Liu H He L-X Dai S-L You
2083 Stereocontrolled Synthesis of 13-Amino Alcohols by Reduction of Substituted 2-1-[(tert-Butylsulfinyl)amino]alkylcyclohexanones J C Gonzaacutelez-Goacutemez F Foubelo M Yus
2089 Tunable Phosphoramidite Ligands for Asymmetric Hydrovinylation Ligands par excellence for Generation of All-Carbon Quaternary Centers C R Smith H J Lim A ZhangT V RajanBabu
2101 Copper-Catalyzed Asymmetric Ring-Opening Reaction of Oxabenzonorbornadienes with Grignard and Aluminum Reagents R Millet L Gremaud T Bernardez L Palais A Alexakis
2113 A Simplified Synthesis of Takemotorsquos Catalyst A Berkessel B Seelig 2116 Pharmaceutical Substances Syntheses Patents and Applications of the
Most Relevant AIPs Edited by Axel Kleeman Juumlrgen Engel Bernhard Kutscher Dietmar Reichert Reviewed by I Agranat
XV Forthcoming Articles
no 13 2117 Recent Advances in the Aza-Claisen Rearrangement K C Majumdar
T Bhattacharyya B Chattopadhyay B Sinha 2143 A Novel and Convenient Synthesis of lsquoReversedrsquo Diamidino 25-Aryl- and
25-Azaheterocycle-Substituted Furans L Hu D W Boykin 2146 Efficient and General Preparation of Pyranostilbenes First Total Synthesis
of Artocarbene and Pawhuskin B B H Park Y R Lee W S Lyoo 2155 Mild Oxidation of Diarylacetylenes to 12-Diketones Using Oxone in
Trifluoroacetic Acid J-H Chu Y-J Chen M-J Wu 2163 One-Pot Microwave-Assisted Selective Azido ReductionTandem Cyclization
in Condensed and Solid Phase with Nickel Boride N Shankaraiah N Markandeya M Espinoza-Moraga C Arancibia A Kamal L Silva Santos
2171 Pyrrolo[321-ij]quinolin-4-one and Pyrrolo[321-ij]quinolin-6-one H McNab D J Nelson E J Rozgowska
2175 Practical Synthesis of 5-Substituted Tetrazoles under Microwave Irradiation J Roh T V Artamonova K Vaacutevrovaacute G I Koldobskii A Hrabaacutelek
2179 A Simple Method for the Synthesis of 3-Arylthieno[23-b]pyridines via Iodine-Mediated Cyclization of 3-(1-Arylalkenyl)-2-[(1-phenylethyl)sulfanyl]pyridines K Kobayashi D Nakamura Y Shiroyama S Fukamachi H Konishi
2184 Synthesis of Four Lysine-Linked Cereulide Analogues Showing Ionophoric Activity Towards Potassium Cations as Lead Compounds for Emetic Toxin-Detection by Immunoassays A Makarasen T Nishikawa M Isobe
2205 Synthesis of α-Aliphatic and β-Aromatic Substituted Taurines via Regioselective Ring Opening of Thiiranes with Ammonia H Yu S Cao L Zhang G Liu J Xu
2210 Stability of 5(6)-Carboxyfluorescein in Microwave-Assisted Synthesis of Fluorescein-Labelled O-Dimannosylated Peptides R Kowalczyk P W R Harris R P Dunbar M A Brimble
2223 Diversity-Oriented Synthesis of Functionalized Diaryl Sulfones by Regioselective [3+3] Cyclizations of 13-Bis(siloxy)buta-13-dienes with 2-(Arylsulfonyl)-3-ethoxy-2-en-1-ones Scope and Limitations M Shkoor A Riahi O Fatunsin H Reinke C Fischer P Langer
2236 Synthesis of Functionalized Salicylates by Formal [3+3] Cyclocondensation of 13-Bis(silyloxy)buta-13-dienes with 3-Alkoxy-2-en-1-ones G Mroszlig S Ladzik H Reinke A Spannenberg C Fischer P Langer
2249 Synthetic Approach to Alkoxy-β-(trifluoromethyl)styrenes and Their Application in the Synthesis of New Trifluoromethylated Heterocycles V M Muzalevskiy V G Nenajdenko A V Shastin E S Balenkova G Haufe
2260 o-Benzenedisulfonimide as a Powerful and Recyclable Organocatalyst for the Nazarov Reaction M Barbero S Cadamuro A Deagostino S Dughera P Larini E G Occhiato C Prandi S Tabasso R Vulcano P Venturello
2267 The Catalytic Potential of 4-Guanidinylpyridines in Acylation Reactions I Held E Larionov C Bozler F Wagner H Zipse
2278 Iron(III) Chloride in EthanolndashWater Highly Efficient Catalytic System for the Synthesis of Garcia Gonzalez Polyhydroxyalkyl- and C-Glycosylfurans L Nagarapu M V Chary A Satyender B Supriya R Bantu
2283 Ruthenium-Catalyzed Addition of Primary Amides to Alkynes A Stereoselective Synthesis of Secondary Enamides L J Gooszligen M Blanchot K S M Salih K Gooszligen
2289 Binaphthyl-Modified Quaternary Phosphonium Salts as Chiral Phase Transfer Catalysts Application to Asymmetric Amination of β-Keto Esters R He K Maruoka
X Table of Contents XI Forthcoming Articles
no 14 2293 Direct Methods for Stereoselective Polypropionate Synthesis A Survey
J Li D Menche 2316 Synthesis of Symmetrical Ketones from Grignard Reagents and
11-Carbonyldiimidazole D Bottalico V Fiandanese G Marchese A Punzi
2319 Synthesis of 45-Substituted Imidazoles by a Fast Condensation of 12-Diketones and Urotropine in Heterogeneous Medium G Bratulescu
2321 (Arylsulfonyl)acetones and -acetonitriles New Activated Methylenic Building Blocks for Synthesis of 123-Triazoles N T Pokhodylo V S Matiychuk M D Obushak
2324 A Safe Convenient and Efficient One-Pot Synthesis of α-Chloroketone Acetals Directly from Ketones Using Iodobenzene Dichloride J Yu C Zhang
2329 An Efficient Oxidative Conversion of Aldehydes into 2-Substituted 2-Oxazolines Using 13-Diiodo-55-dimethylhydantoin S Takahashi H Togo
2333 A Novel Procedure for the Synthesis of Benzo[b][18]naphthyridine-3-carboxylate Derivatives from MoritandashBaylisndashHillman Adduct Acetates W Zhong F Lin R Chen W Su
2341 An Improved Synthesis of 147-Triazacyclononanes (tacns) and 14710-Tetraazacyclododecanes (cyclens) J Huang Z Zhou T H Chan
2345 The Ullmann Coupling between 2-Chlorobenzoic Acids and Amino Acids A Valuable Reaction for Preparing 2-Substituted 1-Acetyl-1H-indol-3-yl Acetates J C Rodriguez Dominguez X Gang G Kirsch
2349 gem-Dibromomethyl Aromatics Efficient Aldehyde Equivalents in the KnoevenagelndashDoebner Reaction J K Augustine Y A Naik S Poojari N Chowdappa B S Sherigara K Areppa
2357 Synthesis of Novel α-Aminophosphonates Containing Adamantyl Fragment M M Kabachnik L I Minaeva I P Beletskaya
2361 Efficient Fluoride-Mediated Synthesis of 5-Amino-Substituted Isothiazoles Y S Zubenko V I Potkin
2365 Phosphine-Catalyzed Reaction of Cyanohydrins with Activated Alkynes A Siby O Loreau F Taran
2371 Sulfanyl-Substituted [3]Cumulenes and Buta-13-dienes from a Tetrakis(pyridinium)-Substituted Butadiene A Schmidt A Rahimi M Gjikaj
2379 Efficient Synthesis of 2-Substituted Pyrido[32-d]pyrimidines Involving SNAr and Palladium-Catalyzed Cross-Coupling Reactions A Tikad S Routier M Akssira J-M Leacuteger C Jarry G Guillaumet
2385 Novel Synthesis of Medium-Sized Heterocycles by Palladium-Catalyzed Intramolecular Heck Reaction via 9-endo-trig Mode of Cyclization K C Majumdar B Chattopadhyay
2393 Facile Synthesis of Fluorinated Benzofuro- and Benzothieno[23-b]pyridines α-Carbolines and Nucleosides Containing the α-Carboline Framework V O Iaroshenko Y Wang B Zhang D Volochnyuk V Ya Sosnovskikh
2403 Synthesis of Functionalized N-Vinyl Nitrogen-Containing Heterocycles S M M Lopes A M Beja M Ramos Silva J A Paixatildeo F Palacios T M V D Pinho e Melo
2408 Kumada Cross-Coupling of Aryl Grignard Reagents with Aryl Halides Catalyzed by an Immobilized Nickel Catalyst X Chen L Wang J Liu
2413 Highly Enantioselective Synthesis of Heteroaromatic Alcohols Catalyzed by Chiral DiaminodiphosphinendashRuthenium(II) Complexes W-Y Shen Y-Y Li Z-R Dong J-X Gao
2418 Concise Total Synthesis of (+)-Disparlure and its trans-Isomer Using Asymmetric Organocatalysis S-G Kim
2423 Rhodium Carbenoid Induced [12]-Migration in an L-Lyxo-Configured α-Diazo β-Keto Ester Synthesis of a New Griseolic Acid Analogue N N Bhujbal K S A Kumar D D Dhavale
2430 Synthesis of 5-Arylthio-3-hydroxyphthalates by the First [4+2] Cycloadditions of 3-Arylthio-1-silyloxy-13-butadienes with Dimethyl Acetylenedicarboxylate I Iqbal M Imran P Langer
2435 Synthesis of Highly Functionalized Proline Derivatives via a One-Pot MichaelSN-AdditionCyclization Approach U Kazmaier C Schmidt
2440 RhodiumGraphite-Catalyzed Hydrogenation of Carbocyclic and Heterocyclic Aromatic Compounds G Falini A Gualandi D Savoia
2447 Potassium [1-(tert-Butoxycarbonyl)-1H-indol-2-yl]trifluoroborate as an Efficient Building Block in Palladium-Catalyzed SuzukindashMiyaura Cross Couplings P Kassis V Beacuteneacuteteau J-Y Meacuterour S Routier
2454 Syntheses of Substituted Furans and Pyrroles by Platinum-Catalyzed Cyclizations of Propargylic Oxiranes and Aziridines in Aqueous Media M Yoshida M Al-Amin K Shishido
2467 Transition-Metal-Free Oxidative Homocoupling of Aryl Alkenyl and Alkynyl Grignard Reagents with TEMPO M S Maji A Studer
XIII Forthcoming Articles
no 15 2471 Advances in Synthetic Approaches for the Preparation of Combretastatin-
Based Anti-Cancer Agents R Singh H Kaur 2492 Synthesis of Unsymmetrical Ureas by Sulfur-Assisted Carbonylation with
Carbon Monoxide and Oxidation with Molecular Oxygen under Mild Conditions T Mizuno T Nakai M Mihara
2497 Ring-OpeningRecyclization Reactions of (Dimethylamino)propenoyl-Substituted Cyclopropanes Facile Synthesis of Halogenated Pyridin-2(1H)-ones R Zhang Y Zhou Y Liang Z Jiang D Dong
2501 Facile and Efficient Total Synthesis of Taspine B Cheng S Zhang L Zhu J Zhang Q Li A Shan L He
2505 Oligomeric Iodosylbenzene Sulfate A Convenient Hypervalent Iodine Reagent for Oxidation of Organic Sulfides and Alkenes M S Yusubov R Y Yusubova T V Funk K-W Chi V V Zhdankin
2509 Pyrrolidine-Based Organocatalysts for Enantioselective Michael Addition of Cyclohexanone to trans-β-Nitrostyrene A P Carley S Dixon J D Kilburn
2517 CundashAl Hydrotalcite An Efficient and Reusable Ligand-Free Catalyst for the Coupling of Aryl Chlorides with Aliphatic Aromatic and N(H)-Heterocyclic Amines B Sreedhar R Arundhathi P L Reddy M A Reddy M L Kantam
2523 Highly Efficient Synthesis of trans-βγ-Unsaturated a-Keto Amides C Allais T Constantieux J Rodriguez
2531 Gas-Phase Synthesis of N-Unsubstituted 3-Hydroxypyrroles and 1H-Pyrrol-3(2H)-ones L Hill G A Hunter S H Imam H McNab W J OrsquoNeill
2535 3-Hydroxy-1H-pyrrole L Hill S H Imam H McNab W J OrsquoNeill 2539 123-Thiadiazoles with Unsaturated Side Chains Synthesis
Polymerization and Photocrosslinking M Al-Smadi N Hanold H Kalbitz H Meier
2547 Synthesis of 1112-Didehydrodibenzo[ae]cycloocten-5(6H)-one A Strained Eight-Membered Alkyne S C Kornmayer F Rominger R Gleiter
2553 Stannous Chloride Dihydrate A Novel and Efficient Catalyst for the Synthesis of gem-Dihydroperoxides from Ketones and Aldehydes D Azarifar K Khosravi F Soleimanei
2557 Synthesis of a Novel Class of Azacrown Macrocycles and Lariat Crown Ethers Containing Two 124-Triazole Rings as Subunits N Foroughifar A Mobinikhaledi S Ebrahimi
2561 Enantioselective Synthesis of the 3C-Protease Inhibitor (ndash)-Thysanone by a StauntonndashWeinreb Annulation Strategy J Sperry T Y Yuen M A Brimble
2570 Stereoselective Synthesis of Unnatural β-Amino Acids from Nitroethane via 56-Dihydro-4H-12-oxazin-3-ylacetates A Yu Sukhorukov A V Lesiv O L Eliseev Y A Khomutova S L Ioffe
2579 A Versatile Unexpected One-Pot Regioselective Synthesis of a New Class of 13-Diazepinoindolones by Reaction of Pyranoindolones with Monosubstituted Ureas D Livadiotou C A Tsoleridis J Stephanidou-Stephanatou
2584 Synthesis of a Trisaccharide and a Tetrasaccharide from the Cell-Wall Lipopolysaccharides of Azospirillum brasilense S17 S Pandey S Ghosh A K Misra
2591 Synthesis of Isoindoline Nitroxides by Electrocyclic Reactions T Kaacutelai J Jekı K Hideg
2596 Glycosylations of Tertiary Alcohols Synthesis of Fully Protected Disaccharides with Sterically Demanding Groups Attached to the Sugar Core A Holkenbrink J B Vicente D B Werz
2605 Copper-Catalyzed [13]-Dipolar Cycloaddition for the Synthesis of Macrocycles Containing Acyclic Aromatic and Steroidal Moieties G V Latyshev M S Baranom A V Kazantsev A D Averin N V Lukashev I P Beletskaya
2616 Aryl Ring Migration Reaction in the Synthesis of 24-Diaryl-4H-31-benzothiazines A V Butin F A Tsiunchik V T Abaev A V Gutnov D A Cheshkov
2627 Hydrogenation of β-N-Substituted and β-NN-Disubstituted Enamino Esters in the Presence of Iridium(I) Catalyst H Hebbache Z Hank C Bruneau J-L Renaud
2634 Stereoselective Olefination Reactions Promoted by Rieke Manganese J M Concelloacuten H Rodriacuteguez-Solla V del Amo P Diacuteaz
2646 Synthesis of Piperidinones through a Radical Cascade E Godineau Y Landais
2650 Asymmetric Organic Synthesis with Enzymes Edited by V Gotor I Alfonso E Garciacutea-Urdiales Reviewed by Steve Collier
XVII Forthcoming Articles
no 16 2651 Synthesis of Spirocyclic Ethers S Rosenberg R Leino 2674 Bimetallic PalladiumndashPlatinum-on-Carbon-Catalyzed HndashD Exchange
Reaction Synergistic Effect on Multiple Deuterium Incorporation T Maegawa N Ito K Oono Y Monguchi H Sajiki
2679 Efficient Copper-Catalyzed Synthesis of 2-Amino-4(3H)-quinazolinone and 2-Aminoquinazoline Derivatives X Huang H Yang H Fu R Qiao Y Zhao
2689 Synthesis and Chemoselective N- and O-Alkylation of Thiadiazolopyrimidine Nucleosides and Uridines A M L Hossion R Islam R K Kandahary T Nagamatsu
2697 Facile and Efficient Synthesis of a New Class of Indole-Substituted Pyridine Derivatives via One-Pot Multicomponent Reactions K Zhao X-P Xu S-L Zhu D-Q Shi Y Zhang S-J Ji
2709 Studies toward a Total Synthesis of Rhizoxin D Stereoselective Preparation of the C11ndashC19 Fragment S Padakanti C K Kumar E Ashok P Das
2715 A Short Synthesis of Enantiomeric Phytoprostanes B1 Type I W Perlikowska M Mikołajczyk
2719 Chemistry of Polyhalogenated Nitrobutadienes Part 7 A Novel Synthetic Access to Chlorinated Nitrile Oxides E Nutz V A Zapolrsquoskii D E Kaufmann
2725 Microwave-Assisted Silver(I)-Mediated Selective O-Alkylation of Aromatic Imidate Systems B K Singh C Cavalluzzo M De Maeyer Z Debyser V S Parmar E Van der Eycken
2729 Iodogen A Novel Reagent for the Oxidation of Urazoles under Heterogeneous Conditions A Khoramabadi A Shiri M A Zolfigol S Mallakpour
2733 An Unprecedented Synthesis of Eight-Membered-Ring Cyclic Thioimidic Esters by a Three-Component Reaction A Alizadeh R Hosseinpour
2737 A Novel Diastereoselective Synthesis of β-Phosphonato Unsaturated Thioimidates A Alizadeh N Zohreh
2741 Synthesis of 21-Benzisoxazoles by Nucleophilic Substitution of Hydrogen in Nitroarenes Activated by the Azole Ring N T Pokhodylo Y O Teslenko V S Matiychuk M D Obushak
2749 A Facile Synthesis of Two Series of Multifunctional Carbon Compounds from αα-Dihalo Ketones Using Allylsamarium Bromide X Liu S Zhang J Di
2756 Stereocontrolled Formation of Protected Aminodeoxyalditols from Simple Carbohydrate Precursors by Debenzylating Cycloetherification Y Jiang Z Fang Q Zheng H Jia J Cheng B Zheng
2761 trans-Stilbene as a Starting Material for the Synthesis of Tamoxifen Based on Palladium-Catalyzed Cross-Coupling Reactions C M Nunes J Limberger S Poersch M Seferin A L Monteiro
2766 Synthesis and Biological Evaluation of 6-Substituted Purinylcarbanucleosides with a Cyclopenta[b]thiophene Pseudosugar P Abeijoacuten J M Blanco O Caamantildeo F Fernaacutendez M D Garciacutea X Garciacutea-Mera J E Rodriacuteguez-Borges J Balzarini E De Clercq
2773 Synthesis and Electrochemical Signature of Novel Norbornyl-ferrocene Hybrids F A Khan S K Upadhyay
2778 A Regioselective TsujindashTrost Pentadienylation of 3-Allyltetronic Acid R Schobert B Barnickel
2785 Copper(I)-Catalyzed CarylndashCalkynyl Bond Formation of Aryl Iodides with Terminal Alkynes K G Thakur G Sekar
2790 Aminolysis of Epoxides Using Iridium Trichloride as an Efficient Catalyst J Agarwal A Duley R Rani R K Peddinti
2797 Preparation of Several Active N-Chloro Compounds from Trichloroisocyanuric Acid A Shiri A Khoramabadi-zad
2802 The First Mineral-Catalyzed One-Pot [3+1+2] Coupling Protocol for Multifunctionalized Fused-Ring Pyrimidines L D S Yadav A Rai
2809 Efficient Synthesis of Tetrahydro-β-carbolin-1-one and Dihydroisoquinolin-1-one Derivatives as Versatile Intermediates K E Judd M F Mahon L Caggiano
2818 A Concise Synthesis of ortho-Iodobenzyl Alcohols via Addition of ortho-Iodophenyl Grignard Reagent to Aldehydes and Ketones J Cvengroš D Stolz A Togni
XIII Forthcoming Articles
no 17 2825 Reactivity of Oxazol-5-(4H)-ones and Their Application toward Natural
Product Synthesis N M Hewlett C D Hupp J J Tepe 2840 Towards the Total Synthesis of 3-Hydroxyvibsanin E B D Schwartz
J R Denton P V Bernhardt H M L Davies C M Williams 2847 Structure Investigations of (ent)-Cladospolide D by De Novo Synthesis and
Kinetic and Thermodynamic Isomerization Y Xing J H Penn G A OrsquoDoherty
2855 New Applications of PhI(OAc)2 in Synthesis Total Synthesis and SAR Development of Potent Antitumor Natural Product PsymberinIrciniastatin A N Shao X Huang A Palani R Aslanian A Buevich J Piwinski R Huryk C Seidel-Dugan
2873 Total Synthesis of Largazole ndash Devolution of a Novel Synthetic Strategy B Wang C J Forsyth
2881 Formal Total Synthesis of Palmerolide A J Jaumlgel M E Maier 2893 Total Synthesis of Bongkrekic Acid via Sequential SuzukindashMiyaura Coupling
Reactions M Kanematsu M Shindo M Yoshida K Shishido 2905 Stereodivergent Approach to Both C28a-syn and C28a-anti Relative
Stereochemical Manifolds in the Lepadin Family via a TiCl4-Promoted G Li L J Carlson I K Sagamanova B W Slafer R P Hsung C Gilardi H M Sklenicka N Sydorenko
2915 Enantioselective Aldol Reaction of Tetrasubstituted Ketene Silyl Acetals with Achiral Aldehydes for the Construction of Asymmetric Tertiary Alcohols An Application for the Divergent Total Syntheses of Buergerinins F and G I Shiina T Iizumi Y-s Yamai Y-i Kawakita K Yokoyama Y-k Yamada
2927 Second-Generation Biomimetic Total Synthesis of Chaetominine A Coste G Karthikeyan F Couty G Evano
2935 Total Synthesis of (+)-Fostriecin and (+)-Phoslactomycin B S Shibahara M Fujino Y Tashiro N Okamoto T Esumi K Takahashi J Ishihara S Hatakeyama
2954 Stereochemical Assignments of the Chlorinated Residues in Victorin C A C Durow C Butts C L Willis
2963 Studies of the Asymmetric Total Synthesis of Clavilactone D by the lsquoLariatrsquo Cyclization Strategy T Yoshimitsu S Nojima M Hashimoto K Tsukamoto T Tanaka
2970 Total Synthesis of the Leucetta-Derived Alkaloid Calcaridine A P B Koswatta R Sivappa H V R Dias C J Lovely
2983 Formal Synthesis of Salinosporamide A Starting from D-Glucose T Momose Y Kaiya J-i Hasegawa T Sato N Chida
2992 Synthesis of Bioactive Natural Products by Asymmetric syn- and anti-Aldol Reactions A K Ghosh Z L Dawson
no 18 3003 Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural
Products B M Trost M K Brennan 3026 One-Pot Synthesis of Furo[34-b]pyridin-5(7H)-ones from 2-
Bromopyridine-3-carboxylic Acid and Carbonyl Compounds K Kobayashi T Kozuki H Konishi
3029 Iodocyclization of N-[2-(Methylthio)phenyl]propiolamides Selective Synthesis of 3-Iodo-15-benzothiazepin-4-ones T-S Jiang X-G Zhang J-H Li
3039 A Facile Synthetic Method for Fluorine-Containing 17-Phenanthrolines Pyridine-Ring Formation Reaction of N-Propargyl-68-bis(trifluoroacetyl)-quinolin-5-amine with Various Nucleophiles D Shibata E Okada M Hinoshita M Meacutedebielle
3047 Enantiotopic Discrimination in Palladium-Mediated Nucleophilic Substitutions on Achiral Substrates Chiral Ligand versus Chiral Nucleophile O Jacquet F Charnay J-C Fiaud J Ollivier
3051 Studies on the Chemistry of 2-[3-(2-Nitrophenyl)-2-oxopropyl]benzaldehydes Novel Syntheses of 5H-Benzo[b]carbazole-611-diones and Indolo[12-b]isoquinoline-611-diones M Fernaacutendez
3061 Studies on the C22ndashC23 Aldol Coupling of Spirangien M Lorenz N Bluhm M Kalesse
3067 One-Pot Synthesis of N-Alkyl Purine Pyrimidine and Azole Derivatives from Alcohols using Ph3PCCl4 A Rapid Route to Carboacyclic Nucleoside Synthesis M N Soltani Rad A Khalafi-Nezhad S Behrouz Z Asrari M Behrouz Z Amini
3077 Synthesis of 2-Amino-34-dihydroquinazolines and Imidazo[21-b]quinazoline-2-ones A Mishra S Batra
3089 Studies on the Reaction of Diimines with Thiourea Synthesis and Solvent-Induced cistrans-Isomerization of 135-Triazinane-2-thiones B Kaboudin T Ghasemi T Yokomatsu
3094 Suzuki Coupling of Heteroaromatic Chlorides Using Highly Electron-Donating ClickPhos Ligands S M Spinella Z-H Guan J Chen X Zhang
3099 Reaction of NN-Dioxyenamines with Anhydrides of Carboxylic and Sulfonic Acids A New Method for the Synthesis of a-Hydroxyoxime Derivatives A A Tabolin A V Lesiv S L Ioffe
3106 Directed ortho Metallation Chemistry and Phosphine Synthesis New Ligands for the SuzukindashMiyaura Reaction D B G Williams S J Evans H de Bod M S Mokhadinyana T Hughes
3113 New Functional Derivatives of 9-Phenylquinine P J Boratyński J SkarŜewski
3120 On the Synthesis of Asymmetric and Dissymmetric Amino Analogues of Troumlgerrsquos Base J Artacho K Waumlrnmark
3127 Synthesis of Polycyclic Sultams by Palladium-Catalyzed Intramolecular Cyclization K C Majumdar S Mondal N De
3136 Synthesis of Functionalized L-Cysteine and L-Methionine by Reaction with Electron-Deficient Acetylenes B A Trofimov A G Malrsquokina O A Shemyakina V V Nosyreva A P Borisova S S Khutsishvili L B Krivdin
3143 A lsquoClickrsquo Approach to the Synthesis of 3-[2-(1-Alkyltriazol-4-yl)ethyl]indoles M Petrini R R Shaikh
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
2066 Enantioselective Copper-Catalyzed Conjugate Addition of Dimethylzinc to 5-(1-Arylalkylidene) Meldrumrsquos Acids A Wilsily T Lou E Fillion
2073 SuzukindashMiyaura Coupling Reactions Using Phosphite Ligands M Jang Y Jo I-K Oh H M Jung S Lee
2076 Synthesis of 2-Methylindoline- and 2-Methyl-1234-tetrahydroquinoline-Derived Phosphoramidites and Their Applications in Iridium-Catalyzed Allylic Alkylation of Indoles W-B Liu H He L-X Dai S-L You
2083 Stereocontrolled Synthesis of 13-Amino Alcohols by Reduction of Substituted 2-1-[(tert-Butylsulfinyl)amino]alkylcyclohexanones J C Gonzaacutelez-Goacutemez F Foubelo M Yus
2089 Tunable Phosphoramidite Ligands for Asymmetric Hydrovinylation Ligands par excellence for Generation of All-Carbon Quaternary Centers C R Smith H J Lim A ZhangT V RajanBabu
2101 Copper-Catalyzed Asymmetric Ring-Opening Reaction of Oxabenzonorbornadienes with Grignard and Aluminum Reagents R Millet L Gremaud T Bernardez L Palais A Alexakis
2113 A Simplified Synthesis of Takemotorsquos Catalyst A Berkessel B Seelig 2116 Pharmaceutical Substances Syntheses Patents and Applications of the
Most Relevant AIPs Edited by Axel Kleeman Juumlrgen Engel Bernhard Kutscher Dietmar Reichert Reviewed by I Agranat
XV Forthcoming Articles
no 13 2117 Recent Advances in the Aza-Claisen Rearrangement K C Majumdar
T Bhattacharyya B Chattopadhyay B Sinha 2143 A Novel and Convenient Synthesis of lsquoReversedrsquo Diamidino 25-Aryl- and
25-Azaheterocycle-Substituted Furans L Hu D W Boykin 2146 Efficient and General Preparation of Pyranostilbenes First Total Synthesis
of Artocarbene and Pawhuskin B B H Park Y R Lee W S Lyoo 2155 Mild Oxidation of Diarylacetylenes to 12-Diketones Using Oxone in
Trifluoroacetic Acid J-H Chu Y-J Chen M-J Wu 2163 One-Pot Microwave-Assisted Selective Azido ReductionTandem Cyclization
in Condensed and Solid Phase with Nickel Boride N Shankaraiah N Markandeya M Espinoza-Moraga C Arancibia A Kamal L Silva Santos
2171 Pyrrolo[321-ij]quinolin-4-one and Pyrrolo[321-ij]quinolin-6-one H McNab D J Nelson E J Rozgowska
2175 Practical Synthesis of 5-Substituted Tetrazoles under Microwave Irradiation J Roh T V Artamonova K Vaacutevrovaacute G I Koldobskii A Hrabaacutelek
2179 A Simple Method for the Synthesis of 3-Arylthieno[23-b]pyridines via Iodine-Mediated Cyclization of 3-(1-Arylalkenyl)-2-[(1-phenylethyl)sulfanyl]pyridines K Kobayashi D Nakamura Y Shiroyama S Fukamachi H Konishi
2184 Synthesis of Four Lysine-Linked Cereulide Analogues Showing Ionophoric Activity Towards Potassium Cations as Lead Compounds for Emetic Toxin-Detection by Immunoassays A Makarasen T Nishikawa M Isobe
2205 Synthesis of α-Aliphatic and β-Aromatic Substituted Taurines via Regioselective Ring Opening of Thiiranes with Ammonia H Yu S Cao L Zhang G Liu J Xu
2210 Stability of 5(6)-Carboxyfluorescein in Microwave-Assisted Synthesis of Fluorescein-Labelled O-Dimannosylated Peptides R Kowalczyk P W R Harris R P Dunbar M A Brimble
2223 Diversity-Oriented Synthesis of Functionalized Diaryl Sulfones by Regioselective [3+3] Cyclizations of 13-Bis(siloxy)buta-13-dienes with 2-(Arylsulfonyl)-3-ethoxy-2-en-1-ones Scope and Limitations M Shkoor A Riahi O Fatunsin H Reinke C Fischer P Langer
2236 Synthesis of Functionalized Salicylates by Formal [3+3] Cyclocondensation of 13-Bis(silyloxy)buta-13-dienes with 3-Alkoxy-2-en-1-ones G Mroszlig S Ladzik H Reinke A Spannenberg C Fischer P Langer
2249 Synthetic Approach to Alkoxy-β-(trifluoromethyl)styrenes and Their Application in the Synthesis of New Trifluoromethylated Heterocycles V M Muzalevskiy V G Nenajdenko A V Shastin E S Balenkova G Haufe
2260 o-Benzenedisulfonimide as a Powerful and Recyclable Organocatalyst for the Nazarov Reaction M Barbero S Cadamuro A Deagostino S Dughera P Larini E G Occhiato C Prandi S Tabasso R Vulcano P Venturello
2267 The Catalytic Potential of 4-Guanidinylpyridines in Acylation Reactions I Held E Larionov C Bozler F Wagner H Zipse
2278 Iron(III) Chloride in EthanolndashWater Highly Efficient Catalytic System for the Synthesis of Garcia Gonzalez Polyhydroxyalkyl- and C-Glycosylfurans L Nagarapu M V Chary A Satyender B Supriya R Bantu
2283 Ruthenium-Catalyzed Addition of Primary Amides to Alkynes A Stereoselective Synthesis of Secondary Enamides L J Gooszligen M Blanchot K S M Salih K Gooszligen
2289 Binaphthyl-Modified Quaternary Phosphonium Salts as Chiral Phase Transfer Catalysts Application to Asymmetric Amination of β-Keto Esters R He K Maruoka
X Table of Contents XI Forthcoming Articles
no 14 2293 Direct Methods for Stereoselective Polypropionate Synthesis A Survey
J Li D Menche 2316 Synthesis of Symmetrical Ketones from Grignard Reagents and
11-Carbonyldiimidazole D Bottalico V Fiandanese G Marchese A Punzi
2319 Synthesis of 45-Substituted Imidazoles by a Fast Condensation of 12-Diketones and Urotropine in Heterogeneous Medium G Bratulescu
2321 (Arylsulfonyl)acetones and -acetonitriles New Activated Methylenic Building Blocks for Synthesis of 123-Triazoles N T Pokhodylo V S Matiychuk M D Obushak
2324 A Safe Convenient and Efficient One-Pot Synthesis of α-Chloroketone Acetals Directly from Ketones Using Iodobenzene Dichloride J Yu C Zhang
2329 An Efficient Oxidative Conversion of Aldehydes into 2-Substituted 2-Oxazolines Using 13-Diiodo-55-dimethylhydantoin S Takahashi H Togo
2333 A Novel Procedure for the Synthesis of Benzo[b][18]naphthyridine-3-carboxylate Derivatives from MoritandashBaylisndashHillman Adduct Acetates W Zhong F Lin R Chen W Su
2341 An Improved Synthesis of 147-Triazacyclononanes (tacns) and 14710-Tetraazacyclododecanes (cyclens) J Huang Z Zhou T H Chan
2345 The Ullmann Coupling between 2-Chlorobenzoic Acids and Amino Acids A Valuable Reaction for Preparing 2-Substituted 1-Acetyl-1H-indol-3-yl Acetates J C Rodriguez Dominguez X Gang G Kirsch
2349 gem-Dibromomethyl Aromatics Efficient Aldehyde Equivalents in the KnoevenagelndashDoebner Reaction J K Augustine Y A Naik S Poojari N Chowdappa B S Sherigara K Areppa
2357 Synthesis of Novel α-Aminophosphonates Containing Adamantyl Fragment M M Kabachnik L I Minaeva I P Beletskaya
2361 Efficient Fluoride-Mediated Synthesis of 5-Amino-Substituted Isothiazoles Y S Zubenko V I Potkin
2365 Phosphine-Catalyzed Reaction of Cyanohydrins with Activated Alkynes A Siby O Loreau F Taran
2371 Sulfanyl-Substituted [3]Cumulenes and Buta-13-dienes from a Tetrakis(pyridinium)-Substituted Butadiene A Schmidt A Rahimi M Gjikaj
2379 Efficient Synthesis of 2-Substituted Pyrido[32-d]pyrimidines Involving SNAr and Palladium-Catalyzed Cross-Coupling Reactions A Tikad S Routier M Akssira J-M Leacuteger C Jarry G Guillaumet
2385 Novel Synthesis of Medium-Sized Heterocycles by Palladium-Catalyzed Intramolecular Heck Reaction via 9-endo-trig Mode of Cyclization K C Majumdar B Chattopadhyay
2393 Facile Synthesis of Fluorinated Benzofuro- and Benzothieno[23-b]pyridines α-Carbolines and Nucleosides Containing the α-Carboline Framework V O Iaroshenko Y Wang B Zhang D Volochnyuk V Ya Sosnovskikh
2403 Synthesis of Functionalized N-Vinyl Nitrogen-Containing Heterocycles S M M Lopes A M Beja M Ramos Silva J A Paixatildeo F Palacios T M V D Pinho e Melo
2408 Kumada Cross-Coupling of Aryl Grignard Reagents with Aryl Halides Catalyzed by an Immobilized Nickel Catalyst X Chen L Wang J Liu
2413 Highly Enantioselective Synthesis of Heteroaromatic Alcohols Catalyzed by Chiral DiaminodiphosphinendashRuthenium(II) Complexes W-Y Shen Y-Y Li Z-R Dong J-X Gao
2418 Concise Total Synthesis of (+)-Disparlure and its trans-Isomer Using Asymmetric Organocatalysis S-G Kim
2423 Rhodium Carbenoid Induced [12]-Migration in an L-Lyxo-Configured α-Diazo β-Keto Ester Synthesis of a New Griseolic Acid Analogue N N Bhujbal K S A Kumar D D Dhavale
2430 Synthesis of 5-Arylthio-3-hydroxyphthalates by the First [4+2] Cycloadditions of 3-Arylthio-1-silyloxy-13-butadienes with Dimethyl Acetylenedicarboxylate I Iqbal M Imran P Langer
2435 Synthesis of Highly Functionalized Proline Derivatives via a One-Pot MichaelSN-AdditionCyclization Approach U Kazmaier C Schmidt
2440 RhodiumGraphite-Catalyzed Hydrogenation of Carbocyclic and Heterocyclic Aromatic Compounds G Falini A Gualandi D Savoia
2447 Potassium [1-(tert-Butoxycarbonyl)-1H-indol-2-yl]trifluoroborate as an Efficient Building Block in Palladium-Catalyzed SuzukindashMiyaura Cross Couplings P Kassis V Beacuteneacuteteau J-Y Meacuterour S Routier
2454 Syntheses of Substituted Furans and Pyrroles by Platinum-Catalyzed Cyclizations of Propargylic Oxiranes and Aziridines in Aqueous Media M Yoshida M Al-Amin K Shishido
2467 Transition-Metal-Free Oxidative Homocoupling of Aryl Alkenyl and Alkynyl Grignard Reagents with TEMPO M S Maji A Studer
XIII Forthcoming Articles
no 15 2471 Advances in Synthetic Approaches for the Preparation of Combretastatin-
Based Anti-Cancer Agents R Singh H Kaur 2492 Synthesis of Unsymmetrical Ureas by Sulfur-Assisted Carbonylation with
Carbon Monoxide and Oxidation with Molecular Oxygen under Mild Conditions T Mizuno T Nakai M Mihara
2497 Ring-OpeningRecyclization Reactions of (Dimethylamino)propenoyl-Substituted Cyclopropanes Facile Synthesis of Halogenated Pyridin-2(1H)-ones R Zhang Y Zhou Y Liang Z Jiang D Dong
2501 Facile and Efficient Total Synthesis of Taspine B Cheng S Zhang L Zhu J Zhang Q Li A Shan L He
2505 Oligomeric Iodosylbenzene Sulfate A Convenient Hypervalent Iodine Reagent for Oxidation of Organic Sulfides and Alkenes M S Yusubov R Y Yusubova T V Funk K-W Chi V V Zhdankin
2509 Pyrrolidine-Based Organocatalysts for Enantioselective Michael Addition of Cyclohexanone to trans-β-Nitrostyrene A P Carley S Dixon J D Kilburn
2517 CundashAl Hydrotalcite An Efficient and Reusable Ligand-Free Catalyst for the Coupling of Aryl Chlorides with Aliphatic Aromatic and N(H)-Heterocyclic Amines B Sreedhar R Arundhathi P L Reddy M A Reddy M L Kantam
2523 Highly Efficient Synthesis of trans-βγ-Unsaturated a-Keto Amides C Allais T Constantieux J Rodriguez
2531 Gas-Phase Synthesis of N-Unsubstituted 3-Hydroxypyrroles and 1H-Pyrrol-3(2H)-ones L Hill G A Hunter S H Imam H McNab W J OrsquoNeill
2535 3-Hydroxy-1H-pyrrole L Hill S H Imam H McNab W J OrsquoNeill 2539 123-Thiadiazoles with Unsaturated Side Chains Synthesis
Polymerization and Photocrosslinking M Al-Smadi N Hanold H Kalbitz H Meier
2547 Synthesis of 1112-Didehydrodibenzo[ae]cycloocten-5(6H)-one A Strained Eight-Membered Alkyne S C Kornmayer F Rominger R Gleiter
2553 Stannous Chloride Dihydrate A Novel and Efficient Catalyst for the Synthesis of gem-Dihydroperoxides from Ketones and Aldehydes D Azarifar K Khosravi F Soleimanei
2557 Synthesis of a Novel Class of Azacrown Macrocycles and Lariat Crown Ethers Containing Two 124-Triazole Rings as Subunits N Foroughifar A Mobinikhaledi S Ebrahimi
2561 Enantioselective Synthesis of the 3C-Protease Inhibitor (ndash)-Thysanone by a StauntonndashWeinreb Annulation Strategy J Sperry T Y Yuen M A Brimble
2570 Stereoselective Synthesis of Unnatural β-Amino Acids from Nitroethane via 56-Dihydro-4H-12-oxazin-3-ylacetates A Yu Sukhorukov A V Lesiv O L Eliseev Y A Khomutova S L Ioffe
2579 A Versatile Unexpected One-Pot Regioselective Synthesis of a New Class of 13-Diazepinoindolones by Reaction of Pyranoindolones with Monosubstituted Ureas D Livadiotou C A Tsoleridis J Stephanidou-Stephanatou
2584 Synthesis of a Trisaccharide and a Tetrasaccharide from the Cell-Wall Lipopolysaccharides of Azospirillum brasilense S17 S Pandey S Ghosh A K Misra
2591 Synthesis of Isoindoline Nitroxides by Electrocyclic Reactions T Kaacutelai J Jekı K Hideg
2596 Glycosylations of Tertiary Alcohols Synthesis of Fully Protected Disaccharides with Sterically Demanding Groups Attached to the Sugar Core A Holkenbrink J B Vicente D B Werz
2605 Copper-Catalyzed [13]-Dipolar Cycloaddition for the Synthesis of Macrocycles Containing Acyclic Aromatic and Steroidal Moieties G V Latyshev M S Baranom A V Kazantsev A D Averin N V Lukashev I P Beletskaya
2616 Aryl Ring Migration Reaction in the Synthesis of 24-Diaryl-4H-31-benzothiazines A V Butin F A Tsiunchik V T Abaev A V Gutnov D A Cheshkov
2627 Hydrogenation of β-N-Substituted and β-NN-Disubstituted Enamino Esters in the Presence of Iridium(I) Catalyst H Hebbache Z Hank C Bruneau J-L Renaud
2634 Stereoselective Olefination Reactions Promoted by Rieke Manganese J M Concelloacuten H Rodriacuteguez-Solla V del Amo P Diacuteaz
2646 Synthesis of Piperidinones through a Radical Cascade E Godineau Y Landais
2650 Asymmetric Organic Synthesis with Enzymes Edited by V Gotor I Alfonso E Garciacutea-Urdiales Reviewed by Steve Collier
XVII Forthcoming Articles
no 16 2651 Synthesis of Spirocyclic Ethers S Rosenberg R Leino 2674 Bimetallic PalladiumndashPlatinum-on-Carbon-Catalyzed HndashD Exchange
Reaction Synergistic Effect on Multiple Deuterium Incorporation T Maegawa N Ito K Oono Y Monguchi H Sajiki
2679 Efficient Copper-Catalyzed Synthesis of 2-Amino-4(3H)-quinazolinone and 2-Aminoquinazoline Derivatives X Huang H Yang H Fu R Qiao Y Zhao
2689 Synthesis and Chemoselective N- and O-Alkylation of Thiadiazolopyrimidine Nucleosides and Uridines A M L Hossion R Islam R K Kandahary T Nagamatsu
2697 Facile and Efficient Synthesis of a New Class of Indole-Substituted Pyridine Derivatives via One-Pot Multicomponent Reactions K Zhao X-P Xu S-L Zhu D-Q Shi Y Zhang S-J Ji
2709 Studies toward a Total Synthesis of Rhizoxin D Stereoselective Preparation of the C11ndashC19 Fragment S Padakanti C K Kumar E Ashok P Das
2715 A Short Synthesis of Enantiomeric Phytoprostanes B1 Type I W Perlikowska M Mikołajczyk
2719 Chemistry of Polyhalogenated Nitrobutadienes Part 7 A Novel Synthetic Access to Chlorinated Nitrile Oxides E Nutz V A Zapolrsquoskii D E Kaufmann
2725 Microwave-Assisted Silver(I)-Mediated Selective O-Alkylation of Aromatic Imidate Systems B K Singh C Cavalluzzo M De Maeyer Z Debyser V S Parmar E Van der Eycken
2729 Iodogen A Novel Reagent for the Oxidation of Urazoles under Heterogeneous Conditions A Khoramabadi A Shiri M A Zolfigol S Mallakpour
2733 An Unprecedented Synthesis of Eight-Membered-Ring Cyclic Thioimidic Esters by a Three-Component Reaction A Alizadeh R Hosseinpour
2737 A Novel Diastereoselective Synthesis of β-Phosphonato Unsaturated Thioimidates A Alizadeh N Zohreh
2741 Synthesis of 21-Benzisoxazoles by Nucleophilic Substitution of Hydrogen in Nitroarenes Activated by the Azole Ring N T Pokhodylo Y O Teslenko V S Matiychuk M D Obushak
2749 A Facile Synthesis of Two Series of Multifunctional Carbon Compounds from αα-Dihalo Ketones Using Allylsamarium Bromide X Liu S Zhang J Di
2756 Stereocontrolled Formation of Protected Aminodeoxyalditols from Simple Carbohydrate Precursors by Debenzylating Cycloetherification Y Jiang Z Fang Q Zheng H Jia J Cheng B Zheng
2761 trans-Stilbene as a Starting Material for the Synthesis of Tamoxifen Based on Palladium-Catalyzed Cross-Coupling Reactions C M Nunes J Limberger S Poersch M Seferin A L Monteiro
2766 Synthesis and Biological Evaluation of 6-Substituted Purinylcarbanucleosides with a Cyclopenta[b]thiophene Pseudosugar P Abeijoacuten J M Blanco O Caamantildeo F Fernaacutendez M D Garciacutea X Garciacutea-Mera J E Rodriacuteguez-Borges J Balzarini E De Clercq
2773 Synthesis and Electrochemical Signature of Novel Norbornyl-ferrocene Hybrids F A Khan S K Upadhyay
2778 A Regioselective TsujindashTrost Pentadienylation of 3-Allyltetronic Acid R Schobert B Barnickel
2785 Copper(I)-Catalyzed CarylndashCalkynyl Bond Formation of Aryl Iodides with Terminal Alkynes K G Thakur G Sekar
2790 Aminolysis of Epoxides Using Iridium Trichloride as an Efficient Catalyst J Agarwal A Duley R Rani R K Peddinti
2797 Preparation of Several Active N-Chloro Compounds from Trichloroisocyanuric Acid A Shiri A Khoramabadi-zad
2802 The First Mineral-Catalyzed One-Pot [3+1+2] Coupling Protocol for Multifunctionalized Fused-Ring Pyrimidines L D S Yadav A Rai
2809 Efficient Synthesis of Tetrahydro-β-carbolin-1-one and Dihydroisoquinolin-1-one Derivatives as Versatile Intermediates K E Judd M F Mahon L Caggiano
2818 A Concise Synthesis of ortho-Iodobenzyl Alcohols via Addition of ortho-Iodophenyl Grignard Reagent to Aldehydes and Ketones J Cvengroš D Stolz A Togni
XIII Forthcoming Articles
no 17 2825 Reactivity of Oxazol-5-(4H)-ones and Their Application toward Natural
Product Synthesis N M Hewlett C D Hupp J J Tepe 2840 Towards the Total Synthesis of 3-Hydroxyvibsanin E B D Schwartz
J R Denton P V Bernhardt H M L Davies C M Williams 2847 Structure Investigations of (ent)-Cladospolide D by De Novo Synthesis and
Kinetic and Thermodynamic Isomerization Y Xing J H Penn G A OrsquoDoherty
2855 New Applications of PhI(OAc)2 in Synthesis Total Synthesis and SAR Development of Potent Antitumor Natural Product PsymberinIrciniastatin A N Shao X Huang A Palani R Aslanian A Buevich J Piwinski R Huryk C Seidel-Dugan
2873 Total Synthesis of Largazole ndash Devolution of a Novel Synthetic Strategy B Wang C J Forsyth
2881 Formal Total Synthesis of Palmerolide A J Jaumlgel M E Maier 2893 Total Synthesis of Bongkrekic Acid via Sequential SuzukindashMiyaura Coupling
Reactions M Kanematsu M Shindo M Yoshida K Shishido 2905 Stereodivergent Approach to Both C28a-syn and C28a-anti Relative
Stereochemical Manifolds in the Lepadin Family via a TiCl4-Promoted G Li L J Carlson I K Sagamanova B W Slafer R P Hsung C Gilardi H M Sklenicka N Sydorenko
2915 Enantioselective Aldol Reaction of Tetrasubstituted Ketene Silyl Acetals with Achiral Aldehydes for the Construction of Asymmetric Tertiary Alcohols An Application for the Divergent Total Syntheses of Buergerinins F and G I Shiina T Iizumi Y-s Yamai Y-i Kawakita K Yokoyama Y-k Yamada
2927 Second-Generation Biomimetic Total Synthesis of Chaetominine A Coste G Karthikeyan F Couty G Evano
2935 Total Synthesis of (+)-Fostriecin and (+)-Phoslactomycin B S Shibahara M Fujino Y Tashiro N Okamoto T Esumi K Takahashi J Ishihara S Hatakeyama
2954 Stereochemical Assignments of the Chlorinated Residues in Victorin C A C Durow C Butts C L Willis
2963 Studies of the Asymmetric Total Synthesis of Clavilactone D by the lsquoLariatrsquo Cyclization Strategy T Yoshimitsu S Nojima M Hashimoto K Tsukamoto T Tanaka
2970 Total Synthesis of the Leucetta-Derived Alkaloid Calcaridine A P B Koswatta R Sivappa H V R Dias C J Lovely
2983 Formal Synthesis of Salinosporamide A Starting from D-Glucose T Momose Y Kaiya J-i Hasegawa T Sato N Chida
2992 Synthesis of Bioactive Natural Products by Asymmetric syn- and anti-Aldol Reactions A K Ghosh Z L Dawson
no 18 3003 Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural
Products B M Trost M K Brennan 3026 One-Pot Synthesis of Furo[34-b]pyridin-5(7H)-ones from 2-
Bromopyridine-3-carboxylic Acid and Carbonyl Compounds K Kobayashi T Kozuki H Konishi
3029 Iodocyclization of N-[2-(Methylthio)phenyl]propiolamides Selective Synthesis of 3-Iodo-15-benzothiazepin-4-ones T-S Jiang X-G Zhang J-H Li
3039 A Facile Synthetic Method for Fluorine-Containing 17-Phenanthrolines Pyridine-Ring Formation Reaction of N-Propargyl-68-bis(trifluoroacetyl)-quinolin-5-amine with Various Nucleophiles D Shibata E Okada M Hinoshita M Meacutedebielle
3047 Enantiotopic Discrimination in Palladium-Mediated Nucleophilic Substitutions on Achiral Substrates Chiral Ligand versus Chiral Nucleophile O Jacquet F Charnay J-C Fiaud J Ollivier
3051 Studies on the Chemistry of 2-[3-(2-Nitrophenyl)-2-oxopropyl]benzaldehydes Novel Syntheses of 5H-Benzo[b]carbazole-611-diones and Indolo[12-b]isoquinoline-611-diones M Fernaacutendez
3061 Studies on the C22ndashC23 Aldol Coupling of Spirangien M Lorenz N Bluhm M Kalesse
3067 One-Pot Synthesis of N-Alkyl Purine Pyrimidine and Azole Derivatives from Alcohols using Ph3PCCl4 A Rapid Route to Carboacyclic Nucleoside Synthesis M N Soltani Rad A Khalafi-Nezhad S Behrouz Z Asrari M Behrouz Z Amini
3077 Synthesis of 2-Amino-34-dihydroquinazolines and Imidazo[21-b]quinazoline-2-ones A Mishra S Batra
3089 Studies on the Reaction of Diimines with Thiourea Synthesis and Solvent-Induced cistrans-Isomerization of 135-Triazinane-2-thiones B Kaboudin T Ghasemi T Yokomatsu
3094 Suzuki Coupling of Heteroaromatic Chlorides Using Highly Electron-Donating ClickPhos Ligands S M Spinella Z-H Guan J Chen X Zhang
3099 Reaction of NN-Dioxyenamines with Anhydrides of Carboxylic and Sulfonic Acids A New Method for the Synthesis of a-Hydroxyoxime Derivatives A A Tabolin A V Lesiv S L Ioffe
3106 Directed ortho Metallation Chemistry and Phosphine Synthesis New Ligands for the SuzukindashMiyaura Reaction D B G Williams S J Evans H de Bod M S Mokhadinyana T Hughes
3113 New Functional Derivatives of 9-Phenylquinine P J Boratyński J SkarŜewski
3120 On the Synthesis of Asymmetric and Dissymmetric Amino Analogues of Troumlgerrsquos Base J Artacho K Waumlrnmark
3127 Synthesis of Polycyclic Sultams by Palladium-Catalyzed Intramolecular Cyclization K C Majumdar S Mondal N De
3136 Synthesis of Functionalized L-Cysteine and L-Methionine by Reaction with Electron-Deficient Acetylenes B A Trofimov A G Malrsquokina O A Shemyakina V V Nosyreva A P Borisova S S Khutsishvili L B Krivdin
3143 A lsquoClickrsquo Approach to the Synthesis of 3-[2-(1-Alkyltriazol-4-yl)ethyl]indoles M Petrini R R Shaikh
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
no 13 2117 Recent Advances in the Aza-Claisen Rearrangement K C Majumdar
T Bhattacharyya B Chattopadhyay B Sinha 2143 A Novel and Convenient Synthesis of lsquoReversedrsquo Diamidino 25-Aryl- and
25-Azaheterocycle-Substituted Furans L Hu D W Boykin 2146 Efficient and General Preparation of Pyranostilbenes First Total Synthesis
of Artocarbene and Pawhuskin B B H Park Y R Lee W S Lyoo 2155 Mild Oxidation of Diarylacetylenes to 12-Diketones Using Oxone in
Trifluoroacetic Acid J-H Chu Y-J Chen M-J Wu 2163 One-Pot Microwave-Assisted Selective Azido ReductionTandem Cyclization
in Condensed and Solid Phase with Nickel Boride N Shankaraiah N Markandeya M Espinoza-Moraga C Arancibia A Kamal L Silva Santos
2171 Pyrrolo[321-ij]quinolin-4-one and Pyrrolo[321-ij]quinolin-6-one H McNab D J Nelson E J Rozgowska
2175 Practical Synthesis of 5-Substituted Tetrazoles under Microwave Irradiation J Roh T V Artamonova K Vaacutevrovaacute G I Koldobskii A Hrabaacutelek
2179 A Simple Method for the Synthesis of 3-Arylthieno[23-b]pyridines via Iodine-Mediated Cyclization of 3-(1-Arylalkenyl)-2-[(1-phenylethyl)sulfanyl]pyridines K Kobayashi D Nakamura Y Shiroyama S Fukamachi H Konishi
2184 Synthesis of Four Lysine-Linked Cereulide Analogues Showing Ionophoric Activity Towards Potassium Cations as Lead Compounds for Emetic Toxin-Detection by Immunoassays A Makarasen T Nishikawa M Isobe
2205 Synthesis of α-Aliphatic and β-Aromatic Substituted Taurines via Regioselective Ring Opening of Thiiranes with Ammonia H Yu S Cao L Zhang G Liu J Xu
2210 Stability of 5(6)-Carboxyfluorescein in Microwave-Assisted Synthesis of Fluorescein-Labelled O-Dimannosylated Peptides R Kowalczyk P W R Harris R P Dunbar M A Brimble
2223 Diversity-Oriented Synthesis of Functionalized Diaryl Sulfones by Regioselective [3+3] Cyclizations of 13-Bis(siloxy)buta-13-dienes with 2-(Arylsulfonyl)-3-ethoxy-2-en-1-ones Scope and Limitations M Shkoor A Riahi O Fatunsin H Reinke C Fischer P Langer
2236 Synthesis of Functionalized Salicylates by Formal [3+3] Cyclocondensation of 13-Bis(silyloxy)buta-13-dienes with 3-Alkoxy-2-en-1-ones G Mroszlig S Ladzik H Reinke A Spannenberg C Fischer P Langer
2249 Synthetic Approach to Alkoxy-β-(trifluoromethyl)styrenes and Their Application in the Synthesis of New Trifluoromethylated Heterocycles V M Muzalevskiy V G Nenajdenko A V Shastin E S Balenkova G Haufe
2260 o-Benzenedisulfonimide as a Powerful and Recyclable Organocatalyst for the Nazarov Reaction M Barbero S Cadamuro A Deagostino S Dughera P Larini E G Occhiato C Prandi S Tabasso R Vulcano P Venturello
2267 The Catalytic Potential of 4-Guanidinylpyridines in Acylation Reactions I Held E Larionov C Bozler F Wagner H Zipse
2278 Iron(III) Chloride in EthanolndashWater Highly Efficient Catalytic System for the Synthesis of Garcia Gonzalez Polyhydroxyalkyl- and C-Glycosylfurans L Nagarapu M V Chary A Satyender B Supriya R Bantu
2283 Ruthenium-Catalyzed Addition of Primary Amides to Alkynes A Stereoselective Synthesis of Secondary Enamides L J Gooszligen M Blanchot K S M Salih K Gooszligen
2289 Binaphthyl-Modified Quaternary Phosphonium Salts as Chiral Phase Transfer Catalysts Application to Asymmetric Amination of β-Keto Esters R He K Maruoka
X Table of Contents XI Forthcoming Articles
no 14 2293 Direct Methods for Stereoselective Polypropionate Synthesis A Survey
J Li D Menche 2316 Synthesis of Symmetrical Ketones from Grignard Reagents and
11-Carbonyldiimidazole D Bottalico V Fiandanese G Marchese A Punzi
2319 Synthesis of 45-Substituted Imidazoles by a Fast Condensation of 12-Diketones and Urotropine in Heterogeneous Medium G Bratulescu
2321 (Arylsulfonyl)acetones and -acetonitriles New Activated Methylenic Building Blocks for Synthesis of 123-Triazoles N T Pokhodylo V S Matiychuk M D Obushak
2324 A Safe Convenient and Efficient One-Pot Synthesis of α-Chloroketone Acetals Directly from Ketones Using Iodobenzene Dichloride J Yu C Zhang
2329 An Efficient Oxidative Conversion of Aldehydes into 2-Substituted 2-Oxazolines Using 13-Diiodo-55-dimethylhydantoin S Takahashi H Togo
2333 A Novel Procedure for the Synthesis of Benzo[b][18]naphthyridine-3-carboxylate Derivatives from MoritandashBaylisndashHillman Adduct Acetates W Zhong F Lin R Chen W Su
2341 An Improved Synthesis of 147-Triazacyclononanes (tacns) and 14710-Tetraazacyclododecanes (cyclens) J Huang Z Zhou T H Chan
2345 The Ullmann Coupling between 2-Chlorobenzoic Acids and Amino Acids A Valuable Reaction for Preparing 2-Substituted 1-Acetyl-1H-indol-3-yl Acetates J C Rodriguez Dominguez X Gang G Kirsch
2349 gem-Dibromomethyl Aromatics Efficient Aldehyde Equivalents in the KnoevenagelndashDoebner Reaction J K Augustine Y A Naik S Poojari N Chowdappa B S Sherigara K Areppa
2357 Synthesis of Novel α-Aminophosphonates Containing Adamantyl Fragment M M Kabachnik L I Minaeva I P Beletskaya
2361 Efficient Fluoride-Mediated Synthesis of 5-Amino-Substituted Isothiazoles Y S Zubenko V I Potkin
2365 Phosphine-Catalyzed Reaction of Cyanohydrins with Activated Alkynes A Siby O Loreau F Taran
2371 Sulfanyl-Substituted [3]Cumulenes and Buta-13-dienes from a Tetrakis(pyridinium)-Substituted Butadiene A Schmidt A Rahimi M Gjikaj
2379 Efficient Synthesis of 2-Substituted Pyrido[32-d]pyrimidines Involving SNAr and Palladium-Catalyzed Cross-Coupling Reactions A Tikad S Routier M Akssira J-M Leacuteger C Jarry G Guillaumet
2385 Novel Synthesis of Medium-Sized Heterocycles by Palladium-Catalyzed Intramolecular Heck Reaction via 9-endo-trig Mode of Cyclization K C Majumdar B Chattopadhyay
2393 Facile Synthesis of Fluorinated Benzofuro- and Benzothieno[23-b]pyridines α-Carbolines and Nucleosides Containing the α-Carboline Framework V O Iaroshenko Y Wang B Zhang D Volochnyuk V Ya Sosnovskikh
2403 Synthesis of Functionalized N-Vinyl Nitrogen-Containing Heterocycles S M M Lopes A M Beja M Ramos Silva J A Paixatildeo F Palacios T M V D Pinho e Melo
2408 Kumada Cross-Coupling of Aryl Grignard Reagents with Aryl Halides Catalyzed by an Immobilized Nickel Catalyst X Chen L Wang J Liu
2413 Highly Enantioselective Synthesis of Heteroaromatic Alcohols Catalyzed by Chiral DiaminodiphosphinendashRuthenium(II) Complexes W-Y Shen Y-Y Li Z-R Dong J-X Gao
2418 Concise Total Synthesis of (+)-Disparlure and its trans-Isomer Using Asymmetric Organocatalysis S-G Kim
2423 Rhodium Carbenoid Induced [12]-Migration in an L-Lyxo-Configured α-Diazo β-Keto Ester Synthesis of a New Griseolic Acid Analogue N N Bhujbal K S A Kumar D D Dhavale
2430 Synthesis of 5-Arylthio-3-hydroxyphthalates by the First [4+2] Cycloadditions of 3-Arylthio-1-silyloxy-13-butadienes with Dimethyl Acetylenedicarboxylate I Iqbal M Imran P Langer
2435 Synthesis of Highly Functionalized Proline Derivatives via a One-Pot MichaelSN-AdditionCyclization Approach U Kazmaier C Schmidt
2440 RhodiumGraphite-Catalyzed Hydrogenation of Carbocyclic and Heterocyclic Aromatic Compounds G Falini A Gualandi D Savoia
2447 Potassium [1-(tert-Butoxycarbonyl)-1H-indol-2-yl]trifluoroborate as an Efficient Building Block in Palladium-Catalyzed SuzukindashMiyaura Cross Couplings P Kassis V Beacuteneacuteteau J-Y Meacuterour S Routier
2454 Syntheses of Substituted Furans and Pyrroles by Platinum-Catalyzed Cyclizations of Propargylic Oxiranes and Aziridines in Aqueous Media M Yoshida M Al-Amin K Shishido
2467 Transition-Metal-Free Oxidative Homocoupling of Aryl Alkenyl and Alkynyl Grignard Reagents with TEMPO M S Maji A Studer
XIII Forthcoming Articles
no 15 2471 Advances in Synthetic Approaches for the Preparation of Combretastatin-
Based Anti-Cancer Agents R Singh H Kaur 2492 Synthesis of Unsymmetrical Ureas by Sulfur-Assisted Carbonylation with
Carbon Monoxide and Oxidation with Molecular Oxygen under Mild Conditions T Mizuno T Nakai M Mihara
2497 Ring-OpeningRecyclization Reactions of (Dimethylamino)propenoyl-Substituted Cyclopropanes Facile Synthesis of Halogenated Pyridin-2(1H)-ones R Zhang Y Zhou Y Liang Z Jiang D Dong
2501 Facile and Efficient Total Synthesis of Taspine B Cheng S Zhang L Zhu J Zhang Q Li A Shan L He
2505 Oligomeric Iodosylbenzene Sulfate A Convenient Hypervalent Iodine Reagent for Oxidation of Organic Sulfides and Alkenes M S Yusubov R Y Yusubova T V Funk K-W Chi V V Zhdankin
2509 Pyrrolidine-Based Organocatalysts for Enantioselective Michael Addition of Cyclohexanone to trans-β-Nitrostyrene A P Carley S Dixon J D Kilburn
2517 CundashAl Hydrotalcite An Efficient and Reusable Ligand-Free Catalyst for the Coupling of Aryl Chlorides with Aliphatic Aromatic and N(H)-Heterocyclic Amines B Sreedhar R Arundhathi P L Reddy M A Reddy M L Kantam
2523 Highly Efficient Synthesis of trans-βγ-Unsaturated a-Keto Amides C Allais T Constantieux J Rodriguez
2531 Gas-Phase Synthesis of N-Unsubstituted 3-Hydroxypyrroles and 1H-Pyrrol-3(2H)-ones L Hill G A Hunter S H Imam H McNab W J OrsquoNeill
2535 3-Hydroxy-1H-pyrrole L Hill S H Imam H McNab W J OrsquoNeill 2539 123-Thiadiazoles with Unsaturated Side Chains Synthesis
Polymerization and Photocrosslinking M Al-Smadi N Hanold H Kalbitz H Meier
2547 Synthesis of 1112-Didehydrodibenzo[ae]cycloocten-5(6H)-one A Strained Eight-Membered Alkyne S C Kornmayer F Rominger R Gleiter
2553 Stannous Chloride Dihydrate A Novel and Efficient Catalyst for the Synthesis of gem-Dihydroperoxides from Ketones and Aldehydes D Azarifar K Khosravi F Soleimanei
2557 Synthesis of a Novel Class of Azacrown Macrocycles and Lariat Crown Ethers Containing Two 124-Triazole Rings as Subunits N Foroughifar A Mobinikhaledi S Ebrahimi
2561 Enantioselective Synthesis of the 3C-Protease Inhibitor (ndash)-Thysanone by a StauntonndashWeinreb Annulation Strategy J Sperry T Y Yuen M A Brimble
2570 Stereoselective Synthesis of Unnatural β-Amino Acids from Nitroethane via 56-Dihydro-4H-12-oxazin-3-ylacetates A Yu Sukhorukov A V Lesiv O L Eliseev Y A Khomutova S L Ioffe
2579 A Versatile Unexpected One-Pot Regioselective Synthesis of a New Class of 13-Diazepinoindolones by Reaction of Pyranoindolones with Monosubstituted Ureas D Livadiotou C A Tsoleridis J Stephanidou-Stephanatou
2584 Synthesis of a Trisaccharide and a Tetrasaccharide from the Cell-Wall Lipopolysaccharides of Azospirillum brasilense S17 S Pandey S Ghosh A K Misra
2591 Synthesis of Isoindoline Nitroxides by Electrocyclic Reactions T Kaacutelai J Jekı K Hideg
2596 Glycosylations of Tertiary Alcohols Synthesis of Fully Protected Disaccharides with Sterically Demanding Groups Attached to the Sugar Core A Holkenbrink J B Vicente D B Werz
2605 Copper-Catalyzed [13]-Dipolar Cycloaddition for the Synthesis of Macrocycles Containing Acyclic Aromatic and Steroidal Moieties G V Latyshev M S Baranom A V Kazantsev A D Averin N V Lukashev I P Beletskaya
2616 Aryl Ring Migration Reaction in the Synthesis of 24-Diaryl-4H-31-benzothiazines A V Butin F A Tsiunchik V T Abaev A V Gutnov D A Cheshkov
2627 Hydrogenation of β-N-Substituted and β-NN-Disubstituted Enamino Esters in the Presence of Iridium(I) Catalyst H Hebbache Z Hank C Bruneau J-L Renaud
2634 Stereoselective Olefination Reactions Promoted by Rieke Manganese J M Concelloacuten H Rodriacuteguez-Solla V del Amo P Diacuteaz
2646 Synthesis of Piperidinones through a Radical Cascade E Godineau Y Landais
2650 Asymmetric Organic Synthesis with Enzymes Edited by V Gotor I Alfonso E Garciacutea-Urdiales Reviewed by Steve Collier
XVII Forthcoming Articles
no 16 2651 Synthesis of Spirocyclic Ethers S Rosenberg R Leino 2674 Bimetallic PalladiumndashPlatinum-on-Carbon-Catalyzed HndashD Exchange
Reaction Synergistic Effect on Multiple Deuterium Incorporation T Maegawa N Ito K Oono Y Monguchi H Sajiki
2679 Efficient Copper-Catalyzed Synthesis of 2-Amino-4(3H)-quinazolinone and 2-Aminoquinazoline Derivatives X Huang H Yang H Fu R Qiao Y Zhao
2689 Synthesis and Chemoselective N- and O-Alkylation of Thiadiazolopyrimidine Nucleosides and Uridines A M L Hossion R Islam R K Kandahary T Nagamatsu
2697 Facile and Efficient Synthesis of a New Class of Indole-Substituted Pyridine Derivatives via One-Pot Multicomponent Reactions K Zhao X-P Xu S-L Zhu D-Q Shi Y Zhang S-J Ji
2709 Studies toward a Total Synthesis of Rhizoxin D Stereoselective Preparation of the C11ndashC19 Fragment S Padakanti C K Kumar E Ashok P Das
2715 A Short Synthesis of Enantiomeric Phytoprostanes B1 Type I W Perlikowska M Mikołajczyk
2719 Chemistry of Polyhalogenated Nitrobutadienes Part 7 A Novel Synthetic Access to Chlorinated Nitrile Oxides E Nutz V A Zapolrsquoskii D E Kaufmann
2725 Microwave-Assisted Silver(I)-Mediated Selective O-Alkylation of Aromatic Imidate Systems B K Singh C Cavalluzzo M De Maeyer Z Debyser V S Parmar E Van der Eycken
2729 Iodogen A Novel Reagent for the Oxidation of Urazoles under Heterogeneous Conditions A Khoramabadi A Shiri M A Zolfigol S Mallakpour
2733 An Unprecedented Synthesis of Eight-Membered-Ring Cyclic Thioimidic Esters by a Three-Component Reaction A Alizadeh R Hosseinpour
2737 A Novel Diastereoselective Synthesis of β-Phosphonato Unsaturated Thioimidates A Alizadeh N Zohreh
2741 Synthesis of 21-Benzisoxazoles by Nucleophilic Substitution of Hydrogen in Nitroarenes Activated by the Azole Ring N T Pokhodylo Y O Teslenko V S Matiychuk M D Obushak
2749 A Facile Synthesis of Two Series of Multifunctional Carbon Compounds from αα-Dihalo Ketones Using Allylsamarium Bromide X Liu S Zhang J Di
2756 Stereocontrolled Formation of Protected Aminodeoxyalditols from Simple Carbohydrate Precursors by Debenzylating Cycloetherification Y Jiang Z Fang Q Zheng H Jia J Cheng B Zheng
2761 trans-Stilbene as a Starting Material for the Synthesis of Tamoxifen Based on Palladium-Catalyzed Cross-Coupling Reactions C M Nunes J Limberger S Poersch M Seferin A L Monteiro
2766 Synthesis and Biological Evaluation of 6-Substituted Purinylcarbanucleosides with a Cyclopenta[b]thiophene Pseudosugar P Abeijoacuten J M Blanco O Caamantildeo F Fernaacutendez M D Garciacutea X Garciacutea-Mera J E Rodriacuteguez-Borges J Balzarini E De Clercq
2773 Synthesis and Electrochemical Signature of Novel Norbornyl-ferrocene Hybrids F A Khan S K Upadhyay
2778 A Regioselective TsujindashTrost Pentadienylation of 3-Allyltetronic Acid R Schobert B Barnickel
2785 Copper(I)-Catalyzed CarylndashCalkynyl Bond Formation of Aryl Iodides with Terminal Alkynes K G Thakur G Sekar
2790 Aminolysis of Epoxides Using Iridium Trichloride as an Efficient Catalyst J Agarwal A Duley R Rani R K Peddinti
2797 Preparation of Several Active N-Chloro Compounds from Trichloroisocyanuric Acid A Shiri A Khoramabadi-zad
2802 The First Mineral-Catalyzed One-Pot [3+1+2] Coupling Protocol for Multifunctionalized Fused-Ring Pyrimidines L D S Yadav A Rai
2809 Efficient Synthesis of Tetrahydro-β-carbolin-1-one and Dihydroisoquinolin-1-one Derivatives as Versatile Intermediates K E Judd M F Mahon L Caggiano
2818 A Concise Synthesis of ortho-Iodobenzyl Alcohols via Addition of ortho-Iodophenyl Grignard Reagent to Aldehydes and Ketones J Cvengroš D Stolz A Togni
XIII Forthcoming Articles
no 17 2825 Reactivity of Oxazol-5-(4H)-ones and Their Application toward Natural
Product Synthesis N M Hewlett C D Hupp J J Tepe 2840 Towards the Total Synthesis of 3-Hydroxyvibsanin E B D Schwartz
J R Denton P V Bernhardt H M L Davies C M Williams 2847 Structure Investigations of (ent)-Cladospolide D by De Novo Synthesis and
Kinetic and Thermodynamic Isomerization Y Xing J H Penn G A OrsquoDoherty
2855 New Applications of PhI(OAc)2 in Synthesis Total Synthesis and SAR Development of Potent Antitumor Natural Product PsymberinIrciniastatin A N Shao X Huang A Palani R Aslanian A Buevich J Piwinski R Huryk C Seidel-Dugan
2873 Total Synthesis of Largazole ndash Devolution of a Novel Synthetic Strategy B Wang C J Forsyth
2881 Formal Total Synthesis of Palmerolide A J Jaumlgel M E Maier 2893 Total Synthesis of Bongkrekic Acid via Sequential SuzukindashMiyaura Coupling
Reactions M Kanematsu M Shindo M Yoshida K Shishido 2905 Stereodivergent Approach to Both C28a-syn and C28a-anti Relative
Stereochemical Manifolds in the Lepadin Family via a TiCl4-Promoted G Li L J Carlson I K Sagamanova B W Slafer R P Hsung C Gilardi H M Sklenicka N Sydorenko
2915 Enantioselective Aldol Reaction of Tetrasubstituted Ketene Silyl Acetals with Achiral Aldehydes for the Construction of Asymmetric Tertiary Alcohols An Application for the Divergent Total Syntheses of Buergerinins F and G I Shiina T Iizumi Y-s Yamai Y-i Kawakita K Yokoyama Y-k Yamada
2927 Second-Generation Biomimetic Total Synthesis of Chaetominine A Coste G Karthikeyan F Couty G Evano
2935 Total Synthesis of (+)-Fostriecin and (+)-Phoslactomycin B S Shibahara M Fujino Y Tashiro N Okamoto T Esumi K Takahashi J Ishihara S Hatakeyama
2954 Stereochemical Assignments of the Chlorinated Residues in Victorin C A C Durow C Butts C L Willis
2963 Studies of the Asymmetric Total Synthesis of Clavilactone D by the lsquoLariatrsquo Cyclization Strategy T Yoshimitsu S Nojima M Hashimoto K Tsukamoto T Tanaka
2970 Total Synthesis of the Leucetta-Derived Alkaloid Calcaridine A P B Koswatta R Sivappa H V R Dias C J Lovely
2983 Formal Synthesis of Salinosporamide A Starting from D-Glucose T Momose Y Kaiya J-i Hasegawa T Sato N Chida
2992 Synthesis of Bioactive Natural Products by Asymmetric syn- and anti-Aldol Reactions A K Ghosh Z L Dawson
no 18 3003 Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural
Products B M Trost M K Brennan 3026 One-Pot Synthesis of Furo[34-b]pyridin-5(7H)-ones from 2-
Bromopyridine-3-carboxylic Acid and Carbonyl Compounds K Kobayashi T Kozuki H Konishi
3029 Iodocyclization of N-[2-(Methylthio)phenyl]propiolamides Selective Synthesis of 3-Iodo-15-benzothiazepin-4-ones T-S Jiang X-G Zhang J-H Li
3039 A Facile Synthetic Method for Fluorine-Containing 17-Phenanthrolines Pyridine-Ring Formation Reaction of N-Propargyl-68-bis(trifluoroacetyl)-quinolin-5-amine with Various Nucleophiles D Shibata E Okada M Hinoshita M Meacutedebielle
3047 Enantiotopic Discrimination in Palladium-Mediated Nucleophilic Substitutions on Achiral Substrates Chiral Ligand versus Chiral Nucleophile O Jacquet F Charnay J-C Fiaud J Ollivier
3051 Studies on the Chemistry of 2-[3-(2-Nitrophenyl)-2-oxopropyl]benzaldehydes Novel Syntheses of 5H-Benzo[b]carbazole-611-diones and Indolo[12-b]isoquinoline-611-diones M Fernaacutendez
3061 Studies on the C22ndashC23 Aldol Coupling of Spirangien M Lorenz N Bluhm M Kalesse
3067 One-Pot Synthesis of N-Alkyl Purine Pyrimidine and Azole Derivatives from Alcohols using Ph3PCCl4 A Rapid Route to Carboacyclic Nucleoside Synthesis M N Soltani Rad A Khalafi-Nezhad S Behrouz Z Asrari M Behrouz Z Amini
3077 Synthesis of 2-Amino-34-dihydroquinazolines and Imidazo[21-b]quinazoline-2-ones A Mishra S Batra
3089 Studies on the Reaction of Diimines with Thiourea Synthesis and Solvent-Induced cistrans-Isomerization of 135-Triazinane-2-thiones B Kaboudin T Ghasemi T Yokomatsu
3094 Suzuki Coupling of Heteroaromatic Chlorides Using Highly Electron-Donating ClickPhos Ligands S M Spinella Z-H Guan J Chen X Zhang
3099 Reaction of NN-Dioxyenamines with Anhydrides of Carboxylic and Sulfonic Acids A New Method for the Synthesis of a-Hydroxyoxime Derivatives A A Tabolin A V Lesiv S L Ioffe
3106 Directed ortho Metallation Chemistry and Phosphine Synthesis New Ligands for the SuzukindashMiyaura Reaction D B G Williams S J Evans H de Bod M S Mokhadinyana T Hughes
3113 New Functional Derivatives of 9-Phenylquinine P J Boratyński J SkarŜewski
3120 On the Synthesis of Asymmetric and Dissymmetric Amino Analogues of Troumlgerrsquos Base J Artacho K Waumlrnmark
3127 Synthesis of Polycyclic Sultams by Palladium-Catalyzed Intramolecular Cyclization K C Majumdar S Mondal N De
3136 Synthesis of Functionalized L-Cysteine and L-Methionine by Reaction with Electron-Deficient Acetylenes B A Trofimov A G Malrsquokina O A Shemyakina V V Nosyreva A P Borisova S S Khutsishvili L B Krivdin
3143 A lsquoClickrsquo Approach to the Synthesis of 3-[2-(1-Alkyltriazol-4-yl)ethyl]indoles M Petrini R R Shaikh
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
2283 Ruthenium-Catalyzed Addition of Primary Amides to Alkynes A Stereoselective Synthesis of Secondary Enamides L J Gooszligen M Blanchot K S M Salih K Gooszligen
2289 Binaphthyl-Modified Quaternary Phosphonium Salts as Chiral Phase Transfer Catalysts Application to Asymmetric Amination of β-Keto Esters R He K Maruoka
X Table of Contents XI Forthcoming Articles
no 14 2293 Direct Methods for Stereoselective Polypropionate Synthesis A Survey
J Li D Menche 2316 Synthesis of Symmetrical Ketones from Grignard Reagents and
11-Carbonyldiimidazole D Bottalico V Fiandanese G Marchese A Punzi
2319 Synthesis of 45-Substituted Imidazoles by a Fast Condensation of 12-Diketones and Urotropine in Heterogeneous Medium G Bratulescu
2321 (Arylsulfonyl)acetones and -acetonitriles New Activated Methylenic Building Blocks for Synthesis of 123-Triazoles N T Pokhodylo V S Matiychuk M D Obushak
2324 A Safe Convenient and Efficient One-Pot Synthesis of α-Chloroketone Acetals Directly from Ketones Using Iodobenzene Dichloride J Yu C Zhang
2329 An Efficient Oxidative Conversion of Aldehydes into 2-Substituted 2-Oxazolines Using 13-Diiodo-55-dimethylhydantoin S Takahashi H Togo
2333 A Novel Procedure for the Synthesis of Benzo[b][18]naphthyridine-3-carboxylate Derivatives from MoritandashBaylisndashHillman Adduct Acetates W Zhong F Lin R Chen W Su
2341 An Improved Synthesis of 147-Triazacyclononanes (tacns) and 14710-Tetraazacyclododecanes (cyclens) J Huang Z Zhou T H Chan
2345 The Ullmann Coupling between 2-Chlorobenzoic Acids and Amino Acids A Valuable Reaction for Preparing 2-Substituted 1-Acetyl-1H-indol-3-yl Acetates J C Rodriguez Dominguez X Gang G Kirsch
2349 gem-Dibromomethyl Aromatics Efficient Aldehyde Equivalents in the KnoevenagelndashDoebner Reaction J K Augustine Y A Naik S Poojari N Chowdappa B S Sherigara K Areppa
2357 Synthesis of Novel α-Aminophosphonates Containing Adamantyl Fragment M M Kabachnik L I Minaeva I P Beletskaya
2361 Efficient Fluoride-Mediated Synthesis of 5-Amino-Substituted Isothiazoles Y S Zubenko V I Potkin
2365 Phosphine-Catalyzed Reaction of Cyanohydrins with Activated Alkynes A Siby O Loreau F Taran
2371 Sulfanyl-Substituted [3]Cumulenes and Buta-13-dienes from a Tetrakis(pyridinium)-Substituted Butadiene A Schmidt A Rahimi M Gjikaj
2379 Efficient Synthesis of 2-Substituted Pyrido[32-d]pyrimidines Involving SNAr and Palladium-Catalyzed Cross-Coupling Reactions A Tikad S Routier M Akssira J-M Leacuteger C Jarry G Guillaumet
2385 Novel Synthesis of Medium-Sized Heterocycles by Palladium-Catalyzed Intramolecular Heck Reaction via 9-endo-trig Mode of Cyclization K C Majumdar B Chattopadhyay
2393 Facile Synthesis of Fluorinated Benzofuro- and Benzothieno[23-b]pyridines α-Carbolines and Nucleosides Containing the α-Carboline Framework V O Iaroshenko Y Wang B Zhang D Volochnyuk V Ya Sosnovskikh
2403 Synthesis of Functionalized N-Vinyl Nitrogen-Containing Heterocycles S M M Lopes A M Beja M Ramos Silva J A Paixatildeo F Palacios T M V D Pinho e Melo
2408 Kumada Cross-Coupling of Aryl Grignard Reagents with Aryl Halides Catalyzed by an Immobilized Nickel Catalyst X Chen L Wang J Liu
2413 Highly Enantioselective Synthesis of Heteroaromatic Alcohols Catalyzed by Chiral DiaminodiphosphinendashRuthenium(II) Complexes W-Y Shen Y-Y Li Z-R Dong J-X Gao
2418 Concise Total Synthesis of (+)-Disparlure and its trans-Isomer Using Asymmetric Organocatalysis S-G Kim
2423 Rhodium Carbenoid Induced [12]-Migration in an L-Lyxo-Configured α-Diazo β-Keto Ester Synthesis of a New Griseolic Acid Analogue N N Bhujbal K S A Kumar D D Dhavale
2430 Synthesis of 5-Arylthio-3-hydroxyphthalates by the First [4+2] Cycloadditions of 3-Arylthio-1-silyloxy-13-butadienes with Dimethyl Acetylenedicarboxylate I Iqbal M Imran P Langer
2435 Synthesis of Highly Functionalized Proline Derivatives via a One-Pot MichaelSN-AdditionCyclization Approach U Kazmaier C Schmidt
2440 RhodiumGraphite-Catalyzed Hydrogenation of Carbocyclic and Heterocyclic Aromatic Compounds G Falini A Gualandi D Savoia
2447 Potassium [1-(tert-Butoxycarbonyl)-1H-indol-2-yl]trifluoroborate as an Efficient Building Block in Palladium-Catalyzed SuzukindashMiyaura Cross Couplings P Kassis V Beacuteneacuteteau J-Y Meacuterour S Routier
2454 Syntheses of Substituted Furans and Pyrroles by Platinum-Catalyzed Cyclizations of Propargylic Oxiranes and Aziridines in Aqueous Media M Yoshida M Al-Amin K Shishido
2467 Transition-Metal-Free Oxidative Homocoupling of Aryl Alkenyl and Alkynyl Grignard Reagents with TEMPO M S Maji A Studer
XIII Forthcoming Articles
no 15 2471 Advances in Synthetic Approaches for the Preparation of Combretastatin-
Based Anti-Cancer Agents R Singh H Kaur 2492 Synthesis of Unsymmetrical Ureas by Sulfur-Assisted Carbonylation with
Carbon Monoxide and Oxidation with Molecular Oxygen under Mild Conditions T Mizuno T Nakai M Mihara
2497 Ring-OpeningRecyclization Reactions of (Dimethylamino)propenoyl-Substituted Cyclopropanes Facile Synthesis of Halogenated Pyridin-2(1H)-ones R Zhang Y Zhou Y Liang Z Jiang D Dong
2501 Facile and Efficient Total Synthesis of Taspine B Cheng S Zhang L Zhu J Zhang Q Li A Shan L He
2505 Oligomeric Iodosylbenzene Sulfate A Convenient Hypervalent Iodine Reagent for Oxidation of Organic Sulfides and Alkenes M S Yusubov R Y Yusubova T V Funk K-W Chi V V Zhdankin
2509 Pyrrolidine-Based Organocatalysts for Enantioselective Michael Addition of Cyclohexanone to trans-β-Nitrostyrene A P Carley S Dixon J D Kilburn
2517 CundashAl Hydrotalcite An Efficient and Reusable Ligand-Free Catalyst for the Coupling of Aryl Chlorides with Aliphatic Aromatic and N(H)-Heterocyclic Amines B Sreedhar R Arundhathi P L Reddy M A Reddy M L Kantam
2523 Highly Efficient Synthesis of trans-βγ-Unsaturated a-Keto Amides C Allais T Constantieux J Rodriguez
2531 Gas-Phase Synthesis of N-Unsubstituted 3-Hydroxypyrroles and 1H-Pyrrol-3(2H)-ones L Hill G A Hunter S H Imam H McNab W J OrsquoNeill
2535 3-Hydroxy-1H-pyrrole L Hill S H Imam H McNab W J OrsquoNeill 2539 123-Thiadiazoles with Unsaturated Side Chains Synthesis
Polymerization and Photocrosslinking M Al-Smadi N Hanold H Kalbitz H Meier
2547 Synthesis of 1112-Didehydrodibenzo[ae]cycloocten-5(6H)-one A Strained Eight-Membered Alkyne S C Kornmayer F Rominger R Gleiter
2553 Stannous Chloride Dihydrate A Novel and Efficient Catalyst for the Synthesis of gem-Dihydroperoxides from Ketones and Aldehydes D Azarifar K Khosravi F Soleimanei
2557 Synthesis of a Novel Class of Azacrown Macrocycles and Lariat Crown Ethers Containing Two 124-Triazole Rings as Subunits N Foroughifar A Mobinikhaledi S Ebrahimi
2561 Enantioselective Synthesis of the 3C-Protease Inhibitor (ndash)-Thysanone by a StauntonndashWeinreb Annulation Strategy J Sperry T Y Yuen M A Brimble
2570 Stereoselective Synthesis of Unnatural β-Amino Acids from Nitroethane via 56-Dihydro-4H-12-oxazin-3-ylacetates A Yu Sukhorukov A V Lesiv O L Eliseev Y A Khomutova S L Ioffe
2579 A Versatile Unexpected One-Pot Regioselective Synthesis of a New Class of 13-Diazepinoindolones by Reaction of Pyranoindolones with Monosubstituted Ureas D Livadiotou C A Tsoleridis J Stephanidou-Stephanatou
2584 Synthesis of a Trisaccharide and a Tetrasaccharide from the Cell-Wall Lipopolysaccharides of Azospirillum brasilense S17 S Pandey S Ghosh A K Misra
2591 Synthesis of Isoindoline Nitroxides by Electrocyclic Reactions T Kaacutelai J Jekı K Hideg
2596 Glycosylations of Tertiary Alcohols Synthesis of Fully Protected Disaccharides with Sterically Demanding Groups Attached to the Sugar Core A Holkenbrink J B Vicente D B Werz
2605 Copper-Catalyzed [13]-Dipolar Cycloaddition for the Synthesis of Macrocycles Containing Acyclic Aromatic and Steroidal Moieties G V Latyshev M S Baranom A V Kazantsev A D Averin N V Lukashev I P Beletskaya
2616 Aryl Ring Migration Reaction in the Synthesis of 24-Diaryl-4H-31-benzothiazines A V Butin F A Tsiunchik V T Abaev A V Gutnov D A Cheshkov
2627 Hydrogenation of β-N-Substituted and β-NN-Disubstituted Enamino Esters in the Presence of Iridium(I) Catalyst H Hebbache Z Hank C Bruneau J-L Renaud
2634 Stereoselective Olefination Reactions Promoted by Rieke Manganese J M Concelloacuten H Rodriacuteguez-Solla V del Amo P Diacuteaz
2646 Synthesis of Piperidinones through a Radical Cascade E Godineau Y Landais
2650 Asymmetric Organic Synthesis with Enzymes Edited by V Gotor I Alfonso E Garciacutea-Urdiales Reviewed by Steve Collier
XVII Forthcoming Articles
no 16 2651 Synthesis of Spirocyclic Ethers S Rosenberg R Leino 2674 Bimetallic PalladiumndashPlatinum-on-Carbon-Catalyzed HndashD Exchange
Reaction Synergistic Effect on Multiple Deuterium Incorporation T Maegawa N Ito K Oono Y Monguchi H Sajiki
2679 Efficient Copper-Catalyzed Synthesis of 2-Amino-4(3H)-quinazolinone and 2-Aminoquinazoline Derivatives X Huang H Yang H Fu R Qiao Y Zhao
2689 Synthesis and Chemoselective N- and O-Alkylation of Thiadiazolopyrimidine Nucleosides and Uridines A M L Hossion R Islam R K Kandahary T Nagamatsu
2697 Facile and Efficient Synthesis of a New Class of Indole-Substituted Pyridine Derivatives via One-Pot Multicomponent Reactions K Zhao X-P Xu S-L Zhu D-Q Shi Y Zhang S-J Ji
2709 Studies toward a Total Synthesis of Rhizoxin D Stereoselective Preparation of the C11ndashC19 Fragment S Padakanti C K Kumar E Ashok P Das
2715 A Short Synthesis of Enantiomeric Phytoprostanes B1 Type I W Perlikowska M Mikołajczyk
2719 Chemistry of Polyhalogenated Nitrobutadienes Part 7 A Novel Synthetic Access to Chlorinated Nitrile Oxides E Nutz V A Zapolrsquoskii D E Kaufmann
2725 Microwave-Assisted Silver(I)-Mediated Selective O-Alkylation of Aromatic Imidate Systems B K Singh C Cavalluzzo M De Maeyer Z Debyser V S Parmar E Van der Eycken
2729 Iodogen A Novel Reagent for the Oxidation of Urazoles under Heterogeneous Conditions A Khoramabadi A Shiri M A Zolfigol S Mallakpour
2733 An Unprecedented Synthesis of Eight-Membered-Ring Cyclic Thioimidic Esters by a Three-Component Reaction A Alizadeh R Hosseinpour
2737 A Novel Diastereoselective Synthesis of β-Phosphonato Unsaturated Thioimidates A Alizadeh N Zohreh
2741 Synthesis of 21-Benzisoxazoles by Nucleophilic Substitution of Hydrogen in Nitroarenes Activated by the Azole Ring N T Pokhodylo Y O Teslenko V S Matiychuk M D Obushak
2749 A Facile Synthesis of Two Series of Multifunctional Carbon Compounds from αα-Dihalo Ketones Using Allylsamarium Bromide X Liu S Zhang J Di
2756 Stereocontrolled Formation of Protected Aminodeoxyalditols from Simple Carbohydrate Precursors by Debenzylating Cycloetherification Y Jiang Z Fang Q Zheng H Jia J Cheng B Zheng
2761 trans-Stilbene as a Starting Material for the Synthesis of Tamoxifen Based on Palladium-Catalyzed Cross-Coupling Reactions C M Nunes J Limberger S Poersch M Seferin A L Monteiro
2766 Synthesis and Biological Evaluation of 6-Substituted Purinylcarbanucleosides with a Cyclopenta[b]thiophene Pseudosugar P Abeijoacuten J M Blanco O Caamantildeo F Fernaacutendez M D Garciacutea X Garciacutea-Mera J E Rodriacuteguez-Borges J Balzarini E De Clercq
2773 Synthesis and Electrochemical Signature of Novel Norbornyl-ferrocene Hybrids F A Khan S K Upadhyay
2778 A Regioselective TsujindashTrost Pentadienylation of 3-Allyltetronic Acid R Schobert B Barnickel
2785 Copper(I)-Catalyzed CarylndashCalkynyl Bond Formation of Aryl Iodides with Terminal Alkynes K G Thakur G Sekar
2790 Aminolysis of Epoxides Using Iridium Trichloride as an Efficient Catalyst J Agarwal A Duley R Rani R K Peddinti
2797 Preparation of Several Active N-Chloro Compounds from Trichloroisocyanuric Acid A Shiri A Khoramabadi-zad
2802 The First Mineral-Catalyzed One-Pot [3+1+2] Coupling Protocol for Multifunctionalized Fused-Ring Pyrimidines L D S Yadav A Rai
2809 Efficient Synthesis of Tetrahydro-β-carbolin-1-one and Dihydroisoquinolin-1-one Derivatives as Versatile Intermediates K E Judd M F Mahon L Caggiano
2818 A Concise Synthesis of ortho-Iodobenzyl Alcohols via Addition of ortho-Iodophenyl Grignard Reagent to Aldehydes and Ketones J Cvengroš D Stolz A Togni
XIII Forthcoming Articles
no 17 2825 Reactivity of Oxazol-5-(4H)-ones and Their Application toward Natural
Product Synthesis N M Hewlett C D Hupp J J Tepe 2840 Towards the Total Synthesis of 3-Hydroxyvibsanin E B D Schwartz
J R Denton P V Bernhardt H M L Davies C M Williams 2847 Structure Investigations of (ent)-Cladospolide D by De Novo Synthesis and
Kinetic and Thermodynamic Isomerization Y Xing J H Penn G A OrsquoDoherty
2855 New Applications of PhI(OAc)2 in Synthesis Total Synthesis and SAR Development of Potent Antitumor Natural Product PsymberinIrciniastatin A N Shao X Huang A Palani R Aslanian A Buevich J Piwinski R Huryk C Seidel-Dugan
2873 Total Synthesis of Largazole ndash Devolution of a Novel Synthetic Strategy B Wang C J Forsyth
2881 Formal Total Synthesis of Palmerolide A J Jaumlgel M E Maier 2893 Total Synthesis of Bongkrekic Acid via Sequential SuzukindashMiyaura Coupling
Reactions M Kanematsu M Shindo M Yoshida K Shishido 2905 Stereodivergent Approach to Both C28a-syn and C28a-anti Relative
Stereochemical Manifolds in the Lepadin Family via a TiCl4-Promoted G Li L J Carlson I K Sagamanova B W Slafer R P Hsung C Gilardi H M Sklenicka N Sydorenko
2915 Enantioselective Aldol Reaction of Tetrasubstituted Ketene Silyl Acetals with Achiral Aldehydes for the Construction of Asymmetric Tertiary Alcohols An Application for the Divergent Total Syntheses of Buergerinins F and G I Shiina T Iizumi Y-s Yamai Y-i Kawakita K Yokoyama Y-k Yamada
2927 Second-Generation Biomimetic Total Synthesis of Chaetominine A Coste G Karthikeyan F Couty G Evano
2935 Total Synthesis of (+)-Fostriecin and (+)-Phoslactomycin B S Shibahara M Fujino Y Tashiro N Okamoto T Esumi K Takahashi J Ishihara S Hatakeyama
2954 Stereochemical Assignments of the Chlorinated Residues in Victorin C A C Durow C Butts C L Willis
2963 Studies of the Asymmetric Total Synthesis of Clavilactone D by the lsquoLariatrsquo Cyclization Strategy T Yoshimitsu S Nojima M Hashimoto K Tsukamoto T Tanaka
2970 Total Synthesis of the Leucetta-Derived Alkaloid Calcaridine A P B Koswatta R Sivappa H V R Dias C J Lovely
2983 Formal Synthesis of Salinosporamide A Starting from D-Glucose T Momose Y Kaiya J-i Hasegawa T Sato N Chida
2992 Synthesis of Bioactive Natural Products by Asymmetric syn- and anti-Aldol Reactions A K Ghosh Z L Dawson
no 18 3003 Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural
Products B M Trost M K Brennan 3026 One-Pot Synthesis of Furo[34-b]pyridin-5(7H)-ones from 2-
Bromopyridine-3-carboxylic Acid and Carbonyl Compounds K Kobayashi T Kozuki H Konishi
3029 Iodocyclization of N-[2-(Methylthio)phenyl]propiolamides Selective Synthesis of 3-Iodo-15-benzothiazepin-4-ones T-S Jiang X-G Zhang J-H Li
3039 A Facile Synthetic Method for Fluorine-Containing 17-Phenanthrolines Pyridine-Ring Formation Reaction of N-Propargyl-68-bis(trifluoroacetyl)-quinolin-5-amine with Various Nucleophiles D Shibata E Okada M Hinoshita M Meacutedebielle
3047 Enantiotopic Discrimination in Palladium-Mediated Nucleophilic Substitutions on Achiral Substrates Chiral Ligand versus Chiral Nucleophile O Jacquet F Charnay J-C Fiaud J Ollivier
3051 Studies on the Chemistry of 2-[3-(2-Nitrophenyl)-2-oxopropyl]benzaldehydes Novel Syntheses of 5H-Benzo[b]carbazole-611-diones and Indolo[12-b]isoquinoline-611-diones M Fernaacutendez
3061 Studies on the C22ndashC23 Aldol Coupling of Spirangien M Lorenz N Bluhm M Kalesse
3067 One-Pot Synthesis of N-Alkyl Purine Pyrimidine and Azole Derivatives from Alcohols using Ph3PCCl4 A Rapid Route to Carboacyclic Nucleoside Synthesis M N Soltani Rad A Khalafi-Nezhad S Behrouz Z Asrari M Behrouz Z Amini
3077 Synthesis of 2-Amino-34-dihydroquinazolines and Imidazo[21-b]quinazoline-2-ones A Mishra S Batra
3089 Studies on the Reaction of Diimines with Thiourea Synthesis and Solvent-Induced cistrans-Isomerization of 135-Triazinane-2-thiones B Kaboudin T Ghasemi T Yokomatsu
3094 Suzuki Coupling of Heteroaromatic Chlorides Using Highly Electron-Donating ClickPhos Ligands S M Spinella Z-H Guan J Chen X Zhang
3099 Reaction of NN-Dioxyenamines with Anhydrides of Carboxylic and Sulfonic Acids A New Method for the Synthesis of a-Hydroxyoxime Derivatives A A Tabolin A V Lesiv S L Ioffe
3106 Directed ortho Metallation Chemistry and Phosphine Synthesis New Ligands for the SuzukindashMiyaura Reaction D B G Williams S J Evans H de Bod M S Mokhadinyana T Hughes
3113 New Functional Derivatives of 9-Phenylquinine P J Boratyński J SkarŜewski
3120 On the Synthesis of Asymmetric and Dissymmetric Amino Analogues of Troumlgerrsquos Base J Artacho K Waumlrnmark
3127 Synthesis of Polycyclic Sultams by Palladium-Catalyzed Intramolecular Cyclization K C Majumdar S Mondal N De
3136 Synthesis of Functionalized L-Cysteine and L-Methionine by Reaction with Electron-Deficient Acetylenes B A Trofimov A G Malrsquokina O A Shemyakina V V Nosyreva A P Borisova S S Khutsishvili L B Krivdin
3143 A lsquoClickrsquo Approach to the Synthesis of 3-[2-(1-Alkyltriazol-4-yl)ethyl]indoles M Petrini R R Shaikh
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
no 14 2293 Direct Methods for Stereoselective Polypropionate Synthesis A Survey
J Li D Menche 2316 Synthesis of Symmetrical Ketones from Grignard Reagents and
11-Carbonyldiimidazole D Bottalico V Fiandanese G Marchese A Punzi
2319 Synthesis of 45-Substituted Imidazoles by a Fast Condensation of 12-Diketones and Urotropine in Heterogeneous Medium G Bratulescu
2321 (Arylsulfonyl)acetones and -acetonitriles New Activated Methylenic Building Blocks for Synthesis of 123-Triazoles N T Pokhodylo V S Matiychuk M D Obushak
2324 A Safe Convenient and Efficient One-Pot Synthesis of α-Chloroketone Acetals Directly from Ketones Using Iodobenzene Dichloride J Yu C Zhang
2329 An Efficient Oxidative Conversion of Aldehydes into 2-Substituted 2-Oxazolines Using 13-Diiodo-55-dimethylhydantoin S Takahashi H Togo
2333 A Novel Procedure for the Synthesis of Benzo[b][18]naphthyridine-3-carboxylate Derivatives from MoritandashBaylisndashHillman Adduct Acetates W Zhong F Lin R Chen W Su
2341 An Improved Synthesis of 147-Triazacyclononanes (tacns) and 14710-Tetraazacyclododecanes (cyclens) J Huang Z Zhou T H Chan
2345 The Ullmann Coupling between 2-Chlorobenzoic Acids and Amino Acids A Valuable Reaction for Preparing 2-Substituted 1-Acetyl-1H-indol-3-yl Acetates J C Rodriguez Dominguez X Gang G Kirsch
2349 gem-Dibromomethyl Aromatics Efficient Aldehyde Equivalents in the KnoevenagelndashDoebner Reaction J K Augustine Y A Naik S Poojari N Chowdappa B S Sherigara K Areppa
2357 Synthesis of Novel α-Aminophosphonates Containing Adamantyl Fragment M M Kabachnik L I Minaeva I P Beletskaya
2361 Efficient Fluoride-Mediated Synthesis of 5-Amino-Substituted Isothiazoles Y S Zubenko V I Potkin
2365 Phosphine-Catalyzed Reaction of Cyanohydrins with Activated Alkynes A Siby O Loreau F Taran
2371 Sulfanyl-Substituted [3]Cumulenes and Buta-13-dienes from a Tetrakis(pyridinium)-Substituted Butadiene A Schmidt A Rahimi M Gjikaj
2379 Efficient Synthesis of 2-Substituted Pyrido[32-d]pyrimidines Involving SNAr and Palladium-Catalyzed Cross-Coupling Reactions A Tikad S Routier M Akssira J-M Leacuteger C Jarry G Guillaumet
2385 Novel Synthesis of Medium-Sized Heterocycles by Palladium-Catalyzed Intramolecular Heck Reaction via 9-endo-trig Mode of Cyclization K C Majumdar B Chattopadhyay
2393 Facile Synthesis of Fluorinated Benzofuro- and Benzothieno[23-b]pyridines α-Carbolines and Nucleosides Containing the α-Carboline Framework V O Iaroshenko Y Wang B Zhang D Volochnyuk V Ya Sosnovskikh
2403 Synthesis of Functionalized N-Vinyl Nitrogen-Containing Heterocycles S M M Lopes A M Beja M Ramos Silva J A Paixatildeo F Palacios T M V D Pinho e Melo
2408 Kumada Cross-Coupling of Aryl Grignard Reagents with Aryl Halides Catalyzed by an Immobilized Nickel Catalyst X Chen L Wang J Liu
2413 Highly Enantioselective Synthesis of Heteroaromatic Alcohols Catalyzed by Chiral DiaminodiphosphinendashRuthenium(II) Complexes W-Y Shen Y-Y Li Z-R Dong J-X Gao
2418 Concise Total Synthesis of (+)-Disparlure and its trans-Isomer Using Asymmetric Organocatalysis S-G Kim
2423 Rhodium Carbenoid Induced [12]-Migration in an L-Lyxo-Configured α-Diazo β-Keto Ester Synthesis of a New Griseolic Acid Analogue N N Bhujbal K S A Kumar D D Dhavale
2430 Synthesis of 5-Arylthio-3-hydroxyphthalates by the First [4+2] Cycloadditions of 3-Arylthio-1-silyloxy-13-butadienes with Dimethyl Acetylenedicarboxylate I Iqbal M Imran P Langer
2435 Synthesis of Highly Functionalized Proline Derivatives via a One-Pot MichaelSN-AdditionCyclization Approach U Kazmaier C Schmidt
2440 RhodiumGraphite-Catalyzed Hydrogenation of Carbocyclic and Heterocyclic Aromatic Compounds G Falini A Gualandi D Savoia
2447 Potassium [1-(tert-Butoxycarbonyl)-1H-indol-2-yl]trifluoroborate as an Efficient Building Block in Palladium-Catalyzed SuzukindashMiyaura Cross Couplings P Kassis V Beacuteneacuteteau J-Y Meacuterour S Routier
2454 Syntheses of Substituted Furans and Pyrroles by Platinum-Catalyzed Cyclizations of Propargylic Oxiranes and Aziridines in Aqueous Media M Yoshida M Al-Amin K Shishido
2467 Transition-Metal-Free Oxidative Homocoupling of Aryl Alkenyl and Alkynyl Grignard Reagents with TEMPO M S Maji A Studer
XIII Forthcoming Articles
no 15 2471 Advances in Synthetic Approaches for the Preparation of Combretastatin-
Based Anti-Cancer Agents R Singh H Kaur 2492 Synthesis of Unsymmetrical Ureas by Sulfur-Assisted Carbonylation with
Carbon Monoxide and Oxidation with Molecular Oxygen under Mild Conditions T Mizuno T Nakai M Mihara
2497 Ring-OpeningRecyclization Reactions of (Dimethylamino)propenoyl-Substituted Cyclopropanes Facile Synthesis of Halogenated Pyridin-2(1H)-ones R Zhang Y Zhou Y Liang Z Jiang D Dong
2501 Facile and Efficient Total Synthesis of Taspine B Cheng S Zhang L Zhu J Zhang Q Li A Shan L He
2505 Oligomeric Iodosylbenzene Sulfate A Convenient Hypervalent Iodine Reagent for Oxidation of Organic Sulfides and Alkenes M S Yusubov R Y Yusubova T V Funk K-W Chi V V Zhdankin
2509 Pyrrolidine-Based Organocatalysts for Enantioselective Michael Addition of Cyclohexanone to trans-β-Nitrostyrene A P Carley S Dixon J D Kilburn
2517 CundashAl Hydrotalcite An Efficient and Reusable Ligand-Free Catalyst for the Coupling of Aryl Chlorides with Aliphatic Aromatic and N(H)-Heterocyclic Amines B Sreedhar R Arundhathi P L Reddy M A Reddy M L Kantam
2523 Highly Efficient Synthesis of trans-βγ-Unsaturated a-Keto Amides C Allais T Constantieux J Rodriguez
2531 Gas-Phase Synthesis of N-Unsubstituted 3-Hydroxypyrroles and 1H-Pyrrol-3(2H)-ones L Hill G A Hunter S H Imam H McNab W J OrsquoNeill
2535 3-Hydroxy-1H-pyrrole L Hill S H Imam H McNab W J OrsquoNeill 2539 123-Thiadiazoles with Unsaturated Side Chains Synthesis
Polymerization and Photocrosslinking M Al-Smadi N Hanold H Kalbitz H Meier
2547 Synthesis of 1112-Didehydrodibenzo[ae]cycloocten-5(6H)-one A Strained Eight-Membered Alkyne S C Kornmayer F Rominger R Gleiter
2553 Stannous Chloride Dihydrate A Novel and Efficient Catalyst for the Synthesis of gem-Dihydroperoxides from Ketones and Aldehydes D Azarifar K Khosravi F Soleimanei
2557 Synthesis of a Novel Class of Azacrown Macrocycles and Lariat Crown Ethers Containing Two 124-Triazole Rings as Subunits N Foroughifar A Mobinikhaledi S Ebrahimi
2561 Enantioselective Synthesis of the 3C-Protease Inhibitor (ndash)-Thysanone by a StauntonndashWeinreb Annulation Strategy J Sperry T Y Yuen M A Brimble
2570 Stereoselective Synthesis of Unnatural β-Amino Acids from Nitroethane via 56-Dihydro-4H-12-oxazin-3-ylacetates A Yu Sukhorukov A V Lesiv O L Eliseev Y A Khomutova S L Ioffe
2579 A Versatile Unexpected One-Pot Regioselective Synthesis of a New Class of 13-Diazepinoindolones by Reaction of Pyranoindolones with Monosubstituted Ureas D Livadiotou C A Tsoleridis J Stephanidou-Stephanatou
2584 Synthesis of a Trisaccharide and a Tetrasaccharide from the Cell-Wall Lipopolysaccharides of Azospirillum brasilense S17 S Pandey S Ghosh A K Misra
2591 Synthesis of Isoindoline Nitroxides by Electrocyclic Reactions T Kaacutelai J Jekı K Hideg
2596 Glycosylations of Tertiary Alcohols Synthesis of Fully Protected Disaccharides with Sterically Demanding Groups Attached to the Sugar Core A Holkenbrink J B Vicente D B Werz
2605 Copper-Catalyzed [13]-Dipolar Cycloaddition for the Synthesis of Macrocycles Containing Acyclic Aromatic and Steroidal Moieties G V Latyshev M S Baranom A V Kazantsev A D Averin N V Lukashev I P Beletskaya
2616 Aryl Ring Migration Reaction in the Synthesis of 24-Diaryl-4H-31-benzothiazines A V Butin F A Tsiunchik V T Abaev A V Gutnov D A Cheshkov
2627 Hydrogenation of β-N-Substituted and β-NN-Disubstituted Enamino Esters in the Presence of Iridium(I) Catalyst H Hebbache Z Hank C Bruneau J-L Renaud
2634 Stereoselective Olefination Reactions Promoted by Rieke Manganese J M Concelloacuten H Rodriacuteguez-Solla V del Amo P Diacuteaz
2646 Synthesis of Piperidinones through a Radical Cascade E Godineau Y Landais
2650 Asymmetric Organic Synthesis with Enzymes Edited by V Gotor I Alfonso E Garciacutea-Urdiales Reviewed by Steve Collier
XVII Forthcoming Articles
no 16 2651 Synthesis of Spirocyclic Ethers S Rosenberg R Leino 2674 Bimetallic PalladiumndashPlatinum-on-Carbon-Catalyzed HndashD Exchange
Reaction Synergistic Effect on Multiple Deuterium Incorporation T Maegawa N Ito K Oono Y Monguchi H Sajiki
2679 Efficient Copper-Catalyzed Synthesis of 2-Amino-4(3H)-quinazolinone and 2-Aminoquinazoline Derivatives X Huang H Yang H Fu R Qiao Y Zhao
2689 Synthesis and Chemoselective N- and O-Alkylation of Thiadiazolopyrimidine Nucleosides and Uridines A M L Hossion R Islam R K Kandahary T Nagamatsu
2697 Facile and Efficient Synthesis of a New Class of Indole-Substituted Pyridine Derivatives via One-Pot Multicomponent Reactions K Zhao X-P Xu S-L Zhu D-Q Shi Y Zhang S-J Ji
2709 Studies toward a Total Synthesis of Rhizoxin D Stereoselective Preparation of the C11ndashC19 Fragment S Padakanti C K Kumar E Ashok P Das
2715 A Short Synthesis of Enantiomeric Phytoprostanes B1 Type I W Perlikowska M Mikołajczyk
2719 Chemistry of Polyhalogenated Nitrobutadienes Part 7 A Novel Synthetic Access to Chlorinated Nitrile Oxides E Nutz V A Zapolrsquoskii D E Kaufmann
2725 Microwave-Assisted Silver(I)-Mediated Selective O-Alkylation of Aromatic Imidate Systems B K Singh C Cavalluzzo M De Maeyer Z Debyser V S Parmar E Van der Eycken
2729 Iodogen A Novel Reagent for the Oxidation of Urazoles under Heterogeneous Conditions A Khoramabadi A Shiri M A Zolfigol S Mallakpour
2733 An Unprecedented Synthesis of Eight-Membered-Ring Cyclic Thioimidic Esters by a Three-Component Reaction A Alizadeh R Hosseinpour
2737 A Novel Diastereoselective Synthesis of β-Phosphonato Unsaturated Thioimidates A Alizadeh N Zohreh
2741 Synthesis of 21-Benzisoxazoles by Nucleophilic Substitution of Hydrogen in Nitroarenes Activated by the Azole Ring N T Pokhodylo Y O Teslenko V S Matiychuk M D Obushak
2749 A Facile Synthesis of Two Series of Multifunctional Carbon Compounds from αα-Dihalo Ketones Using Allylsamarium Bromide X Liu S Zhang J Di
2756 Stereocontrolled Formation of Protected Aminodeoxyalditols from Simple Carbohydrate Precursors by Debenzylating Cycloetherification Y Jiang Z Fang Q Zheng H Jia J Cheng B Zheng
2761 trans-Stilbene as a Starting Material for the Synthesis of Tamoxifen Based on Palladium-Catalyzed Cross-Coupling Reactions C M Nunes J Limberger S Poersch M Seferin A L Monteiro
2766 Synthesis and Biological Evaluation of 6-Substituted Purinylcarbanucleosides with a Cyclopenta[b]thiophene Pseudosugar P Abeijoacuten J M Blanco O Caamantildeo F Fernaacutendez M D Garciacutea X Garciacutea-Mera J E Rodriacuteguez-Borges J Balzarini E De Clercq
2773 Synthesis and Electrochemical Signature of Novel Norbornyl-ferrocene Hybrids F A Khan S K Upadhyay
2778 A Regioselective TsujindashTrost Pentadienylation of 3-Allyltetronic Acid R Schobert B Barnickel
2785 Copper(I)-Catalyzed CarylndashCalkynyl Bond Formation of Aryl Iodides with Terminal Alkynes K G Thakur G Sekar
2790 Aminolysis of Epoxides Using Iridium Trichloride as an Efficient Catalyst J Agarwal A Duley R Rani R K Peddinti
2797 Preparation of Several Active N-Chloro Compounds from Trichloroisocyanuric Acid A Shiri A Khoramabadi-zad
2802 The First Mineral-Catalyzed One-Pot [3+1+2] Coupling Protocol for Multifunctionalized Fused-Ring Pyrimidines L D S Yadav A Rai
2809 Efficient Synthesis of Tetrahydro-β-carbolin-1-one and Dihydroisoquinolin-1-one Derivatives as Versatile Intermediates K E Judd M F Mahon L Caggiano
2818 A Concise Synthesis of ortho-Iodobenzyl Alcohols via Addition of ortho-Iodophenyl Grignard Reagent to Aldehydes and Ketones J Cvengroš D Stolz A Togni
XIII Forthcoming Articles
no 17 2825 Reactivity of Oxazol-5-(4H)-ones and Their Application toward Natural
Product Synthesis N M Hewlett C D Hupp J J Tepe 2840 Towards the Total Synthesis of 3-Hydroxyvibsanin E B D Schwartz
J R Denton P V Bernhardt H M L Davies C M Williams 2847 Structure Investigations of (ent)-Cladospolide D by De Novo Synthesis and
Kinetic and Thermodynamic Isomerization Y Xing J H Penn G A OrsquoDoherty
2855 New Applications of PhI(OAc)2 in Synthesis Total Synthesis and SAR Development of Potent Antitumor Natural Product PsymberinIrciniastatin A N Shao X Huang A Palani R Aslanian A Buevich J Piwinski R Huryk C Seidel-Dugan
2873 Total Synthesis of Largazole ndash Devolution of a Novel Synthetic Strategy B Wang C J Forsyth
2881 Formal Total Synthesis of Palmerolide A J Jaumlgel M E Maier 2893 Total Synthesis of Bongkrekic Acid via Sequential SuzukindashMiyaura Coupling
Reactions M Kanematsu M Shindo M Yoshida K Shishido 2905 Stereodivergent Approach to Both C28a-syn and C28a-anti Relative
Stereochemical Manifolds in the Lepadin Family via a TiCl4-Promoted G Li L J Carlson I K Sagamanova B W Slafer R P Hsung C Gilardi H M Sklenicka N Sydorenko
2915 Enantioselective Aldol Reaction of Tetrasubstituted Ketene Silyl Acetals with Achiral Aldehydes for the Construction of Asymmetric Tertiary Alcohols An Application for the Divergent Total Syntheses of Buergerinins F and G I Shiina T Iizumi Y-s Yamai Y-i Kawakita K Yokoyama Y-k Yamada
2927 Second-Generation Biomimetic Total Synthesis of Chaetominine A Coste G Karthikeyan F Couty G Evano
2935 Total Synthesis of (+)-Fostriecin and (+)-Phoslactomycin B S Shibahara M Fujino Y Tashiro N Okamoto T Esumi K Takahashi J Ishihara S Hatakeyama
2954 Stereochemical Assignments of the Chlorinated Residues in Victorin C A C Durow C Butts C L Willis
2963 Studies of the Asymmetric Total Synthesis of Clavilactone D by the lsquoLariatrsquo Cyclization Strategy T Yoshimitsu S Nojima M Hashimoto K Tsukamoto T Tanaka
2970 Total Synthesis of the Leucetta-Derived Alkaloid Calcaridine A P B Koswatta R Sivappa H V R Dias C J Lovely
2983 Formal Synthesis of Salinosporamide A Starting from D-Glucose T Momose Y Kaiya J-i Hasegawa T Sato N Chida
2992 Synthesis of Bioactive Natural Products by Asymmetric syn- and anti-Aldol Reactions A K Ghosh Z L Dawson
no 18 3003 Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural
Products B M Trost M K Brennan 3026 One-Pot Synthesis of Furo[34-b]pyridin-5(7H)-ones from 2-
Bromopyridine-3-carboxylic Acid and Carbonyl Compounds K Kobayashi T Kozuki H Konishi
3029 Iodocyclization of N-[2-(Methylthio)phenyl]propiolamides Selective Synthesis of 3-Iodo-15-benzothiazepin-4-ones T-S Jiang X-G Zhang J-H Li
3039 A Facile Synthetic Method for Fluorine-Containing 17-Phenanthrolines Pyridine-Ring Formation Reaction of N-Propargyl-68-bis(trifluoroacetyl)-quinolin-5-amine with Various Nucleophiles D Shibata E Okada M Hinoshita M Meacutedebielle
3047 Enantiotopic Discrimination in Palladium-Mediated Nucleophilic Substitutions on Achiral Substrates Chiral Ligand versus Chiral Nucleophile O Jacquet F Charnay J-C Fiaud J Ollivier
3051 Studies on the Chemistry of 2-[3-(2-Nitrophenyl)-2-oxopropyl]benzaldehydes Novel Syntheses of 5H-Benzo[b]carbazole-611-diones and Indolo[12-b]isoquinoline-611-diones M Fernaacutendez
3061 Studies on the C22ndashC23 Aldol Coupling of Spirangien M Lorenz N Bluhm M Kalesse
3067 One-Pot Synthesis of N-Alkyl Purine Pyrimidine and Azole Derivatives from Alcohols using Ph3PCCl4 A Rapid Route to Carboacyclic Nucleoside Synthesis M N Soltani Rad A Khalafi-Nezhad S Behrouz Z Asrari M Behrouz Z Amini
3077 Synthesis of 2-Amino-34-dihydroquinazolines and Imidazo[21-b]quinazoline-2-ones A Mishra S Batra
3089 Studies on the Reaction of Diimines with Thiourea Synthesis and Solvent-Induced cistrans-Isomerization of 135-Triazinane-2-thiones B Kaboudin T Ghasemi T Yokomatsu
3094 Suzuki Coupling of Heteroaromatic Chlorides Using Highly Electron-Donating ClickPhos Ligands S M Spinella Z-H Guan J Chen X Zhang
3099 Reaction of NN-Dioxyenamines with Anhydrides of Carboxylic and Sulfonic Acids A New Method for the Synthesis of a-Hydroxyoxime Derivatives A A Tabolin A V Lesiv S L Ioffe
3106 Directed ortho Metallation Chemistry and Phosphine Synthesis New Ligands for the SuzukindashMiyaura Reaction D B G Williams S J Evans H de Bod M S Mokhadinyana T Hughes
3113 New Functional Derivatives of 9-Phenylquinine P J Boratyński J SkarŜewski
3120 On the Synthesis of Asymmetric and Dissymmetric Amino Analogues of Troumlgerrsquos Base J Artacho K Waumlrnmark
3127 Synthesis of Polycyclic Sultams by Palladium-Catalyzed Intramolecular Cyclization K C Majumdar S Mondal N De
3136 Synthesis of Functionalized L-Cysteine and L-Methionine by Reaction with Electron-Deficient Acetylenes B A Trofimov A G Malrsquokina O A Shemyakina V V Nosyreva A P Borisova S S Khutsishvili L B Krivdin
3143 A lsquoClickrsquo Approach to the Synthesis of 3-[2-(1-Alkyltriazol-4-yl)ethyl]indoles M Petrini R R Shaikh
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
2408 Kumada Cross-Coupling of Aryl Grignard Reagents with Aryl Halides Catalyzed by an Immobilized Nickel Catalyst X Chen L Wang J Liu
2413 Highly Enantioselective Synthesis of Heteroaromatic Alcohols Catalyzed by Chiral DiaminodiphosphinendashRuthenium(II) Complexes W-Y Shen Y-Y Li Z-R Dong J-X Gao
2418 Concise Total Synthesis of (+)-Disparlure and its trans-Isomer Using Asymmetric Organocatalysis S-G Kim
2423 Rhodium Carbenoid Induced [12]-Migration in an L-Lyxo-Configured α-Diazo β-Keto Ester Synthesis of a New Griseolic Acid Analogue N N Bhujbal K S A Kumar D D Dhavale
2430 Synthesis of 5-Arylthio-3-hydroxyphthalates by the First [4+2] Cycloadditions of 3-Arylthio-1-silyloxy-13-butadienes with Dimethyl Acetylenedicarboxylate I Iqbal M Imran P Langer
2435 Synthesis of Highly Functionalized Proline Derivatives via a One-Pot MichaelSN-AdditionCyclization Approach U Kazmaier C Schmidt
2440 RhodiumGraphite-Catalyzed Hydrogenation of Carbocyclic and Heterocyclic Aromatic Compounds G Falini A Gualandi D Savoia
2447 Potassium [1-(tert-Butoxycarbonyl)-1H-indol-2-yl]trifluoroborate as an Efficient Building Block in Palladium-Catalyzed SuzukindashMiyaura Cross Couplings P Kassis V Beacuteneacuteteau J-Y Meacuterour S Routier
2454 Syntheses of Substituted Furans and Pyrroles by Platinum-Catalyzed Cyclizations of Propargylic Oxiranes and Aziridines in Aqueous Media M Yoshida M Al-Amin K Shishido
2467 Transition-Metal-Free Oxidative Homocoupling of Aryl Alkenyl and Alkynyl Grignard Reagents with TEMPO M S Maji A Studer
XIII Forthcoming Articles
no 15 2471 Advances in Synthetic Approaches for the Preparation of Combretastatin-
Based Anti-Cancer Agents R Singh H Kaur 2492 Synthesis of Unsymmetrical Ureas by Sulfur-Assisted Carbonylation with
Carbon Monoxide and Oxidation with Molecular Oxygen under Mild Conditions T Mizuno T Nakai M Mihara
2497 Ring-OpeningRecyclization Reactions of (Dimethylamino)propenoyl-Substituted Cyclopropanes Facile Synthesis of Halogenated Pyridin-2(1H)-ones R Zhang Y Zhou Y Liang Z Jiang D Dong
2501 Facile and Efficient Total Synthesis of Taspine B Cheng S Zhang L Zhu J Zhang Q Li A Shan L He
2505 Oligomeric Iodosylbenzene Sulfate A Convenient Hypervalent Iodine Reagent for Oxidation of Organic Sulfides and Alkenes M S Yusubov R Y Yusubova T V Funk K-W Chi V V Zhdankin
2509 Pyrrolidine-Based Organocatalysts for Enantioselective Michael Addition of Cyclohexanone to trans-β-Nitrostyrene A P Carley S Dixon J D Kilburn
2517 CundashAl Hydrotalcite An Efficient and Reusable Ligand-Free Catalyst for the Coupling of Aryl Chlorides with Aliphatic Aromatic and N(H)-Heterocyclic Amines B Sreedhar R Arundhathi P L Reddy M A Reddy M L Kantam
2523 Highly Efficient Synthesis of trans-βγ-Unsaturated a-Keto Amides C Allais T Constantieux J Rodriguez
2531 Gas-Phase Synthesis of N-Unsubstituted 3-Hydroxypyrroles and 1H-Pyrrol-3(2H)-ones L Hill G A Hunter S H Imam H McNab W J OrsquoNeill
2535 3-Hydroxy-1H-pyrrole L Hill S H Imam H McNab W J OrsquoNeill 2539 123-Thiadiazoles with Unsaturated Side Chains Synthesis
Polymerization and Photocrosslinking M Al-Smadi N Hanold H Kalbitz H Meier
2547 Synthesis of 1112-Didehydrodibenzo[ae]cycloocten-5(6H)-one A Strained Eight-Membered Alkyne S C Kornmayer F Rominger R Gleiter
2553 Stannous Chloride Dihydrate A Novel and Efficient Catalyst for the Synthesis of gem-Dihydroperoxides from Ketones and Aldehydes D Azarifar K Khosravi F Soleimanei
2557 Synthesis of a Novel Class of Azacrown Macrocycles and Lariat Crown Ethers Containing Two 124-Triazole Rings as Subunits N Foroughifar A Mobinikhaledi S Ebrahimi
2561 Enantioselective Synthesis of the 3C-Protease Inhibitor (ndash)-Thysanone by a StauntonndashWeinreb Annulation Strategy J Sperry T Y Yuen M A Brimble
2570 Stereoselective Synthesis of Unnatural β-Amino Acids from Nitroethane via 56-Dihydro-4H-12-oxazin-3-ylacetates A Yu Sukhorukov A V Lesiv O L Eliseev Y A Khomutova S L Ioffe
2579 A Versatile Unexpected One-Pot Regioselective Synthesis of a New Class of 13-Diazepinoindolones by Reaction of Pyranoindolones with Monosubstituted Ureas D Livadiotou C A Tsoleridis J Stephanidou-Stephanatou
2584 Synthesis of a Trisaccharide and a Tetrasaccharide from the Cell-Wall Lipopolysaccharides of Azospirillum brasilense S17 S Pandey S Ghosh A K Misra
2591 Synthesis of Isoindoline Nitroxides by Electrocyclic Reactions T Kaacutelai J Jekı K Hideg
2596 Glycosylations of Tertiary Alcohols Synthesis of Fully Protected Disaccharides with Sterically Demanding Groups Attached to the Sugar Core A Holkenbrink J B Vicente D B Werz
2605 Copper-Catalyzed [13]-Dipolar Cycloaddition for the Synthesis of Macrocycles Containing Acyclic Aromatic and Steroidal Moieties G V Latyshev M S Baranom A V Kazantsev A D Averin N V Lukashev I P Beletskaya
2616 Aryl Ring Migration Reaction in the Synthesis of 24-Diaryl-4H-31-benzothiazines A V Butin F A Tsiunchik V T Abaev A V Gutnov D A Cheshkov
2627 Hydrogenation of β-N-Substituted and β-NN-Disubstituted Enamino Esters in the Presence of Iridium(I) Catalyst H Hebbache Z Hank C Bruneau J-L Renaud
2634 Stereoselective Olefination Reactions Promoted by Rieke Manganese J M Concelloacuten H Rodriacuteguez-Solla V del Amo P Diacuteaz
2646 Synthesis of Piperidinones through a Radical Cascade E Godineau Y Landais
2650 Asymmetric Organic Synthesis with Enzymes Edited by V Gotor I Alfonso E Garciacutea-Urdiales Reviewed by Steve Collier
XVII Forthcoming Articles
no 16 2651 Synthesis of Spirocyclic Ethers S Rosenberg R Leino 2674 Bimetallic PalladiumndashPlatinum-on-Carbon-Catalyzed HndashD Exchange
Reaction Synergistic Effect on Multiple Deuterium Incorporation T Maegawa N Ito K Oono Y Monguchi H Sajiki
2679 Efficient Copper-Catalyzed Synthesis of 2-Amino-4(3H)-quinazolinone and 2-Aminoquinazoline Derivatives X Huang H Yang H Fu R Qiao Y Zhao
2689 Synthesis and Chemoselective N- and O-Alkylation of Thiadiazolopyrimidine Nucleosides and Uridines A M L Hossion R Islam R K Kandahary T Nagamatsu
2697 Facile and Efficient Synthesis of a New Class of Indole-Substituted Pyridine Derivatives via One-Pot Multicomponent Reactions K Zhao X-P Xu S-L Zhu D-Q Shi Y Zhang S-J Ji
2709 Studies toward a Total Synthesis of Rhizoxin D Stereoselective Preparation of the C11ndashC19 Fragment S Padakanti C K Kumar E Ashok P Das
2715 A Short Synthesis of Enantiomeric Phytoprostanes B1 Type I W Perlikowska M Mikołajczyk
2719 Chemistry of Polyhalogenated Nitrobutadienes Part 7 A Novel Synthetic Access to Chlorinated Nitrile Oxides E Nutz V A Zapolrsquoskii D E Kaufmann
2725 Microwave-Assisted Silver(I)-Mediated Selective O-Alkylation of Aromatic Imidate Systems B K Singh C Cavalluzzo M De Maeyer Z Debyser V S Parmar E Van der Eycken
2729 Iodogen A Novel Reagent for the Oxidation of Urazoles under Heterogeneous Conditions A Khoramabadi A Shiri M A Zolfigol S Mallakpour
2733 An Unprecedented Synthesis of Eight-Membered-Ring Cyclic Thioimidic Esters by a Three-Component Reaction A Alizadeh R Hosseinpour
2737 A Novel Diastereoselective Synthesis of β-Phosphonato Unsaturated Thioimidates A Alizadeh N Zohreh
2741 Synthesis of 21-Benzisoxazoles by Nucleophilic Substitution of Hydrogen in Nitroarenes Activated by the Azole Ring N T Pokhodylo Y O Teslenko V S Matiychuk M D Obushak
2749 A Facile Synthesis of Two Series of Multifunctional Carbon Compounds from αα-Dihalo Ketones Using Allylsamarium Bromide X Liu S Zhang J Di
2756 Stereocontrolled Formation of Protected Aminodeoxyalditols from Simple Carbohydrate Precursors by Debenzylating Cycloetherification Y Jiang Z Fang Q Zheng H Jia J Cheng B Zheng
2761 trans-Stilbene as a Starting Material for the Synthesis of Tamoxifen Based on Palladium-Catalyzed Cross-Coupling Reactions C M Nunes J Limberger S Poersch M Seferin A L Monteiro
2766 Synthesis and Biological Evaluation of 6-Substituted Purinylcarbanucleosides with a Cyclopenta[b]thiophene Pseudosugar P Abeijoacuten J M Blanco O Caamantildeo F Fernaacutendez M D Garciacutea X Garciacutea-Mera J E Rodriacuteguez-Borges J Balzarini E De Clercq
2773 Synthesis and Electrochemical Signature of Novel Norbornyl-ferrocene Hybrids F A Khan S K Upadhyay
2778 A Regioselective TsujindashTrost Pentadienylation of 3-Allyltetronic Acid R Schobert B Barnickel
2785 Copper(I)-Catalyzed CarylndashCalkynyl Bond Formation of Aryl Iodides with Terminal Alkynes K G Thakur G Sekar
2790 Aminolysis of Epoxides Using Iridium Trichloride as an Efficient Catalyst J Agarwal A Duley R Rani R K Peddinti
2797 Preparation of Several Active N-Chloro Compounds from Trichloroisocyanuric Acid A Shiri A Khoramabadi-zad
2802 The First Mineral-Catalyzed One-Pot [3+1+2] Coupling Protocol for Multifunctionalized Fused-Ring Pyrimidines L D S Yadav A Rai
2809 Efficient Synthesis of Tetrahydro-β-carbolin-1-one and Dihydroisoquinolin-1-one Derivatives as Versatile Intermediates K E Judd M F Mahon L Caggiano
2818 A Concise Synthesis of ortho-Iodobenzyl Alcohols via Addition of ortho-Iodophenyl Grignard Reagent to Aldehydes and Ketones J Cvengroš D Stolz A Togni
XIII Forthcoming Articles
no 17 2825 Reactivity of Oxazol-5-(4H)-ones and Their Application toward Natural
Product Synthesis N M Hewlett C D Hupp J J Tepe 2840 Towards the Total Synthesis of 3-Hydroxyvibsanin E B D Schwartz
J R Denton P V Bernhardt H M L Davies C M Williams 2847 Structure Investigations of (ent)-Cladospolide D by De Novo Synthesis and
Kinetic and Thermodynamic Isomerization Y Xing J H Penn G A OrsquoDoherty
2855 New Applications of PhI(OAc)2 in Synthesis Total Synthesis and SAR Development of Potent Antitumor Natural Product PsymberinIrciniastatin A N Shao X Huang A Palani R Aslanian A Buevich J Piwinski R Huryk C Seidel-Dugan
2873 Total Synthesis of Largazole ndash Devolution of a Novel Synthetic Strategy B Wang C J Forsyth
2881 Formal Total Synthesis of Palmerolide A J Jaumlgel M E Maier 2893 Total Synthesis of Bongkrekic Acid via Sequential SuzukindashMiyaura Coupling
Reactions M Kanematsu M Shindo M Yoshida K Shishido 2905 Stereodivergent Approach to Both C28a-syn and C28a-anti Relative
Stereochemical Manifolds in the Lepadin Family via a TiCl4-Promoted G Li L J Carlson I K Sagamanova B W Slafer R P Hsung C Gilardi H M Sklenicka N Sydorenko
2915 Enantioselective Aldol Reaction of Tetrasubstituted Ketene Silyl Acetals with Achiral Aldehydes for the Construction of Asymmetric Tertiary Alcohols An Application for the Divergent Total Syntheses of Buergerinins F and G I Shiina T Iizumi Y-s Yamai Y-i Kawakita K Yokoyama Y-k Yamada
2927 Second-Generation Biomimetic Total Synthesis of Chaetominine A Coste G Karthikeyan F Couty G Evano
2935 Total Synthesis of (+)-Fostriecin and (+)-Phoslactomycin B S Shibahara M Fujino Y Tashiro N Okamoto T Esumi K Takahashi J Ishihara S Hatakeyama
2954 Stereochemical Assignments of the Chlorinated Residues in Victorin C A C Durow C Butts C L Willis
2963 Studies of the Asymmetric Total Synthesis of Clavilactone D by the lsquoLariatrsquo Cyclization Strategy T Yoshimitsu S Nojima M Hashimoto K Tsukamoto T Tanaka
2970 Total Synthesis of the Leucetta-Derived Alkaloid Calcaridine A P B Koswatta R Sivappa H V R Dias C J Lovely
2983 Formal Synthesis of Salinosporamide A Starting from D-Glucose T Momose Y Kaiya J-i Hasegawa T Sato N Chida
2992 Synthesis of Bioactive Natural Products by Asymmetric syn- and anti-Aldol Reactions A K Ghosh Z L Dawson
no 18 3003 Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural
Products B M Trost M K Brennan 3026 One-Pot Synthesis of Furo[34-b]pyridin-5(7H)-ones from 2-
Bromopyridine-3-carboxylic Acid and Carbonyl Compounds K Kobayashi T Kozuki H Konishi
3029 Iodocyclization of N-[2-(Methylthio)phenyl]propiolamides Selective Synthesis of 3-Iodo-15-benzothiazepin-4-ones T-S Jiang X-G Zhang J-H Li
3039 A Facile Synthetic Method for Fluorine-Containing 17-Phenanthrolines Pyridine-Ring Formation Reaction of N-Propargyl-68-bis(trifluoroacetyl)-quinolin-5-amine with Various Nucleophiles D Shibata E Okada M Hinoshita M Meacutedebielle
3047 Enantiotopic Discrimination in Palladium-Mediated Nucleophilic Substitutions on Achiral Substrates Chiral Ligand versus Chiral Nucleophile O Jacquet F Charnay J-C Fiaud J Ollivier
3051 Studies on the Chemistry of 2-[3-(2-Nitrophenyl)-2-oxopropyl]benzaldehydes Novel Syntheses of 5H-Benzo[b]carbazole-611-diones and Indolo[12-b]isoquinoline-611-diones M Fernaacutendez
3061 Studies on the C22ndashC23 Aldol Coupling of Spirangien M Lorenz N Bluhm M Kalesse
3067 One-Pot Synthesis of N-Alkyl Purine Pyrimidine and Azole Derivatives from Alcohols using Ph3PCCl4 A Rapid Route to Carboacyclic Nucleoside Synthesis M N Soltani Rad A Khalafi-Nezhad S Behrouz Z Asrari M Behrouz Z Amini
3077 Synthesis of 2-Amino-34-dihydroquinazolines and Imidazo[21-b]quinazoline-2-ones A Mishra S Batra
3089 Studies on the Reaction of Diimines with Thiourea Synthesis and Solvent-Induced cistrans-Isomerization of 135-Triazinane-2-thiones B Kaboudin T Ghasemi T Yokomatsu
3094 Suzuki Coupling of Heteroaromatic Chlorides Using Highly Electron-Donating ClickPhos Ligands S M Spinella Z-H Guan J Chen X Zhang
3099 Reaction of NN-Dioxyenamines with Anhydrides of Carboxylic and Sulfonic Acids A New Method for the Synthesis of a-Hydroxyoxime Derivatives A A Tabolin A V Lesiv S L Ioffe
3106 Directed ortho Metallation Chemistry and Phosphine Synthesis New Ligands for the SuzukindashMiyaura Reaction D B G Williams S J Evans H de Bod M S Mokhadinyana T Hughes
3113 New Functional Derivatives of 9-Phenylquinine P J Boratyński J SkarŜewski
3120 On the Synthesis of Asymmetric and Dissymmetric Amino Analogues of Troumlgerrsquos Base J Artacho K Waumlrnmark
3127 Synthesis of Polycyclic Sultams by Palladium-Catalyzed Intramolecular Cyclization K C Majumdar S Mondal N De
3136 Synthesis of Functionalized L-Cysteine and L-Methionine by Reaction with Electron-Deficient Acetylenes B A Trofimov A G Malrsquokina O A Shemyakina V V Nosyreva A P Borisova S S Khutsishvili L B Krivdin
3143 A lsquoClickrsquo Approach to the Synthesis of 3-[2-(1-Alkyltriazol-4-yl)ethyl]indoles M Petrini R R Shaikh
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
no 15 2471 Advances in Synthetic Approaches for the Preparation of Combretastatin-
Based Anti-Cancer Agents R Singh H Kaur 2492 Synthesis of Unsymmetrical Ureas by Sulfur-Assisted Carbonylation with
Carbon Monoxide and Oxidation with Molecular Oxygen under Mild Conditions T Mizuno T Nakai M Mihara
2497 Ring-OpeningRecyclization Reactions of (Dimethylamino)propenoyl-Substituted Cyclopropanes Facile Synthesis of Halogenated Pyridin-2(1H)-ones R Zhang Y Zhou Y Liang Z Jiang D Dong
2501 Facile and Efficient Total Synthesis of Taspine B Cheng S Zhang L Zhu J Zhang Q Li A Shan L He
2505 Oligomeric Iodosylbenzene Sulfate A Convenient Hypervalent Iodine Reagent for Oxidation of Organic Sulfides and Alkenes M S Yusubov R Y Yusubova T V Funk K-W Chi V V Zhdankin
2509 Pyrrolidine-Based Organocatalysts for Enantioselective Michael Addition of Cyclohexanone to trans-β-Nitrostyrene A P Carley S Dixon J D Kilburn
2517 CundashAl Hydrotalcite An Efficient and Reusable Ligand-Free Catalyst for the Coupling of Aryl Chlorides with Aliphatic Aromatic and N(H)-Heterocyclic Amines B Sreedhar R Arundhathi P L Reddy M A Reddy M L Kantam
2523 Highly Efficient Synthesis of trans-βγ-Unsaturated a-Keto Amides C Allais T Constantieux J Rodriguez
2531 Gas-Phase Synthesis of N-Unsubstituted 3-Hydroxypyrroles and 1H-Pyrrol-3(2H)-ones L Hill G A Hunter S H Imam H McNab W J OrsquoNeill
2535 3-Hydroxy-1H-pyrrole L Hill S H Imam H McNab W J OrsquoNeill 2539 123-Thiadiazoles with Unsaturated Side Chains Synthesis
Polymerization and Photocrosslinking M Al-Smadi N Hanold H Kalbitz H Meier
2547 Synthesis of 1112-Didehydrodibenzo[ae]cycloocten-5(6H)-one A Strained Eight-Membered Alkyne S C Kornmayer F Rominger R Gleiter
2553 Stannous Chloride Dihydrate A Novel and Efficient Catalyst for the Synthesis of gem-Dihydroperoxides from Ketones and Aldehydes D Azarifar K Khosravi F Soleimanei
2557 Synthesis of a Novel Class of Azacrown Macrocycles and Lariat Crown Ethers Containing Two 124-Triazole Rings as Subunits N Foroughifar A Mobinikhaledi S Ebrahimi
2561 Enantioselective Synthesis of the 3C-Protease Inhibitor (ndash)-Thysanone by a StauntonndashWeinreb Annulation Strategy J Sperry T Y Yuen M A Brimble
2570 Stereoselective Synthesis of Unnatural β-Amino Acids from Nitroethane via 56-Dihydro-4H-12-oxazin-3-ylacetates A Yu Sukhorukov A V Lesiv O L Eliseev Y A Khomutova S L Ioffe
2579 A Versatile Unexpected One-Pot Regioselective Synthesis of a New Class of 13-Diazepinoindolones by Reaction of Pyranoindolones with Monosubstituted Ureas D Livadiotou C A Tsoleridis J Stephanidou-Stephanatou
2584 Synthesis of a Trisaccharide and a Tetrasaccharide from the Cell-Wall Lipopolysaccharides of Azospirillum brasilense S17 S Pandey S Ghosh A K Misra
2591 Synthesis of Isoindoline Nitroxides by Electrocyclic Reactions T Kaacutelai J Jekı K Hideg
2596 Glycosylations of Tertiary Alcohols Synthesis of Fully Protected Disaccharides with Sterically Demanding Groups Attached to the Sugar Core A Holkenbrink J B Vicente D B Werz
2605 Copper-Catalyzed [13]-Dipolar Cycloaddition for the Synthesis of Macrocycles Containing Acyclic Aromatic and Steroidal Moieties G V Latyshev M S Baranom A V Kazantsev A D Averin N V Lukashev I P Beletskaya
2616 Aryl Ring Migration Reaction in the Synthesis of 24-Diaryl-4H-31-benzothiazines A V Butin F A Tsiunchik V T Abaev A V Gutnov D A Cheshkov
2627 Hydrogenation of β-N-Substituted and β-NN-Disubstituted Enamino Esters in the Presence of Iridium(I) Catalyst H Hebbache Z Hank C Bruneau J-L Renaud
2634 Stereoselective Olefination Reactions Promoted by Rieke Manganese J M Concelloacuten H Rodriacuteguez-Solla V del Amo P Diacuteaz
2646 Synthesis of Piperidinones through a Radical Cascade E Godineau Y Landais
2650 Asymmetric Organic Synthesis with Enzymes Edited by V Gotor I Alfonso E Garciacutea-Urdiales Reviewed by Steve Collier
XVII Forthcoming Articles
no 16 2651 Synthesis of Spirocyclic Ethers S Rosenberg R Leino 2674 Bimetallic PalladiumndashPlatinum-on-Carbon-Catalyzed HndashD Exchange
Reaction Synergistic Effect on Multiple Deuterium Incorporation T Maegawa N Ito K Oono Y Monguchi H Sajiki
2679 Efficient Copper-Catalyzed Synthesis of 2-Amino-4(3H)-quinazolinone and 2-Aminoquinazoline Derivatives X Huang H Yang H Fu R Qiao Y Zhao
2689 Synthesis and Chemoselective N- and O-Alkylation of Thiadiazolopyrimidine Nucleosides and Uridines A M L Hossion R Islam R K Kandahary T Nagamatsu
2697 Facile and Efficient Synthesis of a New Class of Indole-Substituted Pyridine Derivatives via One-Pot Multicomponent Reactions K Zhao X-P Xu S-L Zhu D-Q Shi Y Zhang S-J Ji
2709 Studies toward a Total Synthesis of Rhizoxin D Stereoselective Preparation of the C11ndashC19 Fragment S Padakanti C K Kumar E Ashok P Das
2715 A Short Synthesis of Enantiomeric Phytoprostanes B1 Type I W Perlikowska M Mikołajczyk
2719 Chemistry of Polyhalogenated Nitrobutadienes Part 7 A Novel Synthetic Access to Chlorinated Nitrile Oxides E Nutz V A Zapolrsquoskii D E Kaufmann
2725 Microwave-Assisted Silver(I)-Mediated Selective O-Alkylation of Aromatic Imidate Systems B K Singh C Cavalluzzo M De Maeyer Z Debyser V S Parmar E Van der Eycken
2729 Iodogen A Novel Reagent for the Oxidation of Urazoles under Heterogeneous Conditions A Khoramabadi A Shiri M A Zolfigol S Mallakpour
2733 An Unprecedented Synthesis of Eight-Membered-Ring Cyclic Thioimidic Esters by a Three-Component Reaction A Alizadeh R Hosseinpour
2737 A Novel Diastereoselective Synthesis of β-Phosphonato Unsaturated Thioimidates A Alizadeh N Zohreh
2741 Synthesis of 21-Benzisoxazoles by Nucleophilic Substitution of Hydrogen in Nitroarenes Activated by the Azole Ring N T Pokhodylo Y O Teslenko V S Matiychuk M D Obushak
2749 A Facile Synthesis of Two Series of Multifunctional Carbon Compounds from αα-Dihalo Ketones Using Allylsamarium Bromide X Liu S Zhang J Di
2756 Stereocontrolled Formation of Protected Aminodeoxyalditols from Simple Carbohydrate Precursors by Debenzylating Cycloetherification Y Jiang Z Fang Q Zheng H Jia J Cheng B Zheng
2761 trans-Stilbene as a Starting Material for the Synthesis of Tamoxifen Based on Palladium-Catalyzed Cross-Coupling Reactions C M Nunes J Limberger S Poersch M Seferin A L Monteiro
2766 Synthesis and Biological Evaluation of 6-Substituted Purinylcarbanucleosides with a Cyclopenta[b]thiophene Pseudosugar P Abeijoacuten J M Blanco O Caamantildeo F Fernaacutendez M D Garciacutea X Garciacutea-Mera J E Rodriacuteguez-Borges J Balzarini E De Clercq
2773 Synthesis and Electrochemical Signature of Novel Norbornyl-ferrocene Hybrids F A Khan S K Upadhyay
2778 A Regioselective TsujindashTrost Pentadienylation of 3-Allyltetronic Acid R Schobert B Barnickel
2785 Copper(I)-Catalyzed CarylndashCalkynyl Bond Formation of Aryl Iodides with Terminal Alkynes K G Thakur G Sekar
2790 Aminolysis of Epoxides Using Iridium Trichloride as an Efficient Catalyst J Agarwal A Duley R Rani R K Peddinti
2797 Preparation of Several Active N-Chloro Compounds from Trichloroisocyanuric Acid A Shiri A Khoramabadi-zad
2802 The First Mineral-Catalyzed One-Pot [3+1+2] Coupling Protocol for Multifunctionalized Fused-Ring Pyrimidines L D S Yadav A Rai
2809 Efficient Synthesis of Tetrahydro-β-carbolin-1-one and Dihydroisoquinolin-1-one Derivatives as Versatile Intermediates K E Judd M F Mahon L Caggiano
2818 A Concise Synthesis of ortho-Iodobenzyl Alcohols via Addition of ortho-Iodophenyl Grignard Reagent to Aldehydes and Ketones J Cvengroš D Stolz A Togni
XIII Forthcoming Articles
no 17 2825 Reactivity of Oxazol-5-(4H)-ones and Their Application toward Natural
Product Synthesis N M Hewlett C D Hupp J J Tepe 2840 Towards the Total Synthesis of 3-Hydroxyvibsanin E B D Schwartz
J R Denton P V Bernhardt H M L Davies C M Williams 2847 Structure Investigations of (ent)-Cladospolide D by De Novo Synthesis and
Kinetic and Thermodynamic Isomerization Y Xing J H Penn G A OrsquoDoherty
2855 New Applications of PhI(OAc)2 in Synthesis Total Synthesis and SAR Development of Potent Antitumor Natural Product PsymberinIrciniastatin A N Shao X Huang A Palani R Aslanian A Buevich J Piwinski R Huryk C Seidel-Dugan
2873 Total Synthesis of Largazole ndash Devolution of a Novel Synthetic Strategy B Wang C J Forsyth
2881 Formal Total Synthesis of Palmerolide A J Jaumlgel M E Maier 2893 Total Synthesis of Bongkrekic Acid via Sequential SuzukindashMiyaura Coupling
Reactions M Kanematsu M Shindo M Yoshida K Shishido 2905 Stereodivergent Approach to Both C28a-syn and C28a-anti Relative
Stereochemical Manifolds in the Lepadin Family via a TiCl4-Promoted G Li L J Carlson I K Sagamanova B W Slafer R P Hsung C Gilardi H M Sklenicka N Sydorenko
2915 Enantioselective Aldol Reaction of Tetrasubstituted Ketene Silyl Acetals with Achiral Aldehydes for the Construction of Asymmetric Tertiary Alcohols An Application for the Divergent Total Syntheses of Buergerinins F and G I Shiina T Iizumi Y-s Yamai Y-i Kawakita K Yokoyama Y-k Yamada
2927 Second-Generation Biomimetic Total Synthesis of Chaetominine A Coste G Karthikeyan F Couty G Evano
2935 Total Synthesis of (+)-Fostriecin and (+)-Phoslactomycin B S Shibahara M Fujino Y Tashiro N Okamoto T Esumi K Takahashi J Ishihara S Hatakeyama
2954 Stereochemical Assignments of the Chlorinated Residues in Victorin C A C Durow C Butts C L Willis
2963 Studies of the Asymmetric Total Synthesis of Clavilactone D by the lsquoLariatrsquo Cyclization Strategy T Yoshimitsu S Nojima M Hashimoto K Tsukamoto T Tanaka
2970 Total Synthesis of the Leucetta-Derived Alkaloid Calcaridine A P B Koswatta R Sivappa H V R Dias C J Lovely
2983 Formal Synthesis of Salinosporamide A Starting from D-Glucose T Momose Y Kaiya J-i Hasegawa T Sato N Chida
2992 Synthesis of Bioactive Natural Products by Asymmetric syn- and anti-Aldol Reactions A K Ghosh Z L Dawson
no 18 3003 Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural
Products B M Trost M K Brennan 3026 One-Pot Synthesis of Furo[34-b]pyridin-5(7H)-ones from 2-
Bromopyridine-3-carboxylic Acid and Carbonyl Compounds K Kobayashi T Kozuki H Konishi
3029 Iodocyclization of N-[2-(Methylthio)phenyl]propiolamides Selective Synthesis of 3-Iodo-15-benzothiazepin-4-ones T-S Jiang X-G Zhang J-H Li
3039 A Facile Synthetic Method for Fluorine-Containing 17-Phenanthrolines Pyridine-Ring Formation Reaction of N-Propargyl-68-bis(trifluoroacetyl)-quinolin-5-amine with Various Nucleophiles D Shibata E Okada M Hinoshita M Meacutedebielle
3047 Enantiotopic Discrimination in Palladium-Mediated Nucleophilic Substitutions on Achiral Substrates Chiral Ligand versus Chiral Nucleophile O Jacquet F Charnay J-C Fiaud J Ollivier
3051 Studies on the Chemistry of 2-[3-(2-Nitrophenyl)-2-oxopropyl]benzaldehydes Novel Syntheses of 5H-Benzo[b]carbazole-611-diones and Indolo[12-b]isoquinoline-611-diones M Fernaacutendez
3061 Studies on the C22ndashC23 Aldol Coupling of Spirangien M Lorenz N Bluhm M Kalesse
3067 One-Pot Synthesis of N-Alkyl Purine Pyrimidine and Azole Derivatives from Alcohols using Ph3PCCl4 A Rapid Route to Carboacyclic Nucleoside Synthesis M N Soltani Rad A Khalafi-Nezhad S Behrouz Z Asrari M Behrouz Z Amini
3077 Synthesis of 2-Amino-34-dihydroquinazolines and Imidazo[21-b]quinazoline-2-ones A Mishra S Batra
3089 Studies on the Reaction of Diimines with Thiourea Synthesis and Solvent-Induced cistrans-Isomerization of 135-Triazinane-2-thiones B Kaboudin T Ghasemi T Yokomatsu
3094 Suzuki Coupling of Heteroaromatic Chlorides Using Highly Electron-Donating ClickPhos Ligands S M Spinella Z-H Guan J Chen X Zhang
3099 Reaction of NN-Dioxyenamines with Anhydrides of Carboxylic and Sulfonic Acids A New Method for the Synthesis of a-Hydroxyoxime Derivatives A A Tabolin A V Lesiv S L Ioffe
3106 Directed ortho Metallation Chemistry and Phosphine Synthesis New Ligands for the SuzukindashMiyaura Reaction D B G Williams S J Evans H de Bod M S Mokhadinyana T Hughes
3113 New Functional Derivatives of 9-Phenylquinine P J Boratyński J SkarŜewski
3120 On the Synthesis of Asymmetric and Dissymmetric Amino Analogues of Troumlgerrsquos Base J Artacho K Waumlrnmark
3127 Synthesis of Polycyclic Sultams by Palladium-Catalyzed Intramolecular Cyclization K C Majumdar S Mondal N De
3136 Synthesis of Functionalized L-Cysteine and L-Methionine by Reaction with Electron-Deficient Acetylenes B A Trofimov A G Malrsquokina O A Shemyakina V V Nosyreva A P Borisova S S Khutsishvili L B Krivdin
3143 A lsquoClickrsquo Approach to the Synthesis of 3-[2-(1-Alkyltriazol-4-yl)ethyl]indoles M Petrini R R Shaikh
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
2584 Synthesis of a Trisaccharide and a Tetrasaccharide from the Cell-Wall Lipopolysaccharides of Azospirillum brasilense S17 S Pandey S Ghosh A K Misra
2591 Synthesis of Isoindoline Nitroxides by Electrocyclic Reactions T Kaacutelai J Jekı K Hideg
2596 Glycosylations of Tertiary Alcohols Synthesis of Fully Protected Disaccharides with Sterically Demanding Groups Attached to the Sugar Core A Holkenbrink J B Vicente D B Werz
2605 Copper-Catalyzed [13]-Dipolar Cycloaddition for the Synthesis of Macrocycles Containing Acyclic Aromatic and Steroidal Moieties G V Latyshev M S Baranom A V Kazantsev A D Averin N V Lukashev I P Beletskaya
2616 Aryl Ring Migration Reaction in the Synthesis of 24-Diaryl-4H-31-benzothiazines A V Butin F A Tsiunchik V T Abaev A V Gutnov D A Cheshkov
2627 Hydrogenation of β-N-Substituted and β-NN-Disubstituted Enamino Esters in the Presence of Iridium(I) Catalyst H Hebbache Z Hank C Bruneau J-L Renaud
2634 Stereoselective Olefination Reactions Promoted by Rieke Manganese J M Concelloacuten H Rodriacuteguez-Solla V del Amo P Diacuteaz
2646 Synthesis of Piperidinones through a Radical Cascade E Godineau Y Landais
2650 Asymmetric Organic Synthesis with Enzymes Edited by V Gotor I Alfonso E Garciacutea-Urdiales Reviewed by Steve Collier
XVII Forthcoming Articles
no 16 2651 Synthesis of Spirocyclic Ethers S Rosenberg R Leino 2674 Bimetallic PalladiumndashPlatinum-on-Carbon-Catalyzed HndashD Exchange
Reaction Synergistic Effect on Multiple Deuterium Incorporation T Maegawa N Ito K Oono Y Monguchi H Sajiki
2679 Efficient Copper-Catalyzed Synthesis of 2-Amino-4(3H)-quinazolinone and 2-Aminoquinazoline Derivatives X Huang H Yang H Fu R Qiao Y Zhao
2689 Synthesis and Chemoselective N- and O-Alkylation of Thiadiazolopyrimidine Nucleosides and Uridines A M L Hossion R Islam R K Kandahary T Nagamatsu
2697 Facile and Efficient Synthesis of a New Class of Indole-Substituted Pyridine Derivatives via One-Pot Multicomponent Reactions K Zhao X-P Xu S-L Zhu D-Q Shi Y Zhang S-J Ji
2709 Studies toward a Total Synthesis of Rhizoxin D Stereoselective Preparation of the C11ndashC19 Fragment S Padakanti C K Kumar E Ashok P Das
2715 A Short Synthesis of Enantiomeric Phytoprostanes B1 Type I W Perlikowska M Mikołajczyk
2719 Chemistry of Polyhalogenated Nitrobutadienes Part 7 A Novel Synthetic Access to Chlorinated Nitrile Oxides E Nutz V A Zapolrsquoskii D E Kaufmann
2725 Microwave-Assisted Silver(I)-Mediated Selective O-Alkylation of Aromatic Imidate Systems B K Singh C Cavalluzzo M De Maeyer Z Debyser V S Parmar E Van der Eycken
2729 Iodogen A Novel Reagent for the Oxidation of Urazoles under Heterogeneous Conditions A Khoramabadi A Shiri M A Zolfigol S Mallakpour
2733 An Unprecedented Synthesis of Eight-Membered-Ring Cyclic Thioimidic Esters by a Three-Component Reaction A Alizadeh R Hosseinpour
2737 A Novel Diastereoselective Synthesis of β-Phosphonato Unsaturated Thioimidates A Alizadeh N Zohreh
2741 Synthesis of 21-Benzisoxazoles by Nucleophilic Substitution of Hydrogen in Nitroarenes Activated by the Azole Ring N T Pokhodylo Y O Teslenko V S Matiychuk M D Obushak
2749 A Facile Synthesis of Two Series of Multifunctional Carbon Compounds from αα-Dihalo Ketones Using Allylsamarium Bromide X Liu S Zhang J Di
2756 Stereocontrolled Formation of Protected Aminodeoxyalditols from Simple Carbohydrate Precursors by Debenzylating Cycloetherification Y Jiang Z Fang Q Zheng H Jia J Cheng B Zheng
2761 trans-Stilbene as a Starting Material for the Synthesis of Tamoxifen Based on Palladium-Catalyzed Cross-Coupling Reactions C M Nunes J Limberger S Poersch M Seferin A L Monteiro
2766 Synthesis and Biological Evaluation of 6-Substituted Purinylcarbanucleosides with a Cyclopenta[b]thiophene Pseudosugar P Abeijoacuten J M Blanco O Caamantildeo F Fernaacutendez M D Garciacutea X Garciacutea-Mera J E Rodriacuteguez-Borges J Balzarini E De Clercq
2773 Synthesis and Electrochemical Signature of Novel Norbornyl-ferrocene Hybrids F A Khan S K Upadhyay
2778 A Regioselective TsujindashTrost Pentadienylation of 3-Allyltetronic Acid R Schobert B Barnickel
2785 Copper(I)-Catalyzed CarylndashCalkynyl Bond Formation of Aryl Iodides with Terminal Alkynes K G Thakur G Sekar
2790 Aminolysis of Epoxides Using Iridium Trichloride as an Efficient Catalyst J Agarwal A Duley R Rani R K Peddinti
2797 Preparation of Several Active N-Chloro Compounds from Trichloroisocyanuric Acid A Shiri A Khoramabadi-zad
2802 The First Mineral-Catalyzed One-Pot [3+1+2] Coupling Protocol for Multifunctionalized Fused-Ring Pyrimidines L D S Yadav A Rai
2809 Efficient Synthesis of Tetrahydro-β-carbolin-1-one and Dihydroisoquinolin-1-one Derivatives as Versatile Intermediates K E Judd M F Mahon L Caggiano
2818 A Concise Synthesis of ortho-Iodobenzyl Alcohols via Addition of ortho-Iodophenyl Grignard Reagent to Aldehydes and Ketones J Cvengroš D Stolz A Togni
XIII Forthcoming Articles
no 17 2825 Reactivity of Oxazol-5-(4H)-ones and Their Application toward Natural
Product Synthesis N M Hewlett C D Hupp J J Tepe 2840 Towards the Total Synthesis of 3-Hydroxyvibsanin E B D Schwartz
J R Denton P V Bernhardt H M L Davies C M Williams 2847 Structure Investigations of (ent)-Cladospolide D by De Novo Synthesis and
Kinetic and Thermodynamic Isomerization Y Xing J H Penn G A OrsquoDoherty
2855 New Applications of PhI(OAc)2 in Synthesis Total Synthesis and SAR Development of Potent Antitumor Natural Product PsymberinIrciniastatin A N Shao X Huang A Palani R Aslanian A Buevich J Piwinski R Huryk C Seidel-Dugan
2873 Total Synthesis of Largazole ndash Devolution of a Novel Synthetic Strategy B Wang C J Forsyth
2881 Formal Total Synthesis of Palmerolide A J Jaumlgel M E Maier 2893 Total Synthesis of Bongkrekic Acid via Sequential SuzukindashMiyaura Coupling
Reactions M Kanematsu M Shindo M Yoshida K Shishido 2905 Stereodivergent Approach to Both C28a-syn and C28a-anti Relative
Stereochemical Manifolds in the Lepadin Family via a TiCl4-Promoted G Li L J Carlson I K Sagamanova B W Slafer R P Hsung C Gilardi H M Sklenicka N Sydorenko
2915 Enantioselective Aldol Reaction of Tetrasubstituted Ketene Silyl Acetals with Achiral Aldehydes for the Construction of Asymmetric Tertiary Alcohols An Application for the Divergent Total Syntheses of Buergerinins F and G I Shiina T Iizumi Y-s Yamai Y-i Kawakita K Yokoyama Y-k Yamada
2927 Second-Generation Biomimetic Total Synthesis of Chaetominine A Coste G Karthikeyan F Couty G Evano
2935 Total Synthesis of (+)-Fostriecin and (+)-Phoslactomycin B S Shibahara M Fujino Y Tashiro N Okamoto T Esumi K Takahashi J Ishihara S Hatakeyama
2954 Stereochemical Assignments of the Chlorinated Residues in Victorin C A C Durow C Butts C L Willis
2963 Studies of the Asymmetric Total Synthesis of Clavilactone D by the lsquoLariatrsquo Cyclization Strategy T Yoshimitsu S Nojima M Hashimoto K Tsukamoto T Tanaka
2970 Total Synthesis of the Leucetta-Derived Alkaloid Calcaridine A P B Koswatta R Sivappa H V R Dias C J Lovely
2983 Formal Synthesis of Salinosporamide A Starting from D-Glucose T Momose Y Kaiya J-i Hasegawa T Sato N Chida
2992 Synthesis of Bioactive Natural Products by Asymmetric syn- and anti-Aldol Reactions A K Ghosh Z L Dawson
no 18 3003 Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural
Products B M Trost M K Brennan 3026 One-Pot Synthesis of Furo[34-b]pyridin-5(7H)-ones from 2-
Bromopyridine-3-carboxylic Acid and Carbonyl Compounds K Kobayashi T Kozuki H Konishi
3029 Iodocyclization of N-[2-(Methylthio)phenyl]propiolamides Selective Synthesis of 3-Iodo-15-benzothiazepin-4-ones T-S Jiang X-G Zhang J-H Li
3039 A Facile Synthetic Method for Fluorine-Containing 17-Phenanthrolines Pyridine-Ring Formation Reaction of N-Propargyl-68-bis(trifluoroacetyl)-quinolin-5-amine with Various Nucleophiles D Shibata E Okada M Hinoshita M Meacutedebielle
3047 Enantiotopic Discrimination in Palladium-Mediated Nucleophilic Substitutions on Achiral Substrates Chiral Ligand versus Chiral Nucleophile O Jacquet F Charnay J-C Fiaud J Ollivier
3051 Studies on the Chemistry of 2-[3-(2-Nitrophenyl)-2-oxopropyl]benzaldehydes Novel Syntheses of 5H-Benzo[b]carbazole-611-diones and Indolo[12-b]isoquinoline-611-diones M Fernaacutendez
3061 Studies on the C22ndashC23 Aldol Coupling of Spirangien M Lorenz N Bluhm M Kalesse
3067 One-Pot Synthesis of N-Alkyl Purine Pyrimidine and Azole Derivatives from Alcohols using Ph3PCCl4 A Rapid Route to Carboacyclic Nucleoside Synthesis M N Soltani Rad A Khalafi-Nezhad S Behrouz Z Asrari M Behrouz Z Amini
3077 Synthesis of 2-Amino-34-dihydroquinazolines and Imidazo[21-b]quinazoline-2-ones A Mishra S Batra
3089 Studies on the Reaction of Diimines with Thiourea Synthesis and Solvent-Induced cistrans-Isomerization of 135-Triazinane-2-thiones B Kaboudin T Ghasemi T Yokomatsu
3094 Suzuki Coupling of Heteroaromatic Chlorides Using Highly Electron-Donating ClickPhos Ligands S M Spinella Z-H Guan J Chen X Zhang
3099 Reaction of NN-Dioxyenamines with Anhydrides of Carboxylic and Sulfonic Acids A New Method for the Synthesis of a-Hydroxyoxime Derivatives A A Tabolin A V Lesiv S L Ioffe
3106 Directed ortho Metallation Chemistry and Phosphine Synthesis New Ligands for the SuzukindashMiyaura Reaction D B G Williams S J Evans H de Bod M S Mokhadinyana T Hughes
3113 New Functional Derivatives of 9-Phenylquinine P J Boratyński J SkarŜewski
3120 On the Synthesis of Asymmetric and Dissymmetric Amino Analogues of Troumlgerrsquos Base J Artacho K Waumlrnmark
3127 Synthesis of Polycyclic Sultams by Palladium-Catalyzed Intramolecular Cyclization K C Majumdar S Mondal N De
3136 Synthesis of Functionalized L-Cysteine and L-Methionine by Reaction with Electron-Deficient Acetylenes B A Trofimov A G Malrsquokina O A Shemyakina V V Nosyreva A P Borisova S S Khutsishvili L B Krivdin
3143 A lsquoClickrsquo Approach to the Synthesis of 3-[2-(1-Alkyltriazol-4-yl)ethyl]indoles M Petrini R R Shaikh
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
no 16 2651 Synthesis of Spirocyclic Ethers S Rosenberg R Leino 2674 Bimetallic PalladiumndashPlatinum-on-Carbon-Catalyzed HndashD Exchange
Reaction Synergistic Effect on Multiple Deuterium Incorporation T Maegawa N Ito K Oono Y Monguchi H Sajiki
2679 Efficient Copper-Catalyzed Synthesis of 2-Amino-4(3H)-quinazolinone and 2-Aminoquinazoline Derivatives X Huang H Yang H Fu R Qiao Y Zhao
2689 Synthesis and Chemoselective N- and O-Alkylation of Thiadiazolopyrimidine Nucleosides and Uridines A M L Hossion R Islam R K Kandahary T Nagamatsu
2697 Facile and Efficient Synthesis of a New Class of Indole-Substituted Pyridine Derivatives via One-Pot Multicomponent Reactions K Zhao X-P Xu S-L Zhu D-Q Shi Y Zhang S-J Ji
2709 Studies toward a Total Synthesis of Rhizoxin D Stereoselective Preparation of the C11ndashC19 Fragment S Padakanti C K Kumar E Ashok P Das
2715 A Short Synthesis of Enantiomeric Phytoprostanes B1 Type I W Perlikowska M Mikołajczyk
2719 Chemistry of Polyhalogenated Nitrobutadienes Part 7 A Novel Synthetic Access to Chlorinated Nitrile Oxides E Nutz V A Zapolrsquoskii D E Kaufmann
2725 Microwave-Assisted Silver(I)-Mediated Selective O-Alkylation of Aromatic Imidate Systems B K Singh C Cavalluzzo M De Maeyer Z Debyser V S Parmar E Van der Eycken
2729 Iodogen A Novel Reagent for the Oxidation of Urazoles under Heterogeneous Conditions A Khoramabadi A Shiri M A Zolfigol S Mallakpour
2733 An Unprecedented Synthesis of Eight-Membered-Ring Cyclic Thioimidic Esters by a Three-Component Reaction A Alizadeh R Hosseinpour
2737 A Novel Diastereoselective Synthesis of β-Phosphonato Unsaturated Thioimidates A Alizadeh N Zohreh
2741 Synthesis of 21-Benzisoxazoles by Nucleophilic Substitution of Hydrogen in Nitroarenes Activated by the Azole Ring N T Pokhodylo Y O Teslenko V S Matiychuk M D Obushak
2749 A Facile Synthesis of Two Series of Multifunctional Carbon Compounds from αα-Dihalo Ketones Using Allylsamarium Bromide X Liu S Zhang J Di
2756 Stereocontrolled Formation of Protected Aminodeoxyalditols from Simple Carbohydrate Precursors by Debenzylating Cycloetherification Y Jiang Z Fang Q Zheng H Jia J Cheng B Zheng
2761 trans-Stilbene as a Starting Material for the Synthesis of Tamoxifen Based on Palladium-Catalyzed Cross-Coupling Reactions C M Nunes J Limberger S Poersch M Seferin A L Monteiro
2766 Synthesis and Biological Evaluation of 6-Substituted Purinylcarbanucleosides with a Cyclopenta[b]thiophene Pseudosugar P Abeijoacuten J M Blanco O Caamantildeo F Fernaacutendez M D Garciacutea X Garciacutea-Mera J E Rodriacuteguez-Borges J Balzarini E De Clercq
2773 Synthesis and Electrochemical Signature of Novel Norbornyl-ferrocene Hybrids F A Khan S K Upadhyay
2778 A Regioselective TsujindashTrost Pentadienylation of 3-Allyltetronic Acid R Schobert B Barnickel
2785 Copper(I)-Catalyzed CarylndashCalkynyl Bond Formation of Aryl Iodides with Terminal Alkynes K G Thakur G Sekar
2790 Aminolysis of Epoxides Using Iridium Trichloride as an Efficient Catalyst J Agarwal A Duley R Rani R K Peddinti
2797 Preparation of Several Active N-Chloro Compounds from Trichloroisocyanuric Acid A Shiri A Khoramabadi-zad
2802 The First Mineral-Catalyzed One-Pot [3+1+2] Coupling Protocol for Multifunctionalized Fused-Ring Pyrimidines L D S Yadav A Rai
2809 Efficient Synthesis of Tetrahydro-β-carbolin-1-one and Dihydroisoquinolin-1-one Derivatives as Versatile Intermediates K E Judd M F Mahon L Caggiano
2818 A Concise Synthesis of ortho-Iodobenzyl Alcohols via Addition of ortho-Iodophenyl Grignard Reagent to Aldehydes and Ketones J Cvengroš D Stolz A Togni
XIII Forthcoming Articles
no 17 2825 Reactivity of Oxazol-5-(4H)-ones and Their Application toward Natural
Product Synthesis N M Hewlett C D Hupp J J Tepe 2840 Towards the Total Synthesis of 3-Hydroxyvibsanin E B D Schwartz
J R Denton P V Bernhardt H M L Davies C M Williams 2847 Structure Investigations of (ent)-Cladospolide D by De Novo Synthesis and
Kinetic and Thermodynamic Isomerization Y Xing J H Penn G A OrsquoDoherty
2855 New Applications of PhI(OAc)2 in Synthesis Total Synthesis and SAR Development of Potent Antitumor Natural Product PsymberinIrciniastatin A N Shao X Huang A Palani R Aslanian A Buevich J Piwinski R Huryk C Seidel-Dugan
2873 Total Synthesis of Largazole ndash Devolution of a Novel Synthetic Strategy B Wang C J Forsyth
2881 Formal Total Synthesis of Palmerolide A J Jaumlgel M E Maier 2893 Total Synthesis of Bongkrekic Acid via Sequential SuzukindashMiyaura Coupling
Reactions M Kanematsu M Shindo M Yoshida K Shishido 2905 Stereodivergent Approach to Both C28a-syn and C28a-anti Relative
Stereochemical Manifolds in the Lepadin Family via a TiCl4-Promoted G Li L J Carlson I K Sagamanova B W Slafer R P Hsung C Gilardi H M Sklenicka N Sydorenko
2915 Enantioselective Aldol Reaction of Tetrasubstituted Ketene Silyl Acetals with Achiral Aldehydes for the Construction of Asymmetric Tertiary Alcohols An Application for the Divergent Total Syntheses of Buergerinins F and G I Shiina T Iizumi Y-s Yamai Y-i Kawakita K Yokoyama Y-k Yamada
2927 Second-Generation Biomimetic Total Synthesis of Chaetominine A Coste G Karthikeyan F Couty G Evano
2935 Total Synthesis of (+)-Fostriecin and (+)-Phoslactomycin B S Shibahara M Fujino Y Tashiro N Okamoto T Esumi K Takahashi J Ishihara S Hatakeyama
2954 Stereochemical Assignments of the Chlorinated Residues in Victorin C A C Durow C Butts C L Willis
2963 Studies of the Asymmetric Total Synthesis of Clavilactone D by the lsquoLariatrsquo Cyclization Strategy T Yoshimitsu S Nojima M Hashimoto K Tsukamoto T Tanaka
2970 Total Synthesis of the Leucetta-Derived Alkaloid Calcaridine A P B Koswatta R Sivappa H V R Dias C J Lovely
2983 Formal Synthesis of Salinosporamide A Starting from D-Glucose T Momose Y Kaiya J-i Hasegawa T Sato N Chida
2992 Synthesis of Bioactive Natural Products by Asymmetric syn- and anti-Aldol Reactions A K Ghosh Z L Dawson
no 18 3003 Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural
Products B M Trost M K Brennan 3026 One-Pot Synthesis of Furo[34-b]pyridin-5(7H)-ones from 2-
Bromopyridine-3-carboxylic Acid and Carbonyl Compounds K Kobayashi T Kozuki H Konishi
3029 Iodocyclization of N-[2-(Methylthio)phenyl]propiolamides Selective Synthesis of 3-Iodo-15-benzothiazepin-4-ones T-S Jiang X-G Zhang J-H Li
3039 A Facile Synthetic Method for Fluorine-Containing 17-Phenanthrolines Pyridine-Ring Formation Reaction of N-Propargyl-68-bis(trifluoroacetyl)-quinolin-5-amine with Various Nucleophiles D Shibata E Okada M Hinoshita M Meacutedebielle
3047 Enantiotopic Discrimination in Palladium-Mediated Nucleophilic Substitutions on Achiral Substrates Chiral Ligand versus Chiral Nucleophile O Jacquet F Charnay J-C Fiaud J Ollivier
3051 Studies on the Chemistry of 2-[3-(2-Nitrophenyl)-2-oxopropyl]benzaldehydes Novel Syntheses of 5H-Benzo[b]carbazole-611-diones and Indolo[12-b]isoquinoline-611-diones M Fernaacutendez
3061 Studies on the C22ndashC23 Aldol Coupling of Spirangien M Lorenz N Bluhm M Kalesse
3067 One-Pot Synthesis of N-Alkyl Purine Pyrimidine and Azole Derivatives from Alcohols using Ph3PCCl4 A Rapid Route to Carboacyclic Nucleoside Synthesis M N Soltani Rad A Khalafi-Nezhad S Behrouz Z Asrari M Behrouz Z Amini
3077 Synthesis of 2-Amino-34-dihydroquinazolines and Imidazo[21-b]quinazoline-2-ones A Mishra S Batra
3089 Studies on the Reaction of Diimines with Thiourea Synthesis and Solvent-Induced cistrans-Isomerization of 135-Triazinane-2-thiones B Kaboudin T Ghasemi T Yokomatsu
3094 Suzuki Coupling of Heteroaromatic Chlorides Using Highly Electron-Donating ClickPhos Ligands S M Spinella Z-H Guan J Chen X Zhang
3099 Reaction of NN-Dioxyenamines with Anhydrides of Carboxylic and Sulfonic Acids A New Method for the Synthesis of a-Hydroxyoxime Derivatives A A Tabolin A V Lesiv S L Ioffe
3106 Directed ortho Metallation Chemistry and Phosphine Synthesis New Ligands for the SuzukindashMiyaura Reaction D B G Williams S J Evans H de Bod M S Mokhadinyana T Hughes
3113 New Functional Derivatives of 9-Phenylquinine P J Boratyński J SkarŜewski
3120 On the Synthesis of Asymmetric and Dissymmetric Amino Analogues of Troumlgerrsquos Base J Artacho K Waumlrnmark
3127 Synthesis of Polycyclic Sultams by Palladium-Catalyzed Intramolecular Cyclization K C Majumdar S Mondal N De
3136 Synthesis of Functionalized L-Cysteine and L-Methionine by Reaction with Electron-Deficient Acetylenes B A Trofimov A G Malrsquokina O A Shemyakina V V Nosyreva A P Borisova S S Khutsishvili L B Krivdin
3143 A lsquoClickrsquo Approach to the Synthesis of 3-[2-(1-Alkyltriazol-4-yl)ethyl]indoles M Petrini R R Shaikh
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
2778 A Regioselective TsujindashTrost Pentadienylation of 3-Allyltetronic Acid R Schobert B Barnickel
2785 Copper(I)-Catalyzed CarylndashCalkynyl Bond Formation of Aryl Iodides with Terminal Alkynes K G Thakur G Sekar
2790 Aminolysis of Epoxides Using Iridium Trichloride as an Efficient Catalyst J Agarwal A Duley R Rani R K Peddinti
2797 Preparation of Several Active N-Chloro Compounds from Trichloroisocyanuric Acid A Shiri A Khoramabadi-zad
2802 The First Mineral-Catalyzed One-Pot [3+1+2] Coupling Protocol for Multifunctionalized Fused-Ring Pyrimidines L D S Yadav A Rai
2809 Efficient Synthesis of Tetrahydro-β-carbolin-1-one and Dihydroisoquinolin-1-one Derivatives as Versatile Intermediates K E Judd M F Mahon L Caggiano
2818 A Concise Synthesis of ortho-Iodobenzyl Alcohols via Addition of ortho-Iodophenyl Grignard Reagent to Aldehydes and Ketones J Cvengroš D Stolz A Togni
XIII Forthcoming Articles
no 17 2825 Reactivity of Oxazol-5-(4H)-ones and Their Application toward Natural
Product Synthesis N M Hewlett C D Hupp J J Tepe 2840 Towards the Total Synthesis of 3-Hydroxyvibsanin E B D Schwartz
J R Denton P V Bernhardt H M L Davies C M Williams 2847 Structure Investigations of (ent)-Cladospolide D by De Novo Synthesis and
Kinetic and Thermodynamic Isomerization Y Xing J H Penn G A OrsquoDoherty
2855 New Applications of PhI(OAc)2 in Synthesis Total Synthesis and SAR Development of Potent Antitumor Natural Product PsymberinIrciniastatin A N Shao X Huang A Palani R Aslanian A Buevich J Piwinski R Huryk C Seidel-Dugan
2873 Total Synthesis of Largazole ndash Devolution of a Novel Synthetic Strategy B Wang C J Forsyth
2881 Formal Total Synthesis of Palmerolide A J Jaumlgel M E Maier 2893 Total Synthesis of Bongkrekic Acid via Sequential SuzukindashMiyaura Coupling
Reactions M Kanematsu M Shindo M Yoshida K Shishido 2905 Stereodivergent Approach to Both C28a-syn and C28a-anti Relative
Stereochemical Manifolds in the Lepadin Family via a TiCl4-Promoted G Li L J Carlson I K Sagamanova B W Slafer R P Hsung C Gilardi H M Sklenicka N Sydorenko
2915 Enantioselective Aldol Reaction of Tetrasubstituted Ketene Silyl Acetals with Achiral Aldehydes for the Construction of Asymmetric Tertiary Alcohols An Application for the Divergent Total Syntheses of Buergerinins F and G I Shiina T Iizumi Y-s Yamai Y-i Kawakita K Yokoyama Y-k Yamada
2927 Second-Generation Biomimetic Total Synthesis of Chaetominine A Coste G Karthikeyan F Couty G Evano
2935 Total Synthesis of (+)-Fostriecin and (+)-Phoslactomycin B S Shibahara M Fujino Y Tashiro N Okamoto T Esumi K Takahashi J Ishihara S Hatakeyama
2954 Stereochemical Assignments of the Chlorinated Residues in Victorin C A C Durow C Butts C L Willis
2963 Studies of the Asymmetric Total Synthesis of Clavilactone D by the lsquoLariatrsquo Cyclization Strategy T Yoshimitsu S Nojima M Hashimoto K Tsukamoto T Tanaka
2970 Total Synthesis of the Leucetta-Derived Alkaloid Calcaridine A P B Koswatta R Sivappa H V R Dias C J Lovely
2983 Formal Synthesis of Salinosporamide A Starting from D-Glucose T Momose Y Kaiya J-i Hasegawa T Sato N Chida
2992 Synthesis of Bioactive Natural Products by Asymmetric syn- and anti-Aldol Reactions A K Ghosh Z L Dawson
no 18 3003 Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural
Products B M Trost M K Brennan 3026 One-Pot Synthesis of Furo[34-b]pyridin-5(7H)-ones from 2-
Bromopyridine-3-carboxylic Acid and Carbonyl Compounds K Kobayashi T Kozuki H Konishi
3029 Iodocyclization of N-[2-(Methylthio)phenyl]propiolamides Selective Synthesis of 3-Iodo-15-benzothiazepin-4-ones T-S Jiang X-G Zhang J-H Li
3039 A Facile Synthetic Method for Fluorine-Containing 17-Phenanthrolines Pyridine-Ring Formation Reaction of N-Propargyl-68-bis(trifluoroacetyl)-quinolin-5-amine with Various Nucleophiles D Shibata E Okada M Hinoshita M Meacutedebielle
3047 Enantiotopic Discrimination in Palladium-Mediated Nucleophilic Substitutions on Achiral Substrates Chiral Ligand versus Chiral Nucleophile O Jacquet F Charnay J-C Fiaud J Ollivier
3051 Studies on the Chemistry of 2-[3-(2-Nitrophenyl)-2-oxopropyl]benzaldehydes Novel Syntheses of 5H-Benzo[b]carbazole-611-diones and Indolo[12-b]isoquinoline-611-diones M Fernaacutendez
3061 Studies on the C22ndashC23 Aldol Coupling of Spirangien M Lorenz N Bluhm M Kalesse
3067 One-Pot Synthesis of N-Alkyl Purine Pyrimidine and Azole Derivatives from Alcohols using Ph3PCCl4 A Rapid Route to Carboacyclic Nucleoside Synthesis M N Soltani Rad A Khalafi-Nezhad S Behrouz Z Asrari M Behrouz Z Amini
3077 Synthesis of 2-Amino-34-dihydroquinazolines and Imidazo[21-b]quinazoline-2-ones A Mishra S Batra
3089 Studies on the Reaction of Diimines with Thiourea Synthesis and Solvent-Induced cistrans-Isomerization of 135-Triazinane-2-thiones B Kaboudin T Ghasemi T Yokomatsu
3094 Suzuki Coupling of Heteroaromatic Chlorides Using Highly Electron-Donating ClickPhos Ligands S M Spinella Z-H Guan J Chen X Zhang
3099 Reaction of NN-Dioxyenamines with Anhydrides of Carboxylic and Sulfonic Acids A New Method for the Synthesis of a-Hydroxyoxime Derivatives A A Tabolin A V Lesiv S L Ioffe
3106 Directed ortho Metallation Chemistry and Phosphine Synthesis New Ligands for the SuzukindashMiyaura Reaction D B G Williams S J Evans H de Bod M S Mokhadinyana T Hughes
3113 New Functional Derivatives of 9-Phenylquinine P J Boratyński J SkarŜewski
3120 On the Synthesis of Asymmetric and Dissymmetric Amino Analogues of Troumlgerrsquos Base J Artacho K Waumlrnmark
3127 Synthesis of Polycyclic Sultams by Palladium-Catalyzed Intramolecular Cyclization K C Majumdar S Mondal N De
3136 Synthesis of Functionalized L-Cysteine and L-Methionine by Reaction with Electron-Deficient Acetylenes B A Trofimov A G Malrsquokina O A Shemyakina V V Nosyreva A P Borisova S S Khutsishvili L B Krivdin
3143 A lsquoClickrsquo Approach to the Synthesis of 3-[2-(1-Alkyltriazol-4-yl)ethyl]indoles M Petrini R R Shaikh
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
no 17 2825 Reactivity of Oxazol-5-(4H)-ones and Their Application toward Natural
Product Synthesis N M Hewlett C D Hupp J J Tepe 2840 Towards the Total Synthesis of 3-Hydroxyvibsanin E B D Schwartz
J R Denton P V Bernhardt H M L Davies C M Williams 2847 Structure Investigations of (ent)-Cladospolide D by De Novo Synthesis and
Kinetic and Thermodynamic Isomerization Y Xing J H Penn G A OrsquoDoherty
2855 New Applications of PhI(OAc)2 in Synthesis Total Synthesis and SAR Development of Potent Antitumor Natural Product PsymberinIrciniastatin A N Shao X Huang A Palani R Aslanian A Buevich J Piwinski R Huryk C Seidel-Dugan
2873 Total Synthesis of Largazole ndash Devolution of a Novel Synthetic Strategy B Wang C J Forsyth
2881 Formal Total Synthesis of Palmerolide A J Jaumlgel M E Maier 2893 Total Synthesis of Bongkrekic Acid via Sequential SuzukindashMiyaura Coupling
Reactions M Kanematsu M Shindo M Yoshida K Shishido 2905 Stereodivergent Approach to Both C28a-syn and C28a-anti Relative
Stereochemical Manifolds in the Lepadin Family via a TiCl4-Promoted G Li L J Carlson I K Sagamanova B W Slafer R P Hsung C Gilardi H M Sklenicka N Sydorenko
2915 Enantioselective Aldol Reaction of Tetrasubstituted Ketene Silyl Acetals with Achiral Aldehydes for the Construction of Asymmetric Tertiary Alcohols An Application for the Divergent Total Syntheses of Buergerinins F and G I Shiina T Iizumi Y-s Yamai Y-i Kawakita K Yokoyama Y-k Yamada
2927 Second-Generation Biomimetic Total Synthesis of Chaetominine A Coste G Karthikeyan F Couty G Evano
2935 Total Synthesis of (+)-Fostriecin and (+)-Phoslactomycin B S Shibahara M Fujino Y Tashiro N Okamoto T Esumi K Takahashi J Ishihara S Hatakeyama
2954 Stereochemical Assignments of the Chlorinated Residues in Victorin C A C Durow C Butts C L Willis
2963 Studies of the Asymmetric Total Synthesis of Clavilactone D by the lsquoLariatrsquo Cyclization Strategy T Yoshimitsu S Nojima M Hashimoto K Tsukamoto T Tanaka
2970 Total Synthesis of the Leucetta-Derived Alkaloid Calcaridine A P B Koswatta R Sivappa H V R Dias C J Lovely
2983 Formal Synthesis of Salinosporamide A Starting from D-Glucose T Momose Y Kaiya J-i Hasegawa T Sato N Chida
2992 Synthesis of Bioactive Natural Products by Asymmetric syn- and anti-Aldol Reactions A K Ghosh Z L Dawson
no 18 3003 Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural
Products B M Trost M K Brennan 3026 One-Pot Synthesis of Furo[34-b]pyridin-5(7H)-ones from 2-
Bromopyridine-3-carboxylic Acid and Carbonyl Compounds K Kobayashi T Kozuki H Konishi
3029 Iodocyclization of N-[2-(Methylthio)phenyl]propiolamides Selective Synthesis of 3-Iodo-15-benzothiazepin-4-ones T-S Jiang X-G Zhang J-H Li
3039 A Facile Synthetic Method for Fluorine-Containing 17-Phenanthrolines Pyridine-Ring Formation Reaction of N-Propargyl-68-bis(trifluoroacetyl)-quinolin-5-amine with Various Nucleophiles D Shibata E Okada M Hinoshita M Meacutedebielle
3047 Enantiotopic Discrimination in Palladium-Mediated Nucleophilic Substitutions on Achiral Substrates Chiral Ligand versus Chiral Nucleophile O Jacquet F Charnay J-C Fiaud J Ollivier
3051 Studies on the Chemistry of 2-[3-(2-Nitrophenyl)-2-oxopropyl]benzaldehydes Novel Syntheses of 5H-Benzo[b]carbazole-611-diones and Indolo[12-b]isoquinoline-611-diones M Fernaacutendez
3061 Studies on the C22ndashC23 Aldol Coupling of Spirangien M Lorenz N Bluhm M Kalesse
3067 One-Pot Synthesis of N-Alkyl Purine Pyrimidine and Azole Derivatives from Alcohols using Ph3PCCl4 A Rapid Route to Carboacyclic Nucleoside Synthesis M N Soltani Rad A Khalafi-Nezhad S Behrouz Z Asrari M Behrouz Z Amini
3077 Synthesis of 2-Amino-34-dihydroquinazolines and Imidazo[21-b]quinazoline-2-ones A Mishra S Batra
3089 Studies on the Reaction of Diimines with Thiourea Synthesis and Solvent-Induced cistrans-Isomerization of 135-Triazinane-2-thiones B Kaboudin T Ghasemi T Yokomatsu
3094 Suzuki Coupling of Heteroaromatic Chlorides Using Highly Electron-Donating ClickPhos Ligands S M Spinella Z-H Guan J Chen X Zhang
3099 Reaction of NN-Dioxyenamines with Anhydrides of Carboxylic and Sulfonic Acids A New Method for the Synthesis of a-Hydroxyoxime Derivatives A A Tabolin A V Lesiv S L Ioffe
3106 Directed ortho Metallation Chemistry and Phosphine Synthesis New Ligands for the SuzukindashMiyaura Reaction D B G Williams S J Evans H de Bod M S Mokhadinyana T Hughes
3113 New Functional Derivatives of 9-Phenylquinine P J Boratyński J SkarŜewski
3120 On the Synthesis of Asymmetric and Dissymmetric Amino Analogues of Troumlgerrsquos Base J Artacho K Waumlrnmark
3127 Synthesis of Polycyclic Sultams by Palladium-Catalyzed Intramolecular Cyclization K C Majumdar S Mondal N De
3136 Synthesis of Functionalized L-Cysteine and L-Methionine by Reaction with Electron-Deficient Acetylenes B A Trofimov A G Malrsquokina O A Shemyakina V V Nosyreva A P Borisova S S Khutsishvili L B Krivdin
3143 A lsquoClickrsquo Approach to the Synthesis of 3-[2-(1-Alkyltriazol-4-yl)ethyl]indoles M Petrini R R Shaikh
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
no 18 3003 Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural
Products B M Trost M K Brennan 3026 One-Pot Synthesis of Furo[34-b]pyridin-5(7H)-ones from 2-
Bromopyridine-3-carboxylic Acid and Carbonyl Compounds K Kobayashi T Kozuki H Konishi
3029 Iodocyclization of N-[2-(Methylthio)phenyl]propiolamides Selective Synthesis of 3-Iodo-15-benzothiazepin-4-ones T-S Jiang X-G Zhang J-H Li
3039 A Facile Synthetic Method for Fluorine-Containing 17-Phenanthrolines Pyridine-Ring Formation Reaction of N-Propargyl-68-bis(trifluoroacetyl)-quinolin-5-amine with Various Nucleophiles D Shibata E Okada M Hinoshita M Meacutedebielle
3047 Enantiotopic Discrimination in Palladium-Mediated Nucleophilic Substitutions on Achiral Substrates Chiral Ligand versus Chiral Nucleophile O Jacquet F Charnay J-C Fiaud J Ollivier
3051 Studies on the Chemistry of 2-[3-(2-Nitrophenyl)-2-oxopropyl]benzaldehydes Novel Syntheses of 5H-Benzo[b]carbazole-611-diones and Indolo[12-b]isoquinoline-611-diones M Fernaacutendez
3061 Studies on the C22ndashC23 Aldol Coupling of Spirangien M Lorenz N Bluhm M Kalesse
3067 One-Pot Synthesis of N-Alkyl Purine Pyrimidine and Azole Derivatives from Alcohols using Ph3PCCl4 A Rapid Route to Carboacyclic Nucleoside Synthesis M N Soltani Rad A Khalafi-Nezhad S Behrouz Z Asrari M Behrouz Z Amini
3077 Synthesis of 2-Amino-34-dihydroquinazolines and Imidazo[21-b]quinazoline-2-ones A Mishra S Batra
3089 Studies on the Reaction of Diimines with Thiourea Synthesis and Solvent-Induced cistrans-Isomerization of 135-Triazinane-2-thiones B Kaboudin T Ghasemi T Yokomatsu
3094 Suzuki Coupling of Heteroaromatic Chlorides Using Highly Electron-Donating ClickPhos Ligands S M Spinella Z-H Guan J Chen X Zhang
3099 Reaction of NN-Dioxyenamines with Anhydrides of Carboxylic and Sulfonic Acids A New Method for the Synthesis of a-Hydroxyoxime Derivatives A A Tabolin A V Lesiv S L Ioffe
3106 Directed ortho Metallation Chemistry and Phosphine Synthesis New Ligands for the SuzukindashMiyaura Reaction D B G Williams S J Evans H de Bod M S Mokhadinyana T Hughes
3113 New Functional Derivatives of 9-Phenylquinine P J Boratyński J SkarŜewski
3120 On the Synthesis of Asymmetric and Dissymmetric Amino Analogues of Troumlgerrsquos Base J Artacho K Waumlrnmark
3127 Synthesis of Polycyclic Sultams by Palladium-Catalyzed Intramolecular Cyclization K C Majumdar S Mondal N De
3136 Synthesis of Functionalized L-Cysteine and L-Methionine by Reaction with Electron-Deficient Acetylenes B A Trofimov A G Malrsquokina O A Shemyakina V V Nosyreva A P Borisova S S Khutsishvili L B Krivdin
3143 A lsquoClickrsquo Approach to the Synthesis of 3-[2-(1-Alkyltriazol-4-yl)ethyl]indoles M Petrini R R Shaikh
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
3150 Efficient Microwave-Assisted Palladium-Catalyzed SuzukindashMiyaura Cross-Coupling Reactions in 5-Nitroimidazole Series M D Crozet L Zink V Remusat C Curti P Vanelle
3157 Total Synthesis of Xestodecalactone C from L-Malic Acid J S Yadav Y Gopala Rao K Ravindar B V Subba Reddy A V Narsaiah
3162 Synthesis of Dibromophakellin Dibromophakellstatin and Dibromoagelaspongin via Oxidative Cyclization of Dihydrooroidin Derivatives dibromoagelaspongin K S Feldman M D Fodor A P Skoumbourdis
3174 A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride T B Nguyen A Martel R Dhal G Dujardin
3177 Addendum and Erratum XIII Forthcoming Articles
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